Target (Institution) | Ligand | Target Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kcal/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Alpha-1A adrenergic receptor (Rattus norvegicus (Rat)) | BDBM50131411![]() (4-(4-Chloro-benzyl)-2-methyl-2H-phthalazin-1-one |...) | KEGG UniProtKB/SwissProt GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars AffyNet ![]() | Article PubMed | n/a | n/a | n/a | n/a | 810 | n/a | n/a | n/a | n/a |
Universidad de Salamanca Curated by ChEMBL | Assay Description Vasorelaxation of noradrenaline-stimulated Wistar rat vas deferens contraction | Bioorg Med Chem Lett 16: 2786-90 (2006) | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Alpha-1A adrenergic receptor (Rattus norvegicus (Rat)) | BDBM50131423![]() (4-Benzyl-2-methyl-2H-phthalazin-1-one | 4-benzyl-2...) | KEGG UniProtKB/SwissProt GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Patents Similars AffyNet ![]() | Article PubMed | n/a | n/a | n/a | n/a | 1.50E+3 | n/a | n/a | n/a | n/a |
Universidad de Salamanca Curated by ChEMBL | Assay Description Vasorelaxation of noradrenaline-stimulated Wistar rat vas deferens contraction | Bioorg Med Chem Lett 16: 2786-90 (2006) | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Alpha-1A adrenergic receptor (Rattus norvegicus (Rat)) | BDBM50131414![]() (4-(benzo[d][1,3]dioxol-5-ylmethyl)phthalazin-1(2H)...) | KEGG UniProtKB/SwissProt GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars AffyNet ![]() | Article PubMed | n/a | n/a | n/a | n/a | 3.00E+3 | n/a | n/a | n/a | n/a |
Universidad de Salamanca Curated by ChEMBL | Assay Description Vasorelaxation of noradrenaline-stimulated Wistar rat vas deferens contraction | Bioorg Med Chem Lett 16: 2786-90 (2006) | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Alpha-1A adrenergic receptor (Rattus norvegicus (Rat)) | BDBM56339![]() (4-(4-chlorobenzyl)-1(2H)-phthalazinone | 4-(4-chlo...) | KEGG UniProtKB/SwissProt GoogleScholar AffyNet ![]() | Purchase CHEMBL PC cid PC sid UniChem Patents Similars AffyNet ![]() | Article PubMed | n/a | n/a | n/a | n/a | 3.90E+3 | n/a | n/a | n/a | n/a |
Universidad de Salamanca Curated by ChEMBL | Assay Description Vasorelaxation of noradrenaline-stimulated Wistar rat vas deferens contraction | Bioorg Med Chem Lett 16: 2786-90 (2006) | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Alpha-1A adrenergic receptor (Rattus norvegicus (Rat)) | BDBM50183665![]() (4-(4-chlorobenzyl)-2-allylphthalazin-1(2H)-one | C...) | KEGG UniProtKB/SwissProt GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars AffyNet ![]() | Article PubMed | n/a | n/a | n/a | n/a | 4.40E+3 | n/a | n/a | n/a | n/a |
Universidad de Salamanca Curated by ChEMBL | Assay Description Vasorelaxation of noradrenaline-stimulated Wistar rat vas deferens contraction | Bioorg Med Chem Lett 16: 2786-90 (2006) | |||||||||||
More data for this Ligand-Target Pair |