Compile Data Set for Download or QSAR
maximum 50k data
Found 33 of ic50 data for polymerid = 49000595,49000596
TargetGalanin receptor type 1(Homo sapiens (Human))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50208989(CHEMBL506553)
Affinity DataIC50:  0.0790nMAssay Description:Displacement of [125I]galanin from human recombinant GAL1 receptor expressed in HEK293 cells measured after 60 mins by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalanin receptor type 1(Homo sapiens (Human))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50378616(GALANIN)
Affinity DataIC50:  0.160nMAssay Description:Binding affinity to human GAL1 receptor by radioligand displacement assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalanin receptor type 1(Homo sapiens (Human))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50378616(GALANIN)
Affinity DataIC50:  0.770nMAssay Description:Binding affinity to human GAL1 receptor by radioligand displacement assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalanin receptor type 1(RAT)
Taisho Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50149871((R)-2-((3-(biphenyl-4-yloxy)-3-(4-fluorophenyl)pro...)
Affinity DataIC50:  3nMAssay Description:Inhibition of [3H]glycine uptake at rat glycine transporter 1 expressed in african green monkey COS7 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalanin receptor type 1(RAT)
Taisho Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50256665((3S,6S,9S,12S)-3-benzyl-9,12-di-sec-butyl-6-((2S,3...)
Affinity DataIC50:  3nMAssay Description:Inhibition of [3H]glycine uptake at rat glycine transporter 1 expressed in african green monkey COS7 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalanin receptor type 1(RAT)
Taisho Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50256666((3S,6S,9S,12S)-3-benzyl-12-sec-butyl-6-((2S,3R)-3-...)
Affinity DataIC50:  10.2nMAssay Description:Inhibition of [3H]glycine uptake at rat glycine transporter 1 expressed in african green monkey COS7 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalanin receptor type 1(RAT)
Taisho Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50256705((3S,6S,9S,12S)-3-benzyl-6-((2S,3R)-3-hydroxybutan-...)
Affinity DataIC50:  11.1nMAssay Description:Inhibition of [3H]glycine uptake at rat glycine transporter 1 expressed in african green monkey COS7 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalanin receptor type 1(RAT)
Taisho Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50256704((3S,6S,9S,12S)-3-benzyl-9-sec-butyl-6-((2S,3R)-3-h...)
Affinity DataIC50:  11.4nMAssay Description:Inhibition of [3H]glycine uptake at rat glycine transporter 1 expressed in african green monkey COS7 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalanin receptor type 1(RAT)
Taisho Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50256664((S)-2-((2S,5S,8S,11S)-5-benzyl-8,11-di-sec-butyl-3...)
Affinity DataIC50:  20.4nMAssay Description:Inhibition of [3H]glycine uptake at rat glycine transporter 1 expressed in african green monkey COS7 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalanin receptor type 1(RAT)
Taisho Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50256706((3S,6S,9S,12S)-3-benzyl-6,9,12-tri-sec-butyl-1,4,7...)
Affinity DataIC50:  29.6nMAssay Description:Inhibition of [3H]glycine uptake at rat glycine transporter 1 expressed in african green monkey COS7 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalanin receptor type 1(RAT)
Taisho Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50256746((3S,6S,9S,15aR)-9-sec-butyl-6-((1-methoxy-1H-indol...)
Affinity DataIC50:  94.6nMAssay Description:Inhibition of [3H]glycine uptake at rat glycine transporter 1 expressed in african green monkey COS7 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalanin receptor type 1(Homo sapiens (Human))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50358662(CHEMBL1922003)
Affinity DataIC50:  1.30E+3nMAssay Description:Displacement of [125I]galanin from GalR1 by gamma countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalanin receptor type 1(Homo sapiens (Human))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50358673(CHEMBL1922025)
Affinity DataIC50:  2.82E+3nMAssay Description:Displacement of [125I]galanin from GalR1 by gamma countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalanin receptor type 1(Homo sapiens (Human))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50358659(CHEMBL1922000)
Affinity DataIC50:  3.35E+3nMAssay Description:Displacement of [125I]galanin from GalR1 by gamma countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalanin receptor type 1(Homo sapiens (Human))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50358669(CHEMBL1922021)
Affinity DataIC50:  3.84E+3nMAssay Description:Displacement of [125I]galanin from GalR1 by gamma countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalanin receptor type 1(Homo sapiens (Human))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50358670(CHEMBL1922022)
Affinity DataIC50:  3.84E+3nMAssay Description:Displacement of [125I]galanin from GalR1 by gamma countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalanin receptor type 1(Homo sapiens (Human))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50358660(CHEMBL1922001)
Affinity DataIC50:  3.90E+3nMAssay Description:Displacement of [125I]galanin from GalR1 by gamma countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalanin receptor type 1(Homo sapiens (Human))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50358653(CHEMBL1921993)
Affinity DataIC50:  4.60E+3nMAssay Description:Displacement of [125I]galanin from GalR1 by gamma countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalanin receptor type 1(Homo sapiens (Human))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50358655(CHEMBL1921996)
Affinity DataIC50:  5.03E+3nMAssay Description:Displacement of [125I]galanin from GalR1 by gamma countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalanin receptor type 1(Homo sapiens (Human))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50358667(CHEMBL1922016)
Affinity DataIC50:  5.48E+3nMAssay Description:Displacement of [125I]galanin from GalR1 by gamma countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalanin receptor type 1(Homo sapiens (Human))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50358657(CHEMBL1921998)
Affinity DataIC50:  5.62E+3nMAssay Description:Displacement of [125I]galanin from GalR1 by gamma countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalanin receptor type 1(Homo sapiens (Human))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50358656(CHEMBL1921997)
Affinity DataIC50:  5.93E+3nMAssay Description:Displacement of [125I]galanin from GalR1 by gamma countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalanin receptor type 1(Homo sapiens (Human))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50358661(CHEMBL1922002)
Affinity DataIC50:  6.32E+3nMAssay Description:Displacement of [125I]galanin from GalR1 by gamma countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalanin receptor type 1(Homo sapiens (Human))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50358651(CHEMBL1921991)
Affinity DataIC50:  6.77E+3nMAssay Description:Displacement of [125I]galanin from GalR1 by gamma countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalanin receptor type 1(Homo sapiens (Human))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50358668(CHEMBL1922019)
Affinity DataIC50:  6.78E+3nMAssay Description:Displacement of [125I]galanin from GalR1 by gamma countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalanin receptor type 1(Homo sapiens (Human))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50358671(CHEMBL1922023)
Affinity DataIC50:  6.82E+3nMAssay Description:Displacement of [125I]galanin from GalR1 by gamma countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalanin receptor type 1(Homo sapiens (Human))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50358658(CHEMBL1921999)
Affinity DataIC50:  6.82E+3nMAssay Description:Displacement of [125I]galanin from GalR1 by gamma countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalanin receptor type 1(Homo sapiens (Human))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50358650(CHEMBL1921989)
Affinity DataIC50:  6.90E+3nMAssay Description:Displacement of [125I]galanin from GalR1 by gamma countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalanin receptor type 1(Homo sapiens (Human))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50358648(CHEMBL1921902)
Affinity DataIC50:  8.59E+3nMAssay Description:Displacement of [125I]galanin from GalR1 by gamma countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalanin receptor type 1(Homo sapiens (Human))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50358652(CHEMBL1921992)
Affinity DataIC50:  1.28E+4nMAssay Description:Displacement of [125I]galanin from GalR1 by gamma countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalanin receptor type 1(Homo sapiens (Human))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50358672(CHEMBL1922024)
Affinity DataIC50:  1.60E+4nMAssay Description:Displacement of [125I]galanin from GalR1 by gamma countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalanin receptor type 1(Homo sapiens (Human))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50358654(CHEMBL1921995)
Affinity DataIC50:  2.75E+4nMAssay Description:Displacement of [125I]galanin from GalR1 by gamma countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalanin receptor type 1(Homo sapiens (Human))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50358649(CHEMBL1921903)
Affinity DataIC50:  3.49E+4nMAssay Description:Displacement of [125I]galanin from GalR1 by gamma countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed