Compile Data Set for Download or QSAR
maximum 50k data
Found 7 of ec50 for UniProtKB: P02753
TargetRetinol-binding protein 4(Homo sapiens (Human))
National University Of Ireland

Curated by ChEMBL
LigandPNGBDBM50347597(CHEMBL60405)
Affinity DataEC50:  145nMAssay Description:Antagonist activity at His-tagged recombinant human sRBP expressed in Escherichia coli BL21(DE3) assessed as disruption of ROH-sRBP-TTR protein inter...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinol-binding protein 4(Homo sapiens (Human))
National University Of Ireland

Curated by ChEMBL
LigandPNGBDBM50347599(CHEMBL1802454)
Affinity DataEC50:  154nMAssay Description:Antagonist activity at His-tagged recombinant human sRBP expressed in Escherichia coli BL21(DE3) assessed as disruption of ROH-sRBP-TTR protein inter...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinol-binding protein 4(Homo sapiens (Human))
National University Of Ireland

Curated by ChEMBL
LigandPNGBDBM50347596(CHEMBL1803043)
Affinity DataEC50:  171nMAssay Description:Antagonist activity at His-tagged recombinant human sRBP expressed in Escherichia coli BL21(DE3) assessed as disruption of ROH-sRBP-TTR protein inter...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinol-binding protein 4(Homo sapiens (Human))
National University Of Ireland

Curated by ChEMBL
LigandPNGBDBM50347595(CHEMBL58106)
Affinity DataEC50:  245nMAssay Description:Antagonist activity at His-tagged recombinant human sRBP expressed in Escherichia coli BL21(DE3) assessed as disruption of ROH-sRBP-TTR protein inter...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinol-binding protein 4(Homo sapiens (Human))
National University Of Ireland

Curated by ChEMBL
LigandPNGBDBM50347598(CHEMBL1802450)
Affinity DataEC50:  954nMAssay Description:Antagonist activity at His-tagged recombinant human sRBP expressed in Escherichia coli BL21(DE3) assessed as disruption of ROH-sRBP-TTR protein inter...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinol-binding protein 4(Homo sapiens (Human))
National University Of Ireland

Curated by ChEMBL
LigandPNGBDBM50347594(CHEMBL1801542)
Affinity DataEC50:  1.26E+3nMAssay Description:Antagonist activity at His-tagged recombinant human sRBP expressed in Escherichia coli BL21(DE3) assessed as disruption of ROH-sRBP-TTR protein inter...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinol-binding protein 4(Homo sapiens (Human))
National University Of Ireland

Curated by ChEMBL
LigandPNGBDBM50092055((2E,4E,6E,8E)-3,7-Dimethyl-9-(2,6,6-trimethyl-cycl...)
Affinity DataEC50:  2.37E+3nMAssay Description:Antagonist activity at His-tagged recombinant human sRBP expressed in Escherichia coli BL21(DE3) assessed as disruption of ROH-sRBP-TTR protein inter...More data for this Ligand-Target Pair