Target (Institution) | Ligand | Target Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kcal/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Human diphtheria toxin-like ADP-ribosyltransferase (ARTD8 or PARP14) (Homo sapiens (Human)) | BDBM50397960![]() (CHEMBL2179989) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid PDB UniChem Similars AffyNet ![]() | PDB Article PubMed | n/a | n/a | n/a | 7.60E+3 | n/a | n/a | n/a | n/a | n/a |
Ume£ University Curated by ChEMBL | Assay Description Binding affinity at human recombinant ARTD8 expressed in Escherichia coli BL21 (DE3) R3 pRARE cells by isothermal titration calorimetry | J Med Chem 55: 7706-18 (2012) | |||||||||||
More data for this Ligand-Target Pair | ![]() 3D Structure (crystal) | ||||||||||||
Human diphtheria toxin-like ADP-ribosyltransferase (ARTD8 or PARP14) (Homo sapiens (Human)) | BDBM50397961![]() (CHEMBL2179988) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet ![]() | Purchase CHEMBL PC cid PC sid PDB UniChem Similars AffyNet ![]() | PDB Article PubMed | n/a | n/a | n/a | 1.12E+4 | n/a | n/a | n/a | n/a | n/a |
Ume£ University Curated by ChEMBL | Assay Description Binding affinity at human recombinant ARTD8 expressed in Escherichia coli BL21 (DE3) R3 pRARE cells by isothermal titration calorimetry | J Med Chem 55: 7706-18 (2012) | |||||||||||
More data for this Ligand-Target Pair | ![]() 3D Structure (crystal) |