Compile Data Set for Download or QSAR
maximum 50k data
Found 101 of ic50 data for polymerid = 50004749
TargetP2Y purinoceptor 14(Mus musculus)
Merck Frosst Center For Therapeutic Research

Curated by ChEMBL
LigandPNGBDBM50343131(2-(2-cyanopyrimidin-5-yl)-N-(3-ethylphenyl)-4-o-to...)
Affinity DataIC50:  1nMAssay Description:Antagonist activity at mouse P2Y14 expressed in human HEK cells coexpressing Galphai5 assessed as inhibition of UDP-glucose stimulated calcium releas...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 14(Mus musculus)
Merck Frosst Center For Therapeutic Research

Curated by ChEMBL
LigandPNGBDBM50343129(2-(4-cyanopyridin-3-yl)-N-(3-ethylphenyl)-4-o-toly...)
Affinity DataIC50:  3nMAssay Description:Antagonist activity at mouse P2Y14 expressed in human HEK cells coexpressing Galphai5 assessed as inhibition of UDP-glucose stimulated calcium releas...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 14(Mus musculus)
Merck Frosst Center For Therapeutic Research

Curated by ChEMBL
LigandPNGBDBM50343132(2-(3,5-dimethylisoxazol-4-yl)-N-(3-ethylphenyl)-4-...)
Affinity DataIC50:  4nMAssay Description:Antagonist activity at mouse P2Y14 expressed in human HEK cells coexpressing Galphai5 assessed as inhibition of UDP-glucose stimulated calcium releas...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 14(Mus musculus)
Merck Frosst Center For Therapeutic Research

Curated by ChEMBL
LigandPNGBDBM50343886((R)-4-(4-(2,2,2-trifluoro-1-hydroxyethyl)phenyl)-7...)
Affinity DataIC50:  4nMAssay Description:Antagonist activity at mouse P2Y14 receptor expressed in HEK293 cells assessed as calcium flux by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 14(Mus musculus)
Merck Frosst Center For Therapeutic Research

Curated by ChEMBL
LigandPNGBDBM50343888((R)-4-(4-(2,2-difluoro-1-hydroxyethyl)phenyl)-7-(4...)
Affinity DataIC50:  8nMAssay Description:Antagonist activity at mouse P2Y14 receptor expressed in HEK293 cells assessed as calcium flux by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 14(Mus musculus)
Merck Frosst Center For Therapeutic Research

Curated by ChEMBL
LigandPNGBDBM50343120(4-(2,6-dimethylphenyl)-N-(3-ethylphenyl)-2-(pyridi...)
Affinity DataIC50:  9nMAssay Description:Antagonist activity at mouse P2Y14 expressed in human HEK cells coexpressing Galphai5 assessed as inhibition of UDP-glucose stimulated calcium releas...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 14(Mus musculus)
Merck Frosst Center For Therapeutic Research

Curated by ChEMBL
LigandPNGBDBM50343128(2-(benzo[d][1,3]dioxol-5-yl)-N-(3-ethylphenyl)-4-o...)
Affinity DataIC50:  10nMAssay Description:Antagonist activity at mouse P2Y14 expressed in human HEK cells coexpressing Galphai5 assessed as inhibition of UDP-glucose stimulated calcium releas...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 14(Mus musculus)
Merck Frosst Center For Therapeutic Research

Curated by ChEMBL
LigandPNGBDBM50343130(CHEMBL1771458 | N-(3-ethylphenyl)-2-(pyrimidin-5-y...)
Affinity DataIC50:  12nMAssay Description:Antagonist activity at mouse P2Y14 expressed in human HEK cells coexpressing Galphai5 assessed as inhibition of UDP-glucose stimulated calcium releas...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 14(Mus musculus)
Merck Frosst Center For Therapeutic Research

Curated by ChEMBL
LigandPNGBDBM50343885(4-(4-(2,2,2-trifluoro-1-hydroxyethyl)phenyl)-7-(4-...)
Affinity DataIC50:  13nMAssay Description:Antagonist activity at mouse P2Y14 receptor expressed in HEK293 cells assessed as calcium flux by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 14(Mus musculus)
Merck Frosst Center For Therapeutic Research

Curated by ChEMBL
LigandPNGBDBM50584883(CHEMBL5074765)
Affinity DataIC50:  13nMAssay Description:Inhibition of fluorescent antagonist binding to mouse P2Y14R expressed in HEK293 cells preincubated for 30 mins followed by addition of 6-amino-9-(2-...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 14(Mus musculus)
Merck Frosst Center For Therapeutic Research

Curated by ChEMBL
LigandPNGBDBM50343127(CHEMBL1771455 | N-(3-ethylphenyl)-2-(quinolin-3-yl...)
Affinity DataIC50:  13nMAssay Description:Antagonist activity at mouse P2Y14 expressed in human HEK cells coexpressing Galphai5 assessed as inhibition of UDP-glucose stimulated calcium releas...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 14(Mus musculus)
Merck Frosst Center For Therapeutic Research

Curated by ChEMBL
LigandPNGBDBM50343877(7-(4-fluoro-2,6-dimethylbenzyloxy)-4-(thiophen-3-y...)
Affinity DataIC50:  14nMAssay Description:Antagonist activity at mouse P2Y14 receptor expressed in HEK293 cells assessed as calcium flux by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 14(Mus musculus)
Merck Frosst Center For Therapeutic Research

Curated by ChEMBL
LigandPNGBDBM50343877(7-(4-fluoro-2,6-dimethylbenzyloxy)-4-(thiophen-3-y...)
Affinity DataIC50:  14nMAssay Description:Inhibition of mouse P2Y14 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 14(Mus musculus)
Merck Frosst Center For Therapeutic Research

Curated by ChEMBL
LigandPNGBDBM50584890(CHEMBL5079102)
Affinity DataIC50:  16nMAssay Description:Inhibition of fluorescent antagonist binding to mouse P2Y14R expressed in HEK293 cells preincubated for 30 mins followed by addition of 6-amino-9-(2-...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 14(Mus musculus)
Merck Frosst Center For Therapeutic Research

Curated by ChEMBL
LigandPNGBDBM50343094(2-(4-cyanophenyl)-N-(3-ethylphenyl)-4-o-tolyl-7,8-...)
Affinity DataIC50:  16nMAssay Description:Antagonist activity at mouse P2Y14 expressed in human HEK cells coexpressing Galphai5 assessed as inhibition of UDP-glucose stimulated calcium releas...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 14(Mus musculus)
Merck Frosst Center For Therapeutic Research

Curated by ChEMBL
LigandPNGBDBM50584893(CHEMBL5083619)
Affinity DataIC50:  18nMAssay Description:Inhibition of fluorescent antagonist binding to mouse P2Y14R expressed in HEK293 cells preincubated for 30 mins followed by addition of 6-amino-9-(2-...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 14(Mus musculus)
Merck Frosst Center For Therapeutic Research

Curated by ChEMBL
LigandPNGBDBM50566405(CHEMBL4864408)
Affinity DataIC50:  19nMAssay Description:Inhibition of fluorescent antagonist binding to mouse P2Y14 receptor expressed in HEK293 cells preincubated with compound for 30 mins followed by flu...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 14(Mus musculus)
Merck Frosst Center For Therapeutic Research

Curated by ChEMBL
LigandPNGBDBM50343884(4-(4-(methylsulfonyl)phenyl)-7-(4-(trifluoromethyl...)
Affinity DataIC50:  20nMAssay Description:Antagonist activity at mouse P2Y14 receptor expressed in HEK293 cells assessed as calcium flux by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 14(Mus musculus)
Merck Frosst Center For Therapeutic Research

Curated by ChEMBL
LigandPNGBDBM50543257(CHEMBL4645216)
Affinity DataIC50:  21nMAssay Description:Inhibition of MRS4174 binding to mouse P2Y14R expressed in HEK293 cells pre-incubated for 30 mins before MRS4174 addition and further incubated for 3...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 14(Mus musculus)
Merck Frosst Center For Therapeutic Research

Curated by ChEMBL
LigandPNGBDBM50456168(CHEMBL1800685)
Affinity DataIC50:  22nMAssay Description:Inhibition of MRS4174 binding to mouse P2Y14R expressed in HEK293 cells pre-incubated for 30 mins before MRS4174 addition and further incubated for 3...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 14(Mus musculus)
Merck Frosst Center For Therapeutic Research

Curated by ChEMBL
LigandPNGBDBM50456168(CHEMBL1800685)
Affinity DataIC50:  22nMAssay Description:Displacement of Alexafluor488 labeled 4-(4-(1-(4-(1-(6-(4-(6-amino-3-imino-4,5-disulfo-3H-xanthen-9-yl)-3-carboxybenzamido)hexyl)-1H-1,2,3-triazol-4-...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 14(Mus musculus)
Merck Frosst Center For Therapeutic Research

Curated by ChEMBL
LigandPNGBDBM50343095(CHEMBL1771452 | N-(3-ethylphenyl)-2-(4-fluoropheny...)
Affinity DataIC50:  25nMAssay Description:Antagonist activity at mouse P2Y14 expressed in human HEK cells coexpressing Galphai5 assessed as inhibition of UDP-glucose stimulated calcium releas...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 14(Mus musculus)
Merck Frosst Center For Therapeutic Research

Curated by ChEMBL
LigandPNGBDBM50343876(7-(2,6-dimethylbenzyloxy)-4-(thiophen-3-yl)-2-naph...)
Affinity DataIC50:  26nMAssay Description:Antagonist activity at mouse P2Y14 receptor expressed in HEK293 cells assessed as calcium flux by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 14(Mus musculus)
Merck Frosst Center For Therapeutic Research

Curated by ChEMBL
LigandPNGBDBM50584894(CHEMBL5076127)
Affinity DataIC50:  26nMAssay Description:Inhibition of fluorescent antagonist binding to mouse P2Y14R expressed in HEK293 cells preincubated for 30 mins followed by addition of 6-amino-9-(2-...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 14(Mus musculus)
Merck Frosst Center For Therapeutic Research

Curated by ChEMBL
LigandPNGBDBM50343109(CHEMBL1771244 | N-(3-(1-fluoroethyl)phenyl)-2-(pyr...)
Affinity DataIC50:  29nMAssay Description:Antagonist activity at mouse P2Y14 expressed in human HEK cells coexpressing Galphai5 assessed as inhibition of UDP-glucose stimulated calcium releas...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 14(Mus musculus)
Merck Frosst Center For Therapeutic Research

Curated by ChEMBL
LigandPNGBDBM50343125(CHEMBL1771453 | N-(3-ethylphenyl)-2-(3-fluoropheny...)
Affinity DataIC50:  30nMAssay Description:Antagonist activity at mouse P2Y14 expressed in human HEK cells coexpressing Galphai5 assessed as inhibition of UDP-glucose stimulated calcium releas...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 14(Mus musculus)
Merck Frosst Center For Therapeutic Research

Curated by ChEMBL
LigandPNGBDBM50541998(CHEMBL4642592)
Affinity DataIC50:  30nMAssay Description:Displacement of Alexafluor488 labeled 4-(4-(1-(4-(1-(6-(4-(6-amino-3-imino-4,5-disulfo-3H-xanthen-9-yl)-3-carboxybenzamido)hexyl)-1H-1,2,3-triazol-4-...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 14(Mus musculus)
Merck Frosst Center For Therapeutic Research

Curated by ChEMBL
LigandPNGBDBM50541998(CHEMBL4642592)
Affinity DataIC50:  30nMAssay Description:Inhibition of MRS4174 binding to mouse P2Y14R expressed in HEK293 cells pre-incubated for 30 mins before MRS4174 addition and further incubated for 3...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 14(Mus musculus)
Merck Frosst Center For Therapeutic Research

Curated by ChEMBL
LigandPNGBDBM50584891(CHEMBL5085823)
Affinity DataIC50:  34nMAssay Description:Inhibition of fluorescent antagonist binding to mouse P2Y14R expressed in HEK293 cells preincubated for 30 mins followed by addition of 6-amino-9-(2-...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 14(Mus musculus)
Merck Frosst Center For Therapeutic Research

Curated by ChEMBL
LigandPNGBDBM50541997(CHEMBL4649855)
Affinity DataIC50:  38nMAssay Description:Displacement of Alexafluor488 labeled 4-(4-(1-(4-(1-(6-(4-(6-amino-3-imino-4,5-disulfo-3H-xanthen-9-yl)-3-carboxybenzamido)hexyl)-1H-1,2,3-triazol-4-...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 14(Mus musculus)
Merck Frosst Center For Therapeutic Research

Curated by ChEMBL
LigandPNGBDBM50584895(CHEMBL5076678)
Affinity DataIC50:  41nMAssay Description:Inhibition of fluorescent antagonist binding to mouse P2Y14R expressed in HEK293 cells preincubated for 30 mins followed by addition of 6-amino-9-(2-...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 14(Mus musculus)
Merck Frosst Center For Therapeutic Research

Curated by ChEMBL
LigandPNGBDBM50584889(CHEMBL5083773)
Affinity DataIC50:  43nMAssay Description:Inhibition of fluorescent antagonist binding to mouse P2Y14R expressed in HEK293 cells preincubated for 30 mins followed by addition of 6-amino-9-(2-...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 14(Mus musculus)
Merck Frosst Center For Therapeutic Research

Curated by ChEMBL
LigandPNGBDBM50343121(4-(2-chloro-6-methylphenyl)-N-(3-ethylphenyl)-2-(p...)
Affinity DataIC50:  50nMAssay Description:Antagonist activity at mouse P2Y14 expressed in human HEK cells coexpressing Galphai5 assessed as inhibition of UDP-glucose stimulated calcium releas...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 14(Mus musculus)
Merck Frosst Center For Therapeutic Research

Curated by ChEMBL
LigandPNGBDBM50343887((S)-4-(4-(2,2,2-trifluoro-1-hydroxyethyl)phenyl)-7...)
Affinity DataIC50:  51nMAssay Description:Antagonist activity at mouse P2Y14 receptor expressed in HEK293 cells assessed as calcium flux by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 14(Mus musculus)
Merck Frosst Center For Therapeutic Research

Curated by ChEMBL
LigandPNGBDBM50343122(4-(2,6-dichlorophenyl)-N-(3-ethylphenyl)-2-(pyridi...)
Affinity DataIC50:  51nMAssay Description:Antagonist activity at mouse P2Y14 expressed in human HEK cells coexpressing Galphai5 assessed as inhibition of UDP-glucose stimulated calcium releas...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 14(Mus musculus)
Merck Frosst Center For Therapeutic Research

Curated by ChEMBL
LigandPNGBDBM50343878(4-(thiophen-3-yl)-7-(4-(trifluoromethoxy)phenyl)-2...)
Affinity DataIC50:  54nMAssay Description:Antagonist activity at mouse P2Y14 receptor expressed in HEK293 cells assessed as calcium flux by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 14(Mus musculus)
Merck Frosst Center For Therapeutic Research

Curated by ChEMBL
LigandPNGBDBM50543255(CHEMBL4640370)
Affinity DataIC50:  56nMAssay Description:Inhibition of MRS4174 binding to mouse P2Y14R expressed in HEK293 cells pre-incubated for 30 mins before MRS4174 addition and further incubated for 3...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 14(Mus musculus)
Merck Frosst Center For Therapeutic Research

Curated by ChEMBL
LigandPNGBDBM50343090(CHEMBL1771446 | N-(3-ethylphenyl)-4-o-tolyl-2-p-to...)
Affinity DataIC50:  62nMAssay Description:Antagonist activity at mouse P2Y14 expressed in human HEK cells coexpressing Galphai5 assessed as inhibition of UDP-glucose stimulated calcium releas...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 14(Mus musculus)
Merck Frosst Center For Therapeutic Research

Curated by ChEMBL
LigandPNGBDBM50343103(CHEMBL1771238 | N-(3-ethylphenyl)-2-(pyridin-3-yl)...)
Affinity DataIC50:  81nMAssay Description:Antagonist activity at mouse P2Y14 expressed in human HEK cells coexpressing Galphai5 assessed as inhibition of UDP-glucose stimulated calcium releas...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 14(Mus musculus)
Merck Frosst Center For Therapeutic Research

Curated by ChEMBL
LigandPNGBDBM50343089(CHEMBL1771445 | N-(3-ethylphenyl)-2-phenyl-4-o-tol...)
Affinity DataIC50:  87nMAssay Description:Antagonist activity at mouse P2Y14 expressed in human HEK cells coexpressing Galphai5 assessed as inhibition of UDP-glucose stimulated calcium releas...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 14(Mus musculus)
Merck Frosst Center For Therapeutic Research

