TargetO94806/P05129/P05771/P17252/P24723/P41743/Q02156/Q04759/Q05513/Q05655/Q15139(Homo sapiens (Human))
Toho University
Curated by ChEMBL
Toho University
Curated by ChEMBL
Affinity DataEC50: 0.190nMAssay Description:Agonist activity at Protein kinase C in human U1 cells infected with HIV-1 NL4-3 assessed as induction of HIV-1 p24 production after 72 hrs by ELISAMore data for this Ligand-Target Pair
TargetO94806/P05129/P05771/P17252/P24723/P41743/Q02156/Q04759/Q05513/Q05655/Q15139(Homo sapiens (Human))
Toho University
Curated by ChEMBL
Toho University
Curated by ChEMBL
Affinity DataEC50: 0.550nMAssay Description:Agonist activity at Protein kinase C in human U1 cells infected with HIV-1 NL4-3 assessed as induction of HIV-1 p24 production after 72 hrs by ELISAMore data for this Ligand-Target Pair
TargetO94806/P05129/P05771/P17252/P24723/P41743/Q02156/Q04759/Q05513/Q05655/Q15139(Homo sapiens (Human))
Toho University
Curated by ChEMBL
Toho University
Curated by ChEMBL
Affinity DataEC50: 0.600nMAssay Description:Agonist activity at Protein kinase C in human U1 cells infected with HIV-1 NL4-3 assessed as induction of HIV-1 p24 production after 72 hrs by ELISAMore data for this Ligand-Target Pair
Affinity DataEC50: 2.5nMAssay Description:Activation of PKCdelta (unknown origin) after 40 minsMore data for this Ligand-Target Pair
Affinity DataEC50: 2.90nMAssay Description:Activation of PKCdelta (unknown origin) using phosphatidylserine as substrateMore data for this Ligand-Target Pair
Affinity DataEC50: 3.30nMAssay Description:Activation of PKCdelta (unknown origin) after 40 minsMore data for this Ligand-Target Pair
Affinity DataEC50: 3.70nMAssay Description:Activation of PKCdelta (unknown origin) after 40 minsMore data for this Ligand-Target Pair
Affinity DataEC50: 3.80nMAssay Description:Activation of PKCdelta (unknown origin) after 40 minsMore data for this Ligand-Target Pair
TargetO94806/P05129/P05771/P17252/P24723/P41743/Q02156/Q04759/Q05513/Q05655/Q15139(Homo sapiens (Human))
Toho University
Curated by ChEMBL
Toho University
Curated by ChEMBL
Affinity DataEC50: >3.90nMAssay Description:Agonist activity at Protein kinase C in human U1 cells infected with HIV-1 NL4-3 assessed as induction of HIV-1 p24 production after 72 hrs by ELISAMore data for this Ligand-Target Pair
Affinity DataEC50: 4.10nMAssay Description:Activation of PKCdelta (unknown origin) using phosphatidylserine as substrateMore data for this Ligand-Target Pair
Affinity DataEC50: 4.10nMAssay Description:Activation of PKCdelta (unknown origin) after 40 minsMore data for this Ligand-Target Pair
Affinity DataEC50: 4.20nMAssay Description:Activation of PKCdelta (unknown origin) after 40 minsMore data for this Ligand-Target Pair
Affinity DataEC50: 4.5nMAssay Description:Activation of PKCdelta (unknown origin) using phosphatidylserine as substrateMore data for this Ligand-Target Pair
Affinity DataEC50: 4.70nMAssay Description:Activation of PKCdelta (unknown origin) using phosphatidylserine as substrateMore data for this Ligand-Target Pair
Affinity DataEC50: 5.20nMAssay Description:Activation of PKCdelta (unknown origin) using phosphatidylserine as substrateMore data for this Ligand-Target Pair
Affinity DataEC50: 5.30nMAssay Description:Activation of PKCdelta (unknown origin) using phosphatidylserine as substrateMore data for this Ligand-Target Pair
Affinity DataEC50: 5.30nMAssay Description:Activation of PKCdelta (unknown origin) using phosphatidylserine as substrateMore data for this Ligand-Target Pair
