Compile Data Set for Download or QSAR
maximum 50k data
Found 113 of ic50 data for polymerid = 9822
TargetNAD-dependent protein deacylase sirtuin-6(Homo sapiens (Human))
Nagoya City University

Curated by ChEMBL
LigandPNGBDBM50502278(CHEMBL4438193)
Affinity DataIC50:  250nMAssay Description:Inhibition of recombinant human N-terminal polyhis-tagged SIRT6 (1 to 355 residues) defatty-acylase activity expressed in Escherichia coli using SFP3...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNAD-dependent protein deacylase sirtuin-6(Homo sapiens (Human))
Nagoya City University

Curated by ChEMBL
LigandPNGBDBM50408842(CHEMBL5277251)
Affinity DataIC50:  256nMAssay Description:Inhibition of human recombinant FAAHMore data for this Ligand-Target Pair
In DepthDetails
TargetNAD-dependent protein deacylase sirtuin-6(Homo sapiens (Human))
Nagoya City University

Curated by ChEMBL
LigandPNGBDBM50408843(CHEMBL5274589)
Affinity DataIC50:  282nMAssay Description:Inhibition of human recombinant FAAHMore data for this Ligand-Target Pair
In DepthDetails
TargetNAD-dependent protein deacylase sirtuin-6(Homo sapiens (Human))
Nagoya City University

Curated by ChEMBL
LigandPNGBDBM50408841(CHEMBL5281352)
Affinity DataIC50:  319nMAssay Description:Inhibition of human recombinant FAAHMore data for this Ligand-Target Pair
In DepthDetails
TargetNAD-dependent protein deacylase sirtuin-6(Homo sapiens (Human))
Nagoya City University

Curated by ChEMBL
LigandPNGBDBM50408845(CHEMBL5267327)
Affinity DataIC50:  319nMAssay Description:Inhibition of human recombinant FAAHMore data for this Ligand-Target Pair
In DepthDetails
TargetNAD-dependent protein deacylase sirtuin-6(Homo sapiens (Human))
Nagoya City University

Curated by ChEMBL
LigandPNGBDBM50408841(CHEMBL5281352)
Affinity DataIC50:  319nMAssay Description:Inhibition of human recombinant MGLMore data for this Ligand-Target Pair
In DepthDetails
TargetNAD-dependent protein deacylase sirtuin-6(Homo sapiens (Human))
Nagoya City University

Curated by ChEMBL
LigandPNGBDBM50408844(CHEMBL5280037)
Affinity DataIC50:  368nMAssay Description:Inhibition of rat brain FAAHMore data for this Ligand-Target Pair
In DepthDetails
TargetNAD-dependent protein deacylase sirtuin-6(Homo sapiens (Human))
Nagoya City University

Curated by ChEMBL
LigandPNGBDBM50408846(CHEMBL5270531)
Affinity DataIC50:  495nMAssay Description:Antagonist activity at human adenosine A1 receptor expressed in CHO FlpIn cells assessed as inhibition of of N(6)-(R-phenylisopropyl)adenosine-induce...More data for this Ligand-Target Pair
In DepthDetails
TargetNAD-dependent protein deacylase sirtuin-6(Homo sapiens (Human))
Nagoya City University

Curated by ChEMBL
LigandPNGBDBM50540059(CHEMBL4645806)
Affinity DataIC50:  1.70E+3nMAssay Description:Inhibition of sirtuin 6 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNAD-dependent protein deacylase sirtuin-6(Homo sapiens (Human))
Nagoya City University

Curated by ChEMBL
LigandPNGBDBM7459(2-(3,4-dihydroxyphenyl)-5,7-dihydroxy-4H-chromen-4...)
Affinity DataIC50:  1.90E+3nMAssay Description:Antagonist activity at histamine H3 receptor in electrically-stimulated guinea pig ileumMore data for this Ligand-Target Pair
In DepthDetails
TargetNAD-dependent protein deacylase sirtuin-6(Homo sapiens (Human))
Nagoya City University

Curated by ChEMBL
LigandPNGBDBM7460(2-(3,4-dihydroxyphenyl)-3,5,7-trihydroxy-4H-chrome...)
Affinity DataIC50:  1.90E+3nMAssay Description:Antagonist activity at histamine H3 receptor in electrically-stimulated guinea pig ileumMore data for this Ligand-Target Pair
In DepthDetails PDB3D3D Structure (crystal)
TargetNAD-dependent protein deacylase sirtuin-6(Homo sapiens (Human))
Nagoya City University

Curated by ChEMBL
LigandPNGBDBM50135169((-)-Catechin gallate | (2S,3R)-2-(3,4-dihydroxyphe...)
Affinity DataIC50:  2.50E+3nMAssay Description:Antagonist activity at adrenergic Alpha-1B receptor in guinea pig spleenMore data for this Ligand-Target Pair
In DepthDetails
TargetNAD-dependent protein deacylase sirtuin-6(Homo sapiens (Human))
Nagoya City University

Curated by ChEMBL
LigandPNGBDBM50135169((-)-Catechin gallate | (2S,3R)-2-(3,4-dihydroxyphe...)
Affinity DataIC50:  2.50E+3nMAssay Description:Antagonist activity at adrenergic alpha1A receptor in rat tail arteryMore data for this Ligand-Target Pair
In DepthDetails
TargetNAD-dependent protein deacylase sirtuin-6(Homo sapiens (Human))
Nagoya City University

Curated by ChEMBL
LigandPNGBDBM50276143(CHEMBL4128547)
Affinity DataIC50:  2.80E+3nMAssay Description:Inhibition of sirtuin 6 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNAD-dependent protein deacylase sirtuin-6(Homo sapiens (Human))
Nagoya City University

Curated by ChEMBL
LigandPNGBDBM50276143(CHEMBL4128547)
Affinity DataIC50:  2.80E+3nMAssay Description:Inhibition of human SIRT6 (1 to 294 residues) expressed in Escherichia coli Rosetta (DE3) using H3K9AcWW as substrate preincubated for 15 mins follow...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNAD-dependent protein deacylase sirtuin-6(Homo sapiens (Human))
Nagoya City University

Curated by ChEMBL
LigandPNGBDBM50544037(CHEMBL1370863)
Affinity DataIC50:  4.93E+3nMAssay Description:Inhibition of SIRT6 (unknown origin) using Ac-RYQK(Ac)-AMC as substrate by Fluor de Lys assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNAD-dependent protein deacylase sirtuin-6(Homo sapiens (Human))
Nagoya City University

Curated by ChEMBL
LigandPNGBDBM50236531((-)-gallocatechin gallate | (2R,3S)-5,7-dihydroxy-...)
Affinity DataIC50:  5.40E+3nMAssay Description:Antagonist activity at adrenergic Alpha-1B receptor in guinea pig spleenMore data for this Ligand-Target Pair
In DepthDetails
TargetNAD-dependent protein deacylase sirtuin-6(Homo sapiens (Human))
Nagoya City University

Curated by ChEMBL
LigandPNGBDBM50408847(CHEMBL5281841)
Affinity DataIC50:  6.70E+3nMAssay Description:Antagonist activity at adrenergic alpha1A receptor in rat tail arteryMore data for this Ligand-Target Pair
In DepthDetails
TargetNAD-dependent protein deacylase sirtuin-6(Homo sapiens (Human))
Nagoya City University

Curated by ChEMBL
LigandPNGBDBM50518647(CHEMBL4440955)
Affinity DataIC50:  7.90E+3nMAssay Description:Inhibition of demyristoylation activity of recombinant human full length N-terminal His6-tagged SIRT6 expressed in Escherichia coli using H2N-EALPK-[...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNAD-dependent protein deacylase sirtuin-6(Homo sapiens (Human))
Nagoya City University

Curated by ChEMBL
LigandPNGBDBM50408836(CHEMBL5270371)
Affinity DataIC50:  8.10E+3nMAssay Description:Antagonist activity at histamine H3 receptor in electrically-stimulated guinea pig ileumMore data for this Ligand-Target Pair
In DepthDetails
TargetNAD-dependent protein deacylase sirtuin-6(Homo sapiens (Human))
Nagoya City University

Curated by ChEMBL
LigandPNGBDBM50544040(CHEMBL4638368)
Affinity DataIC50:  9.09E+3nMAssay Description:Inhibition of SIRT6 (unknown origin) using Ac-RYQK(Ac)-AMC as substrate by Fluor de Lys assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNAD-dependent protein deacylase sirtuin-6(Homo sapiens (Human))
Nagoya City University

Curated by ChEMBL
LigandPNGBDBM50544045(CHEMBL4636099)
Affinity DataIC50:  9.46E+3nMAssay Description:Inhibition of SIRT6 (unknown origin) using Ac-RYQK(Ac)-AMC as substrate by Fluor de Lys assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNAD-dependent protein deacylase sirtuin-6(Homo sapiens (Human))
Nagoya City University

Curated by ChEMBL
LigandPNGBDBM50544039(CHEMBL4638821)
Affinity DataIC50:  1.10E+4nMAssay Description:Inhibition of SIRT6 (unknown origin) using Ac-RYQK(Ac)-AMC as substrate by Fluor de Lys assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNAD-dependent protein deacylase sirtuin-6(Homo sapiens (Human))
Nagoya City University

Curated by ChEMBL
LigandPNGBDBM50518648(CHEMBL4438364)
Affinity DataIC50:  1.12E+4nMAssay Description:Inhibition of demyristoylation activity of recombinant human full length N-terminal His6-tagged SIRT6 expressed in Escherichia coli using H2N-EALPK-[...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNAD-dependent protein deacylase sirtuin-6(Homo sapiens (Human))
Nagoya City University

Curated by ChEMBL
LigandPNGBDBM50544041(CHEMBL4642889)
Affinity DataIC50:  1.24E+4nMAssay Description:Inhibition of SIRT6 (unknown origin) using Ac-RYQK(Ac)-AMC as substrate by Fluor de Lys assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNAD-dependent protein deacylase sirtuin-6(Homo sapiens (Human))
Nagoya City University

Curated by ChEMBL
LigandPNGBDBM50544038(CHEMBL249033 | US11459308, Compound 3514)
Affinity DataIC50:  1.25E+4nMAssay Description:Inhibition of SIRT6 (unknown origin) using Ac-RYQK(Ac)-AMC as substrate by Fluor de Lys assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNAD-dependent protein deacylase sirtuin-6(Homo sapiens (Human))
Nagoya City University

Curated by ChEMBL
LigandPNGBDBM50544042(CHEMBL4637552)
Affinity DataIC50:  1.68E+4nMAssay Description:Inhibition of SIRT6 (unknown origin) using Ac-RYQK(Ac)-AMC as substrate by Fluor de Lys assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNAD-dependent protein deacylase sirtuin-6(Homo sapiens (Human))
Nagoya City University

Curated by ChEMBL
LigandPNGBDBM50544044(CHEMBL4641736)
Affinity DataIC50:  1.75E+4nMAssay Description:Inhibition of SIRT6 (unknown origin) using Ac-RYQK(Ac)-AMC as substrate by Fluor de Lys assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNAD-dependent protein deacylase sirtuin-6(Homo sapiens (Human))
Nagoya City University

Curated by ChEMBL
LigandPNGBDBM50276139(CHEMBL4128509)
Affinity DataIC50: >2.00E+4nMAssay Description:Inhibition of human SIRT6 (1 to 294 residues) expressed in Escherichia coli Rosetta (DE3) using H3K9AcWW as substrate preincubated for 15 mins follow...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNAD-dependent protein deacylase sirtuin-6(Homo sapiens (Human))
Nagoya City University

Curated by ChEMBL
LigandPNGBDBM50451276(CHEMBL4217987)
Affinity DataIC50:  2.00E+4nMAssay Description:Inhibition of human recombinant SIRT6 assessed as reduction in NAD+-dependent deacetylase activity using Arg-His-Lys-Lys(epsilon-acetyl)-AMC substrat...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNAD-dependent protein deacylase sirtuin-6(Homo sapiens (Human))
Nagoya City University

