Compile Data Set for Download or QSAR
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Found 5 of ec50 for UniProtKB: P11716
TargetRyanodine receptor 1(Oryctolagus cuniculus)
University Of California

Curated by ChEMBL
LigandPNGBDBM50191286(Bastadin-5 | CHEMBL439151 | bastadin 5)
Affinity DataEC50:  2.00E+3nMAssay Description:Displacement of [3H]ryanodine from Ry1R/FKBP12 receptor complex in rabbit sarcoplasmic reticulumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRyanodine receptor 1(Oryctolagus cuniculus)
University Of California

Curated by ChEMBL
LigandPNGBDBM50292367(15,34-O-disulfatobastadin 7 | CHEMBL509326)
Affinity DataEC50:  1.36E+4nMAssay Description:Displacement of [3H]ryanodine from Ry1R/FKBP12 receptor complex in rabbit sarcoplasmic reticulumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRyanodine receptor 1(Oryctolagus cuniculus)
University Of California

Curated by ChEMBL
LigandPNGBDBM50292368(CHEMBL498932 | bastadin 20)
Affinity DataEC50:  2.06E+4nMAssay Description:Displacement of [3H]ryanodine from Ry1R/FKBP12 receptor complex in rabbit sarcoplasmic reticulumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRyanodine receptor 1(Oryctolagus cuniculus)
University Of California

Curated by ChEMBL
LigandPNGBDBM50241985((E,Z)bastadin-19 | Bastadin-19 | CHEMBL506286 | CH...)
Affinity DataEC50: >1.00E+5nMAssay Description:Displacement of [3H]ryanodine from Ry1R/FKBP12 receptor complex in rabbit sarcoplasmic reticulumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRyanodine receptor 1(Oryctolagus cuniculus)
University Of California

Curated by ChEMBL
LigandPNGBDBM50292366(10-sulfatobastadin 3 | CHEMBL450681)
Affinity DataEC50:  1.00E+5nMAssay Description:Displacement of [3H]ryanodine from Ry1R/FKBP12 receptor complex in rabbit sarcoplasmic reticulumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed