TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
University Of Missouri-Columbia
Curated by ChEMBL
University Of Missouri-Columbia
Curated by ChEMBL
Affinity DataIC50: 1.47nMAssay Description:Displacement of [3H]pentazocine from sigma1 receptor in guinea pig membraneMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
University Of Missouri-Columbia
Curated by ChEMBL
University Of Missouri-Columbia
Curated by ChEMBL
Affinity DataIC50: 1.89nMAssay Description:Displacement of [3H]pentazocine from sigma1 receptor in guinea pig membrane in presence of phenytoinMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
University Of Missouri-Columbia
Curated by ChEMBL
University Of Missouri-Columbia
Curated by ChEMBL
Affinity DataIC50: 3.90nMAssay Description:Displacement of [3H](+)pentazocine from guinea-pig cerebral cortex sigma 1 receptor after 150 minsMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
University Of Missouri-Columbia
Curated by ChEMBL
University Of Missouri-Columbia
Curated by ChEMBL
Affinity DataIC50: 15.2nMAssay Description:Displacement of [3H]pentazocine from sigma1 receptor in guinea pig membrane in presence of phenytoinMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
University Of Missouri-Columbia
Curated by ChEMBL
University Of Missouri-Columbia
Curated by ChEMBL
Affinity DataIC50: 17nMAssay Description:Displacement of [3H]-(+)-pentazocine from sigma1 receptor in guinea pig brain membranes by scintillation counting methodMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
University Of Missouri-Columbia
Curated by ChEMBL
University Of Missouri-Columbia
Curated by ChEMBL
Affinity DataIC50: 232nMAssay Description:Displacement of [3H]pentazocine from sigma1 receptor in guinea pig membraneMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
University Of Missouri-Columbia
Curated by ChEMBL
University Of Missouri-Columbia
Curated by ChEMBL
Affinity DataIC50: 960nMAssay Description:Displacement of [3H]pentazocine from sigma1 receptor in guinea pig membraneMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
University Of Missouri-Columbia
Curated by ChEMBL
University Of Missouri-Columbia
Curated by ChEMBL
Affinity DataIC50: 1.09E+3nMAssay Description:Displacement of [3H]pentazocine from sigma1 receptor in guinea pig membrane in presence of phenytoinMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
University Of Missouri-Columbia
Curated by ChEMBL
University Of Missouri-Columbia
Curated by ChEMBL
Affinity DataIC50: 1.90E+3nMpH: 8.0Assay Description:Displacement of [3H]-(+)-pentazocine from sigma 1 receptor in guinea pig brain membrane at pH 8.0 at 25 degCMore data for this Ligand-Target Pair