TargetCalcitonin gene-related peptide 1(Homo sapiens (Human))
Bristol-Myers Squibb Discovery
Curated by ChEMBL
Bristol-Myers Squibb Discovery
Curated by ChEMBL
Affinity DataIC50: 0.110nMAssay Description:Displacement of [125I]CGRP from alpha CGRP in human SK-N-MC cells after 2 hrs by scintillation counterMore data for this Ligand-Target Pair
TargetCalcitonin gene-related peptide 1(Homo sapiens (Human))
Bristol-Myers Squibb Discovery
Curated by ChEMBL
Bristol-Myers Squibb Discovery
Curated by ChEMBL
Affinity DataIC50: 0.120nMAssay Description:Inhibition of human CGRP receptor expressed in huamn HEK293 cells coexpressing CLR/RAMP1 assessed as inhibition of CGRP-stimulated cAMP production af...More data for this Ligand-Target Pair
TargetCalcitonin gene-related peptide 1(Homo sapiens (Human))
Bristol-Myers Squibb Discovery
Curated by ChEMBL
Bristol-Myers Squibb Discovery
Curated by ChEMBL
Affinity DataIC50: 0.200nMAssay Description:Antagonist activity at human CGRP1 receptor in human SK-N-MC cells assessed as effect on human alpha-CGRP-induced cAMP accumulationMore data for this Ligand-Target Pair
TargetCalcitonin gene-related peptide 1(Homo sapiens (Human))
Bristol-Myers Squibb Discovery
Curated by ChEMBL
Bristol-Myers Squibb Discovery
Curated by ChEMBL
Affinity DataIC50: 0.230nMAssay Description:Displacement of [125I]CGRP from alpha CGRP in human SK-N-MC cells after 2 hrs by scintillation counterMore data for this Ligand-Target Pair
TargetCalcitonin gene-related peptide 1(Homo sapiens (Human))
Bristol-Myers Squibb Discovery
Curated by ChEMBL
Bristol-Myers Squibb Discovery
Curated by ChEMBL
Affinity DataIC50: 0.530nMAssay Description:Antagonist activity at human CGRP1 receptor in human SK-N-MC cells assessed as effect on human alpha-CGRP-induced cAMP accumulationMore data for this Ligand-Target Pair
TargetCalcitonin gene-related peptide 1(Homo sapiens (Human))
Bristol-Myers Squibb Discovery
Curated by ChEMBL
Bristol-Myers Squibb Discovery
Curated by ChEMBL
Affinity DataIC50: 0.570nMAssay Description:Antagonist activity at human CGRP1 receptor in human SK-N-MC cells assessed as effect on human alpha-CGRP-induced cAMP accumulationMore data for this Ligand-Target Pair
TargetCalcitonin gene-related peptide 1(Homo sapiens (Human))
Bristol-Myers Squibb Discovery
Curated by ChEMBL
Bristol-Myers Squibb Discovery
Curated by ChEMBL
Affinity DataIC50: 0.580nMAssay Description:Antagonist activity at human CGRP1 receptor in human SK-N-MC cells assessed as effect on human alpha-CGRP-induced cAMP accumulationMore data for this Ligand-Target Pair
TargetCalcitonin gene-related peptide 1(Homo sapiens (Human))
Bristol-Myers Squibb Discovery
Curated by ChEMBL
Bristol-Myers Squibb Discovery
Curated by ChEMBL
Affinity DataIC50: 0.640nMAssay Description:Antagonist activity at human CGRP1 receptor in human SK-N-MC cells assessed as effect on human alpha-CGRP-induced cAMP accumulationMore data for this Ligand-Target Pair
TargetCalcitonin gene-related peptide 1(Homo sapiens (Human))
Bristol-Myers Squibb Discovery
Curated by ChEMBL
Bristol-Myers Squibb Discovery
Curated by ChEMBL
Affinity DataIC50: 0.710nMAssay Description:Antagonist activity at human CGRP1 receptor in human SK-N-MC cells assessed as effect on human alpha-CGRP-induced cAMP accumulationMore data for this Ligand-Target Pair
TargetCalcitonin gene-related peptide 1(Homo sapiens (Human))
Bristol-Myers Squibb Discovery
Curated by ChEMBL
Bristol-Myers Squibb Discovery
Curated by ChEMBL
Affinity DataIC50: 0.790nMAssay Description:Antagonist activity at human CGRP1 receptor in human SK-N-MC cells assessed as effect on human alpha-CGRP-induced cAMP accumulationMore data for this Ligand-Target Pair
TargetCalcitonin gene-related peptide 1(Homo sapiens (Human))
Bristol-Myers Squibb Discovery
Curated by ChEMBL
Bristol-Myers Squibb Discovery
Curated by ChEMBL
Affinity DataIC50: 0.850nMAssay Description:Antagonist activity at human CGRP1 receptor in human SK-N-MC cells assessed as effect on human alpha-CGRP-induced cAMP accumulationMore data for this Ligand-Target Pair
TargetCalcitonin gene-related peptide 1(Homo sapiens (Human))
Bristol-Myers Squibb Discovery
Curated by ChEMBL
Bristol-Myers Squibb Discovery
Curated by ChEMBL
Affinity DataIC50: 1nMAssay Description:Antagonist activity at human CGRP1 receptor in human SK-N-MC cells assessed as effect on human alpha-CGRP-induced cAMP accumulationMore data for this Ligand-Target Pair
TargetCalcitonin gene-related peptide 1(Homo sapiens (Human))
Bristol-Myers Squibb Discovery
Curated by ChEMBL
Bristol-Myers Squibb Discovery
Curated by ChEMBL
Affinity DataIC50: 1.10nMAssay Description:Displacement of [125I]CGRP from alpha CGRP in human SK-N-MC cells after 2 hrs by scintillation counterMore data for this Ligand-Target Pair
TargetCalcitonin gene-related peptide 1(Homo sapiens (Human))
Bristol-Myers Squibb Discovery
Curated by ChEMBL
Bristol-Myers Squibb Discovery
Curated by ChEMBL
Affinity DataIC50: 1.30nMAssay Description:Antagonist activity at human CGRP1 receptor in human SK-N-MC cells assessed as effect on human alpha-CGRP-induced cAMP accumulationMore data for this Ligand-Target Pair
TargetCalcitonin gene-related peptide 1(Homo sapiens (Human))
Bristol-Myers Squibb Discovery
Curated by ChEMBL
Bristol-Myers Squibb Discovery
Curated by ChEMBL
Affinity DataIC50: 1.30nMAssay Description:Antagonist activity at human CGRP1 receptor in human SK-N-MC cells assessed as effect on human alpha-CGRP-induced cAMP accumulationMore data for this Ligand-Target Pair
TargetCalcitonin gene-related peptide 1(Homo sapiens (Human))
Bristol-Myers Squibb Discovery
Curated by ChEMBL
Bristol-Myers Squibb Discovery
Curated by ChEMBL
Affinity DataIC50: 1.60nMAssay Description:Antagonist activity at human CGRP1 receptor in human SK-N-MC cells assessed as effect on human alpha-CGRP-induced cAMP accumulationMore data for this Ligand-Target Pair
TargetCalcitonin gene-related peptide 1(Homo sapiens (Human))
Bristol-Myers Squibb Discovery
Curated by ChEMBL
Bristol-Myers Squibb Discovery
Curated by ChEMBL
Affinity DataIC50: 1.70nMAssay Description:Antagonist activity at human CGRP1 receptor in human SK-N-MC cells assessed as effect on human alpha-CGRP-induced cAMP accumulationMore data for this Ligand-Target Pair
TargetCalcitonin gene-related peptide 1(Homo sapiens (Human))
Bristol-Myers Squibb Discovery
Curated by ChEMBL
Bristol-Myers Squibb Discovery
Curated by ChEMBL
Affinity DataIC50: 1.70nMAssay Description:Antagonist activity at human CGRP1 receptor in human SK-N-MC cells assessed as effect on human alpha-CGRP-induced cAMP accumulationMore data for this Ligand-Target Pair
TargetCalcitonin gene-related peptide 1(Homo sapiens (Human))
Bristol-Myers Squibb Discovery
Curated by ChEMBL
Bristol-Myers Squibb Discovery
Curated by ChEMBL
Affinity DataIC50: 1.80nMAssay Description:Antagonist activity at human CGRP1 receptor in human SK-N-MC cells assessed as effect on human alpha-CGRP-induced cAMP accumulationMore data for this Ligand-Target Pair
TargetCalcitonin gene-related peptide 1(Homo sapiens (Human))
Bristol-Myers Squibb Discovery
Curated by ChEMBL
Bristol-Myers Squibb Discovery
Curated by ChEMBL
