TargetTransmembrane domain-containing protein TMIGD3(Homo sapiens (Human))
Georgia Institute of Technology
Curated by ChEMBL
Georgia Institute of Technology
Curated by ChEMBL
Affinity DataIC50: 42nMAssay Description:Antagonist activity at adenosine A3 receptor in human NPE cells assessed as inhibition of adenosine-triggered cell shrinkageMore data for this Ligand-Target Pair
TargetTransmembrane domain-containing protein TMIGD3(Homo sapiens (Human))
Georgia Institute of Technology
Curated by ChEMBL
Georgia Institute of Technology
Curated by ChEMBL
Affinity DataIC50: 73nMAssay Description:Antagonist activity at human A3 receptor expressed in CHO cells assessed as inhibition of CI-IB-MECA-mediated inhibition of cAMP production by [3H]cA...More data for this Ligand-Target Pair
TargetTransmembrane domain-containing protein TMIGD3(Homo sapiens (Human))
Georgia Institute of Technology
Curated by ChEMBL
Georgia Institute of Technology
Curated by ChEMBL
Affinity DataIC50: 163nMAssay Description:Antagonist activity at human A3 receptor expressed in CHO cells assessed as inhibition of CI-IB-MECA-mediated inhibition of cAMP production by [3H]cA...More data for this Ligand-Target Pair
TargetTransmembrane domain-containing protein TMIGD3(Homo sapiens (Human))
Georgia Institute of Technology
Curated by ChEMBL
Georgia Institute of Technology
Curated by ChEMBL
Affinity DataIC50: 172nMAssay Description:Displacement of [125I]AB-MECA from human adenosine A3 receptor expressed in CHO cell membranes after 120 mins by scintillation counting methodMore data for this Ligand-Target Pair
TargetTransmembrane domain-containing protein TMIGD3(Homo sapiens (Human))
Georgia Institute of Technology
Curated by ChEMBL
Georgia Institute of Technology
Curated by ChEMBL
Affinity DataIC50: 187nMAssay Description:Antagonist activity at human A3 receptor expressed in CHO cells assessed as inhibition of CI-IB-MECA-mediated inhibition of cAMP production by [3H]cA...More data for this Ligand-Target Pair
TargetTransmembrane domain-containing protein TMIGD3(Homo sapiens (Human))
Georgia Institute of Technology
Curated by ChEMBL
Georgia Institute of Technology
Curated by ChEMBL
Affinity DataIC50: 235nMAssay Description:Antagonist activity at human A3 receptor expressed in CHO cells assessed as inhibition of CI-IB-MECA-mediated inhibition of cAMP production by [3H]cA...More data for this Ligand-Target Pair