Compile Data Set for Download or QSAR
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Found 75 of ic50 for UniProtKB: P03887
TargetNADH-ubiquinone oxidoreductase chain 1(Bos taurus (Bovine))TBA
LigandPNGBDBM50366820(BULLATACIN)
Affinity DataIC50:  0.800nMAssay Description:Inhibition of Bos taurus (bovine) mitochodrial complex 1 isolated from heart submitochondrial particle by NADH oxidase assayMore data for this Ligand-Target Pair
In DepthDetails Article
TargetNADH-ubiquinone oxidoreductase chain 1(Bos taurus (Bovine))TBA
LigandPNGBDBM92960(Piperazine derivative, 24)
Affinity DataIC50:  1nMAssay Description:Inhibition assay using NADH-ubiquinone oxidoreductase (complex I).More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNADH-ubiquinone oxidoreductase chain 1(Bos taurus (Bovine))TBA
LigandPNGBDBM92945(Piperazine derivative, 10)
Affinity DataIC50:  1.20nMAssay Description:Inhibition assay using NADH-ubiquinone oxidoreductase (complex I).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNADH-ubiquinone oxidoreductase chain 1(Bos taurus (Bovine))TBA
LigandPNGBDBM50004703(Corossoline)
Affinity DataIC50:  1.5nMAssay Description:Inhibition of Bos taurus (bovine) mitochodrial complex 1 isolated from heart submitochondrial particle by NADH oxidase assayMore data for this Ligand-Target Pair
In DepthDetails Article
TargetNADH-ubiquinone oxidoreductase chain 1(Bos taurus (Bovine))TBA
LigandPNGBDBM92946(Piperazine derivative, 9)
Affinity DataIC50:  1.70nMAssay Description:Inhibition assay using NADH-ubiquinone oxidoreductase (complex I).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNADH-ubiquinone oxidoreductase chain 1(Bos taurus (Bovine))TBA
LigandPNGBDBM92949(Piperazine derivative, 13)
Affinity DataIC50:  1.70nMAssay Description:Inhibition assay using NADH-ubiquinone oxidoreductase (complex I).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNADH-ubiquinone oxidoreductase chain 1(Bos taurus (Bovine))TBA
LigandPNGBDBM50004702((10S)-COROSSOLINE)
Affinity DataIC50:  2nMAssay Description:Inhibition of Bos taurus (bovine) mitochodrial complex 1 isolated from heart submitochondrial particle by NADH oxidase assayMore data for this Ligand-Target Pair
In DepthDetails Article
TargetNADH-ubiquinone oxidoreductase chain 1(Bos taurus (Bovine))TBA
LigandPNGBDBM50004705(CIS-SOLAMIN)
Affinity DataIC50:  2.10nMAssay Description:Inhibition of Bos taurus (bovine) mitochodrial complex 1 isolated from heart submitochondrial particle by NADH oxidase assayMore data for this Ligand-Target Pair
In DepthDetails Article
TargetNADH-ubiquinone oxidoreductase chain 1(Bos taurus (Bovine))TBA
LigandPNGBDBM50427137(SOLAMIN)
Affinity DataIC50:  2.10nMAssay Description:Inhibition of bovine heart mitochondrial complex 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNADH-ubiquinone oxidoreductase chain 1(Bos taurus (Bovine))TBA
LigandPNGBDBM50004705(CIS-SOLAMIN)
Affinity DataIC50:  2.20nMAssay Description:Inhibition of Bos taurus (bovine) mitochodrial complex 1 isolated from heart submitochondrial particle by NADH oxidase assayMore data for this Ligand-Target Pair
In DepthDetails Article
TargetNADH-ubiquinone oxidoreductase chain 1(Bos taurus (Bovine))TBA
LigandPNGBDBM92955(Piperazine derivative, 19)
Affinity DataIC50:  2.20nMAssay Description:Inhibition assay using NADH-ubiquinone oxidoreductase (complex I).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNADH-ubiquinone oxidoreductase chain 1(Bos taurus (Bovine))TBA
LigandPNGBDBM92948(Piperazine derivative, 12)
Affinity DataIC50:  2.30nMAssay Description:Inhibition assay using NADH-ubiquinone oxidoreductase (complex I).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNADH-ubiquinone oxidoreductase chain 1(Bos taurus (Bovine))TBA
LigandPNGBDBM92941(Piperazine derivative, 5)
Affinity DataIC50:  2.60nMAssay Description:Inhibition assay using NADH-ubiquinone oxidoreductase (complex I).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNADH-ubiquinone oxidoreductase chain 1(Bos taurus (Bovine))TBA
LigandPNGBDBM92950(Piperazine derivative, 14)
Affinity DataIC50:  2.80nMAssay Description:Inhibition assay using NADH-ubiquinone oxidoreductase (complex I).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNADH-ubiquinone oxidoreductase chain 1(Bos taurus (Bovine))TBA
LigandPNGBDBM50427136(CHEMBL1834283)
Affinity DataIC50:  2.90nMAssay Description:Inhibition of bovine heart mitochondrial complex 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNADH-ubiquinone oxidoreductase chain 1(Bos taurus (Bovine))TBA
LigandPNGBDBM50411905(CHEMBL272733)
Affinity DataIC50:  3nMAssay Description:Inhibition of Bos taurus (bovine) mitochondrial complex 1 assessed as reduction in enzyme activity by NADH-HU oxidoreductase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNADH-ubiquinone oxidoreductase chain 1(Bos taurus (Bovine))TBA
LigandPNGBDBM92956(Piperazine derivative, 20)
Affinity DataIC50:  3.60nMAssay Description:Inhibition assay using NADH-ubiquinone oxidoreductase (complex I).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNADH-ubiquinone oxidoreductase chain 1(Bos taurus (Bovine))TBA
LigandPNGBDBM50135527((-)-cis-rotenone | (-)-rotenone | (2R,6aS,12aS)-8,...)
Affinity DataIC50:  4.40nMAssay Description:Inhibition of Bos taurus (beef) heart NAD1More data for this Ligand-Target Pair
TargetNADH-ubiquinone oxidoreductase chain 1(Bos taurus (Bovine))TBA
LigandPNGBDBM92947(Piperazine derivative, 11)
Affinity DataIC50:  5.90nMAssay Description:Inhibition assay using NADH-ubiquinone oxidoreductase (complex I).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNADH-ubiquinone oxidoreductase chain 1(Bos taurus (Bovine))TBA
LigandPNGBDBM92954(Piperazine derivative, 18)
Affinity DataIC50:  12nMAssay Description:Inhibition assay using NADH-ubiquinone oxidoreductase (complex I).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNADH-ubiquinone oxidoreductase chain 1(Bos taurus (Bovine))TBA
LigandPNGBDBM92944(Piperazine derivative, 8)
Affinity DataIC50:  12nMAssay Description:Inhibition assay using NADH-ubiquinone oxidoreductase (complex I).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNADH-ubiquinone oxidoreductase chain 1(Bos taurus (Bovine))TBA
LigandPNGBDBM50004701((17R,18R,21R,22S)-reticulation-1)
Affinity DataIC50:  16nMAssay Description:Inhibition of Bos taurus (bovine) mitochodrial complex 1 isolated from heart submitochondrial particle by NADH oxidase assayMore data for this Ligand-Target Pair
In DepthDetails Article
TargetNADH-ubiquinone oxidoreductase chain 1(Bos taurus (Bovine))TBA
LigandPNGBDBM50004700((17S, 18S, 21S, 22R)-reticulation-1)
Affinity DataIC50:  17nMAssay Description:Inhibition of Bos taurus (bovine) mitochodrial complex 1 isolated from heart submitochondrial particle by NADH oxidase assayMore data for this Ligand-Target Pair
In DepthDetails Article
TargetNADH-ubiquinone oxidoreductase chain 1(Bos taurus (Bovine))TBA
LigandPNGBDBM92942(Piperazine derivative, 6)
Affinity DataIC50:  26nMAssay Description:Inhibition assay using NADH-ubiquinone oxidoreductase (complex I).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNADH-ubiquinone oxidoreductase chain 1(Bos taurus (Bovine))TBA
LigandPNGBDBM50427135(CHEMBL1834284)
Affinity DataIC50:  31nMAssay Description:Inhibition of bovine heart mitochondrial complex 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNADH-ubiquinone oxidoreductase chain 1(Bos taurus (Bovine))TBA
LigandPNGBDBM50488011(CHEMBL2272021)
