Compile Data Set for Download or QSAR
maximum 50k data
Found 79 of ki for UniProtKB: P07374
TargetUrease(Canavalia ensiformis (Jack bean) (Horse bean))
Institute Of Science

Curated by ChEMBL
LigandPNGBDBM50223161(1-cyclohexyl-1-isopropyl-3,3-dimethylselenourea | ...)
Affinity DataKi:  25nMAssay Description:Inhibition of jack bean ureaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrease(Canavalia ensiformis (Jack bean) (Horse bean))
Institute Of Science

Curated by ChEMBL
LigandPNGBDBM50356190(CHEMBL193474)
Affinity DataKi:  90nMAssay Description:Inhibition of jack bean urease assessed as ammonia production after 30 mins by indophenol methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrease(Canavalia ensiformis (Jack bean) (Horse bean))
Institute Of Science

Curated by ChEMBL
LigandPNGBDBM50223158((S)-1,1-dimethyl-3-(1-(naphthalen-1-yl)ethyl)selen...)
Affinity DataKi:  94nMAssay Description:Inhibition of jack bean ureaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrease(Canavalia ensiformis (Jack bean) (Horse bean))
Institute Of Science

Curated by ChEMBL
LigandPNGBDBM50356195(CHEMBL241902)
Affinity DataKi:  122nMAssay Description:Inhibition of jack bean urease assessed as ammonia production after 30 mins by indophenol methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrease(Canavalia ensiformis (Jack bean) (Horse bean))
Institute Of Science

Curated by ChEMBL
LigandPNGBDBM50223159(3-dodecyl-1,1-dimethylthiourea | CHEMBL251521)
Affinity DataKi:  124nMAssay Description:Inhibition of jack bean ureaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrease(Canavalia ensiformis (Jack bean) (Horse bean))
Institute Of Science

Curated by ChEMBL
LigandPNGBDBM50356192(CHEMBL241894)
Affinity DataKi:  127nMAssay Description:Inhibition of jack bean urease assessed as ammonia production after 30 mins by indophenol methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrease(Canavalia ensiformis (Jack bean) (Horse bean))
Institute Of Science

Curated by ChEMBL
LigandPNGBDBM53627(1-[[(E)-(5-oxidanyl-6-oxidanylidene-cyclohexa-2,4-...)
Affinity DataKi:  127nMAssay Description:Inhibition of jack bean urease assessed as ammonia production after 30 mins by indophenol methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrease(Canavalia ensiformis (Jack bean) (Horse bean))
Institute Of Science

Curated by ChEMBL
LigandPNGBDBM50356201(CHEMBL1910224)
Affinity DataKi:  134nMAssay Description:Inhibition of jack bean urease assessed as ammonia production after 30 mins by indophenol methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrease(Canavalia ensiformis (Jack bean) (Horse bean))
Institute Of Science

Curated by ChEMBL
LigandPNGBDBM50223157(3-(4-bromobenzyl)-1,1-dimethylselenourea | CHEMBL3...)
Affinity DataKi:  135nMAssay Description:Inhibition of jack bean ureaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrease(Canavalia ensiformis (Jack bean) (Horse bean))
Institute Of Science

Curated by ChEMBL
LigandPNGBDBM50356197(CHEMBL1910221)
Affinity DataKi:  152nMAssay Description:Inhibition of jack bean urease assessed as ammonia production after 30 mins by indophenol methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrease(Canavalia ensiformis (Jack bean) (Horse bean))
Institute Of Science

Curated by ChEMBL
LigandPNGBDBM50356186(CHEMBL239452)
Affinity DataKi:  170nMAssay Description:Inhibition of jack bean urease assessed as ammonia production after 30 mins by indophenol methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrease(Canavalia ensiformis (Jack bean) (Horse bean))
Institute Of Science

Curated by ChEMBL
LigandPNGBDBM50356198(CHEMBL1910222)
Affinity DataKi:  191nMAssay Description:Inhibition of jack bean urease assessed as ammonia production after 30 mins by indophenol methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrease(Canavalia ensiformis (Jack bean) (Horse bean))
Institute Of Science

Curated by ChEMBL
LigandPNGBDBM50488912(CHEMBL2298033)
Affinity DataKi:  200nMAssay Description:Inhibition of Canavalia ensiformis (jack bean) urease assessed as release of ammonia after 30 min by indophenol methodMore data for this Ligand-Target Pair
In DepthDetails Article
TargetUrease(Canavalia ensiformis (Jack bean) (Horse bean))
Institute Of Science

Curated by ChEMBL
LigandPNGBDBM50223160(3-(4-bromophenyl)-1,1-dimethylthiourea | CHEMBL249...)
Affinity DataKi:  255nMAssay Description:Inhibition of jack bean ureaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrease(Canavalia ensiformis (Jack bean) (Horse bean))
Institute Of Science

Curated by ChEMBL
LigandPNGBDBM50356199(CHEMBL242113)
Affinity DataKi:  391nMAssay Description:Inhibition of jack bean urease assessed as ammonia production after 30 mins by indophenol methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrease(Canavalia ensiformis (Jack bean) (Horse bean))
Institute Of Science

Curated by ChEMBL
LigandPNGBDBM50356188(CHEMBL391982)
Affinity DataKi:  398nMAssay Description:Inhibition of jack bean urease assessed as ammonia production after 30 mins by indophenol methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrease(Canavalia ensiformis (Jack bean) (Horse bean))
Institute Of Science

Curated by ChEMBL
LigandPNGBDBM50356196(CHEMBL1276230)
Affinity DataKi:  407nMAssay Description:Inhibition of jack bean urease assessed as ammonia production after 30 mins by indophenol methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrease(Canavalia ensiformis (Jack bean) (Horse bean))
Institute Of Science

Curated by ChEMBL
LigandPNGBDBM50356202(CHEMBL1910225)
Affinity DataKi:  430nMAssay Description:Inhibition of jack bean urease assessed as ammonia production after 30 mins by indophenol methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrease(Canavalia ensiformis (Jack bean) (Horse bean))
Institute Of Science

Curated by ChEMBL
LigandPNGBDBM50488911(CHEMBL2298025)
Affinity DataKi:  440nMAssay Description:Inhibition of Canavalia ensiformis (jack bean) urease assessed as release of ammonia after 30 min by indophenol methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
TargetUrease(Canavalia ensiformis (Jack bean) (Horse bean))
Institute Of Science

Curated by ChEMBL
LigandPNGBDBM50488920(CHEMBL2298019)
Affinity DataKi:  450nMAssay Description:Inhibition of Canavalia ensiformis (jack bean) urease assessed as release of ammonia after 30 min by indophenol methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
TargetUrease(Canavalia ensiformis (Jack bean) (Horse bean))
Institute Of Science

Curated by ChEMBL
LigandPNGBDBM50356191(CHEMBL193804)
Affinity DataKi:  497nMAssay Description:Inhibition of jack bean urease assessed as ammonia production after 30 mins by indophenol methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrease(Canavalia ensiformis (Jack bean) (Horse bean))
Institute Of Science

Curated by ChEMBL
LigandPNGBDBM50356187(CHEMBL1269725)
Affinity DataKi:  625nMAssay Description:Inhibition of jack bean urease assessed as ammonia production after 30 mins by indophenol methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrease(Canavalia ensiformis (Jack bean) (Horse bean))
Institute Of Science

Curated by ChEMBL
LigandPNGBDBM50488905(CHEMBL2298023)
Affinity DataKi:  650nMAssay Description:Inhibition of Canavalia ensiformis (jack bean) urease assessed as release of ammonia after 30 min by indophenol methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
TargetUrease(Canavalia ensiformis (Jack bean) (Horse bean))
Institute Of Science

Curated by ChEMBL
LigandPNGBDBM50114665(2-(trifluoromethyl)benzaldehyde thiosemicarbazone ...)
Affinity DataKi:  670nMAssay Description:Inhibition of jack bean urease assessed as ammonia production after 30 mins by indophenol methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrease(Canavalia ensiformis (Jack bean) (Horse bean))
Institute Of Science

Curated by ChEMBL
LigandPNGBDBM50356189(CHEMBL1910220)
Affinity DataKi:  770nMAssay Description:Inhibition of jack bean urease assessed as ammonia production after 30 mins by indophenol methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrease(Canavalia ensiformis (Jack bean) (Horse bean))
Institute Of Science

Curated by ChEMBL
LigandPNGBDBM50356193(CHEMBL398206)
Affinity DataKi:  807nMAssay Description:Inhibition of jack bean urease assessed as ammonia production after 30 mins by indophenol methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrease(Canavalia ensiformis (Jack bean) (Horse bean))
Institute Of Science

Curated by ChEMBL
LigandPNGBDBM50488918(CHEMBL2298024)
Affinity DataKi:  820nMAssay Description:Inhibition of Canavalia ensiformis (jack bean) urease assessed as release of ammonia after 30 min by indophenol methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
TargetUrease(Canavalia ensiformis (Jack bean) (Horse bean))
Institute Of Science

Curated by ChEMBL
LigandPNGBDBM50488919(CHEMBL2298022)
Affinity DataKi:  890nMAssay Description:Inhibition of Canavalia ensiformis (jack bean) urease assessed as release of ammonia after 30 min by indophenol methodMore data for this Ligand-Target Pair
In DepthDetails Article
TargetUrease(Canavalia ensiformis (Jack bean) (Horse bean))
Institute Of Science

Curated by ChEMBL
LigandPNGBDBM50356194(CHEMBL499789)
Affinity DataKi:  910nMAssay Description:Inhibition of jack bean urease assessed as ammonia production after 30 mins by indophenol methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrease(Canavalia ensiformis (Jack bean) (Horse bean))
Institute Of Science

Curated by ChEMBL
LigandPNGBDBM50488914(CHEMBL1370012)
Affinity DataKi:  1.14E+3nMAssay Description:Inhibition of Canavalia ensiformis (jack bean) urease assessed as release of ammonia after 30 min by indophenol methodMore data for this Ligand-Target Pair
In DepthDetails Article
TargetUrease(Canavalia ensiformis (Jack bean) (Horse bean))
Institute Of Science

Curated by ChEMBL
LigandPNGBDBM50488915(CHEMBL2298030)
Affinity DataKi:  1.21E+3nMAssay Description:Inhibition of Canavalia ensiformis (jack bean) urease assessed as release of ammonia after 30 min by indophenol methodMore data for this Ligand-Target Pair
In DepthDetails Article
TargetUrease(Canavalia ensiformis (Jack bean) (Horse bean))
Institute Of Science

Curated by ChEMBL
LigandPNGBDBM50488923(CHEMBL2298031)
Affinity DataKi:  1.23E+3nMAssay Description:Inhibition of Canavalia ensiformis (jack bean) urease assessed as release of ammonia after 30 min by indophenol methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
TargetUrease(Canavalia ensiformis (Jack bean) (Horse bean))
Institute Of Science

Curated by ChEMBL
LigandPNGBDBM50488910(CHEMBL2298029)
Affinity DataKi:  1.30E+3nMAssay Description:Inhibition of Canavalia ensiformis (jack bean) urease assessed as release of ammonia after 30 min by indophenol methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
TargetUrease(Canavalia ensiformis (Jack bean) (Horse bean))
Institute Of Science

Curated by ChEMBL
LigandPNGBDBM50488922(CHEMBL2298032)
Affinity DataKi:  1.31E+3nMAssay Description:Inhibition of Canavalia ensiformis (jack bean) urease assessed as release of ammonia after 30 min by indophenol methodMore data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails Article
TargetUrease(Canavalia ensiformis (Jack bean) (Horse bean))
Institute Of Science

Curated by ChEMBL
LigandPNGBDBM50488908(CHEMBL2298027)
Affinity DataKi:  1.34E+3nMAssay Description:Inhibition of Canavalia ensiformis (jack bean) urease assessed as release of ammonia after 30 min by indophenol methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
TargetUrease(Canavalia ensiformis (Jack bean) (Horse bean))
Institute Of Science

Curated by ChEMBL
LigandPNGBDBM50488917(CHEMBL2298026)
Affinity DataKi:  1.49E+3nMAssay Description:Inhibition of Canavalia ensiformis (jack bean) urease assessed as release of ammonia after 30 min by indophenol methodMore data for this Ligand-Target Pair
In DepthDetails Article
TargetUrease(Canavalia ensiformis (Jack bean) (Horse bean))
Institute Of Science

Curated by ChEMBL
LigandPNGBDBM50488909(CHEMBL2298036)
Affinity DataKi:  1.50E+3nMAssay Description:Inhibition of Canavalia ensiformis (jack bean) urease assessed as release of ammonia after 30 min by indophenol methodMore data for this Ligand-Target Pair
In DepthDetails Article
TargetUrease(Canavalia ensiformis (Jack bean) (Horse bean))
Institute Of Science

Curated by ChEMBL
LigandPNGBDBM50488906(CHEMBL2298020)
Affinity DataKi:  1.60E+3nMAssay Description:Inhibition of Canavalia ensiformis (jack bean) urease assessed as release of ammonia after 30 min by indophenol methodMore data for this Ligand-Target Pair
In DepthDetails Article
TargetUrease(Canavalia ensiformis (Jack bean) (Horse bean))
Institute Of Science

Curated by ChEMBL
LigandPNGBDBM50488913(CHEMBL179559)
Affinity DataKi:  1.91E+3nMAssay Description:Inhibition of Canavalia ensiformis (jack bean) urease assessed as release of ammonia after 30 min by indophenol methodMore data for this Ligand-Target Pair
In DepthDetails Article
TargetUrease(Canavalia ensiformis (Jack bean) (Horse bean))
Institute Of Science

Curated by ChEMBL
LigandPNGBDBM246417(US9447057, 1)
Affinity DataKi:  3.82E+3nM IC50:  2.80E+3nMpH: 6.8Assay Description:Reaction mixtures consisting of 25 μL (1 unit/well) of Jack bean (Canavalia ensiformis) urease, 55 μL of buffer at pH 6.8, 100 mM of urea, ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetUrease(Canavalia ensiformis (Jack bean) (Horse bean))
Institute Of Science

Curated by ChEMBL
LigandPNGBDBM50488907(CHEMBL2298034)
Affinity DataKi:  4.32E+3nMAssay Description:Inhibition of Canavalia ensiformis (jack bean) urease assessed as release of ammonia after 30 min by indophenol methodMore data for this Ligand-Target Pair
In DepthDetails Article
TargetUrease(Canavalia ensiformis (Jack bean) (Horse bean))
Institute Of Science

Curated by ChEMBL
LigandPNGBDBM50488916(CHEMBL2298028)
Affinity DataKi:  5.59E+3nMAssay Description:Inhibition of Canavalia ensiformis (jack bean) urease assessed as release of ammonia after 30 min by indophenol methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
TargetUrease(Canavalia ensiformis (Jack bean) (Horse bean))
Institute Of Science

Curated by ChEMBL
LigandPNGBDBM50488921(CHEMBL2298035)
Affinity DataKi:  7.50E+3nMAssay Description:Inhibition of Canavalia ensiformis (jack bean) urease assessed as release of ammonia after 30 min by indophenol methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
TargetUrease(Canavalia ensiformis (Jack bean) (Horse bean))
Institute Of Science

Curated by ChEMBL
LigandPNGBDBM246422(US9447057, 8)
Affinity DataKi:  7.89E+3nM IC50:  8.13E+3nMpH: 6.8Assay Description:Reaction mixtures consisting of 25 μL (1 unit/well) of Jack bean (Canavalia ensiformis) urease, 55 μL of buffer at pH 6.8, 100 mM of urea, ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetUrease(Canavalia ensiformis (Jack bean) (Horse bean))
Institute Of Science

Curated by ChEMBL
LigandPNGBDBM246420(US9447057, 6)
Affinity DataKi:  8.22E+3nM IC50:  8.80E+3nMpH: 6.8Assay Description:Reaction mixtures consisting of 25 μL (1 unit/well) of Jack bean (Canavalia ensiformis) urease, 55 μL of buffer at pH 6.8, 100 mM of urea, ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetUrease(Canavalia ensiformis (Jack bean) (Horse bean))
Institute Of Science

Curated by ChEMBL
LigandPNGBDBM50448175(CHEMBL3120552)
Affinity DataKi:  8.60E+3nMAssay Description:Competitive inhibition of jack bean urease using urea as substrate assessed as ammonia production after 15 mins by Lineweaver-Burk/Dixon plot analysi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrease(Canavalia ensiformis (Jack bean) (Horse bean))
Institute Of Science

Curated by ChEMBL
LigandPNGBDBM246418(US9447057, 4)
Affinity DataKi:  9.23E+3nM IC50:  1.12E+4nMpH: 6.8Assay Description:Reaction mixtures consisting of 25 μL (1 unit/well) of Jack bean (Canavalia ensiformis) urease, 55 μL of buffer at pH 6.8, 100 mM of urea, ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetUrease(Canavalia ensiformis (Jack bean) (Horse bean))
Institute Of Science

Curated by ChEMBL
LigandPNGBDBM246442(US9447057, 2)
Affinity DataKi:  9.60E+3nM IC50:  8.56E+3nMpH: 6.8Assay Description:Reaction mixtures consisting of 25 μL (1 unit/well) of Jack bean (Canavalia ensiformis) urease, 55 μL of buffer at pH 6.8, 100 mM of urea, ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetUrease(Canavalia ensiformis (Jack bean) (Horse bean))
Institute Of Science

Curated by ChEMBL
LigandPNGBDBM246443(US9447057, 3)
Affinity DataKi:  9.70E+3nM IC50:  7.90E+3nMpH: 6.8Assay Description:Reaction mixtures consisting of 25 μL (1 unit/well) of Jack bean (Canavalia ensiformis) urease, 55 μL of buffer at pH 6.8, 100 mM of urea, ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetUrease(Canavalia ensiformis (Jack bean) (Horse bean))
Institute Of Science

Curated by ChEMBL
LigandPNGBDBM50448176(CHEMBL3120570)
Affinity DataKi:  1.17E+4nMAssay Description:Competitive inhibition of jack bean urease using urea as substrate assessed as ammonia production after 15 mins by Lineweaver-Burk/Dixon plot analysi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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