Affinity DataEC50: 6.10nMAssay Description:Activation of PKCdelta (unknown origin) after 40 minsMore data for this Ligand-Target Pair
Affinity DataEC50: 7nMpH: 7.4Assay Description:On the day at experiment Human Protein Kinase C delta (PKCδ, Millipore cat#14-504) was diluted in 20 mM HEPES, 0.03% Triton X-100. Amount of enz...More data for this Ligand-Target Pair
Affinity DataEC50: 8nMAssay Description:Activation of PKCdelta (unknown origin) after 40 minsMore data for this Ligand-Target Pair
TargetO94806/P05129/P05771/P17252/P24723/P41743/Q02156/Q04759/Q05513/Q05655/Q15139(Homo sapiens (Human))
Toho University
Curated by ChEMBL
Toho University
Curated by ChEMBL
Affinity DataEC50: 9.5nMAssay Description:Activation of PKC in human platelet assessed as induction of platelet aggregation measured within 15 mins by tribidimetric methodMore data for this Ligand-Target Pair
Affinity DataEC50: 11nMAssay Description:Activation of PKCdelta (unknown origin) using phosphatidylserine as substrateMore data for this Ligand-Target Pair
Affinity DataEC50: 11nMAssay Description:Activation of PKCdelta (unknown origin) after 40 minsMore data for this Ligand-Target Pair
Affinity DataEC50: 13nMAssay Description:Activation of PKCdelta (unknown origin) after 40 minsMore data for this Ligand-Target Pair
Affinity DataEC50: 13nMAssay Description:Activation of PKCdelta (unknown origin) after 40 minsMore data for this Ligand-Target Pair
Affinity DataEC50: 20nMAssay Description:Activation of PKCdelta (unknown origin) after 40 minsMore data for this Ligand-Target Pair
Affinity DataEC50: 26nMAssay Description:Activation of PKCdelta (unknown origin) after 40 minsMore data for this Ligand-Target Pair
TargetO94806/P05129/P05771/P17252/P24723/P41743/Q02156/Q04759/Q05513/Q05655/Q15139(Homo sapiens (Human))
Toho University
Curated by ChEMBL
Toho University
Curated by ChEMBL
Affinity DataEC50: 73nMAssay Description:Activation of PKC in human platelet assessed as induction of platelet aggregation measured within 15 mins by tribidimetric methodMore data for this Ligand-Target Pair
Affinity DataEC50: 80nMpH: 7.4Assay Description:On the day at experiment Human Protein Kinase C delta (PKCδ, Millipore cat#14-504) was diluted in 20 mM HEPES, 0.03% Triton X-100. Amount of enz...More data for this Ligand-Target Pair
Affinity DataEC50: 154nMpH: 7.4Assay Description:On the day at experiment Human Protein Kinase C delta (PKCδ, Millipore cat#14-504) was diluted in 20 mM HEPES, 0.03% Triton X-100. Amount of enz...More data for this Ligand-Target Pair
Affinity DataEC50: 156nMAssay Description:Activation of PKCdelta (unknown origin) after 40 minsMore data for this Ligand-Target Pair
Affinity DataEC50: 290nMAssay Description:Activation of PKCdelta (unknown origin) expressed in HEK293 cells harboring GFP-tagged RasGRP3 assessed as phosphorylation at ser299 residues after 3...More data for this Ligand-Target Pair
TargetO94806/P05129/P05771/P17252/P24723/P41743/Q02156/Q04759/Q05513/Q05655/Q15139(Homo sapiens (Human))
Toho University
Curated by ChEMBL
Toho University
Curated by ChEMBL
Affinity DataEC50: 910nMAssay Description:Activation of PKC in human platelet assessed as induction of platelet aggregation measured within 15 mins by tribidimetric methodMore data for this Ligand-Target Pair
Affinity DataEC50: 988nMAssay Description:Activation of PKCdelta (unknown origin) after 40 minsMore data for this Ligand-Target Pair
