BindingDB PrimarySearch_ki

Found 211 of ic50 for UniProtKB: Q9NZ08

Endoplasmic reticulum aminopeptidase 1(Homo sapiens (Human))
National Center For Scientific Research&Quot;Demokritos&Quot

Curated by ChEMBL

PNG

BDBM50076744(CHEMBL3416733)

IC50: 33nMAssay Description:Inhibition of human recombinant ERAP1 expressed in baculovirus infected Sf9 cells using L-leucine-7-amido-4-methyl coumarin as substrate after 5 to 1...More data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
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3D Structure (crystal)

Endoplasmic reticulum aminopeptidase 1(Homo sapiens (Human))
National Center For Scientific Research&Quot;Demokritos&Quot

Curated by ChEMBL

PNG

BDBM50076744(CHEMBL3416733)

IC50: 33nMAssay Description:Inhibition of recombinant human ERAP1 using L-AMC as substrate measured for 15 to 30 mins by fluorescence analysisMore data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
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3D Structure (crystal)

Endoplasmic reticulum aminopeptidase 1(Homo sapiens (Human))
National Center For Scientific Research&Quot;Demokritos&Quot

Curated by ChEMBL

PNG

BDBM50076744(CHEMBL3416733)

IC50: 33nMAssay Description:Inhibition of recombinant human ERAP1 using L-AMC as substrate incubated for 5 to 10 mins by fluorescence based assayMore data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
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3D Structure (crystal)

Endoplasmic reticulum aminopeptidase 1(Homo sapiens (Human))
National Center For Scientific Research&Quot;Demokritos&Quot

Curated by ChEMBL

PNG

BDBM50076744(CHEMBL3416733)

IC50: 33nMAssay Description:Inhibition of human recombinant ERAP1 using L-leucine 7-amido-4-methyl coumarin as substrate after 5 to 10 mins by fluorescence microplate reader met...More data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
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3D Structure (crystal)

Endoplasmic reticulum aminopeptidase 1(Homo sapiens (Human))
National Center For Scientific Research&Quot;Demokritos&Quot

Curated by ChEMBL

PNG

BDBM50245391(CHEMBL4095882)

IC50: 33nMAssay Description:Inhibition of ERAP1 (unknown origin) expressed in Hi5 cells by in vitro fluorimetric assayMore data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD antibodypedia GoogleScholar

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Endoplasmic reticulum aminopeptidase 1(Homo sapiens (Human))
National Center For Scientific Research&Quot;Demokritos&Quot

Curated by ChEMBL

PNG

BDBM50076744(CHEMBL3416733)

IC50: 33nMAssay Description:Inhibition of human recombinant ERAP1 using L-leucine 7-amido-4-methyl coumarin as substrate after 5 to 10 mins by fluorescence microplate reader met...More data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD antibodypedia GoogleScholar

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3D Structure (crystal)

Endoplasmic reticulum aminopeptidase 1(Homo sapiens (Human))
National Center For Scientific Research&Quot;Demokritos&Quot

Curated by ChEMBL

PNG

BDBM50571866(CHEMBL4862557)

IC50: 34nMAssay Description:Inhibition of wild type ERAP1 (unknown origin) using L-Rho-Succ-FKARKF as substrate preincubated for 15 mins followed by substrate addition and measu...More data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD antibodypedia GoogleScholar

Details Article PubMed

Endoplasmic reticulum aminopeptidase 1(Homo sapiens (Human))
National Center For Scientific Research&Quot;Demokritos&Quot

Curated by ChEMBL

PNG

BDBM50245396(CHEMBL4101200)

IC50: 43nMAssay Description:Inhibition of ERAP1 (unknown origin)More data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
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Endoplasmic reticulum aminopeptidase 1(Homo sapiens (Human))
National Center For Scientific Research&Quot;Demokritos&Quot

Curated by ChEMBL

PNG

BDBM50245396(CHEMBL4101200)

IC50: 43nMAssay Description:Inhibition of ERAP1 (unknown origin) expressed in Hi5 cells by in vitro fluorimetric assayMore data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
UniProtKB/SwissProt
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Endoplasmic reticulum aminopeptidase 1(Homo sapiens (Human))
National Center For Scientific Research&Quot;Demokritos&Quot

Curated by ChEMBL

PNG

BDBM50245400(CHEMBL4099107)

IC50: 48nMAssay Description:Inhibition of ERAP1 (unknown origin) expressed in Hi5 cells by in vitro fluorimetric assayMore data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
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Endoplasmic reticulum aminopeptidase 1(Homo sapiens (Human))
National Center For Scientific Research&Quot;Demokritos&Quot

Curated by ChEMBL

PNG

BDBM50076744(CHEMBL3416733)

IC50: 48nMAssay Description:Inhibition of ERAP1 (unknown origin) expressed in Hi5 cells by in vitro fluorimetric assayMore data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
UniProtKB/SwissProt
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3D Structure (crystal)

Endoplasmic reticulum aminopeptidase 1(Homo sapiens (Human))
National Center For Scientific Research&Quot;Demokritos&Quot

Curated by ChEMBL

PNG

BDBM50076744(CHEMBL3416733)

IC50: 52nMAssay Description:Inhibition of wild type ERAP1 (unknown origin) using L-Rho-Succ-FKARKF as substrate preincubated for 15 mins followed by substrate addition and measu...More data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
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3D Structure (crystal)

Endoplasmic reticulum aminopeptidase 1(Homo sapiens (Human))
National Center For Scientific Research&Quot;Demokritos&Quot

Curated by ChEMBL

PNG

BDBM50245390(CHEMBL4077855)

IC50: 65nMAssay Description:Inhibition of ERAP1 (unknown origin) expressed in Hi5 cells by in vitro fluorimetric assayMore data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
UniProtKB/SwissProt
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Endoplasmic reticulum aminopeptidase 1(Homo sapiens (Human))
National Center For Scientific Research&Quot;Demokritos&Quot

Curated by ChEMBL

PNG

BDBM50245401(CHEMBL4103640)

IC50: 71nMAssay Description:Inhibition of ERAP1 (unknown origin) expressed in Hi5 cells by in vitro fluorimetric assayMore data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
UniProtKB/SwissProt
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Endoplasmic reticulum aminopeptidase 1(Homo sapiens (Human))
National Center For Scientific Research&Quot;Demokritos&Quot

Curated by ChEMBL

PNG

BDBM50245383(CHEMBL4104383)

IC50: 98nMAssay Description:Inhibition of ERAP1 (unknown origin) expressed in Hi5 cells by in vitro fluorimetric assayMore data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
UniProtKB/SwissProt
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Endoplasmic reticulum aminopeptidase 1(Homo sapiens (Human))
National Center For Scientific Research&Quot;Demokritos&Quot

Curated by ChEMBL

PNG

BDBM50571865(CHEMBL4863142)

IC50: 99nMAssay Description:Inhibition of wild type ERAP1 (unknown origin) using L-Rho-Succ-FKARKF as substrate preincubated for 15 mins followed by substrate addition and measu...More data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD antibodypedia GoogleScholar

Details Article PubMed

Endoplasmic reticulum aminopeptidase 1(Homo sapiens (Human))
National Center For Scientific Research&Quot;Demokritos&Quot

Curated by ChEMBL

PNG

BDBM50245388(CHEMBL4081073)

IC50: 102nMAssay Description:Inhibition of ERAP1 (unknown origin) expressed in Hi5 cells by in vitro fluorimetric assayMore data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
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Endoplasmic reticulum aminopeptidase 1(Homo sapiens (Human))
National Center For Scientific Research&Quot;Demokritos&Quot

Curated by ChEMBL

PNG

BDBM50571867(CHEMBL4875461)

IC50: 115nMAssay Description:Inhibition of wild type ERAP1 (unknown origin) using L-Rho-Succ-FKARKF as substrate preincubated for 15 mins followed by substrate addition and measu...More data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD antibodypedia GoogleScholar

Details Article PubMed

Endoplasmic reticulum aminopeptidase 1(Homo sapiens (Human))
National Center For Scientific Research&Quot;Demokritos&Quot

Curated by ChEMBL

PNG

BDBM50571872(CHEMBL4864508)

IC50: 120nMAssay Description:Inhibition of wild type ERAP1 (unknown origin) using L-Rho-Succ-FKARKF as substrate preincubated for 15 mins followed by substrate addition and measu...More data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD antibodypedia GoogleScholar

Details Article PubMed

Endoplasmic reticulum aminopeptidase 1(Homo sapiens (Human))
National Center For Scientific Research&Quot;Demokritos&Quot

Curated by ChEMBL

PNG

BDBM50245399(CHEMBL4069425)

IC50: 126nMAssay Description:Inhibition of ERAP1 (unknown origin) expressed in Hi5 cells by in vitro fluorimetric assayMore data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
UniProtKB/SwissProt
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Endoplasmic reticulum aminopeptidase 1(Homo sapiens (Human))
National Center For Scientific Research&Quot;Demokritos&Quot

Curated by ChEMBL

PNG

BDBM50570849(CHEMBL4854733)

IC50: 140nMAssay Description:Inhibition of ERAP1 (unknown origin) using L-AMC as substrateMore data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD antibodypedia GoogleScholar

Details Article PubMed

Endoplasmic reticulum aminopeptidase 1(Homo sapiens (Human))
National Center For Scientific Research&Quot;Demokritos&Quot

Curated by ChEMBL

PNG

BDBM50570849(CHEMBL4854733)

IC50: 141nMAssay Description:Inhibition of ERAP1 (unknown origin) using L-AMC as substrateMore data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD antibodypedia GoogleScholar

Details Article PubMed

Endoplasmic reticulum aminopeptidase 1(Homo sapiens (Human))
National Center For Scientific Research&Quot;Demokritos&Quot

Curated by ChEMBL

PNG

BDBM50245389(CHEMBL4085707)

IC50: 143nMAssay Description:Inhibition of ERAP1 (unknown origin) expressed in Hi5 cells by in vitro fluorimetric assayMore data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD antibodypedia GoogleScholar

CHEMBL PC cid PC sid Similars

Details Article PubMed

Endoplasmic reticulum aminopeptidase 1(Homo sapiens (Human))
National Center For Scientific Research&Quot;Demokritos&Quot

Curated by ChEMBL

PNG

BDBM50571874(CHEMBL4855038)

IC50: 151nMAssay Description:Inhibition of wild type ERAP1 (unknown origin) using L-Rho-Succ-FKARKF as substrate preincubated for 15 mins followed by substrate addition and measu...More data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD antibodypedia GoogleScholar

Details Article PubMed

Endoplasmic reticulum aminopeptidase 1(Homo sapiens (Human))
National Center For Scientific Research&Quot;Demokritos&Quot

Curated by ChEMBL

PNG

BDBM50245348(CHEMBL4099693)

IC50: 155nMAssay Description:Inhibition of ERAP1 (unknown origin) expressed in Hi5 cells by in vitro fluorimetric assayMore data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD antibodypedia GoogleScholar

CHEMBL PC cid PC sid Similars

Details Article PubMed

Endoplasmic reticulum aminopeptidase 1(Homo sapiens (Human))
National Center For Scientific Research&Quot;Demokritos&Quot

Curated by ChEMBL

PNG

BDBM50245382(CHEMBL4080145)

IC50: 178nMAssay Description:Inhibition of ERAP1 (unknown origin) expressed in Hi5 cells by in vitro fluorimetric assayMore data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD antibodypedia GoogleScholar

CHEMBL PC cid PC sid Similars

Details Article PubMed

Endoplasmic reticulum aminopeptidase 1(Homo sapiens (Human))
National Center For Scientific Research&Quot;Demokritos&Quot

Curated by ChEMBL

PNG

BDBM50076744(CHEMBL3416733)

IC50: 186nMAssay Description:Inhibition of ERAP1 (unknown origin) using L-AMC as substrateMore data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
UniProtKB/SwissProt
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3D Structure (crystal)

Endoplasmic reticulum aminopeptidase 1(Homo sapiens (Human))
National Center For Scientific Research&Quot;Demokritos&Quot

Curated by ChEMBL

PNG

BDBM50076744(CHEMBL3416733)

IC50: 190nMAssay Description:Inhibition of ERAP1 (unknown origin) using L-AMC as substrateMore data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD antibodypedia GoogleScholar

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3D Structure (crystal)

Endoplasmic reticulum aminopeptidase 1(Homo sapiens (Human))
National Center For Scientific Research&Quot;Demokritos&Quot

Curated by ChEMBL

PNG

BDBM50571868(CHEMBL4854530)

IC50: 262nMAssay Description:Inhibition of wild type ERAP1 (unknown origin) using L-Rho-Succ-FKARKF as substrate preincubated for 15 mins followed by substrate addition and measu...More data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD antibodypedia GoogleScholar

Details Article PubMed

Endoplasmic reticulum aminopeptidase 1(Homo sapiens (Human))
National Center For Scientific Research&Quot;Demokritos&Quot

Curated by ChEMBL

PNG

BDBM50571862(CHEMBL4847534)

IC50: 275nMAssay Description:Inhibition of wild type ERAP1 (unknown origin) using L-Rho-Succ-FKARKF as substrate preincubated for 15 mins followed by substrate addition and measu...More data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD antibodypedia GoogleScholar

Details Article PubMed

Endoplasmic reticulum aminopeptidase 1(Homo sapiens (Human))
National Center For Scientific Research&Quot;Demokritos&Quot

Curated by ChEMBL

PNG

BDBM50570851(CHEMBL4853049)

IC50: 324nMAssay Description:Inhibition of ERAP1 (unknown origin) using L-AMC as substrateMore data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD antibodypedia GoogleScholar

Details Article PubMed

Endoplasmic reticulum aminopeptidase 1(Homo sapiens (Human))
National Center For Scientific Research&Quot;Demokritos&Quot

Curated by ChEMBL

PNG

BDBM50570851(CHEMBL4853049)

IC50: 330nMAssay Description:Inhibition of ERAP1 (unknown origin) using L-AMC as substrateMore data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD antibodypedia GoogleScholar

Details Article PubMed

Endoplasmic reticulum aminopeptidase 1(Homo sapiens (Human))
National Center For Scientific Research&Quot;Demokritos&Quot

Curated by ChEMBL

PNG

BDBM50245354(CHEMBL4097268)

IC50: 340nMAssay Description:Inhibition of ERAP1 (unknown origin) expressed in Hi5 cells by in vitro fluorimetric assayMore data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD antibodypedia GoogleScholar

CHEMBL PC cid PC sid Similars

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Endoplasmic reticulum aminopeptidase 1(Homo sapiens (Human))
National Center For Scientific Research&Quot;Demokritos&Quot

Curated by ChEMBL

PNG

BDBM50571856(CHEMBL4850551)

IC50: 377nMAssay Description:Inhibition of wild type ERAP1 (unknown origin) using L-Rho-Succ-FKARKF as substrate preincubated for 15 mins followed by substrate addition and measu...More data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD antibodypedia GoogleScholar

Details Article PubMed

Endoplasmic reticulum aminopeptidase 1(Homo sapiens (Human))
National Center For Scientific Research&Quot;Demokritos&Quot

Curated by ChEMBL

PNG

BDBM50570850(CHEMBL4877339)

IC50: 410nMAssay Description:Inhibition of ERAP1 (unknown origin) using L-AMC as substrateMore data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD antibodypedia GoogleScholar

Details Article PubMed

Endoplasmic reticulum aminopeptidase 1(Homo sapiens (Human))
National Center For Scientific Research&Quot;Demokritos&Quot

Curated by ChEMBL

PNG

BDBM50570850(CHEMBL4877339)

IC50: 417nMAssay Description:Inhibition of ERAP1 (unknown origin) using L-AMC as substrateMore data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD antibodypedia GoogleScholar

Details Article PubMed

Endoplasmic reticulum aminopeptidase 1(Homo sapiens (Human))
National Center For Scientific Research&Quot;Demokritos&Quot

Curated by ChEMBL

PNG

BDBM50601035(CHEMBL5194003)

IC50: 480nMAssay Description:Inhibition of recombinant ERAP1 (unknown origin) expressed in baculovirus infected Hi-5 insect cells using L-AMC as substrate by flourescence assayMore data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD antibodypedia GoogleScholar

Endoplasmic reticulum aminopeptidase 1(Homo sapiens (Human))
National Center For Scientific Research&Quot;Demokritos&Quot

Curated by ChEMBL

PNG

BDBM50190107(CHEMBL3827468)

IC50: 520nMAssay Description:Inhibition of recombinant human ERAP1 using L-AMC as substrate measured for 15 to 30 mins by fluorescence analysisMore data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD antibodypedia GoogleScholar

CHEMBL PC cid PC sid Patents Similars

Details Article PubMed

Endoplasmic reticulum aminopeptidase 1(Homo sapiens (Human))
National Center For Scientific Research&Quot;Demokritos&Quot

Curated by ChEMBL

PNG

BDBM50601033(CHEMBL5209483)

IC50: 590nMAssay Description:Inhibition of recombinant ERAP1 (unknown origin) expressed in baculovirus infected Hi-5 insect cells using L-AMC as substrate by flourescence assayMore data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD antibodypedia GoogleScholar

Endoplasmic reticulum aminopeptidase 1(Homo sapiens (Human))
National Center For Scientific Research&Quot;Demokritos&Quot

Curated by ChEMBL

PNG

BDBM50601042(CHEMBL5195885)

IC50: 670nMAssay Description:Inhibition of recombinant ERAP1 (unknown origin) expressed in baculovirus infected Hi-5 insect cells using L-AMC as substrate by flourescence assayMore data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD antibodypedia GoogleScholar

Endoplasmic reticulum aminopeptidase 1(Homo sapiens (Human))
National Center For Scientific Research&Quot;Demokritos&Quot

Curated by ChEMBL

PNG

BDBM50245347(CHEMBL4081682)

IC50: 682nMAssay Description:Inhibition of ERAP1 (unknown origin) expressed in Hi5 cells by in vitro fluorimetric assayMore data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD antibodypedia GoogleScholar

CHEMBL PC cid PC sid Similars

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Endoplasmic reticulum aminopeptidase 1(Homo sapiens (Human))
National Center For Scientific Research&Quot;Demokritos&Quot

Curated by ChEMBL

PNG

BDBM50571857(CHEMBL4854083)

IC50: 698nMAssay Description:Inhibition of wild type ERAP1 (unknown origin) using L-Rho-Succ-FKARKF as substrate preincubated for 15 mins followed by substrate addition and measu...More data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD antibodypedia GoogleScholar

Details Article PubMed

Endoplasmic reticulum aminopeptidase 1(Homo sapiens (Human))
National Center For Scientific Research&Quot;Demokritos&Quot

Curated by ChEMBL

PNG

BDBM50245402(CHEMBL4074464)

IC50: 726nMAssay Description:Inhibition of ERAP1 (unknown origin) expressed in Hi5 cells by in vitro fluorimetric assayMore data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD antibodypedia GoogleScholar

CHEMBL PC cid PC sid Similars

Details Article PubMed

Endoplasmic reticulum aminopeptidase 1(Homo sapiens (Human))
National Center For Scientific Research&Quot;Demokritos&Quot

Curated by ChEMBL

PNG

BDBM50076984(CHEMBL3416720)

IC50: 800nMAssay Description:Inhibition of human recombinant ERAP1 expressed in baculovirus infected Sf9 cells using L-leucine-7-amido-4-methyl coumarin as substrate after 5 to 1...More data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD antibodypedia GoogleScholar

CHEMBL PC cid PC sid Similars

Details Article PubMed

Endoplasmic reticulum aminopeptidase 1(Homo sapiens (Human))
National Center For Scientific Research&Quot;Demokritos&Quot

Curated by ChEMBL

PNG

BDBM50077028(CHEMBL3416692)

IC50: 920nMAssay Description:Inhibition of human recombinant ERAP1 expressed in baculovirus infected Sf9 cells using L-leucine-7-amido-4-methyl coumarin as substrate after 5 to 1...More data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD antibodypedia GoogleScholar

CHEMBL PC cid PC sid Patents Similars

Details Article PubMed

Endoplasmic reticulum aminopeptidase 1(Homo sapiens (Human))
National Center For Scientific Research&Quot;Demokritos&Quot

