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Found 14 Enz. Inhib. hit(s) with all data for entry = 5944
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Merck Sharp & Dohme

US Patent
LigandPNGBDBM9048(US8536193, 10-5)
Affinity DataIC50:  0.340nMAssay Description:Activated Akt isoforms and pleckstrin homology domain deletion constructs were assayed utilizing a GSK-derived biotinylated peptide substrate. The e...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Merck Sharp & Dohme

US Patent
LigandPNGBDBM102310(US8536193, 10-4)
Affinity DataIC50:  0.380nMpH: 7.5Assay Description:Activated Akt isoforms and pleckstrin homology domain deletion constructs were assayed utilizing a GSK-derived biotinylated peptide substrate. The e...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Merck Sharp & Dohme

US Patent
LigandPNGBDBM8727(US8536193, 7-26)
Affinity DataIC50:  0.700nMAssay Description:Activated Akt isoforms and pleckstrin homology domain deletion constructs were assayed utilizing a GSK-derived biotinylated peptide substrate. The e...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetRAC-beta serine/threonine-protein kinase(Homo sapiens (Human))
Merck Sharp & Dohme

US Patent
LigandPNGBDBM102310(US8536193, 10-4)
Affinity DataIC50:  1.70nMpH: 7.5Assay Description:Activated Akt isoforms and pleckstrin homology domain deletion constructs were assayed utilizing a GSK-derived biotinylated peptide substrate. The e...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Merck Sharp & Dohme

US Patent
LigandPNGBDBM102311(US8536193, 2-1)
Affinity DataIC50:  2.30nMpH: 7.5Assay Description:Activated Akt isoforms and pleckstrin homology domain deletion constructs were assayed utilizing a GSK-derived biotinylated peptide substrate. The e...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Merck Sharp & Dohme

US Patent
LigandPNGBDBM102307(US8536193, 3-1)
Affinity DataIC50:  6.10nMpH: 7.5Assay Description:Activated Akt isoforms and pleckstrin homology domain deletion constructs were assayed utilizing a GSK-derived biotinylated peptide substrate. The e...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Merck Sharp & Dohme

US Patent
LigandPNGBDBM102308(US8536193, 4-1)
Affinity DataIC50:  8.20nMpH: 7.5Assay Description:Activated Akt isoforms and pleckstrin homology domain deletion constructs were assayed utilizing a GSK-derived biotinylated peptide substrate. The e...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Merck Sharp & Dohme

US Patent
LigandPNGBDBM102309(US8536193, 5-12)
Affinity DataIC50:  10nMpH: 7.5Assay Description:Activated Akt isoforms and pleckstrin homology domain deletion constructs were assayed utilizing a GSK-derived biotinylated peptide substrate. The e...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetRAC-beta serine/threonine-protein kinase(Homo sapiens (Human))
Merck Sharp & Dohme

US Patent
LigandPNGBDBM102307(US8536193, 3-1)
Affinity DataIC50:  24nMpH: 7.5Assay Description:Activated Akt isoforms and pleckstrin homology domain deletion constructs were assayed utilizing a GSK-derived biotinylated peptide substrate. The e...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetRAC-beta serine/threonine-protein kinase(Homo sapiens (Human))
Merck Sharp & Dohme

US Patent
LigandPNGBDBM102311(US8536193, 2-1)
Affinity DataIC50:  32nMpH: 7.5Assay Description:Activated Akt isoforms and pleckstrin homology domain deletion constructs were assayed utilizing a GSK-derived biotinylated peptide substrate. The e...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Merck Sharp & Dohme

US Patent
LigandPNGBDBM102312(US8536193, 1-9)
Affinity DataIC50:  39nMpH: 7.5Assay Description:Activated Akt isoforms and pleckstrin homology domain deletion constructs were assayed utilizing a GSK-derived biotinylated peptide substrate. The e...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetRAC-beta serine/threonine-protein kinase(Homo sapiens (Human))
Merck Sharp & Dohme

US Patent
LigandPNGBDBM102308(US8536193, 4-1)
Affinity DataIC50:  50nMpH: 7.5Assay Description:Activated Akt isoforms and pleckstrin homology domain deletion constructs were assayed utilizing a GSK-derived biotinylated peptide substrate. The e...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetRAC-beta serine/threonine-protein kinase(Homo sapiens (Human))
Merck Sharp & Dohme

US Patent
LigandPNGBDBM102309(US8536193, 5-12)
Affinity DataIC50:  140nMpH: 7.5Assay Description:Activated Akt isoforms and pleckstrin homology domain deletion constructs were assayed utilizing a GSK-derived biotinylated peptide substrate. The e...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetRAC-beta serine/threonine-protein kinase(Homo sapiens (Human))
Merck Sharp & Dohme

US Patent
LigandPNGBDBM102312(US8536193, 1-9)
Affinity DataIC50:  200nMpH: 7.5Assay Description:Activated Akt isoforms and pleckstrin homology domain deletion constructs were assayed utilizing a GSK-derived biotinylated peptide substrate. The e...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent