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Found 6 of ic50 data for polymerid = 50006943
TargetAmiloride-sensitive sodium channel subunit alpha(Mus musculus)
Temple University School Of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50112167(CHEMBL3608428)
Affinity DataIC50:  6nMAssay Description:Inhibition of ENaC in mouse M1 assessed as effect on trans epithelial electrical resistance by measuring short circuit currents by voltage-clamp base...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmiloride-sensitive sodium channel subunit alpha(Mus musculus)
Temple University School Of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50112170(CHEMBL3608425)
Affinity DataIC50:  6nMAssay Description:Inhibition of ENaC in mouse M1 assessed as effect on trans epithelial electrical resistance by measuring short circuit currents by voltage-clamp base...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmiloride-sensitive sodium channel subunit alpha(Mus musculus)
Temple University School Of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50112171(CHEMBL3608426)
Affinity DataIC50:  9nMAssay Description:Inhibition of ENaC in mouse M1 assessed as effect on trans epithelial electrical resistance by measuring short circuit currents by voltage-clamp base...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmiloride-sensitive sodium channel subunit alpha(Mus musculus)
Temple University School Of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50112172(CHEMBL3608427)
Affinity DataIC50:  13nMAssay Description:Inhibition of ENaC in mouse M1 assessed as effect on trans epithelial electrical resistance by measuring short circuit currents by voltage-clamp base...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmiloride-sensitive sodium channel subunit alpha(Mus musculus)
Temple University School Of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50112169(CHEMBL3608424)
Affinity DataIC50:  20nMAssay Description:Inhibition of ENaC in mouse M1 assessed as effect on trans epithelial electrical resistance by measuring short circuit currents by voltage-clamp base...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmiloride-sensitive sodium channel subunit alpha(Mus musculus)
Temple University School Of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50112168(CHEMBL3608423)
Affinity DataIC50:  70nMAssay Description:Inhibition of ENaC in mouse M1 assessed as effect on trans epithelial electrical resistance by measuring short circuit currents by voltage-clamp base...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed