Compile Data Set for Download or QSAR
maximum 50k data
Found 7 of ic50 data for polymerid = 50006881
TargetEquilibrative nucleoside transporter 2(Homo sapiens (Human))
Monash University Malaysia

Curated by ChEMBL
LigandPNGBDBM56941(6-[[4-(4-fluorophenyl)-1-piperazinyl]methyl]-N2-(3...)
Affinity DataIC50:  570nMAssay Description:Inhibition of human ENT2 transfected in nucleoside transporter-deficient pig PK-15 cells assessed as inhibition of [3H]-uridine uptake by liquid scin...More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetEquilibrative nucleoside transporter 2(Homo sapiens (Human))
Monash University Malaysia

Curated by ChEMBL
LigandPNGBDBM50606918(CHEMBL5219061)
Affinity DataIC50:  1.69E+3nMAssay Description:Inhibition of human ENT2 transfected in nucleoside transporter-deficient pig PK-15 cells assessed as inhibition of [3H]-uridine uptake by liquid scin...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetEquilibrative nucleoside transporter 2(Homo sapiens (Human))
Monash University Malaysia

Curated by ChEMBL
LigandPNGBDBM50606918(CHEMBL5219061)
Affinity DataIC50:  4.36E+3nMAssay Description:Inhibition of human ENT2 transfected in nucleoside transporter-deficient pig PK-15 cells assessed as inhibition of [3H]-adenosine uptake by liquid sc...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetEquilibrative nucleoside transporter 2(Homo sapiens (Human))
Monash University Malaysia

Curated by ChEMBL
LigandPNGBDBM50606919(CHEMBL5219347)
Affinity DataIC50:  7.71E+4nMAssay Description:Inhibition of human ENT2 transfected in nucleoside transporter-deficient pig PK-15 cells assessed as inhibition of [3H]-uridine uptake by liquid scin...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetEquilibrative nucleoside transporter 2(Homo sapiens (Human))
Monash University Malaysia

Curated by ChEMBL
LigandPNGBDBM14487((2R,3R,4S,5R)-2-(6-amino-9H-purin-9-yl)-5-(hydroxy...)
Affinity DataIC50:  1.06E+5nMAssay Description:Binding affinity to recombinant human ENT2 expressed in Saccharomyces cerevisiae assessed as inhibition of [3H]-uridine transport after 15 mins by sc...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEquilibrative nucleoside transporter 2(Homo sapiens (Human))
Monash University Malaysia

Curated by ChEMBL
LigandPNGBDBM50138530((2R,3R,5R)-2-Hydroxymethyl-5-{6-[(R)-(tetrahydro-f...)
Affinity DataIC50:  1.90E+5nMAssay Description:Binding affinity to recombinant human ENT2 expressed in Saccharomyces cerevisiae assessed as inhibition of [3H]-uridine transport after 15 mins by sc...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEquilibrative nucleoside transporter 2(Homo sapiens (Human))
Monash University Malaysia

Curated by ChEMBL
LigandPNGBDBM50088517(CHEBI:16704 | Uridine)
Affinity DataIC50:  2.34E+5nMAssay Description:Binding affinity to recombinant human ENT2 expressed in Saccharomyces cerevisiae assessed as inhibition of [3H]-uridine transport after 15 mins by sc...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed