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Found 968 of ic50 for UniProtKB: P32300
TargetDelta-type opioid receptor(MOUSE)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50422795(CHEMBL202585)
Affinity DataIC50:  0.00100nMAssay Description:Agonist activity at delta opioid receptor in mouse vas deferensMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(MOUSE)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50422811(CHEMBL204716)
Affinity DataIC50:  0.00200nMAssay Description:Agonist activity at delta opioid receptor in mouse vas deferensMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(MOUSE)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50422791(CHEMBL204480)
Affinity DataIC50:  0.00500nMAssay Description:Agonist activity at delta opioid receptor in mouse vas deferensMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(MOUSE)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50121648(2-({2-[2-Amino-3-(4-hydroxy-2,6-dimethyl-phenyl)-p...)
Affinity DataIC50:  0.0150nMAssay Description:In vitro inhibitory activity against electrically evoked contractions of in mouse vas deferens (MVD)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(MOUSE)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50043724((S)-2-({(4R,7S)-13-[(S)-2-Amino-3-(4-hydroxy-pheny...)
Affinity DataIC50:  0.0160nMAssay Description:Inhibitory potency against Opioid receptor delta 1 was determined in electrically induced smooth muscle contractions of mouse vas deferens (MVD)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(MOUSE)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50061295((S)-2-{[(4R,7S,13S)-13-[(S)-2-Amino-3-(4-hydroxy-p...)
Affinity DataIC50:  0.0160nMAssay Description:Inhibitory potency against Opioid receptor delta 1 was determined in electrically induced smooth muscle contractions of mouse vas deferens (MVD)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(MOUSE)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50422809(CHEMBL204136)
Affinity DataIC50:  0.0200nMAssay Description:Agonist activity at delta opioid receptor in mouse vas deferensMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(MOUSE)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50111905((S)-4-[(S)-2-{(S)-2-[(S)-2-Amino-3-(4-hydroxy-phen...)
Affinity DataIC50:  0.0220nMAssay Description:In vitro biological activity by electrically induced smooth muscle contractions in mouse vas deferens (Opioid receptor delta 1); inhibitory concentra...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(MOUSE)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50121645(2-[(2S)-2-amino-3-(4-hydroxy-2,6-dimethylphenyl)pr...)
Affinity DataIC50:  0.0260nMAssay Description:In vitro inhibitory activity against electrically evoked contractions of in mouse vas deferens (MVD)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(MOUSE)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50121645(2-[(2S)-2-amino-3-(4-hydroxy-2,6-dimethylphenyl)pr...)
Affinity DataIC50:  0.0260nMAssay Description:In vitro inhibitory activity against electrically evoked contractions of in mouse vas deferens (MVD)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(MOUSE)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50043721((S)-2-{[(4R,7S)-13-[(S)-2-Amino-3-(4-hydroxy-pheny...)
Affinity DataIC50:  0.0280nMAssay Description:Inhibitory concentration against delta opioid receptor of electrically induced smooth muscle contraction of mouse vas deferensMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(MOUSE)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50334989((R)-2-((S)-2-amino-3-(4-hydroxy-2,6-dimethylphenyl...)
Affinity DataIC50:  0.0290nMAssay Description:Agonist activity at delta opioid receptor in mouse vas deferens assessed as inhibition of electrically-stimulated muscle contractionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(MOUSE)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50179191((S)-N-((1H-benzo[d]imidazol-2-yl)methyl)-2-((S)-2-...)
Affinity DataIC50:  0.0350nMAssay Description:Functional bioactivity against delta opioid receptor in mouse vas deferensMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(MOUSE)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50179191((S)-N-((1H-benzo[d]imidazol-2-yl)methyl)-2-((S)-2-...)
Affinity DataIC50:  0.0350nMAssay Description:In vitro inhibitory activity against electrically evoked contractions of in mouse vas deferens (MVD)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(MOUSE)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50422804(CHEMBL202578)
Affinity DataIC50:  0.0400nMAssay Description:Agonist activity at delta opioid receptor in mouse vas deferensMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(MOUSE)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50001462(3-[(2-{2-[2-Amino-3-(4-hydroxy-phenyl)-propionylam...)
Affinity DataIC50:  0.0803nMAssay Description:Inhibition of electrically evoked contractions in mouse vas deferensMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(MOUSE)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50001468((S)-3-((S)-2-{(R)-2-[(S)-2-Amino-3-(4-hydroxy-phen...)
Affinity DataIC50:  0.110nMAssay Description:Inhibitory activity against Mouse vas deferens smooth muscleMore data for this Ligand-Target Pair
In DepthDetails Article
TargetDelta-type opioid receptor(MOUSE)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50001459(3-[(2-{2-[2-Amino-3-(4-hydroxy-phenyl)-propionylam...)
Affinity DataIC50:  0.115nMAssay Description:Inhibition of electrically evoked contractions in mouse vas deferensMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(MOUSE)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50272169((S)-3-((S)-2-((S)-2-amino-3-(4-hydroxy-2,6-dimethy...)
Affinity DataIC50:  0.120nMAssay Description:In vitro inhibitory activity against electrically evoked contractions of in mouse vas deferens (MVD)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(MOUSE)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50272169((S)-3-((S)-2-((S)-2-amino-3-(4-hydroxy-2,6-dimethy...)
Affinity DataIC50:  0.120nMAssay Description:Agonist activity at delta opioid receptor in mouse vas deferenceMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(MOUSE)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50297288((S)-4-(1H-benzo[d]imidazol-2-yloxy)-3-((S)-2-((S)-...)
Affinity DataIC50:  0.120nMAssay Description:Agonist activity at delta opioid receptor in mouse vas deferens assessed as inhibition of electrically evoked contractionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(MOUSE)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50422803(CHEMBL382024)
Affinity DataIC50:  0.126nMAssay Description:Agonist activity at delta opioid receptor in mouse vas deferensMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(MOUSE)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50010532(13-[2-Amino-3-(4-hydroxy-phenyl)-propionylamino]-7...)
Affinity DataIC50:  0.130nMAssay Description:Evaluated for inhibitory activity against Opioid receptor delta 1 of mouse vas deferens (MVD).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(MOUSE)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50179191((S)-N-((1H-benzo[d]imidazol-2-yl)methyl)-2-((S)-2-...)
Affinity DataIC50:  0.130nMAssay Description:Agonist activity at delta opioid receptor in mouse vas deferenceMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(MOUSE)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50297286(1H-benzo[d]imidazol-2-yl 2-((S)-2-((S)-2-amino-3-(...)
Affinity DataIC50:  0.130nMAssay Description:Agonist activity at delta opioid receptor in mouse vas deferens assessed as inhibition of electrically evoked contractionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(MOUSE)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50027229(CHEMBL2375157)
Affinity DataIC50:  0.130nMAssay Description:Agonist activity at delta opioid receptor by mouse vas deferens assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(MOUSE)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50009142((S)-3-((S)-2-{(S)-2-[(S)-2-Amino-3-(4-hydroxy-phen...)
Affinity DataIC50:  0.140nMAssay Description:In vitro opioid receptor delta mediated mouse vas deferens (MVD) assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(MOUSE)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50001468((S)-3-((S)-2-{(R)-2-[(S)-2-Amino-3-(4-hydroxy-phen...)
Affinity DataIC50:  0.147nMAssay Description:Inhibition of electrically evoked contractions in mouse vas deferensMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(MOUSE)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50009146((S)-4-((S)-2-{(R)-2-[(S)-2-Amino-3-(4-hydroxy-phen...)
Affinity DataIC50:  0.147nMAssay Description:Agonist activity at delta-opioid receptor in mouse vasa deferens assessed as inhibition of electrically induced contractionsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(MOUSE)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50422808(CHEMBL380737)
Affinity DataIC50:  0.158nMAssay Description:Agonist activity at delta opioid receptor in mouse vas deferensMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(MOUSE)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50001468((S)-3-((S)-2-{(R)-2-[(S)-2-Amino-3-(4-hydroxy-phen...)
Affinity DataIC50:  0.160nMAssay Description:Inhibitory concentration against delta opioid receptor of electrically induced smooth muscle contraction of mouse vas deferensMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(MOUSE)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50001459(3-[(2-{2-[2-Amino-3-(4-hydroxy-phenyl)-propionylam...)
Affinity DataIC50:  0.163nMAssay Description:Inhibition of [3H]- ]DAMGO binding to Opioid receptor mu 1 from rat brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(MOUSE)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50061292((S)-2-{[(4R,7S,13S)-13-[(S)-2-Amino-3-(4-hydroxy-p...)
Affinity DataIC50:  0.170nMAssay Description:Inhibitory potency against Opioid receptor delta 1 was determined in electrically induced smooth muscle contractions of mouse vas deferens (MVD)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(MOUSE)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50001468((S)-3-((S)-2-{(R)-2-[(S)-2-Amino-3-(4-hydroxy-phen...)
Affinity DataIC50:  0.170nMAssay Description:Functional bioactivity against delta opioid receptor in mouse vas deferensMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(MOUSE)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50096716(CHEMBL100480 | Enkephalin derivative)
Affinity DataIC50:  0.170nMAssay Description:In vitro inhibitory activity was determined against Opioid receptor delta 1 in mouse vas deferensMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(MOUSE)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50151753(1N-[6-carbamoyl-9-(4-nitrobenzyl)-8,11,14-trioxo-(...)
Affinity DataIC50:  0.180nMAssay Description:Inhibitory concentration against Delta opioid receptor of mouse vas deferensMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(MOUSE)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50061291((S)-2-{[(4R,7S,13S)-13-[(S)-2-Amino-3-(4-hydroxy-p...)
Affinity DataIC50:  0.180nMAssay Description:Inhibitory potency against Opioid receptor delta 1 was determined in electrically induced smooth muscle contractions of mouse vas deferens (MVD)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(MOUSE)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50049376(1-((S)-2-{(S)-2-[(S)-2-Amino-3-(4-hydroxy-phenyl)-...)
Affinity DataIC50:  0.190nMAssay Description:Inhibitory activity against Opioid receptor delta 1 of mouse vas deferens (MVD)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(MOUSE)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50039028(4-[(4-Allyl-2,5-dimethyl-piperazin-1-yl)-(3-hydrox...)
Affinity DataIC50:  0.200nMAssay Description:Tested for agonist activity against delta opioid receptor mouse vas deferensMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(MOUSE)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50492539(CHEMBL2408009)
Affinity DataIC50:  0.210nMAssay Description:Agonist activity at delta opioid receptor in ICR mouse vas deferens assessed as inhibition of electrically-stimulated muscle contractionMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(MOUSE)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50334990((R)-2-((S)-2-amino-3-(4-hydroxy-2,6-dimethylphenyl...)
Affinity DataIC50:  0.210nMAssay Description:Agonist activity at delta opioid receptor in mouse vas deferens assessed as inhibition of electrically-stimulated muscle contractionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(MOUSE)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50008837(CHEMBL3236674)
Affinity DataIC50:  0.220nMAssay Description:Agonist activity at delta opioid receptor in mouse vas deferens assessed as inhibition of electrically-stimulated muscle contractionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(MOUSE)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50043717(CHEMBL289006 | {(4S,7R,10S,13R)-13-[(S)-2-Amino-3-...)
Affinity DataIC50:  0.230nMAssay Description:In vitro inhibition of electrically induced smooth muscle contractions of mouse vas deferensMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(MOUSE)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50280456(CHEMBL153466 | {(4S,7R,10S,13R)-13-[(S)-2-Amino-3-...)
Affinity DataIC50:  0.230nMAssay Description:Inhibitory activity against Mouse vas deferens smooth muscleMore data for this Ligand-Target Pair
In DepthDetails Article
TargetDelta-type opioid receptor(MOUSE)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50207839(CHEMBL396356 | H-Tyr-c[cys-Gly-Phe(p-NO2)-cys]NH2)
Affinity DataIC50:  0.232nMAssay Description:Agonist activity at delta opioid receptor in mouse vas deferensMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(MOUSE)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50070386(CHEMBL3408737)
Affinity DataIC50:  0.240nMAssay Description:Agonist activity at delta opioid receptor in Swiss Webster albino mouse vas deferans assessed as inhibition of electrically-induced longitudinal musc...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(MOUSE)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50070386(CHEMBL3408737)
Affinity DataIC50:  0.240nMAssay Description:Activation of DOR in mouse vas deferensMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(MOUSE)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50043712(CHEMBL286629 | {(4S,7R,10S,13R)-13-[(S)-2-Amino-3-...)
Affinity DataIC50:  0.25nMAssay Description:In vitro inhibition of electrically induced smooth muscle contractions of mouse vas deferensMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(MOUSE)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50297287((S)-1H-benzo[d]imidazol-2-yl 2-((S)-2-((S)-2-amino...)
Affinity DataIC50:  0.260nMAssay Description:Agonist activity at delta opioid receptor in mouse vas deferens assessed as inhibition of electrically evoked contractionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(MOUSE)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50117262(12-[2-Amino-3-(4-hydroxy-phenyl)-propionylamino]-6...)
Affinity DataIC50:  0.260nMAssay Description:Ability to inhibit electrically evoked contractions of isolated muscle preparations of mouse vas deference (MVD, delta receptor)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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