Affinity DataEC50: 1.11E+3nMpH: 7.4Assay Description:On the day at experiment Human Protein Kinase C delta (PKCδ, Millipore cat#14-504) was diluted in 20 mM HEPES, 0.03% Triton X-100. Amount of enz...More data for this Ligand-Target Pair
TargetO94806/P05129/P05771/P17252/P24723/P41743/Q02156/Q04759/Q05513/Q05655/Q15139(Homo sapiens (Human))
Toho University
Curated by ChEMBL
Toho University
Curated by ChEMBL
Affinity DataEC50: 5.04E+3nMAssay Description:Activation of PKC in human platelet assessed as induction of platelet aggregation measured within 15 mins by tribidimetric methodMore data for this Ligand-Target Pair
Affinity DataEC50: 5.17E+3nMAssay Description:Binding affinity to GST-tagged PKCdelta expressed in Escherichia coli BL21(DE3) by fluorescence quenchingMore data for this Ligand-Target Pair
TargetO94806/P05129/P05771/P17252/P24723/P41743/Q02156/Q04759/Q05513/Q05655/Q15139(Homo sapiens (Human))
Toho University
Curated by ChEMBL
Toho University
Curated by ChEMBL
Affinity DataEC50: 6.08E+3nMAssay Description:Activation of PKC in human platelet assessed as induction of platelet aggregation measured within 15 mins by tribidimetric methodMore data for this Ligand-Target Pair
Affinity DataEC50: 7.49E+3nMAssay Description:Binding affinity to GST-tagged PKCdelta expressed in Escherichia coli BL21(DE3) by fluorescence quenchingMore data for this Ligand-Target Pair
Affinity DataEC50: 8.03E+3nMAssay Description:Activation of PKCdelta (unknown origin) expressed in human LNCAP cells harboring GFP-tagged RasGRP1 assessed as phosphorylation at ser299 residues af...More data for this Ligand-Target Pair
Affinity DataEC50: 8.28E+3nMAssay Description:Activation of PKCdelta (unknown origin) expressed in human LNCAP cells harboring GFP-tagged RasGRP3 assessed as phosphorylation at ser299 residues af...More data for this Ligand-Target Pair
Affinity DataEC50: 8.69E+3nMAssay Description:Binding affinity to GST-tagged PKCdelta expressed in Escherichia coli BL21(DE3) by fluorescence quenchingMore data for this Ligand-Target Pair
Affinity DataEC50: 8.98E+3nMAssay Description:Binding affinity to GST-tagged PKCdelta expressed in Escherichia coli BL21(DE3) by fluorescence quenchingMore data for this Ligand-Target Pair
Affinity DataEC50: >1.00E+4nMAssay Description:Activation of PKCdelta (unknown origin) after 40 minsMore data for this Ligand-Target Pair
Affinity DataEC50: 1.07E+4nMAssay Description:Binding affinity to GST-tagged PKCdelta expressed in Escherichia coli BL21(DE3) by fluorescence quenchingMore data for this Ligand-Target Pair
Affinity DataEC50: 1.16E+4nMAssay Description:Binding affinity to PKCdelta C1B subdomain after 1 hr by fluorescence quenching analysisMore data for this Ligand-Target Pair
Affinity DataEC50: 1.25E+4nMAssay Description:Binding affinity to GST-tagged PKCdelta expressed in Escherichia coli BL21(DE3) by fluorescence quenchingMore data for this Ligand-Target Pair
Affinity DataEC50: 1.26E+4nMAssay Description:Activation of PKCdelta (unknown origin) expressed in HEK293 cells harboring GFP-tagged RasGRP1 assessed as phosphorylation at ser299 residues after 3...More data for this Ligand-Target Pair
Affinity DataEC50: 1.50E+4nMAssay Description:Binding affinity to PKCdelta C1B subdomain after 1 hr by fluorescence quenching analysisMore data for this Ligand-Target Pair
Affinity DataEC50: 1.62E+4nMAssay Description:Binding affinity to GST-tagged PKCdelta expressed in Escherichia coli BL21(DE3) by fluorescence quenchingMore data for this Ligand-Target Pair