Affinity DataIC50:  77nMAssay Description:Inhibition of Bos taurus (bovine) mitochondrial complex 1 assessed as reduction in enzyme activity by NADH-HU oxidoreductase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNADH-ubiquinone oxidoreductase chain 1(Bos taurus (Bovine))TBA
LigandPNGBDBM50488011(CHEMBL2272021)
Affinity DataIC50:  88nMAssay Description:Inhibition of Bos taurus (bovine) mitochondrial complex 1 assessed as reduction in enzyme activity by NADH-DU oxidoreductase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNADH-ubiquinone oxidoreductase chain 1(Bos taurus (Bovine))TBA
LigandPNGBDBM92943(Piperazine derivative, 7)
Affinity DataIC50:  110nMAssay Description:Inhibition assay using NADH-ubiquinone oxidoreductase (complex I).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNADH-ubiquinone oxidoreductase chain 1(Bos taurus (Bovine))TBA
LigandPNGBDBM50488037(CHEMBL2269636)
Affinity DataIC50:  270nMAssay Description:Inhibition of Bos taurus (beef) heart NAD1 assessed as NADH oxidase activityMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNADH-ubiquinone oxidoreductase chain 1(Bos taurus (Bovine))TBA
LigandPNGBDBM50427133(CHEMBL2323448)
Affinity DataIC50:  270nMAssay Description:Inhibition of bovine heart mitochondrial complex 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNADH-ubiquinone oxidoreductase chain 1(Bos taurus (Bovine))TBA
LigandPNGBDBM50427134(CHEMBL1834285)
Affinity DataIC50:  310nMAssay Description:Inhibition of bovine heart mitochondrial complex 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNADH-ubiquinone oxidoreductase chain 1(Bos taurus (Bovine))TBA
LigandPNGBDBM50488012(CHEMBL2272023)
Affinity DataIC50:  340nMAssay Description:Inhibition of Bos taurus (bovine) mitochondrial complex 1 assessed as reduction in enzyme activity by NADH-HU oxidoreductase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNADH-ubiquinone oxidoreductase chain 1(Bos taurus (Bovine))TBA
LigandPNGBDBM50488007(CHEMBL2272022)
Affinity DataIC50:  370nMAssay Description:Inhibition of Bos taurus (bovine) mitochondrial complex 1 assessed as reduction in enzyme activity by NADH-HU oxidoreductase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNADH-ubiquinone oxidoreductase chain 1(Bos taurus (Bovine))TBA
LigandPNGBDBM50488008(CHEMBL2272026)
Affinity DataIC50:  470nMAssay Description:Inhibition of Bos taurus (bovine) mitochondrial complex 1 assessed as reduction in enzyme activity by NADH-HU oxidoreductase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNADH-ubiquinone oxidoreductase chain 1(Bos taurus (Bovine))TBA
LigandPNGBDBM50488012(CHEMBL2272023)
Affinity DataIC50:  530nMAssay Description:Inhibition of Bos taurus (bovine) mitochondrial complex 1 assessed as reduction in enzyme activity by NADH-DU oxidoreductase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNADH-ubiquinone oxidoreductase chain 1(Bos taurus (Bovine))TBA
LigandPNGBDBM50427132(CHEMBL2323449)
Affinity DataIC50:  570nMAssay Description:Inhibition of bovine heart mitochondrial complex 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNADH-ubiquinone oxidoreductase chain 1(Bos taurus (Bovine))TBA
LigandPNGBDBM50488009(CHEMBL2272027)
Affinity DataIC50:  610nMAssay Description:Inhibition of Bos taurus (bovine) mitochondrial complex 1 assessed as reduction in enzyme activity by NADH-DU oxidoreductase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNADH-ubiquinone oxidoreductase chain 1(Bos taurus (Bovine))TBA
LigandPNGBDBM50488007(CHEMBL2272022)
Affinity DataIC50:  630nMAssay Description:Inhibition of Bos taurus (bovine) mitochondrial complex 1 assessed as reduction in enzyme activity by NADH-DU oxidoreductase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNADH-ubiquinone oxidoreductase chain 1(Bos taurus (Bovine))TBA
LigandPNGBDBM50488005(CHEMBL2272029)
Affinity DataIC50:  650nMAssay Description:Inhibition of Bos taurus (bovine) mitochondrial complex 1 assessed as reduction in enzyme activity by NADH-HU oxidoreductase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNADH-ubiquinone oxidoreductase chain 1(Bos taurus (Bovine))TBA
LigandPNGBDBM92951(Piperazine derivative, 15)
Affinity DataIC50:  670nMAssay Description:Inhibition assay using NADH-ubiquinone oxidoreductase (complex I).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNADH-ubiquinone oxidoreductase chain 1(Bos taurus (Bovine))TBA
LigandPNGBDBM50488008(CHEMBL2272026)
Affinity DataIC50:  760nMAssay Description:Inhibition of Bos taurus (bovine) mitochondrial complex 1 assessed as reduction in enzyme activity by NADH-DU oxidoreductase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNADH-ubiquinone oxidoreductase chain 1(Bos taurus (Bovine))TBA
LigandPNGBDBM144632(US8952025, Compound 2, table 3)
Affinity DataIC50:  829nMpH: 7.4Assay Description:Beef heart mitochondria were obtained by a large-scale procedure. Inverted submitochondrial particles (SMP) were prepared by the method of Matsuno-Ya...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetNADH-ubiquinone oxidoreductase chain 1(Bos taurus (Bovine))TBA
LigandPNGBDBM50488010(CHEMBL2272025)
Affinity DataIC50:  840nMAssay Description:Inhibition of Bos taurus (bovine) mitochondrial complex 1 assessed as reduction in enzyme activity by NADH-DU oxidoreductase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNADH-ubiquinone oxidoreductase chain 1(Bos taurus (Bovine))TBA
LigandPNGBDBM50488033(CHEMBL2269635)
Affinity DataIC50:  920nMAssay Description:Inhibition of Bos taurus (beef) heart NAD1 assessed as NADH oxidase activityMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNADH-ubiquinone oxidoreductase chain 1(Bos taurus (Bovine))TBA
LigandPNGBDBM92953(Piperazine derivative, 17)
Affinity DataIC50:  930nMAssay Description:Inhibition assay using NADH-ubiquinone oxidoreductase (complex I).More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNADH-ubiquinone oxidoreductase chain 1(Bos taurus (Bovine))TBA
LigandPNGBDBM50488010(CHEMBL2272025)
Affinity DataIC50:  970nMAssay Description:Inhibition of Bos taurus (bovine) mitochondrial complex 1 assessed as reduction in enzyme activity by NADH-HU oxidoreductase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNADH-ubiquinone oxidoreductase chain 1(Bos taurus (Bovine))TBA
LigandPNGBDBM50488009(CHEMBL2272027)
Affinity DataIC50:  1.10E+3nMAssay Description:Inhibition of Bos taurus (bovine) mitochondrial complex 1 assessed as reduction in enzyme activity by NADH-HU oxidoreductase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNADH-ubiquinone oxidoreductase chain 1(Bos taurus (Bovine))TBA
LigandPNGBDBM92958(Piperazine derivative, 22)
Affinity DataIC50:  1.10E+3nMAssay Description:Inhibition assay using NADH-ubiquinone oxidoreductase (complex I).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNADH-ubiquinone oxidoreductase chain 1(Bos taurus (Bovine))TBA
LigandPNGBDBM92957(Piperazine derivative, 21)
Affinity DataIC50:  1.30E+3nMAssay Description:Inhibition assay using NADH-ubiquinone oxidoreductase (complex I).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNADH-ubiquinone oxidoreductase chain 1(Bos taurus (Bovine))TBA
LigandPNGBDBM50488037(CHEMBL2269636)
Affinity DataIC50:  1.52E+3nMAssay Description:Inhibition of Bos taurus (beef) heart NAD1 assessed as NADH-ubiquinone oxidoreductase activityMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
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