Curated by ChEMBL

PNG

BDBM50245349(CHEMBL4089555)

IC50: 949nMAssay Description:Inhibition of ERAP1 (unknown origin) expressed in Hi5 cells by in vitro fluorimetric assayMore data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD antibodypedia GoogleScholar

CHEMBL PC cid PC sid Similars

Details Article PubMed

Endoplasmic reticulum aminopeptidase 1(Homo sapiens (Human))
National Center For Scientific Research&Quot;Demokritos&Quot

Curated by ChEMBL

PNG

BDBM50519953(CHEMBL2140832)

IC50: 1.00E+3nMAssay Description:Inhibition of ERAP1 in human HeLa cells stably expressing H-2 Kb infected with vaccinia virus containing ss-LEQLE-SIINFEKL epitope assessed as suppre...More data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD antibodypedia GoogleScholar

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Endoplasmic reticulum aminopeptidase 1(Homo sapiens (Human))
National Center For Scientific Research&Quot;Demokritos&Quot

Curated by ChEMBL

PNG

BDBM50514671(CHEMBL4532803)

IC50: 1.00E+3nMAssay Description:Inhibition of full length C-terminal His6-tagged ERAP1 (unknown origin)-mediated antigenic epitope destruction assessed as inhibition of trimming of ...More data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD antibodypedia GoogleScholar

Details Article PubMed

Endoplasmic reticulum aminopeptidase 1(Homo sapiens (Human))
National Center For Scientific Research&Quot;Demokritos&Quot

Curated by ChEMBL

PNG

BDBM50514671(CHEMBL4532803)

IC50: 1.00E+3nMAssay Description:Activation of full length C-terminal His6-tagged ERAP1 (unknown origin)-mediated fluorogenic Leu-AMC substrate hydrolysis after 60 mins by Rapidfire-...More data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD antibodypedia GoogleScholar

Details Article PubMed

Endoplasmic reticulum aminopeptidase 1(Homo sapiens (Human))
National Center For Scientific Research&Quot;Demokritos&Quot

Curated by ChEMBL

PNG

BDBM50601032(CHEMBL5183817)

IC50: 1.00E+3nMAssay Description:Inhibition of recombinant ERAP1 (unknown origin) expressed in baculovirus infected Hi-5 insect cells using L-AMC as substrate by flourescence assayMore data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD antibodypedia GoogleScholar

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Filter my 211 hits

Targets 1▿
- Endoplasmic reticulum aminopeptidase 1 211
Publications 14▿
- J Med Chem 58: 1524-43 (2015) 41
- J Med Chem 65: 10098-10117 (2022) 36
- J Med Chem 63: 103-121 (2020) 33
- J Med Chem 59: 9107-9123 (2016) 31
- ACS Med Chem Lett 12: 1137-1142 (2021) 20
- Bioorg Med Chem Lett 42: (2021) 13
- ACS Med Chem Lett 7: 681-5 (2016) 10
- Bioorg Med Chem 27: (2019) 10
- J Med Chem 63: 3348-3358 (2020) 5
- Bioorg Med Chem Lett 23: 4832-6 (2013) 4
- Eur J Med Chem 211: (2021) 3
- Bioorg Med Chem Lett 29: 1031-1042 (2019) 2
- Bioorg Med Chem Lett 26: 4122-6 (2016) 2
- ACS Med Chem Lett 11: 1429-1434 (2020) 1
Institutions 12▿
- National Centre For Scientific Research "Demokritos 46
- National Center For Scientific Research&Quot;Demokritos&Quot 41
- Kansas University Specialized Chemistry Center 33
- National And Kapodistrian University Of Athens 31
- Sanofi 20
- The Institute Of Cancer Research 13
- National Center For Scientific Research Demokritos 11
- Glaxosmithkline 5
- University Of California San Diego 4
- Institut Pasteur De Lille 3
- Wroc?Aw University Of Science And Technology 2
- Wroclaw University Of Technology 2
Affinity: 33 to 5.0E+5 nM▿
- IC50 211
- Affinity ≤ nM
Xtal structures: 3
Docked structures: 0
Catalog Cmpds: 8