Compile Data Set for Download or QSAR
maximum 50k data
Found 258 of ki for UniProtKB: P30536
TargetTranslocator protein(Homo sapiens (Human))
Palack£

Curated by ChEMBL
LigandPNGBDBM50274351(2-(6,8-Dichloro-2-(4-nitrophenyl)imidazo[1,2-a]pyr...)
Affinity DataKi:  0.150nMAssay Description:Inhibition of TSPO (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Homo sapiens (Human))
Palack£

Curated by ChEMBL
LigandPNGBDBM50274351(2-(6,8-Dichloro-2-(4-nitrophenyl)imidazo[1,2-a]pyr...)
Affinity DataKi:  0.150nMAssay Description:Inhibition of TSPO (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Homo sapiens (Human))
Palack£

Curated by ChEMBL
LigandPNGBDBM50122293(CHEMBL401000 | CHEMBL63064 | N-(2,5-Dimethoxy-benz...)
Affinity DataKi:  0.188nMAssay Description:In vitro binding affinity for PBR (peripheral benzodiazepine receptor) in monkey brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Homo sapiens (Human))
Palack£

Curated by ChEMBL
LigandPNGBDBM50122293(CHEMBL401000 | CHEMBL63064 | N-(2,5-Dimethoxy-benz...)
Affinity DataKi:  0.200nMAssay Description:Inhibition of human TSPOMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Homo sapiens (Human))
Palack£

Curated by ChEMBL
LigandPNGBDBM50122293(CHEMBL401000 | CHEMBL63064 | N-(2,5-Dimethoxy-benz...)
Affinity DataKi:  0.242nMAssay Description:Binding affinity to PBR in human mitochondrial tissueMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Homo sapiens (Human))
Palack£

Curated by ChEMBL
LigandPNGBDBM50122293(CHEMBL401000 | CHEMBL63064 | N-(2,5-Dimethoxy-benz...)
Affinity DataKi:  0.242nMAssay Description:Displacement of [3H]PK11195 from human PBR receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Homo sapiens (Human))
Palack£

Curated by ChEMBL
LigandPNGBDBM50421116(CHEMBL2088374)
Affinity DataKi:  0.280nMAssay Description:Binding affinity to TSPO (unknown origin) relative to controlMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetTranslocator protein(Homo sapiens (Human))
Palack£

Curated by ChEMBL
LigandPNGBDBM50060095(2-[6,8-Dichloro-2-(4-chloro-phenyl)-imidazo[1,2-a]...)
Affinity DataKi:  0.410nMAssay Description:Inhibition of TSPO (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Homo sapiens (Human))
Palack£

Curated by ChEMBL
LigandPNGBDBM50060095(2-[6,8-Dichloro-2-(4-chloro-phenyl)-imidazo[1,2-a]...)
Affinity DataKi:  0.410nMAssay Description:Inhibition of TSPO (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Homo sapiens (Human))
Palack£

Curated by ChEMBL
LigandPNGBDBM98172(US8492379, 28)
Affinity DataKi:  0.450nMAssay Description:In vitro binding activity of TSPO.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetTranslocator protein(Homo sapiens (Human))
Palack£

Curated by ChEMBL
LigandPNGBDBM98171(US8492379, 27)
Affinity DataKi:  0.460nMAssay Description:In vitro binding activity of TSPO.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetTranslocator protein(Homo sapiens (Human))
Palack£

Curated by ChEMBL
LigandPNGBDBM22041(2-[6-chloro-2-(4-chlorophenyl)imidazo[1,2-a]pyridi...)
Affinity DataKi:  0.5nMAssay Description:Inhibition of TSPO (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Homo sapiens (Human))
Palack£

Curated by ChEMBL
LigandPNGBDBM22041(2-[6-chloro-2-(4-chlorophenyl)imidazo[1,2-a]pyridi...)
Affinity DataKi:  0.5nMAssay Description:Binding affinity to TSPO (unknown origin)More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetTranslocator protein(Homo sapiens (Human))
Palack£

Curated by ChEMBL
LigandPNGBDBM22041(2-[6-chloro-2-(4-chlorophenyl)imidazo[1,2-a]pyridi...)
Affinity DataKi:  0.5nMAssay Description:Inhibition of TSPO (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Homo sapiens (Human))
Palack£

Curated by ChEMBL
LigandPNGBDBM50274258(2-(6,8-Dichloro-2-(4-methoxyphenyl)imidazo[1,2-a]p...)
Affinity DataKi:  0.537nMAssay Description:Inhibition of TSPO (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Homo sapiens (Human))
Palack£

Curated by ChEMBL
LigandPNGBDBM50274258(2-(6,8-Dichloro-2-(4-methoxyphenyl)imidazo[1,2-a]p...)
Affinity DataKi:  0.537nMAssay Description:Inhibition of TSPO (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Homo sapiens (Human))
Palack£

Curated by ChEMBL
LigandPNGBDBM50274561(4-(2-(4-Chlorophenyl)-3-(2-(dipropylamino)-2-oxoet...)
Affinity DataKi:  0.860nMAssay Description:Inhibition of TSPO (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Homo sapiens (Human))
Palack£

Curated by ChEMBL
LigandPNGBDBM50274561(4-(2-(4-Chlorophenyl)-3-(2-(dipropylamino)-2-oxoet...)
Affinity DataKi:  0.860nMAssay Description:Inhibition of TSPO (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Homo sapiens (Human))
Palack£

Curated by ChEMBL
LigandPNGBDBM50073588(CHEMBL3408974)
Affinity DataKi:  0.870nMAssay Description:Inhibition of TSPO (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Homo sapiens (Human))
Palack£

Curated by ChEMBL
LigandPNGBDBM50274259(CHEMBL521186 | N-Butyl-2-(6,8-dichloro-2-(4-methox...)
Affinity DataKi:  0.882nMAssay Description:Inhibition of TSPO (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Homo sapiens (Human))
Palack£

Curated by ChEMBL
LigandPNGBDBM50274259(CHEMBL521186 | N-Butyl-2-(6,8-dichloro-2-(4-methox...)
Affinity DataKi:  0.882nMAssay Description:Inhibition of TSPO (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Homo sapiens (Human))
Palack£

Curated by ChEMBL
LigandPNGBDBM98173(US8492379, 29)
Affinity DataKi:  0.970nMAssay Description:In vitro binding activity of TSPO.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetTranslocator protein(Homo sapiens (Human))
Palack£

Curated by ChEMBL
LigandPNGBDBM50255877(CHEMBL473435 | N-Fluoroacetyl-N-(2,5-dimethoxybenz...)
Affinity DataKi:  0.997nMAssay Description:Displacement of [3H]PK11195 from human PBR receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Homo sapiens (Human))
Palack£

Curated by ChEMBL
LigandPNGBDBM50350912(CHEMBL1817978)
Affinity DataKi:  1.19nMAssay Description:Displacement of [3H]PK11195 from TSPO in human HEK293 mitochondrial fractionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Homo sapiens (Human))
Palack£

Curated by ChEMBL
LigandPNGBDBM50229593(CHEMBL253596 | N-acetyl-N-(2-methoxycarbonylbenzyl...)
Affinity DataKi:  1.40nMAssay Description:Binding affinity to PBR in human mitochondrial tissueMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Homo sapiens (Human))
Palack£

Curated by ChEMBL
LigandPNGBDBM98176(US8492379, 53)
Affinity DataKi:  1.55nMAssay Description:In vitro binding activity of TSPO.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetTranslocator protein(Homo sapiens (Human))
Palack£

Curated by ChEMBL
LigandPNGBDBM50335270(2-(1-methyl-2-(4-nitrophenyl)-1H-indol-3-yl)-2-oxo...)
Affinity DataKi:  1.57nMAssay Description:Displacement of [11C]PK11195 from high affinity binding site of TSPO in human brain membrane homogenate by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Homo sapiens (Human))
Palack£

Curated by ChEMBL
LigandPNGBDBM50408728(CHEMBL339816)
Affinity DataKi:  1.60nMAssay Description:Inhibition of TSPO (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Homo sapiens (Human))
Palack£

Curated by ChEMBL
LigandPNGBDBM50408728(CHEMBL339816)
Affinity DataKi:  1.60nMAssay Description:Inhibition of TSPO (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Homo sapiens (Human))
Palack£

Curated by ChEMBL
LigandPNGBDBM50335270(2-(1-methyl-2-(4-nitrophenyl)-1H-indol-3-yl)-2-oxo...)
Affinity DataKi:  1.82nMAssay Description:Displacement of [11C]PK11195 from mixed affinity binding site of TSPO in human brain membrane homogenate by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Homo sapiens (Human))
Palack£

Curated by ChEMBL
LigandPNGBDBM98174(US8492379, 30)
Affinity DataKi:  2.40nMAssay Description:In vitro binding activity of TSPO.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetTranslocator protein(Homo sapiens (Human))
Palack£

Curated by ChEMBL
LigandPNGBDBM50229594(CHEMBL253597 | N-(2-methoxybenzyl)-N-(4-phenoxypyr...)
Affinity DataKi:  2.5nMAssay Description:Binding affinity to PBR in human mitochondrial tissueMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Homo sapiens (Human))
Palack£

Curated by ChEMBL
LigandPNGBDBM50229594(CHEMBL253597 | N-(2-methoxybenzyl)-N-(4-phenoxypyr...)
Affinity DataKi:  2.5nMAssay Description:Inhibition of human TSPOMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Homo sapiens (Human))
Palack£

Curated by ChEMBL
LigandPNGBDBM279584(US10035780, Compound 8)
Affinity DataKi:  2.5nMAssay Description:For the assays described herein systemic injections of kainic in rats were applied and also contusion (Veenman et al. 2002; Soustiel et al. Neuropath...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTranslocator protein(Homo sapiens (Human))
Palack£

