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Found 25 of ic50 for UniProtKB: P05193
TargetBeta-lactamase(Citrobacter freundii)TBA
LigandPNGBDBM50212638(CHEMBL302512)
Affinity DataIC50:  37.4nMAssay Description:Inhibitory activity against Citrobacter freundii 87470 Class-I beta-lactamase enzymeMore data for this Ligand-Target Pair
In DepthDetails
TargetBeta-lactamase(Citrobacter freundii)TBA
LigandPNGBDBM50212640(CHEMBL423309)
Affinity DataIC50:  115nMAssay Description:Inhibitory activity against Citrobacter freundii 87470 Class-I beta-lactamase enzymeMore data for this Ligand-Target Pair
In DepthDetails
TargetBeta-lactamase(Citrobacter freundii)TBA
LigandPNGBDBM50212634(CHEMBL309009)
Affinity DataIC50:  130nMAssay Description:Inhibitory activity against Citrobacter freundii 87470 Class-I beta-lactamase enzymeMore data for this Ligand-Target Pair
In DepthDetails
TargetBeta-lactamase(Citrobacter freundii)TBA
LigandPNGBDBM50053173((2S,3S,5R)-3-Methyl-4,4,7-trioxo-3-[1,2,3]triazol-...)
Affinity DataIC50:  166nMAssay Description:Inhibitory activity against Citrobacter freundii 87470 Class-I beta-lactamase enzymeMore data for this Ligand-Target Pair
In DepthDetails
TargetBeta-lactamase(Citrobacter freundii)TBA
LigandPNGBDBM50076680(CHEMBL6461 | Ro-48-1220 | Sodium; (2S,3R,5R)-3-((Z...)
Affinity DataIC50:  210nMAssay Description:Compound was tested for inhibition of Beta-lactamase from Citrobacter freundii 1982More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-lactamase(Citrobacter freundii)TBA
LigandPNGBDBM50076680(CHEMBL6461 | Ro-48-1220 | Sodium; (2S,3R,5R)-3-((Z...)
Affinity DataIC50:  210nMAssay Description:Compound was tested for inhibition of Beta-lactamase from Morganell morgani U1627More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-lactamase(Citrobacter freundii)TBA
LigandPNGBDBM50053181((2S,3S,5R)-3-((Z)-2-Ethoxycarbonyl-vinyl)-3-methyl...)
Affinity DataIC50:  370nMAssay Description:Compound was tested for inhibition of Citrobacter freundii 1928, class C of Beta-lactamaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-lactamase(Citrobacter freundii)TBA
LigandPNGBDBM50053180(CHEMBL332565 | Sodium; (2S,3S,5R)-3-methyl-4,4,7-t...)
Affinity DataIC50:  410nMAssay Description:Compound was tested for inhibition of Citrobacter freundii 1928, class C of Beta-lactamaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-lactamase(Citrobacter freundii)TBA
LigandPNGBDBM50212637(CHEMBL72046)
Affinity DataIC50:  456nMAssay Description:Inhibitory activity against Citrobacter freundii 87470 Class-I beta-lactamase enzymeMore data for this Ligand-Target Pair
In DepthDetails
TargetBeta-lactamase(Citrobacter freundii)TBA
LigandPNGBDBM50212639(CHEMBL302241)
Affinity DataIC50:  463nMAssay Description:Inhibitory activity against Citrobacter freundii 87470 Class-I beta-lactamase enzymeMore data for this Ligand-Target Pair
In DepthDetails
TargetBeta-lactamase(Citrobacter freundii)TBA
LigandPNGBDBM50212646(CHEMBL72972)
Affinity DataIC50:  524nMAssay Description:Inhibitory activity against Citrobacter freundii 87470 Class-I beta-lactamase enzymeMore data for this Ligand-Target Pair
In DepthDetails
TargetBeta-lactamase(Citrobacter freundii)TBA
LigandPNGBDBM50021954((2S,5R)-3,3-Dimethyl-4,4,7-trioxo-4lambda*6*-thia-...)
Affinity DataIC50:  857nMAssay Description:Inhibitory activity against Citrobacter freundii 87470 Class-I beta-lactamase enzymeMore data for this Ligand-Target Pair
In DepthDetails
TargetBeta-lactamase(Citrobacter freundii)TBA
LigandPNGBDBM50053173((2S,3S,5R)-3-Methyl-4,4,7-trioxo-3-[1,2,3]triazol-...)
Affinity DataIC50:  930nMAssay Description:Compound was tested for inhibition of Beta-lactamase from Citrobacter freundii 1982More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-lactamase(Citrobacter freundii)TBA
LigandPNGBDBM50053179(CHEMBL121924 | Sodium; (2S,3S,5R)-3-methyl-4,4,7-t...)
Affinity DataIC50:  1.00E+3nMAssay Description:Compound was tested for inhibition of Citrobacter freundii 1928, class C of Beta-lactamaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-lactamase(Citrobacter freundii)TBA
LigandPNGBDBM50053175((2S,3S,5R)-3-Methyl-4,4,7-trioxo-3-((E)-2-thiazol-...)
Affinity DataIC50:  1.30E+3nMAssay Description:Compound was tested for inhibition of Citrobacter freundii 1928, class C of Beta-lactamaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-lactamase(Citrobacter freundii)TBA
LigandPNGBDBM50212641(Brobactam)
Affinity DataIC50:  1.78E+3nMAssay Description:Inhibitory activity against Citrobacter freundii 87470 Class-I beta-lactamase enzymeMore data for this Ligand-Target Pair
In DepthDetails
TargetBeta-lactamase(Citrobacter freundii)TBA
LigandPNGBDBM50327179((S)-3-(2-(2-aminothiazol-4-yl)-2-((1,5-dihydroxy-4...)
Affinity DataIC50:  2.70E+3nMAssay Description:Inhibition of Citrobacter freundii AmpCMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-lactamase(Citrobacter freundii)TBA
LigandPNGBDBM50212643(CHEMBL308516)
Affinity DataIC50:  5.61E+3nMAssay Description:Inhibitory activity against Citrobacter freundii 87470 Class-I beta-lactamase enzymeMore data for this Ligand-Target Pair
In DepthDetails
TargetBeta-lactamase(Citrobacter freundii)TBA
LigandPNGBDBM50212645(CHEMBL305908)
Affinity DataIC50:  1.05E+4nMAssay Description:Inhibitory activity against Citrobacter freundii 87470 Class-I beta-lactamase enzymeMore data for this Ligand-Target Pair
In DepthDetails
TargetBeta-lactamase(Citrobacter freundii)TBA
LigandPNGBDBM50212642(CHEMBL70269)
Affinity DataIC50:  1.46E+4nMAssay Description:Inhibitory activity against Citrobacter freundii 87470 Class-I beta-lactamase enzymeMore data for this Ligand-Target Pair
In DepthDetails
TargetBeta-lactamase(Citrobacter freundii)TBA
LigandPNGBDBM50021959(CHEMBL777 | MM 14151 | US9120808, Clavulanic acid ...)
Affinity DataIC50:  1.60E+4nMAssay Description:Inhibitory activity against Citrobacter freundii 87470 Class-I beta-lactamase enzymeMore data for this Ligand-Target Pair
In DepthDetails
TargetBeta-lactamase(Citrobacter freundii)TBA
LigandPNGBDBM50053183(CHEMBL123481 | Trifluoro-methanesulfonate1-[(E)-3-...)
Affinity DataIC50:  1.60E+4nMAssay Description:Compound was tested for inhibition of Citrobacter freundii 1928, class C of Beta-lactamaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-lactamase(Citrobacter freundii)TBA
LigandPNGBDBM50212636(CHEMBL310221)
Affinity DataIC50:  5.03E+4nMAssay Description:Inhibitory activity against Citrobacter freundii 87470 Class-I beta-lactamase enzymeMore data for this Ligand-Target Pair
In DepthDetails
TargetBeta-lactamase(Citrobacter freundii)TBA
LigandPNGBDBM50212644(CHEMBL73450)
Affinity DataIC50:  8.15E+4nMAssay Description:Inhibitory activity against Citrobacter freundii 87470 Class-I beta-lactamase enzymeMore data for this Ligand-Target Pair
In DepthDetails
TargetBeta-lactamase(Citrobacter freundii)TBA
LigandPNGBDBM50212635(CHEMBL415266)
Affinity DataIC50:  1.01E+5nMAssay Description:Inhibitory activity against Citrobacter freundii 87470 Class-I beta-lactamase enzymeMore data for this Ligand-Target Pair
In DepthDetails