Curated by ChEMBL
LigandPNGBDBM50276145(CHEMBL4128630)
Affinity DataIC50:  2.09E+4nMAssay Description:Inhibition of human SIRT6 (1 to 294 residues) expressed in Escherichia coli Rosetta (DE3) using H3K9AcWW as substrate preincubated for 15 mins follow...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNAD-dependent protein deacylase sirtuin-6(Homo sapiens (Human))
Nagoya City University

Curated by ChEMBL
LigandPNGBDBM50544043(CHEMBL4640570)
Affinity DataIC50:  2.09E+4nMAssay Description:Inhibition of SIRT6 (unknown origin) using Ac-RYQK(Ac)-AMC as substrate by Fluor de Lys assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNAD-dependent protein deacylase sirtuin-6(Homo sapiens (Human))
Nagoya City University

Curated by ChEMBL
LigandPNGBDBM50544036(CHEMBL4634194)
Affinity DataIC50:  2.11E+4nMAssay Description:Inhibition of SIRT6 (unknown origin) using Ac-RYQK(Ac)-AMC as substrate by Fluor de Lys assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNAD-dependent protein deacylase sirtuin-6(Homo sapiens (Human))
Nagoya City University

Curated by ChEMBL
LigandPNGBDBM50473422(CHEMBL340881)
Affinity DataIC50:  2.19E+4nMAssay Description:Inhibition of SIRT6 (unknown origin) using Ac-RYQK(Ac)-AMC as substrate by Fluor de Lys assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNAD-dependent protein deacylase sirtuin-6(Homo sapiens (Human))
Nagoya City University

Curated by ChEMBL
LigandPNGBDBM50451275(CHEMBL4205716)
Affinity DataIC50:  2.20E+4nMAssay Description:Antagonist activity at human adenosine A1 receptor expressed in CHO FlpIn cells assessed as inhibition of of N(6)-(R-phenylisopropyl)adenosine-induce...More data for this Ligand-Target Pair
In DepthDetails
TargetNAD-dependent protein deacylase sirtuin-6(Homo sapiens (Human))
Nagoya City University

Curated by ChEMBL
LigandPNGBDBM50451275(CHEMBL4205716)
Affinity DataIC50:  2.20E+4nMAssay Description:Inhibition of human recombinant SIRT6 assessed as reduction in NAD+-dependent deacetylase activity using Arg-His-Lys-Lys(epsilon-acetyl)-AMC substrat...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNAD-dependent protein deacylase sirtuin-6(Homo sapiens (Human))
Nagoya City University

Curated by ChEMBL
LigandPNGBDBM228816(5-Cl-PZA)
Affinity DataIC50:  3.32E+4nMAssay Description:Inhibition of His-tagged human SIRT6 expressed in Escherichia coli BL21(DE3) using Ac-p53 as substrate by fluorescence-based coupled-enzyme assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNAD-dependent protein deacylase sirtuin-6(Homo sapiens (Human))
Nagoya City University

Curated by ChEMBL
LigandPNGBDBM228816(5-Cl-PZA)
Affinity DataIC50:  3.32E+4nMAssay Description:Antagonist activity at oxytocin receptor in rat uterine strips assessed as inhibition of oxytocin-induced contractionMore data for this Ligand-Target Pair
In DepthDetails
TargetNAD-dependent protein deacylase sirtuin-6(Homo sapiens (Human))
Nagoya City University

Curated by ChEMBL
LigandPNGBDBM228816(5-Cl-PZA)
Affinity DataIC50:  3.32E+4nMAssay Description:Inhibitory constants (Ki) and IC50 values were determined under saturating substrate conditions by using a fluorimetric assay (components were purcha...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNAD-dependent protein deacylase sirtuin-6(Homo sapiens (Human))
Nagoya City University

Curated by ChEMBL
LigandPNGBDBM228816(5-Cl-PZA)
Affinity DataIC50:  3.32E+4nMAssay Description:Inhibition of human recombinant MGLMore data for this Ligand-Target Pair
In DepthDetails
TargetNAD-dependent protein deacylase sirtuin-6(Homo sapiens (Human))
Nagoya City University

Curated by ChEMBL
LigandPNGBDBM50451274(CHEMBL4206619)
Affinity DataIC50:  3.40E+4nMAssay Description:Inhibition of human recombinant SIRT6 assessed as reduction in NAD+-dependent deacetylase activity using Arg-His-Lys-Lys(epsilon-acetyl)-AMC substrat...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNAD-dependent protein deacylase sirtuin-6(Homo sapiens (Human))
Nagoya City University

Curated by ChEMBL
LigandPNGBDBM50451274(CHEMBL4206619)
Affinity DataIC50:  3.40E+4nMAssay Description:Antagonist activity at human adenosine A1 receptor expressed in CHO FlpIn cells assessed as inhibition of of N(6)-(R-phenylisopropyl)adenosine-induce...More data for this Ligand-Target Pair
In DepthDetails
TargetNAD-dependent protein deacylase sirtuin-6(Homo sapiens (Human))
Nagoya City University

Curated by ChEMBL
LigandPNGBDBM50001908(1-(4-Nitro-phenyl)-piperazine | CHEMBL165012)
Affinity DataIC50:  3.50E+4nMAssay Description:Inhibition of SIRT6 (unknown origin) using Ac-RYQK(Ac)-AMC as substrate by Fluor de Lys assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNAD-dependent protein deacylase sirtuin-6(Homo sapiens (Human))
Nagoya City University

Curated by ChEMBL
LigandPNGBDBM50123364(CHEMBL3622696)
Affinity DataIC50:  3.70E+4nMAssay Description:Inhibition of human SIRT6 deacetylase activity using Arg-His-Lys-Lys(AC)-AMC as a substrate by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNAD-dependent protein deacylase sirtuin-6(Homo sapiens (Human))
Nagoya City University

Curated by ChEMBL
LigandPNGBDBM50123399(CHEMBL3623254)
Affinity DataIC50:  3.80E+4nMAssay Description:Inhibition of human recombinant SIRT6 deacetylase activity using Arg-His-Lys-Lys(AC)-AMC as a substrate by luminescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNAD-dependent protein deacylase sirtuin-6(Homo sapiens (Human))
Nagoya City University

Curated by ChEMBL
LigandPNGBDBM228815(5-MeO-PZA)
Affinity DataIC50:  4.04E+4nMAssay Description:Inhibitory constants (Ki) and IC50 values were determined under saturating substrate conditions by using a fluorimetric assay (components were purcha...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNAD-dependent protein deacylase sirtuin-6(Homo sapiens (Human))
Nagoya City University

Curated by ChEMBL
LigandPNGBDBM228815(5-MeO-PZA)
Affinity DataIC50:  4.04E+4nMAssay Description:Inhibition of human recombinant MGLMore data for this Ligand-Target Pair
In DepthDetails
TargetNAD-dependent protein deacylase sirtuin-6(Homo sapiens (Human))
Nagoya City University

Curated by ChEMBL
LigandPNGBDBM27507(3-Pyridinecarboxamide | CHEMBL1140 | NAM | niacina...)
Affinity DataIC50:  4.50E+4nMAssay Description:Antagonist activity at adrenergic Alpha-1B receptor in guinea pig spleenMore data for this Ligand-Target Pair
In DepthDetails PDB3D3D Structure (crystal)
TargetNAD-dependent protein deacylase sirtuin-6(Homo sapiens (Human))
Nagoya City University

Curated by ChEMBL
LigandPNGBDBM50257405(Ala-Lys-Lys(epsilon-thioAc)Leu-Met | CHEMBL504711)
Affinity DataIC50:  4.70E+4nMAssay Description:Inhibition of human recombinant SIRT6 assessed as 7-amino-4-methylcoumarin labelled Arg-His-Lys-Lys(epsilon-acetyl) substrate deacetylation after 90 ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNAD-dependent protein deacylase sirtuin-6(Homo sapiens (Human))
Nagoya City University

Curated by ChEMBL
LigandPNGBDBM50123399(CHEMBL3623254)
Affinity DataIC50:  4.90E+4nMAssay Description:Inhibition of human SIRT6 deacetylase activity using Arg-His-Lys-Lys(AC)-AMC as a substrate by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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