Affinity DataIC50: 0.900nMAssay Description:Inhibition of [3H]-ATRA-Hl60 binding to Retinoic acid receptor betaMore data for this Ligand-Target Pair
Affinity DataIC50: 0.940nMAssay Description:Binding affinity for Retinoic acid receptor betaMore data for this Ligand-Target Pair
Affinity DataIC50: 2nMAssay Description:Antagonistic activity against RAR beta in transcriptional activation assay with 10 nM TTNPBMore data for this Ligand-Target Pair
Affinity DataIC50: 2.5nMAssay Description:Binding affinity for Retinoic Acid Receptor beta (RAR beta)More data for this Ligand-Target Pair
Affinity DataIC50: 4.5nMAssay Description:Binding affinity for Retinoic Acid Receptor beta (RAR beta)More data for this Ligand-Target Pair
Affinity DataIC50: 5nMAssay Description:Binding affinity against retinoic Acid beta receptor using [3H]- -9-cis-Retinoic Acid in competitive binding assayMore data for this Ligand-Target Pair
Affinity DataIC50: 6.5nMAssay Description:Antagonistic activity against RAR beta in transcriptional activation assay with 10 nM TTNPBMore data for this Ligand-Target Pair
Affinity DataIC50: 7nMAssay Description:Binding affinity against retinoic Acid beta receptor using [3H]- -9-cis-Retinoic Acid in competitive binding assayMore data for this Ligand-Target Pair
Affinity DataIC50: 7.5nMAssay Description:Antagonistic activity against RAR beta in transcriptional activation assay with 10 nM TTNPBMore data for this Ligand-Target Pair
Affinity DataIC50: 13nMAssay Description:Binding affinity against retinoic Acid beta receptor using [3H]- -9-cis-Retinoic Acid in competitive binding assayMore data for this Ligand-Target Pair
Affinity DataIC50: 15nMAssay Description:Antagonistic activity against RAR gamma in transcriptional activation assay with 3.2 nM TTNPBMore data for this Ligand-Target Pair
Affinity DataIC50: 20nMAssay Description:Antagonist activity of TTNPB (10 nM) function at retinoic acid receptor betaMore data for this Ligand-Target Pair
Affinity DataIC50: 21nMAssay Description:Binding affinity for Retinoic Acid Receptor beta (RAR beta)More data for this Ligand-Target Pair
Affinity DataIC50: 22nMAssay Description:Binding affinity towards retinoic acid receptor beta was determined using [3H]-ATRA (5 nM) as radioligandMore data for this Ligand-Target Pair
Affinity DataIC50: 22nMAssay Description:Antagonistic activity against RAR beta in transcriptional activation assay with 10 nM TTNPBMore data for this Ligand-Target Pair
Affinity DataIC50: 25nMAssay Description:Antagonist activity of TTNPB (10 nM) function at retinoic acid receptor gammaMore data for this Ligand-Target Pair
Affinity DataIC50: 36nMAssay Description:Binding affinity for Retinoic Acid Receptor beta (RAR beta)More data for this Ligand-Target Pair
Affinity DataIC50: 39nMAssay Description:Binding affinity for Retinoic Acid Receptor beta (RAR beta)More data for this Ligand-Target Pair
Affinity DataIC50: 40nMAssay Description:Antagonist activity of TTNPB (10 nM) function at retinoic acid receptor betaMore data for this Ligand-Target Pair
Affinity DataIC50: 40nMAssay Description:Displacement of radioligand from RARbeta receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 53nMAssay Description:Antagonist activity of TTNPB (10 nM) function at retinoic acid receptor betaMore data for this Ligand-Target Pair
Affinity DataIC50: 75nMAssay Description:Binding affinity against retinoic Acid beta receptor using [3H]- -9-cis-Retinoic Acid in competitive binding assayMore data for this Ligand-Target Pair
Affinity DataIC50: 100nMAssay Description:Binding affinity for Retinoic Acid Receptor beta (RAR beta)More data for this Ligand-Target Pair
Affinity DataIC50: 140nMAssay Description:Binding affinity for Retinoic Acid Receptor beta (RAR beta)More data for this Ligand-Target Pair
Affinity DataIC50: 150nMAssay Description:Binding affinity against retinoic Acid beta receptor using [3H]- -9-cis-Retinoic Acid in competitive binding assayMore data for this Ligand-Target Pair
Affinity DataIC50: 230nMAssay Description:Binding affinity for Retinoic Acid Receptor beta (RAR beta)More data for this Ligand-Target Pair
Affinity DataIC50: 290nMAssay Description:Binding affinity for Retinoic Acid Receptor beta (RAR beta)More data for this Ligand-Target Pair
Affinity DataIC50: 1.17E+3nMAssay Description:Binding affinity against retinoic Acid beta receptor using [3H]- -9-cis-Retinoic Acid in competitive binding assayMore data for this Ligand-Target Pair
Affinity DataIC50: 3.00E+3nMAssay Description:Displacement of [11,12-3H]ARTA from RARbetaMore data for this Ligand-Target Pair
Affinity DataIC50: >3.00E+3nMAssay Description:Antagonistic activity of the compound was evaluated in terms of inhibition of Retinoic acid receptor beta transactivation by ATRA (50 nM); Not detect...More data for this Ligand-Target Pair
Affinity DataIC50: 9.00E+4nMAssay Description:Displacement of [11,12-3H]ARTA from RARbetaMore data for this Ligand-Target Pair
Affinity DataIC50: 1.75E+5nMAssay Description:Displacement of [11,12-3H]ARTA from RARbetaMore data for this Ligand-Target Pair
Affinity DataIC50: 1.75E+5nMAssay Description:Displacement of [11,12-3H]ARTA from RARbetaMore data for this Ligand-Target Pair
Affinity DataIC50: 2.50E+5nMAssay Description:Displacement of [11,12-3H]ARTA from RARbetaMore data for this Ligand-Target Pair
Affinity DataIC50: 5.00E+5nMAssay Description:Displacement of [11,12-3H]ARTA from RARbetaMore data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+6nMAssay Description:Displacement of [11,12-3H]ARTA from RARbetaMore data for this Ligand-Target Pair