Curated by ChEMBL
LigandPNGBDBM279583(US10035780, Compound 7)
Affinity DataKi:  2.5nMAssay Description:For the assays described herein systemic injections of kainic in rats were applied and also contusion (Veenman et al. 2002; Soustiel et al. Neuropath...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTranslocator protein(Homo sapiens (Human))
Palack£

Curated by ChEMBL
LigandPNGBDBM98170(US8492379, 26)
Affinity DataKi:  2.61nMAssay Description:In vitro binding activity of TSPO.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetTranslocator protein(Homo sapiens (Human))
Palack£

Curated by ChEMBL
LigandPNGBDBM50159089(CHEMBL180523 | N,N-Dibutyl-2-[6,8-dichloro-2-(4-ch...)
Affinity DataKi:  2.70nMAssay Description:Inhibition of TSPO (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Homo sapiens (Human))
Palack£

Curated by ChEMBL
LigandPNGBDBM50509027(CHEMBL4459176)
Affinity DataKi:  3.20nMAssay Description:Displacement of [3H]PK11195 from wild-type human TSPO expressed in HEK293 cells after 90 mins by scintillation counting methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTranslocator protein(Homo sapiens (Human))
Palack£

Curated by ChEMBL
LigandPNGBDBM50045877(2-(2-(4-fluorophenyl)-1H-indol-3-yl)-N,N-dihexylac...)
Affinity DataKi:  3.30nMAssay Description:Inhibition of TSPO (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Homo sapiens (Human))
Palack£

Curated by ChEMBL
LigandPNGBDBM50045880(2-[5-Chloro-2-(4-chloro-phenyl)-1H-indol-3-yl]-N,N...)
Affinity DataKi:  3.90nMAssay Description:Inhibition of TSPO (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Homo sapiens (Human))
Palack£

Curated by ChEMBL
LigandPNGBDBM50045880(2-[5-Chloro-2-(4-chloro-phenyl)-1H-indol-3-yl]-N,N...)
Affinity DataKi:  3.90nMAssay Description:Inhibition of TSPO (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Homo sapiens (Human))
Palack£

Curated by ChEMBL
LigandPNGBDBM98177(US8492379, 54)
Affinity DataKi:  4nMAssay Description:In vitro binding activity of TSPO.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTranslocator protein(Homo sapiens (Human))
Palack£

Curated by ChEMBL
LigandPNGBDBM50598611(CHEMBL5187502)
Affinity DataKi:  4nMAssay Description:Binding affinity to TSPO (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetTranslocator protein(Homo sapiens (Human))
Palack£

Curated by ChEMBL
LigandPNGBDBM22032(1-(2-chlorophenyl)-N-methyl-N-(1-methylpropyl)isoq...)
Affinity DataKi:  4.5nMAssay Description:Inhibition of human TSPOMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Homo sapiens (Human))
Palack£

Curated by ChEMBL
LigandPNGBDBM50229596(1-(2-chlorophenyl)-N-methyl-N-[(1S)-1-methylpropyl...)
Affinity DataKi:  4.5nMAssay Description:Binding affinity to PBR in human mitochondrial tissueMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Homo sapiens (Human))
Palack£

Curated by ChEMBL
LigandPNGBDBM98178(US8492379, 55)
Affinity DataKi:  5nMAssay Description:In vitro binding activity of TSPO.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetTranslocator protein(Homo sapiens (Human))
Palack£

Curated by ChEMBL
LigandPNGBDBM98179(US8492379, 56)
Affinity DataKi:  5.70nMAssay Description:In vitro binding activity of TSPO.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetTranslocator protein(Homo sapiens (Human))
Palack£

Curated by ChEMBL
LigandPNGBDBM50556264(CHEMBL4789235)
Affinity DataKi:  6.20nMAssay Description:Displacement of [3H]-PK11195 from wild type TSPO (unknown origin) expressed in human HEK293T cells assessed as inhibitory constant incubated for 90 m...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTranslocator protein(Homo sapiens (Human))
Palack£

Curated by ChEMBL
LigandPNGBDBM50509027(CHEMBL4459176)
Affinity DataKi:  6.60nMAssay Description:Displacement of [3H]PK11195 from wild-type human TSPO expressed in HEK293 cell membranes after 90 mins by scintillation counting methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTranslocator protein(Homo sapiens (Human))
Palack£

Curated by ChEMBL
LigandPNGBDBM50327238(2-[2-(4'-Methoxyphenyl)-5,7-dimethylpyrazolo[1,5-a...)
Affinity DataKi:  6.70nMAssay Description:Displacement of [3H]PK11195 from TSPO in human T98G cell membranes incubated for 90 mins by competition radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Displayed 1 to 50 (of 258 total ) | Next | Last >>
Jump to: