Compile Data Set for Download or QSAR
maximum 50k data
Found 12 of ic50 for UniProtKB: A0A140VJZ1
TargetUbiquitin carboxyl-terminal hydrolase 5(Homo sapiens (Human))TBA
LigandPNGBDBM50412352(CHEMBL5278336)
Affinity DataIC50:  800nMAssay Description:Inhibition of AChE in organophosphate-susceptible clone of Schizaphis graminum OSS adult or last-instar nymphs homogenates assessed as bimolecular ra...More data for this Ligand-Target Pair
In DepthDetails PDB3D3D Structure (crystal)
TargetUbiquitin carboxyl-terminal hydrolase 5(Homo sapiens (Human))TBA
LigandPNGBDBM50437695(CHEMBL1923233)
Affinity DataIC50:  3.00E+3nMAssay Description:Inhibition of USP5 in human Z138 cells after 1 hr by immunoblotting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUbiquitin carboxyl-terminal hydrolase 5(Homo sapiens (Human))TBA
LigandPNGBDBM50437693(VIALININ A)
Affinity DataIC50:  5.90E+3nMAssay Description:Inhibition of wild type human USP5 expressed in Escherichia coli BL21(DE3) using Ub-AMC as substrate after 60 mins by fluorometric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUbiquitin carboxyl-terminal hydrolase 5(Homo sapiens (Human))TBA
LigandPNGBDBM50412352(CHEMBL5278336)
Affinity DataIC50:  7.00E+3nMAssay Description:Inhibition of AChE in organophosphate-resistant clone of Schizaphis graminum OR1 adult or last-instar nymphs homogenates assessed as bimolecular rate...More data for this Ligand-Target Pair
In DepthDetails PDB3D3D Structure (crystal)
TargetUbiquitin carboxyl-terminal hydrolase 5(Homo sapiens (Human))TBA
LigandPNGBDBM50538571(CHEMBL4635160)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of human 6His-tagged USP5 expressed in Escherichia coli assessed as cleavage of Ubiquitin-Rhodamine110-glycine to Ubiquitin and Rhodamine1...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetUbiquitin carboxyl-terminal hydrolase 5(Homo sapiens (Human))TBA
LigandPNGBDBM50608542(CHEMBL5276142)
Affinity DataIC50:  2.15E+4nMMore data for this Ligand-Target Pair
Ligand InfoPDB
In DepthDetails
TargetUbiquitin carboxyl-terminal hydrolase 5(Homo sapiens (Human))TBA
LigandPNGBDBM50412352(CHEMBL5278336)
Affinity DataIC50:  2.60E+4nMAssay Description:Inhibition of AChE in organophosphate-susceptible clone of Schizaphis graminum OSS adult or last-instar nymphs homogenates assessed as bimolecular ra...More data for this Ligand-Target Pair
In DepthDetails PDB3D3D Structure (crystal)
TargetUbiquitin carboxyl-terminal hydrolase 5(Homo sapiens (Human))TBA
LigandPNGBDBM50608541(CHEMBL1493046)
Affinity DataIC50:  2.91E+4nMMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails
TargetUbiquitin carboxyl-terminal hydrolase 5(Homo sapiens (Human))TBA
LigandPNGBDBM50412352(CHEMBL5278336)
Affinity DataIC50:  4.60E+4nMAssay Description:Inhibition of AChE in organophosphate-resistant clone of Schizaphis graminum OR1 adult or last-instar nymphs homogenates assessed as bimolecular rate...More data for this Ligand-Target Pair
In DepthDetails PDB3D3D Structure (crystal)
TargetUbiquitin carboxyl-terminal hydrolase 5(Homo sapiens (Human))TBA
LigandPNGBDBM50437694(CHEMBL1410015)
Affinity DataIC50:  1.43E+5nMMore data for this Ligand-Target Pair
In DepthDetails
TargetUbiquitin carboxyl-terminal hydrolase 5(Homo sapiens (Human))TBA
LigandPNGBDBM50271098(CHEMBL4129140)
Affinity DataIC50: >2.00E+5nMAssay Description:Inhibition of USP5 (unknown origin) using Ub-AMC as substrate preincubated for 30 mins followed by substrate addition measured after 60 mins by fluor...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUbiquitin carboxyl-terminal hydrolase 5(Homo sapiens (Human))TBA
LigandPNGBDBM50608424(CHEMBL5267683)
Affinity DataIC50: >2.00E+5nMMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails