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Found 51 Enz. Inhib. hit(s) with all data for entry = 4640
TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
TBA

Curated by PDSP Ki Database
LigandPNGBDBM81450(CAS_112184 | Hydroxybenzylpindolol,(+/-) | NSC_112...)
Affinity DataKi:  0.5nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
TBA

Curated by PDSP Ki Database
LigandPNGBDBM25761(Anapriline | Avlocardyl | CHEMBL27 | PROPANOLOL(-)...)
Affinity DataKi:  2.10nMMore data for this Ligand-Target Pair
In DepthDetails PubMedDrugBank

TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
TBA

Curated by PDSP Ki Database
LigandPNGBDBM25764(ALPRENOLOL,(+) | ALPRENOLOL,(-) | Alfeprol | Alphe...)
Affinity DataKi:  2.30nMMore data for this Ligand-Target Pair
In DepthDetails PubMedDrugBank

TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
TBA

Curated by PDSP Ki Database
LigandPNGBDBM81447(CAS_43216 | Dihydroalprenolol,(+/-) | NSC_43216)
Affinity DataKi:  2.60nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
TBA

Curated by PDSP Ki Database
LigandPNGBDBM25392(4-[1-hydroxy-2-(isopropylamino)ethyl]pyrocatechol;...)
Affinity DataKi:  46nMMore data for this Ligand-Target Pair
TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
TBA

Curated by PDSP Ki Database
LigandPNGBDBM50036835(1-(3,4-Dichloro-phenyl)-2-isopropylamino-ethanol |...)
Affinity DataKi:  100nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
TBA

Curated by PDSP Ki Database
LigandPNGBDBM25764(ALPRENOLOL,(+) | ALPRENOLOL,(-) | Alfeprol | Alphe...)
Affinity DataKi:  170nMMore data for this Ligand-Target Pair
In DepthDetails PubMedDrugBank

TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
TBA

Curated by PDSP Ki Database
LigandPNGBDBM81449(CAS_193350 | Cc-25,(+/-) | NSC_193350)
Affinity DataKi:  180nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
TBA

Curated by PDSP Ki Database
LigandPNGBDBM25761(Anapriline | Avlocardyl | CHEMBL27 | PROPANOLOL(-)...)
Affinity DataKi:  400nMMore data for this Ligand-Target Pair
In DepthDetails PubMedDrugBank

TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
TBA

Curated by PDSP Ki Database
LigandPNGBDBM50326545(CHEMBL1243407 | MJ-9184-1,(+/-) | Zinterol)
Affinity DataKi:  460nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
TBA

Curated by PDSP Ki Database
LigandPNGBDBM50167939(3,4-DNH | 5-Hydroxy Tryptamine | BM 613 | Benzen |...)
Affinity DataKi:  490nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
TBA

Curated by PDSP Ki Database
LigandPNGBDBM35234(DL-[7-3H]norepinephrine | NOREPINEPHRINE | Noradre...)
Affinity DataKi:  800nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
TBA

Curated by PDSP Ki Database
LigandPNGBDBM25749(CHEMBL6995 | N-{4-[2-hydroxy-3-(propan-2-ylamino)p...)
Affinity DataKi:  880nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
TBA

Curated by PDSP Ki Database
LigandPNGBDBM84342(4-[1-hydroxy-2-(methylamino)ethyl]benzene-1,2-diol...)
Affinity DataKi:  1.10E+3nMMore data for this Ligand-Target Pair
TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
TBA

Curated by PDSP Ki Database
LigandPNGBDBM25762(CHEMBL471 | N-{4-[1-hydroxy-2-(propan-2-ylamino)et...)
Affinity DataKi:  1.90E+3nMMore data for this Ligand-Target Pair
In DepthDetails PubMedDrugBank

TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
TBA

Curated by PDSP Ki Database
LigandPNGBDBM25769(4-[2-(tert-butylamino)-1-hydroxyethyl]-2-(hydroxym...)
Affinity DataKi:  2.70E+3nMMore data for this Ligand-Target Pair
TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
TBA

Curated by PDSP Ki Database
LigandPNGBDBM25392(4-[1-hydroxy-2-(isopropylamino)ethyl]pyrocatechol;...)
Affinity DataKi:  2.80E+3nMMore data for this Ligand-Target Pair
TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
TBA

Curated by PDSP Ki Database
LigandPNGBDBM84342(4-[1-hydroxy-2-(methylamino)ethyl]benzene-1,2-diol...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
TBA

Curated by PDSP Ki Database
LigandPNGBDBM50027065((5'alpha)-12'-hydroxy-2'-methyl-5'-(phenylmethyl)e...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
TBA

Curated by PDSP Ki Database
LigandPNGBDBM50167939(3,4-DNH | 5-Hydroxy Tryptamine | BM 613 | Benzen |...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
TBA

Curated by PDSP Ki Database
LigandPNGBDBM21398(4-[4-(4-Chloro-phenyl)-4-hydroxy-piperidin-1-yl]-1...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
TBA

Curated by PDSP Ki Database
LigandPNGBDBM50005246(1-Phenylpropan-2-amin | 1-phenyl-2-aminopropane | ...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails PubMedDrugBank

TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
TBA

Curated by PDSP Ki Database
LigandPNGBDBM50010859(CHEMBL11 | IMIPRAMINE HYDROCHLORIDE | IMIPRAMINE P...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
TBA

Curated by PDSP Ki Database
LigandPNGBDBM81448(CAS_5560-72-5 | IPRINDOLE | NSC_21722)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
TBA

Curated by PDSP Ki Database
LigandPNGBDBM50167939(3,4-DNH | 5-Hydroxy Tryptamine | BM 613 | Benzen |...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
TBA

Curated by PDSP Ki Database
LigandPNGBDBM81451(CAS_120852 | MJ-1998,(+/-) | NSC_120852)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
TBA

Curated by PDSP Ki Database
LigandPNGBDBM50130257((3E)-3-(2-chloro-9H-thioxanthen-9-ylidene)-N,N-dim...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
TBA

Curated by PDSP Ki Database
LigandPNGBDBM35234(DL-[7-3H]norepinephrine | NOREPINEPHRINE | Noradre...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
TBA

Curated by PDSP Ki Database
LigandPNGBDBM112777(NORTRIPTYLINE | US8629135, SW-02)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails PubMedDrugBank

TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
TBA

Curated by PDSP Ki Database
LigandPNGBDBM50017679(Benzyl-(2-chloro-ethyl)-(1-methyl-2-phenoxy-ethyl)...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails PubMedDrugBank

TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
TBA

Curated by PDSP Ki Database
LigandPNGBDBM31046(3-[4,5-dihydro-1H-imidazol-2-ylmethyl-(4-methylphe...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
TBA

Curated by PDSP Ki Database
LigandPNGBDBM36024((R)-(-)-phenylephrine | PHENYLEPHRINE | Phenylephr...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
TBA

Curated by PDSP Ki Database
LigandPNGBDBM36024((R)-(-)-phenylephrine | PHENYLEPHRINE | Phenylephr...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
TBA

Curated by PDSP Ki Database
LigandPNGBDBM25749(CHEMBL6995 | N-{4-[2-hydroxy-3-(propan-2-ylamino)p...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
TBA

Curated by PDSP Ki Database
LigandPNGBDBM67545(N,N-dimethyl-3-(10-phenothiazinyl)-1-propanamine;h...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
TBA

Curated by PDSP Ki Database
LigandPNGBDBM50016018((S)-11-methoxy-7-methyl-6,7,7a,8-tetrahydro-5H-ben...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
TBA

Curated by PDSP Ki Database
LigandPNGBDBM50167939(3,4-DNH | 5-Hydroxy Tryptamine | BM 613 | Benzen |...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
TBA

Curated by PDSP Ki Database
LigandPNGBDBM50176062(3-(5H-dibenzo[a,d][7]annulen-5-yl)-N-methylpropan-...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
TBA

Curated by PDSP Ki Database
LigandPNGBDBM36014((1R,2S)-(-)-ephedrine | Ephedrine,(+) | Ephedrine,...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
TBA

Curated by PDSP Ki Database
LigandPNGBDBM50292375((-)-4-hydroxy-alpha-[(methylamino)methyl]benzeneme...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
TBA

Curated by PDSP Ki Database
LigandPNGBDBM25770(5-[2-(tert-butylamino)-1-hydroxyethyl]benzene-1,3-...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails PubMedDrugBank

TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
TBA

Curated by PDSP Ki Database
LigandPNGBDBM50167939(3,4-DNH | 5-Hydroxy Tryptamine | BM 613 | Benzen |...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
TBA

Curated by PDSP Ki Database
LigandPNGBDBM78576(CIS-THIOTHIXENE | MLS000028463 | SMR000058396 | TH...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
TBA

Curated by PDSP Ki Database
LigandPNGBDBM25762(CHEMBL471 | N-{4-[1-hydroxy-2-(propan-2-ylamino)et...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails PubMedDrugBank

TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
TBA

Curated by PDSP Ki Database
LigandPNGBDBM36014((1R,2S)-(-)-ephedrine | Ephedrine,(+) | Ephedrine,...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
TBA

Curated by PDSP Ki Database
LigandPNGBDBM36014((1R,2S)-(-)-ephedrine | Ephedrine,(+) | Ephedrine,...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
TBA

Curated by PDSP Ki Database
LigandPNGBDBM55121(3-HYDROXYTYRAMINE HYDROCHLORIDE | 4-(2-aminoethyl)...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
TBA

Curated by PDSP Ki Database
LigandPNGBDBM81452(CAS_91533 | Dimethindene | NSC_91533)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
TBA

Curated by PDSP Ki Database
LigandPNGBDBM78576(CIS-THIOTHIXENE | MLS000028463 | SMR000058396 | TH...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
TBA

Curated by PDSP Ki Database
LigandPNGBDBM86698(BENZTROPINE | CAS_132-17-2 | CHEMBL116590 | NSC_23...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
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