Curated by ChEMBL
LigandPNGBDBM50584896(CHEMBL5087295)
Affinity DataIC50:  91nMAssay Description:Inhibition of fluorescent antagonist binding to mouse P2Y14R expressed in HEK293 cells preincubated for 30 mins followed by addition of 6-amino-9-(2-...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 14(Mus musculus)
Merck Frosst Center For Therapeutic Research

Curated by ChEMBL
LigandPNGBDBM50584904(CHEMBL5093465)
Affinity DataIC50:  102nMAssay Description:Inhibition of fluorescent antagonist binding to mouse P2Y14R expressed in HEK293 cells preincubated for 30 mins followed by addition of 6-amino-9-(2-...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 14(Mus musculus)
Merck Frosst Center For Therapeutic Research

Curated by ChEMBL
LigandPNGBDBM50584886(CHEMBL5090079)
Affinity DataIC50:  103nMAssay Description:Inhibition of fluorescent antagonist binding to mouse P2Y14R expressed in HEK293 cells preincubated for 30 mins followed by addition of 6-amino-9-(2-...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 14(Mus musculus)
Merck Frosst Center For Therapeutic Research

Curated by ChEMBL
LigandPNGBDBM50343872(7-(2,6-dimethylbenzyloxy)-4-phenyl-2-naphthoic aci...)
Affinity DataIC50:  110nMAssay Description:Antagonist activity at mouse P2Y14 receptor expressed in HEK293 cells assessed as calcium flux by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 14(Mus musculus)
Merck Frosst Center For Therapeutic Research

Curated by ChEMBL
LigandPNGBDBM50343875(4-(benzyloxy)-7-(2,6-dimethylbenzyloxy)-2-naphthoi...)
Affinity DataIC50:  110nMAssay Description:Antagonist activity at mouse P2Y14 receptor expressed in HEK293 cells assessed as calcium flux by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 14(Mus musculus)
Merck Frosst Center For Therapeutic Research

Curated by ChEMBL
LigandPNGBDBM50456170(CHEMBL4212441)
Affinity DataIC50:  130nMAssay Description:Inhibition of MRS4174 binding to mouse P2Y14R expressed in HEK293 cells pre-incubated for 30 mins before MRS4174 addition and further incubated for 3...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 14(Mus musculus)
Merck Frosst Center For Therapeutic Research

Curated by ChEMBL
LigandPNGBDBM50456170(CHEMBL4212441)
Affinity DataIC50:  130nMAssay Description:Displacement of Alexafluor488 labeled 4-(4-(1-(4-(1-(6-(4-(6-amino-3-imino-4,5-disulfo-3H-xanthen-9-yl)-3-carboxybenzamido)hexyl)-1H-1,2,3-triazol-4-...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 14(Mus musculus)
Merck Frosst Center For Therapeutic Research

Curated by ChEMBL
LigandPNGBDBM50343093(2-(3-cyanophenyl)-N-(3-ethylphenyl)-4-o-tolyl-7,8-...)
Affinity DataIC50:  140nMAssay Description:Antagonist activity at mouse P2Y14 expressed in human HEK cells coexpressing Galphai5 assessed as inhibition of UDP-glucose stimulated calcium releas...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 14(Mus musculus)
Merck Frosst Center For Therapeutic Research

Curated by ChEMBL
LigandPNGBDBM50532694(CHEMBL4454538)
Affinity DataIC50:  142nMAssay Description:Inhibition of MRS4174 binding to mouse P2Y14R expressed in HEK293 cells pre-incubated for 30 mins before MRS4174 addition and further incubated for 3...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 14(Mus musculus)
Merck Frosst Center For Therapeutic Research

Curated by ChEMBL
LigandPNGBDBM50532694(CHEMBL4454538)
Affinity DataIC50:  142nMAssay Description:Displacement of Alexafluor488 labeled 4-(4-(1-(4-(1-(6-(4-(6-amino-3-imino-4,5-disulfo-3H-xanthen-9-yl)-3-carboxybenzamido)hexyl)-1H-1,2,3-triazol-4-...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Displayed 1 to 50 (of 101 total ) | Next | Last >>
Jump to: