Compile Data Set for Download or QSAR
maximum 50k data
Found 45 Enz. Inhib. hit(s) with all data for entry = 7299
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Gilead Sciences

US Patent
LigandPNGBDBM187363(US9169243, 11 | US9908875, 11)
Affinity DataIC50:  0.400nMAssay Description:The assay measures the phosphorylation level of a biotinylated peptide substrate by the ASK1 kinase using HTRF detection. This is a competitive, time...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Gilead Sciences

US Patent
LigandPNGBDBM187354(US9169243, 2 | US9908875, 2)
Affinity DataIC50:  0.900nMAssay Description:The assay measures the phosphorylation level of a biotinylated peptide substrate by the ASK1 kinase using HTRF detection. This is a competitive, time...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Gilead Sciences

US Patent
LigandPNGBDBM187369(US9169243, 17 | US9908875, 17)
Affinity DataIC50:  1.10nMAssay Description:The assay measures the phosphorylation level of a biotinylated peptide substrate by the ASK1 kinase using HTRF detection. This is a competitive, time...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Gilead Sciences

US Patent
LigandPNGBDBM187385(US9169243, 33 | US9908875, 33)
Affinity DataIC50:  1.20nMAssay Description:The assay measures the phosphorylation level of a biotinylated peptide substrate by the ASK1 kinase using HTRF detection. This is a competitive, time...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Gilead Sciences

US Patent
LigandPNGBDBM187376(US9169243, 24 | US9908875, 24)
Affinity DataIC50:  1.40nMAssay Description:The assay measures the phosphorylation level of a biotinylated peptide substrate by the ASK1 kinase using HTRF detection. This is a competitive, time...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Gilead Sciences

US Patent
LigandPNGBDBM187384(US9169243, 32 | US9908875, 32)
Affinity DataIC50:  1.5nMAssay Description:The assay measures the phosphorylation level of a biotinylated peptide substrate by the ASK1 kinase using HTRF detection. This is a competitive, time...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Gilead Sciences

US Patent
LigandPNGBDBM187381(US9169243, 29 | US9908875, 29)
Affinity DataIC50:  1.70nMAssay Description:The assay measures the phosphorylation level of a biotinylated peptide substrate by the ASK1 kinase using HTRF detection. This is a competitive, time...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Gilead Sciences

US Patent
LigandPNGBDBM187378(US9169243, 26 | US9908875, 26)
Affinity DataIC50:  1.70nMAssay Description:The assay measures the phosphorylation level of a biotinylated peptide substrate by the ASK1 kinase using HTRF detection. This is a competitive, time...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Gilead Sciences

US Patent
LigandPNGBDBM187386(US9169243, 34 | US9908875, 34)
Affinity DataIC50:  1.70nMAssay Description:The assay measures the phosphorylation level of a biotinylated peptide substrate by the ASK1 kinase using HTRF detection. This is a competitive, time...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Gilead Sciences

US Patent
LigandPNGBDBM187356(US9169243, 4 | US9908875, 4)
Affinity DataIC50:  1.80nMAssay Description:The assay measures the phosphorylation level of a biotinylated peptide substrate by the ASK1 kinase using HTRF detection. This is a competitive, time...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Gilead Sciences

US Patent
LigandPNGBDBM187394(US9169243, 42 | US9908875, 42)
Affinity DataIC50:  1.80nMAssay Description:The assay measures the phosphorylation level of a biotinylated peptide substrate by the ASK1 kinase using HTRF detection. This is a competitive, time...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Gilead Sciences

US Patent
LigandPNGBDBM187389(US9169243, 37)
Affinity DataIC50:  1.80nMAssay Description:The assay measures the phosphorylation level of a biotinylated peptide substrate by the ASK1 kinase using HTRF detection. This is a competitive, time...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Gilead Sciences

US Patent
LigandPNGBDBM187395(US9169243, 43 | US9908875, 43)
Affinity DataIC50:  1.80nMAssay Description:The assay measures the phosphorylation level of a biotinylated peptide substrate by the ASK1 kinase using HTRF detection. This is a competitive, time...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Gilead Sciences

US Patent
LigandPNGBDBM187380(US9169243, 28 | US9908875, 28)
Affinity DataIC50:  1.90nMAssay Description:The assay measures the phosphorylation level of a biotinylated peptide substrate by the ASK1 kinase using HTRF detection. This is a competitive, time...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Gilead Sciences

