Affinity DataIC50: 0.320nMAssay Description:Ability to inhibit OT-induced inositol phosphate accumulation was determined in CHO cells expressing the human OT receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 0.700nMAssay Description:Inhibition of radioligand [3H]-oxytocin binding at the oxytocin (OT) receptor in rat uterine tissueMore data for this Ligand-Target Pair
Affinity DataIC50: 1nMAssay Description:Inhibitory concentration required for antagonist activity against oxytocin receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 1.20nMAssay Description:Inhibition of radioligand [3H]-oxytocin binding at the oxytocin (OT) receptor in rat uterine tissueMore data for this Ligand-Target Pair
Affinity DataIC50: 1.30nMAssay Description:Displacement of [3H]-OT from binding to oxytocin receptor of rat uterusMore data for this Ligand-Target Pair
Affinity DataIC50: 1.40nMAssay Description:Displacement of [3H]-OT from binding to oxytocin receptor of rat uterusMore data for this Ligand-Target Pair
Affinity DataIC50: 1.70nMAssay Description:Inhibition of radioligand [3H]-oxytocin binding at the oxytocin (OT) receptor in rat uterine tissueMore data for this Ligand-Target Pair
Affinity DataIC50: 2.20nMAssay Description:Inhibition of radioligand [3H]-oxytocin binding at the oxytocin (OT) receptor in rat uterine tissueMore data for this Ligand-Target Pair
Affinity DataIC50: 2.20nMAssay Description:Concentration required to displace 50% of [3H]oxytocin from rat uterine receptor.More data for this Ligand-Target Pair
Affinity DataIC50: 2.30nMAssay Description:Inhibition of radioligand [3H]-oxytocin binding at the oxytocin (OT) receptor in rat uterine tissueMore data for this Ligand-Target Pair
Affinity DataIC50: 2.40nMAssay Description:Displacement of [3H]-OT from binding to oxytocin receptor of rat uterusMore data for this Ligand-Target Pair
Affinity DataIC50: 2.60nMAssay Description:Inhibition of radioligand [3H]-oxytocin binding at the oxytocin (OT) receptor in rat uterine tissueMore data for this Ligand-Target Pair
Affinity DataIC50: 2.70nMAssay Description:Displacement of [3H]OT from human OT receptor expressed in HEK cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 2.80nMAssay Description:Displacement of [3H]-OT from binding to oxytocin receptor of rat uterusMore data for this Ligand-Target Pair
Affinity DataIC50: 3.20nMAssay Description:Inhibition of radioligand [3H]-oxytocin binding at the oxytocin (OT) receptor in rat uterine tissueMore data for this Ligand-Target Pair
Affinity DataIC50: 3.70nMAssay Description:Agonist activity at human OTR expressed in CHO cells assessed as inhibition of oxytocin-induced calcium mobilization by FLIPR assayMore data for this Ligand-Target Pair
Affinity DataIC50: 4.10nMAssay Description:Inhibition of radioligand [3H]-oxytocin binding at the oxytocin (OT) receptor in rat uterine tissueMore data for this Ligand-Target Pair
Affinity DataIC50: 4.20nMAssay Description:Inhibition of radioligand [3H]-oxytocin binding at the oxytocin (OT) receptor in rat uterine tissueMore data for this Ligand-Target Pair
Affinity DataIC50: 4.60nMAssay Description:Antagonist activity at human OXTR expressed in CHO-K1 cells by PathHunter beta-arrestin assayMore data for this Ligand-Target Pair
Affinity DataIC50: 4.90nMAssay Description:Inhibition of radioligand [3H]-oxytocin binding at the oxytocin (OT) receptor in rat uterine tissueMore data for this Ligand-Target Pair
Affinity DataIC50: 4.90nMAssay Description:Displacement of [3H]-OT from binding to oxytocin receptor of rat uterusMore data for this Ligand-Target Pair
Affinity DataIC50: 5nMAssay Description:Inhibitory concentration required for antagonist activity against oxytocin receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 5.90nMAssay Description:Inhibition of radioligand [3H]-oxytocin binding at the oxytocin (OT) receptor in rat uterine tissueMore data for this Ligand-Target Pair
Affinity DataIC50: 6nMAssay Description:Inhibition of radioligand [3H]-oxytocin binding at the oxytocin (OT) receptor in rat uterine tissueMore data for this Ligand-Target Pair
Affinity DataIC50: 6nMAssay Description:Concentration required to displace 50% of [3H]oxytocin from rat uterine receptor.More data for this Ligand-Target Pair
Affinity DataIC50: 6.30nMAssay Description:Inhibition of radioligand [3H]-oxytocin binding at the oxytocin (OT) receptor in rat uterine tissueMore data for this Ligand-Target Pair
Affinity DataIC50: 6.70nMAssay Description:Inhibition of radioligand [3H]-oxytocin binding at the oxytocin (OT) receptor in rat uterine tissueMore data for this Ligand-Target Pair
Affinity DataIC50: 7nMAssay Description:Inhibitory activity against human Oxytocin induced intracellular Calcium mobilization in human Oxytocin receptor transfected HEK293-EBNA cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 7nMAssay Description:Inhibitory activity against human Oxytocin induced intracellular Calcium mobilization in human Oxytocin receptor transfected HEK293-EBNA cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 7nMAssay Description:Displacement of [3H]OT from human OT receptor expressed in HEK cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 7nMAssay Description:Inhibition of binding of [3H]-oxytocin to rat uterine oxytocin receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 7.60nMAssay Description:Inhibition of radioligand [3H]-oxytocin binding at the oxytocin (OT) receptor in rat uterine tissueMore data for this Ligand-Target Pair
Affinity DataIC50: 8nMAssay Description:Binding affinity towards oxytocin receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 8nMAssay Description:Inhibitory activity against human Oxytocin induced intracellular Calcium mobilization in human Oxytocin receptor transfected HEK293-EBNA cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 8.30nMAssay Description:Inhibition of radioligand [3H]-oxytocin binding at the oxytocin (OT) receptor in rat uterine tissueMore data for this Ligand-Target Pair
Affinity DataIC50: 8.30nMAssay Description:Concentration required to displace 50% of [3H]oxytocin from rat uterine receptor.More data for this Ligand-Target Pair
Affinity DataIC50: 8.40nMAssay Description:Compound was evaluated for OT receptor affinity by displacement of [3H]OT from binding sites in uterine tissue taken from pregnant ratsMore data for this Ligand-Target Pair
Affinity DataIC50: 8.90nMAssay Description:Inhibition of rat uterus OT receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 8.90nMAssay Description:Displacement of [3H]-OT from binding to oxytocin receptor of rat uterusMore data for this Ligand-Target Pair
Affinity DataIC50: 9nMAssay Description:Inhibition of binding of [3H]-oxytocin to rat uterine oxytocin receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 9.20nMAssay Description:Displacement of [3H]-OT from binding to oxytocin receptor of rat uterusMore data for this Ligand-Target Pair
Affinity DataIC50: 9.20nMAssay Description:Inhibition of rat uterus OT receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 9.20nMAssay Description:Antagonist activity at human OTR expressed in HEK293 cells assessed as decrease in calcium flux measured after 10 mins in presence of vasopressin by ...More data for this Ligand-Target Pair
Affinity DataIC50: 9.30nMAssay Description:Antagonist activity at human OTR expressed in HEK293 cells assessed as decrease in calcium flux measured after 10 mins in presence of vasopressin by ...More data for this Ligand-Target Pair
Affinity DataIC50: 10nMAssay Description:Antagonist activity at human OTR expressed in HEK293 cells assessed as decrease in calcium flux measured after 10 mins in presence of vasopressin by ...More data for this Ligand-Target Pair
Affinity DataIC50: 10nMAssay Description:Concentration required to displace 50% of [3H]oxytocin from rat uterine receptor.More data for this Ligand-Target Pair
Affinity DataIC50: 10nMAssay Description:Inhibition of binding of [3H]-oxytocin to rat uterine oxytocin receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 11nMAssay Description:Inhibition of radioligand [3H]-AVP binding to the vasopressin V2 receptor in rat kidney tissueMore data for this Ligand-Target Pair
Affinity DataIC50: 11nMAssay Description:Inhibition of radioligand [3H]-oxytocin binding at the oxytocin (OT) receptor in rat uterine tissueMore data for this Ligand-Target Pair
Affinity DataIC50: 11nMAssay Description:Inhibition of radioligand [3H]oxytocin binding at the oxytocin (OT) receptor in rat uterine tissueMore data for this Ligand-Target Pair