Affinity DataKi: 0.150nMAssay Description:Inhibition of TSPO (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 0.150nMAssay Description:Inhibition of TSPO (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 0.188nMAssay Description:In vitro binding affinity for PBR (peripheral benzodiazepine receptor) in monkey brainMore data for this Ligand-Target Pair
Affinity DataKi: 0.200nMAssay Description:Inhibition of human TSPOMore data for this Ligand-Target Pair
Affinity DataKi: 0.242nMAssay Description:Binding affinity to PBR in human mitochondrial tissueMore data for this Ligand-Target Pair
Affinity DataKi: 0.242nMAssay Description:Displacement of [3H]PK11195 from human PBR receptorMore data for this Ligand-Target Pair
Affinity DataKi: 0.280nMAssay Description:Binding affinity to TSPO (unknown origin) relative to controlMore data for this Ligand-Target Pair
Affinity DataKi: 0.410nMAssay Description:Inhibition of TSPO (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 0.410nMAssay Description:Inhibition of TSPO (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 0.450nMAssay Description:In vitro binding activity of TSPO.More data for this Ligand-Target Pair
Affinity DataKi: 0.460nMAssay Description:In vitro binding activity of TSPO.More data for this Ligand-Target Pair
Affinity DataKi: 0.5nMAssay Description:Inhibition of TSPO (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 0.5nMAssay Description:Binding affinity to TSPO (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 0.5nMAssay Description:Inhibition of TSPO (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 0.537nMAssay Description:Inhibition of TSPO (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 0.537nMAssay Description:Inhibition of TSPO (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 0.860nMAssay Description:Inhibition of TSPO (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 0.860nMAssay Description:Inhibition of TSPO (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 0.870nMAssay Description:Inhibition of TSPO (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 0.882nMAssay Description:Inhibition of TSPO (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 0.882nMAssay Description:Inhibition of TSPO (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 0.970nMAssay Description:In vitro binding activity of TSPO.More data for this Ligand-Target Pair
Affinity DataKi: 0.997nMAssay Description:Displacement of [3H]PK11195 from human PBR receptorMore data for this Ligand-Target Pair
Affinity DataKi: 1.19nMAssay Description:Displacement of [3H]PK11195 from TSPO in human HEK293 mitochondrial fractionMore data for this Ligand-Target Pair
Affinity DataKi: 1.40nMAssay Description:Binding affinity to PBR in human mitochondrial tissueMore data for this Ligand-Target Pair
Affinity DataKi: 1.55nMAssay Description:In vitro binding activity of TSPO.More data for this Ligand-Target Pair
Affinity DataKi: 1.57nMAssay Description:Displacement of [11C]PK11195 from high affinity binding site of TSPO in human brain membrane homogenate by scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 1.60nMAssay Description:Inhibition of TSPO (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 1.60nMAssay Description:Inhibition of TSPO (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 1.82nMAssay Description:Displacement of [11C]PK11195 from mixed affinity binding site of TSPO in human brain membrane homogenate by scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 2.40nMAssay Description:In vitro binding activity of TSPO.More data for this Ligand-Target Pair
Affinity DataKi: 2.5nMAssay Description:Binding affinity to PBR in human mitochondrial tissueMore data for this Ligand-Target Pair
Affinity DataKi: 2.5nMAssay Description:Inhibition of human TSPOMore data for this Ligand-Target Pair
Affinity DataKi: 2.5nMAssay Description:For the assays described herein systemic injections of kainic in rats were applied and also contusion (Veenman et al. 2002; Soustiel et al. Neuropath...More data for this Ligand-Target Pair
Affinity DataKi: 2.5nMAssay Description:For the assays described herein systemic injections of kainic in rats were applied and also contusion (Veenman et al. 2002; Soustiel et al. Neuropath...More data for this Ligand-Target Pair
Affinity DataKi: 2.61nMAssay Description:In vitro binding activity of TSPO.More data for this Ligand-Target Pair
Affinity DataKi: 2.70nMAssay Description:Inhibition of TSPO (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 3.20nMAssay Description:Displacement of [3H]PK11195 from wild-type human TSPO expressed in HEK293 cells after 90 mins by scintillation counting methodMore data for this Ligand-Target Pair
Affinity DataKi: 3.30nMAssay Description:Inhibition of TSPO (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 3.90nMAssay Description:Inhibition of TSPO (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 3.90nMAssay Description:Inhibition of TSPO (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 4nMAssay Description:In vitro binding activity of TSPO.More data for this Ligand-Target Pair
Affinity DataKi: 4nMAssay Description:Binding affinity to TSPO (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 4.5nMAssay Description:Inhibition of human TSPOMore data for this Ligand-Target Pair
Affinity DataKi: 4.5nMAssay Description:Binding affinity to PBR in human mitochondrial tissueMore data for this Ligand-Target Pair
Affinity DataKi: 5nMAssay Description:In vitro binding activity of TSPO.More data for this Ligand-Target Pair
Affinity DataKi: 5.70nMAssay Description:In vitro binding activity of TSPO.More data for this Ligand-Target Pair
Affinity DataKi: 6.20nMAssay Description:Displacement of [3H]-PK11195 from wild type TSPO (unknown origin) expressed in human HEK293T cells assessed as inhibitory constant incubated for 90 m...More data for this Ligand-Target Pair
Affinity DataKi: 6.60nMAssay Description:Displacement of [3H]PK11195 from wild-type human TSPO expressed in HEK293 cell membranes after 90 mins by scintillation counting methodMore data for this Ligand-Target Pair
Affinity DataKi: 6.70nMAssay Description:Displacement of [3H]PK11195 from TSPO in human T98G cell membranes incubated for 90 mins by competition radioligand binding assayMore data for this Ligand-Target Pair