Affinity DataIC50: 2nMAssay Description:Antagonist activity at human CGRP1 receptor in human SK-N-MC cells assessed as effect on human alpha-CGRP-induced cAMP accumulationMore data for this Ligand-Target Pair
TargetCalcitonin gene-related peptide 1(Homo sapiens (Human))
Bristol-Myers Squibb Discovery
Curated by ChEMBL
Bristol-Myers Squibb Discovery
Curated by ChEMBL
Affinity DataIC50: 2.10nMAssay Description:Antagonist activity at human CGRP1 receptor in human SK-N-MC cells assessed as effect on human alpha-CGRP-induced cAMP accumulationMore data for this Ligand-Target Pair
TargetCalcitonin gene-related peptide 1(Homo sapiens (Human))
Bristol-Myers Squibb Discovery
Curated by ChEMBL
Bristol-Myers Squibb Discovery
Curated by ChEMBL
Affinity DataIC50: 2.20nMAssay Description:Antagonist activity at human CGRP1 receptor in human SK-N-MC cells assessed as effect on human alpha-CGRP-induced cAMP accumulationMore data for this Ligand-Target Pair
TargetCalcitonin gene-related peptide 1(Homo sapiens (Human))
Bristol-Myers Squibb Discovery
Curated by ChEMBL
Bristol-Myers Squibb Discovery
Curated by ChEMBL
Affinity DataIC50: 2.20nMAssay Description:Inhibition of human CGRP receptor expressed in huamn HEK293 cells coexpressing CLR/RAMP1 assessed as inhibition of CGRP-stimulated cAMP production af...More data for this Ligand-Target Pair
TargetCalcitonin gene-related peptide 1(Homo sapiens (Human))
Bristol-Myers Squibb Discovery
Curated by ChEMBL
Bristol-Myers Squibb Discovery
Curated by ChEMBL
Affinity DataIC50: 2.20nMAssay Description:Antagonist activity at human CGRP1 receptor in human SK-N-MC cells assessed as effect on human alpha-CGRP-induced cAMP accumulationMore data for this Ligand-Target Pair
TargetCalcitonin gene-related peptide 1(Homo sapiens (Human))
Bristol-Myers Squibb Discovery
Curated by ChEMBL
Bristol-Myers Squibb Discovery
Curated by ChEMBL
Affinity DataIC50: 2.90nMAssay Description:Displacement of [125I]CGRP from alpha CGRP in human SK-N-MC cells after 2 hrs by scintillation counterMore data for this Ligand-Target Pair
TargetCalcitonin gene-related peptide 1(Homo sapiens (Human))
Bristol-Myers Squibb Discovery
Curated by ChEMBL
Bristol-Myers Squibb Discovery
Curated by ChEMBL
Affinity DataIC50: 3.5nMAssay Description:Antagonist activity at human CGRP1 receptor in human SK-N-MC cells assessed as effect on human alpha-CGRP-induced cAMP accumulationMore data for this Ligand-Target Pair
TargetCalcitonin gene-related peptide 1(Homo sapiens (Human))
Bristol-Myers Squibb Discovery
Curated by ChEMBL
Bristol-Myers Squibb Discovery
Curated by ChEMBL
Affinity DataIC50: 3.5nMAssay Description:Antagonist activity at human CGRP1 receptor in human SK-N-MC cells assessed as effect on human alpha-CGRP-induced cAMP accumulationMore data for this Ligand-Target Pair
TargetCalcitonin gene-related peptide 1(Homo sapiens (Human))
Bristol-Myers Squibb Discovery
Curated by ChEMBL
Bristol-Myers Squibb Discovery
Curated by ChEMBL
Affinity DataIC50: 3.60nMAssay Description:Antagonist activity at human CGRP1 receptor in human SK-N-MC cells assessed as effect on human alpha-CGRP-induced cAMP accumulationMore data for this Ligand-Target Pair
TargetCalcitonin gene-related peptide 1(Homo sapiens (Human))
Bristol-Myers Squibb Discovery
Curated by ChEMBL
Bristol-Myers Squibb Discovery
Curated by ChEMBL
Affinity DataIC50: 3.80nMAssay Description:Antagonist activity at human CGRP1 receptor in human SK-N-MC cells assessed as effect on human alpha-CGRP-induced cAMP accumulationMore data for this Ligand-Target Pair
TargetCalcitonin gene-related peptide 1(Homo sapiens (Human))
Bristol-Myers Squibb Discovery
Curated by ChEMBL
Bristol-Myers Squibb Discovery
Curated by ChEMBL
Affinity DataIC50: 4.20nMAssay Description:Antagonist activity at human CGRP1 receptor in human SK-N-MC cells assessed as effect on human alpha-CGRP-induced cAMP accumulationMore data for this Ligand-Target Pair
TargetCalcitonin gene-related peptide 1(Homo sapiens (Human))
Bristol-Myers Squibb Discovery
Curated by ChEMBL
Bristol-Myers Squibb Discovery
Curated by ChEMBL
Affinity DataIC50: 4.30nMAssay Description:Displacement of [125I]CGRP from alpha CGRP in human SK-N-MC cells after 2 hrs by scintillation counterMore data for this Ligand-Target Pair
TargetCalcitonin gene-related peptide 1(Homo sapiens (Human))
Bristol-Myers Squibb Discovery
Curated by ChEMBL
Bristol-Myers Squibb Discovery
Curated by ChEMBL
Affinity DataIC50: 4.90nMAssay Description:Antagonist activity at human CGRP1 receptor in human SK-N-MC cells assessed as effect on human alpha-CGRP-induced cAMP accumulationMore data for this Ligand-Target Pair
TargetCalcitonin gene-related peptide 1(Homo sapiens (Human))
Bristol-Myers Squibb Discovery
Curated by ChEMBL
Bristol-Myers Squibb Discovery
Curated by ChEMBL
Affinity DataIC50: 5nMAssay Description:Antagonist activity at human CGRP1 receptor in human SK-N-MC cells assessed as effect on human alpha-CGRP-induced cAMP accumulationMore data for this Ligand-Target Pair
TargetCalcitonin gene-related peptide 1(Homo sapiens (Human))
Bristol-Myers Squibb Discovery
Curated by ChEMBL
Bristol-Myers Squibb Discovery
Curated by ChEMBL
Affinity DataIC50: 7nMAssay Description:Displacement of [125I]CGRP from alpha CGRP in human SK-N-MC cells after 2 hrs by scintillation counterMore data for this Ligand-Target Pair
TargetCalcitonin gene-related peptide 1(Homo sapiens (Human))
Bristol-Myers Squibb Discovery
Curated by ChEMBL
Bristol-Myers Squibb Discovery
Curated by ChEMBL
Affinity DataIC50: 8.90nMAssay Description:Displacement of [125I]CGRP from alpha CGRP in human SK-N-MC cells after 2 hrs by scintillation counterMore data for this Ligand-Target Pair
TargetCalcitonin gene-related peptide 1(Homo sapiens (Human))
Bristol-Myers Squibb Discovery
Curated by ChEMBL
Bristol-Myers Squibb Discovery
Curated by ChEMBL
Affinity DataIC50: 9.80nMAssay Description:Displacement of [125I]CGRP from alpha CGRP in human SK-N-MC cells after 2 hrs by scintillation counterMore data for this Ligand-Target Pair
TargetCalcitonin gene-related peptide 1(Homo sapiens (Human))
Bristol-Myers Squibb Discovery
Curated by ChEMBL
Bristol-Myers Squibb Discovery
Curated by ChEMBL
Affinity DataIC50: 11nMAssay Description:Antagonist activity at human CGRP1 receptor in human SK-N-MC cells assessed as effect on human alpha-CGRP-induced cAMP accumulationMore data for this Ligand-Target Pair
TargetCalcitonin gene-related peptide 1(Homo sapiens (Human))
Bristol-Myers Squibb Discovery
Curated by ChEMBL
Bristol-Myers Squibb Discovery
Curated by ChEMBL
Affinity DataIC50: 12nMAssay Description:Displacement of [125I]CGRP from alpha CGRP in human SK-N-MC cells after 2 hrs by scintillation counterMore data for this Ligand-Target Pair
TargetCalcitonin gene-related peptide 1(Homo sapiens (Human))
Bristol-Myers Squibb Discovery
Curated by ChEMBL
Bristol-Myers Squibb Discovery
Curated by ChEMBL
Affinity DataIC50: 12nMAssay Description:Displacement of [125I]CGRP from alpha CGRP in human SK-N-MC cells after 2 hrs by scintillation counterMore data for this Ligand-Target Pair
TargetCalcitonin gene-related peptide 1(Homo sapiens (Human))
Bristol-Myers Squibb Discovery
Curated by ChEMBL
Bristol-Myers Squibb Discovery
Curated by ChEMBL
Affinity DataIC50: 13nMAssay Description:Displacement of [125I]CGRP from alpha CGRP in human SK-N-MC cells after 2 hrs by scintillation counterMore data for this Ligand-Target Pair
TargetCalcitonin gene-related peptide 1(Homo sapiens (Human))
Bristol-Myers Squibb Discovery
Curated by ChEMBL
Bristol-Myers Squibb Discovery
Curated by ChEMBL
Affinity DataIC50: 14nMAssay Description:Displacement of [125I]CGRP from alpha CGRP in human SK-N-MC cells after 2 hrs by scintillation counterMore data for this Ligand-Target Pair
TargetCalcitonin gene-related peptide 1(Homo sapiens (Human))
Bristol-Myers Squibb Discovery
Curated by ChEMBL
Bristol-Myers Squibb Discovery
Curated by ChEMBL
Affinity DataIC50: 15nMAssay Description:Displacement of [125I]CGRP from alpha CGRP in human SK-N-MC cells after 2 hrs by scintillation counterMore data for this Ligand-Target Pair
TargetCalcitonin gene-related peptide 1(Homo sapiens (Human))
Bristol-Myers Squibb Discovery
Curated by ChEMBL
Bristol-Myers Squibb Discovery
Curated by ChEMBL
Affinity DataIC50: 16nMAssay Description:Displacement of [125I]CGRP from alpha CGRP in human SK-N-MC cells after 2 hrs by scintillation counterMore data for this Ligand-Target Pair
TargetCalcitonin gene-related peptide 1(Homo sapiens (Human))
Bristol-Myers Squibb Discovery
Curated by ChEMBL
Bristol-Myers Squibb Discovery
Curated by ChEMBL
Affinity DataIC50: 19nMAssay Description:Displacement of [125I]CGRP from alpha CGRP in human SK-N-MC cells after 2 hrs by scintillation counterMore data for this Ligand-Target Pair
TargetCalcitonin gene-related peptide 1(Homo sapiens (Human))
Bristol-Myers Squibb Discovery
Curated by ChEMBL
Bristol-Myers Squibb Discovery
Curated by ChEMBL
Affinity DataIC50: 19nMAssay Description:Displacement of [125I]CGRP from alpha CGRP in human SK-N-MC cells after 2 hrs by scintillation counterMore data for this Ligand-Target Pair
TargetCalcitonin gene-related peptide 1(Homo sapiens (Human))
Bristol-Myers Squibb Discovery
Curated by ChEMBL
Bristol-Myers Squibb Discovery
Curated by ChEMBL
Affinity DataIC50: 22nMAssay Description:Displacement of [125I]CGRP from alpha CGRP in human SK-N-MC cells after 2 hrs by scintillation counterMore data for this Ligand-Target Pair
TargetCalcitonin gene-related peptide 1(Homo sapiens (Human))
Bristol-Myers Squibb Discovery
Curated by ChEMBL
Bristol-Myers Squibb Discovery
Curated by ChEMBL
Affinity DataIC50: 24nMAssay Description:Displacement of [125I]CGRP from alpha CGRP in human SK-N-MC cells after 2 hrs by scintillation counterMore data for this Ligand-Target Pair
TargetCalcitonin gene-related peptide 1(Homo sapiens (Human))
Bristol-Myers Squibb Discovery
Curated by ChEMBL
Bristol-Myers Squibb Discovery
Curated by ChEMBL
Affinity DataIC50: 30nMAssay Description:Antagonist activity at human CGRP1 receptor in human SK-N-MC cells assessed as effect on human alpha-CGRP-induced cAMP accumulationMore data for this Ligand-Target Pair
TargetCalcitonin gene-related peptide 1(Homo sapiens (Human))
Bristol-Myers Squibb Discovery
Curated by ChEMBL
Bristol-Myers Squibb Discovery
Curated by ChEMBL
Affinity DataIC50: 33nMAssay Description:Displacement of [125I]CGRP from alpha CGRP in human SK-N-MC cells after 2 hrs by scintillation counterMore data for this Ligand-Target Pair
TargetCalcitonin gene-related peptide 1(Homo sapiens (Human))
Bristol-Myers Squibb Discovery
Curated by ChEMBL
Bristol-Myers Squibb Discovery
Curated by ChEMBL
Affinity DataIC50: 34nMAssay Description:Displacement of [125I]CGRP from alpha CGRP in human SK-N-MC cells after 2 hrs by scintillation counterMore data for this Ligand-Target Pair