TargetTubulin alpha-1A chain(Sus scrofa (Pig))
University Of Manchester Institute Of Science And Technology
Curated by ChEMBL
University Of Manchester Institute Of Science And Technology
Curated by ChEMBL
Affinity DataIC50: 12nMAssay Description:Tested for inhibition of polymerization of tubulinMore data for this Ligand-Target Pair
TargetTubulin alpha-1A chain(Sus scrofa (Pig))
University Of Manchester Institute Of Science And Technology
Curated by ChEMBL
University Of Manchester Institute Of Science And Technology
Curated by ChEMBL
Affinity DataIC50: 170nMAssay Description:Ability to inhibit the GTP/glutamate-induced polymerization of tubulinMore data for this Ligand-Target Pair
TargetTubulin alpha-1A chain(Sus scrofa (Pig))
University Of Manchester Institute Of Science And Technology
Curated by ChEMBL
University Of Manchester Institute Of Science And Technology
Curated by ChEMBL
Affinity DataIC50: 220nMAssay Description:The compound was evaluated in vitro for the mammalian brain tubulin polymerization using standard assay.More data for this Ligand-Target Pair
TargetTubulin alpha-1A chain(Sus scrofa (Pig))
University Of Manchester Institute Of Science And Technology
Curated by ChEMBL
University Of Manchester Institute Of Science And Technology
Curated by ChEMBL
Affinity DataIC50: 310nMAssay Description:In vitro mammalian brain tubulin polymerization using standard assay.More data for this Ligand-Target Pair
TargetTubulin alpha-1A chain(Sus scrofa (Pig))
University Of Manchester Institute Of Science And Technology
Curated by ChEMBL
University Of Manchester Institute Of Science And Technology
Curated by ChEMBL
Affinity DataIC50: 363nMAssay Description:Inhibition of tubulin polymerization interacting at the colchicine binding site.More data for this Ligand-Target Pair
TargetTubulin alpha-1A chain(Sus scrofa (Pig))
University Of Manchester Institute Of Science And Technology
Curated by ChEMBL
University Of Manchester Institute Of Science And Technology
Curated by ChEMBL
Affinity DataIC50: 372nMAssay Description:Inhibition of tubulin polymerization interacting at the colchicine binding site.More data for this Ligand-Target Pair
TargetTubulin alpha-1A chain(Sus scrofa (Pig))
University Of Manchester Institute Of Science And Technology
Curated by ChEMBL
University Of Manchester Institute Of Science And Technology
Curated by ChEMBL
Affinity DataIC50: 380nMAssay Description:Inhibition of tubulin polymerization interacting at the colchicine binding site.More data for this Ligand-Target Pair
TargetTubulin alpha-1A chain(Sus scrofa (Pig))
University Of Manchester Institute Of Science And Technology
Curated by ChEMBL
University Of Manchester Institute Of Science And Technology
Curated by ChEMBL
Affinity DataIC50: 437nMAssay Description:Inhibition of tubulin polymerization interacting at the colchicine binding site.More data for this Ligand-Target Pair
TargetTubulin alpha-1A chain(Sus scrofa (Pig))
University Of Manchester Institute Of Science And Technology
Curated by ChEMBL
University Of Manchester Institute Of Science And Technology
Curated by ChEMBL
Affinity DataIC50: 447nMAssay Description:Inhibition of tubulin polymerization interacting at the colchicine binding site.More data for this Ligand-Target Pair
TargetTubulin alpha-1A chain(Sus scrofa (Pig))
University Of Manchester Institute Of Science And Technology
Curated by ChEMBL
University Of Manchester Institute Of Science And Technology
Curated by ChEMBL
Affinity DataIC50: 457nMAssay Description:Inhibition of tubulin polymerization interacting at the colchicine binding site.More data for this Ligand-Target Pair
TargetTubulin alpha-1A chain(Sus scrofa (Pig))
University Of Manchester Institute Of Science And Technology
Curated by ChEMBL
University Of Manchester Institute Of Science And Technology
Curated by ChEMBL
Affinity DataIC50: 460nMAssay Description:Inhibition of tubulin polymerization.(ITP)More data for this Ligand-Target Pair
TargetTubulin alpha-1A chain(Sus scrofa (Pig))
University Of Manchester Institute Of Science And Technology
Curated by ChEMBL
University Of Manchester Institute Of Science And Technology
Curated by ChEMBL
Affinity DataIC50: 468nMAssay Description:Inhibition of tubulin polymerization interacting at the colchicine binding site.More data for this Ligand-Target Pair
TargetTubulin alpha-1A chain(Sus scrofa (Pig))
University Of Manchester Institute Of Science And Technology
Curated by ChEMBL
University Of Manchester Institute Of Science And Technology
Curated by ChEMBL
Affinity DataIC50: 500nMAssay Description:Concentration that cause a 50% inhibition in tubulin assembly as measured by an increase inturbidity using microtubule assembly assayMore data for this Ligand-Target Pair
TargetTubulin alpha-1A chain(Sus scrofa (Pig))
University Of Manchester Institute Of Science And Technology
Curated by ChEMBL
University Of Manchester Institute Of Science And Technology
Curated by ChEMBL
Affinity DataIC50: 525nMAssay Description:Inhibition of tubulin polymerization interacting at the colchicine binding site.More data for this Ligand-Target Pair
TargetTubulin alpha-1A chain(Sus scrofa (Pig))
University Of Manchester Institute Of Science And Technology
Curated by ChEMBL
University Of Manchester Institute Of Science And Technology
Curated by ChEMBL
Affinity DataIC50: 525nMAssay Description:Inhibition of tubulin polymerization interacting at the colchicine binding site.More data for this Ligand-Target Pair
TargetTubulin alpha-1A chain(Sus scrofa (Pig))
University Of Manchester Institute Of Science And Technology
Curated by ChEMBL
University Of Manchester Institute Of Science And Technology
Curated by ChEMBL
Affinity DataIC50: 530nMAssay Description:Inhibition of tubulin polymerization(ITP)More data for this Ligand-Target Pair
TargetTubulin alpha-1A chain(Sus scrofa (Pig))
University Of Manchester Institute Of Science And Technology
Curated by ChEMBL
University Of Manchester Institute Of Science And Technology
Curated by ChEMBL
Affinity DataIC50: 550nMAssay Description:Inhibition of tubulin polymerization interacting at the colchicine binding site.More data for this Ligand-Target Pair
TargetTubulin alpha-1A chain(Sus scrofa (Pig))
University Of Manchester Institute Of Science And Technology
Curated by ChEMBL
University Of Manchester Institute Of Science And Technology
Curated by ChEMBL
Affinity DataIC50: 562nMAssay Description:Inhibition of tubulin polymerization interacting at the colchicine binding site.More data for this Ligand-Target Pair
TargetTubulin alpha-1A chain(Sus scrofa (Pig))
University Of Manchester Institute Of Science And Technology
Curated by ChEMBL
University Of Manchester Institute Of Science And Technology
Curated by ChEMBL
Affinity DataIC50: 575nMAssay Description:Inhibition of tubulin polymerization interacting at the colchicine binding site.More data for this Ligand-Target Pair
Affinity DataIC50: 600nMAssay Description:Effect on tubulin binding and the concentration required to cause 50% decrease in tubulin assembly at 350 nm.More data for this Ligand-Target Pair
TargetTubulin alpha-1A chain(Sus scrofa (Pig))
University Of Manchester Institute Of Science And Technology
Curated by ChEMBL
University Of Manchester Institute Of Science And Technology
Curated by ChEMBL
Affinity DataIC50: 617nMAssay Description:Inhibition of tubulin polymerization interacting at the colchicine binding site.More data for this Ligand-Target Pair
TargetTubulin alpha-1A chain(Sus scrofa (Pig))
University Of Manchester Institute Of Science And Technology
Curated by ChEMBL
University Of Manchester Institute Of Science And Technology
Curated by ChEMBL
Affinity DataIC50: 631nMAssay Description:Inhibition of tubulin polymerization interacting at the colchicine binding siteMore data for this Ligand-Target Pair
TargetTubulin alpha-1A chain(Sus scrofa (Pig))
University Of Manchester Institute Of Science And Technology
Curated by ChEMBL
University Of Manchester Institute Of Science And Technology
Curated by ChEMBL
Affinity DataIC50: 646nMAssay Description:Inhibition of tubulin polymerization interacting at the colchicine binding site.More data for this Ligand-Target Pair
TargetTubulin alpha-1A chain(Sus scrofa (Pig))
University Of Manchester Institute Of Science And Technology
Curated by ChEMBL
University Of Manchester Institute Of Science And Technology
Curated by ChEMBL
Affinity DataIC50: 646nMAssay Description:Inhibition of tubulin polymerization interacting at the colchicine binding site.More data for this Ligand-Target Pair
TargetTubulin alpha-1A chain(Sus scrofa (Pig))
University Of Manchester Institute Of Science And Technology
Curated by ChEMBL
University Of Manchester Institute Of Science And Technology
Curated by ChEMBL
Affinity DataIC50: 661nMAssay Description:Inhibition of tubulin polymerization interacting at the colchicine binding site.More data for this Ligand-Target Pair
TargetTubulin alpha-1A chain(Sus scrofa (Pig))
University Of Manchester Institute Of Science And Technology
Curated by ChEMBL
University Of Manchester Institute Of Science And Technology
Curated by ChEMBL
Affinity DataIC50: 680nMAssay Description:Inhibition of tubulin polymerization(ITP)More data for this Ligand-Target Pair
TargetTubulin alpha-1A chain(Sus scrofa (Pig))
University Of Manchester Institute Of Science And Technology
Curated by ChEMBL
University Of Manchester Institute Of Science And Technology
Curated by ChEMBL
Affinity DataIC50: 692nMAssay Description:Inhibition of tubulin polymerization interacting at the colchicine binding site.More data for this Ligand-Target Pair
TargetTubulin alpha-1A chain(Sus scrofa (Pig))
University Of Manchester Institute Of Science And Technology
Curated by ChEMBL
University Of Manchester Institute Of Science And Technology
Curated by ChEMBL
Affinity DataIC50: 724nMAssay Description:Inhibition of tubulin polymerization interacting at the colchicine binding site.More data for this Ligand-Target Pair
TargetTubulin alpha-1A chain(Sus scrofa (Pig))
University Of Manchester Institute Of Science And Technology
Curated by ChEMBL
University Of Manchester Institute Of Science And Technology
Curated by ChEMBL
Affinity DataIC50: 724nMAssay Description:Inhibition of tubulin polymerization interacting at the colchicine binding site.More data for this Ligand-Target Pair
TargetTubulin alpha-1A chain(Sus scrofa (Pig))
University Of Manchester Institute Of Science And Technology
Curated by ChEMBL
University Of Manchester Institute Of Science And Technology
Curated by ChEMBL
Affinity DataIC50: 724nMAssay Description:Inhibition of tubulin polymerization interacting at the colchicine binding site.More data for this Ligand-Target Pair
TargetTubulin alpha-1A chain(Sus scrofa (Pig))
University Of Manchester Institute Of Science And Technology
Curated by ChEMBL
University Of Manchester Institute Of Science And Technology
Curated by ChEMBL
Affinity DataIC50: 741nMAssay Description:Inhibition of tubulin polymerization interacting at the colchicine binding site.More data for this Ligand-Target Pair
TargetTubulin alpha-1A chain(Sus scrofa (Pig))
University Of Manchester Institute Of Science And Technology
Curated by ChEMBL
University Of Manchester Institute Of Science And Technology
Curated by ChEMBL
Affinity DataIC50: 759nMAssay Description:Inhibition of tubulin polymerization interacting at the colchicine binding site.More data for this Ligand-Target Pair
TargetTubulin alpha-1A chain(Sus scrofa (Pig))
University Of Manchester Institute Of Science And Technology
Curated by ChEMBL
University Of Manchester Institute Of Science And Technology
Curated by ChEMBL
Affinity DataIC50: 759nMAssay Description:Inhibition of tubulin polymerization interacting at the colchicine binding site.More data for this Ligand-Target Pair
TargetTubulin alpha-1A chain(Sus scrofa (Pig))
University Of Manchester Institute Of Science And Technology
Curated by ChEMBL
University Of Manchester Institute Of Science And Technology
Curated by ChEMBL
Affinity DataIC50: 776nMAssay Description:Inhibition of tubulin polymerization interacting at the colchicine binding site.More data for this Ligand-Target Pair
TargetTubulin alpha-1A chain(Sus scrofa (Pig))
University Of Manchester Institute Of Science And Technology
Curated by ChEMBL
University Of Manchester Institute Of Science And Technology
Curated by ChEMBL
Affinity DataIC50: 776nMAssay Description:Inhibition of tubulin polymerization interacting at the colchicine binding site.More data for this Ligand-Target Pair
TargetTubulin alpha-1A chain(Sus scrofa (Pig))
University Of Manchester Institute Of Science And Technology
Curated by ChEMBL
University Of Manchester Institute Of Science And Technology
Curated by ChEMBL
Affinity DataIC50: 794nMAssay Description:Inhibition of tubulin polymerization interacting at the colchicine binding site.More data for this Ligand-Target Pair
TargetTubulin alpha-1A chain(Sus scrofa (Pig))
University Of Manchester Institute Of Science And Technology
Curated by ChEMBL
University Of Manchester Institute Of Science And Technology
Curated by ChEMBL
Affinity DataIC50: 800nMAssay Description:Inhibition of tubulin polymerization(ITP)More data for this Ligand-Target Pair
TargetTubulin alpha-1A chain(Sus scrofa (Pig))
University Of Manchester Institute Of Science And Technology
Curated by ChEMBL
University Of Manchester Institute Of Science And Technology
Curated by ChEMBL
Affinity DataIC50: 813nMAssay Description:Inhibition of tubulin polymerization interacting at the colchicine binding site.More data for this Ligand-Target Pair
TargetTubulin alpha-1A chain(Sus scrofa (Pig))
University Of Manchester Institute Of Science And Technology
Curated by ChEMBL
University Of Manchester Institute Of Science And Technology
Curated by ChEMBL
Affinity DataIC50: 820nMAssay Description:Inhibition of tubulin polymerizationMore data for this Ligand-Target Pair
TargetTubulin alpha-1A chain(Sus scrofa (Pig))
University Of Manchester Institute Of Science And Technology
Curated by ChEMBL
University Of Manchester Institute Of Science And Technology
Curated by ChEMBL
Affinity DataIC50: 860nMAssay Description:Displacement of 5.8 uM [3H]-oncodazole from homogeneous tubulin.More data for this Ligand-Target Pair
TargetTubulin alpha-1A chain(Sus scrofa (Pig))
University Of Manchester Institute Of Science And Technology
Curated by ChEMBL
University Of Manchester Institute Of Science And Technology
Curated by ChEMBL
Affinity DataIC50: 871nMAssay Description:Inhibition of tubulin polymerization interacting at the colchicine binding site.More data for this Ligand-Target Pair
TargetTubulin alpha-1A chain(Sus scrofa (Pig))
University Of Manchester Institute Of Science And Technology
Curated by ChEMBL
University Of Manchester Institute Of Science And Technology
Curated by ChEMBL
Affinity DataIC50: 880nMAssay Description:Displacement of 5.8 uM [3H]-oncodazole from homogeneous tubulin.More data for this Ligand-Target Pair
TargetTubulin alpha-1A chain(Sus scrofa (Pig))
University Of Manchester Institute Of Science And Technology
Curated by ChEMBL
University Of Manchester Institute Of Science And Technology
Curated by ChEMBL
Affinity DataIC50: 891nMAssay Description:Inhibition of tubulin polymerization interacting at the colchicine binding site.More data for this Ligand-Target Pair
TargetTubulin alpha-1A chain(Sus scrofa (Pig))
University Of Manchester Institute Of Science And Technology
Curated by ChEMBL
University Of Manchester Institute Of Science And Technology
Curated by ChEMBL
Affinity DataIC50: 933nMAssay Description:Inhibition of tubulin polymerization interacting at the colchicine binding site.More data for this Ligand-Target Pair
TargetTubulin alpha-1A chain(Sus scrofa (Pig))
University Of Manchester Institute Of Science And Technology
Curated by ChEMBL
University Of Manchester Institute Of Science And Technology
Curated by ChEMBL
Affinity DataIC50: 955nMAssay Description:Inhibition of tubulin polymerization interacting at the colchicine binding site.More data for this Ligand-Target Pair
TargetTubulin alpha-1A chain(Sus scrofa (Pig))
University Of Manchester Institute Of Science And Technology
Curated by ChEMBL
University Of Manchester Institute Of Science And Technology
Curated by ChEMBL
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of tubulin polymerization interacting at the colchicine binding site.More data for this Ligand-Target Pair
TargetTubulin alpha-1A chain(Sus scrofa (Pig))
University Of Manchester Institute Of Science And Technology
Curated by ChEMBL
University Of Manchester Institute Of Science And Technology
Curated by ChEMBL
Affinity DataIC50: 1.00E+3nMAssay Description:Compound was evaluated for inhibition of tubulin polymerizationMore data for this Ligand-Target Pair
TargetTubulin alpha-1A chain(Sus scrofa (Pig))
University Of Manchester Institute Of Science And Technology
Curated by ChEMBL
University Of Manchester Institute Of Science And Technology
Curated by ChEMBL
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of tubulin polymerizationMore data for this Ligand-Target Pair
TargetTubulin alpha-1A chain(Sus scrofa (Pig))
University Of Manchester Institute Of Science And Technology
Curated by ChEMBL
University Of Manchester Institute Of Science And Technology
Curated by ChEMBL
Affinity DataIC50: 1.10E+3nMAssay Description:Inhibition of tubulin polymerization interacting at the colchicine binding site.More data for this Ligand-Target Pair
TargetTubulin alpha-1A chain(Sus scrofa (Pig))
University Of Manchester Institute Of Science And Technology
Curated by ChEMBL
University Of Manchester Institute Of Science And Technology
Curated by ChEMBL
Affinity DataIC50: 1.10E+3nMAssay Description:Inhibition of tubulin polymerizationMore data for this Ligand-Target Pair