US Patent
LigandPNGBDBM187373(US9169243, 21 | US9908875, 21)
Affinity DataIC50:  1.90nMAssay Description:The assay measures the phosphorylation level of a biotinylated peptide substrate by the ASK1 kinase using HTRF detection. This is a competitive, time...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Gilead Sciences

US Patent
LigandPNGBDBM187355(US9169243, 3 | US9908875, 3)
Affinity DataIC50:  1.90nMAssay Description:The assay measures the phosphorylation level of a biotinylated peptide substrate by the ASK1 kinase using HTRF detection. This is a competitive, time...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Gilead Sciences

US Patent
LigandPNGBDBM187388(US9169243, 36 | US9908875, 36)
Affinity DataIC50:  1.90nMAssay Description:The assay measures the phosphorylation level of a biotinylated peptide substrate by the ASK1 kinase using HTRF detection. This is a competitive, time...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Gilead Sciences

US Patent
LigandPNGBDBM187393(US9169243, 41 | US9908875, 41)
Affinity DataIC50:  1.90nMAssay Description:The assay measures the phosphorylation level of a biotinylated peptide substrate by the ASK1 kinase using HTRF detection. This is a competitive, time...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Gilead Sciences

US Patent
LigandPNGBDBM187375(US9169243, 23 | US9908875, 23)
Affinity DataIC50:  2nMAssay Description:The assay measures the phosphorylation level of a biotinylated peptide substrate by the ASK1 kinase using HTRF detection. This is a competitive, time...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Gilead Sciences

US Patent
LigandPNGBDBM187377(US9169243, 25 | US9908875, 25)
Affinity DataIC50:  2nMAssay Description:The assay measures the phosphorylation level of a biotinylated peptide substrate by the ASK1 kinase using HTRF detection. This is a competitive, time...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Gilead Sciences

US Patent
LigandPNGBDBM187379(US9169243, 27 | US9908875, 27)
Affinity DataIC50:  2.10nMAssay Description:The assay measures the phosphorylation level of a biotinylated peptide substrate by the ASK1 kinase using HTRF detection. This is a competitive, time...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Gilead Sciences

US Patent
LigandPNGBDBM187396(US9169243, 44 | US9908875, 44)
Affinity DataIC50:  2.10nMAssay Description:The assay measures the phosphorylation level of a biotinylated peptide substrate by the ASK1 kinase using HTRF detection. This is a competitive, time...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Gilead Sciences

US Patent
LigandPNGBDBM187361(US9169243, 9 | US9908875, 9)
Affinity DataIC50:  2.20nMAssay Description:The assay measures the phosphorylation level of a biotinylated peptide substrate by the ASK1 kinase using HTRF detection. This is a competitive, time...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Gilead Sciences

US Patent
LigandPNGBDBM187392(US9169243, 40 | US9908875, 40)
Affinity DataIC50:  2.20nMAssay Description:The assay measures the phosphorylation level of a biotinylated peptide substrate by the ASK1 kinase using HTRF detection. This is a competitive, time...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Gilead Sciences

US Patent
LigandPNGBDBM187353(US9169243, 1 | US9908875, 1)
Affinity DataIC50:  2.20nMAssay Description:The assay measures the phosphorylation level of a biotinylated peptide substrate by the ASK1 kinase using HTRF detection. This is a competitive, time...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Gilead Sciences

US Patent
LigandPNGBDBM187387(US9169243, 35 | US9908875, 35)
Affinity DataIC50:  2.20nMAssay Description:The assay measures the phosphorylation level of a biotinylated peptide substrate by the ASK1 kinase using HTRF detection. This is a competitive, time...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Gilead Sciences

US Patent
LigandPNGBDBM187383(US9169243, 31 | US9908875, 31)
Affinity DataIC50:  2.30nMAssay Description:The assay measures the phosphorylation level of a biotinylated peptide substrate by the ASK1 kinase using HTRF detection. This is a competitive, time...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Gilead Sciences

US Patent
LigandPNGBDBM187370(US9169243, 18 | US9908875, 18)
Affinity DataIC50:  2.30nMAssay Description:The assay measures the phosphorylation level of a biotinylated peptide substrate by the ASK1 kinase using HTRF detection. This is a competitive, time...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Gilead Sciences

US Patent
LigandPNGBDBM187382(US9169243, 30 | US9908875, 30)
Affinity DataIC50:  2.30nMAssay Description:The assay measures the phosphorylation level of a biotinylated peptide substrate by the ASK1 kinase using HTRF detection. This is a competitive, time...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Gilead Sciences

US Patent
LigandPNGBDBM187391(US9169243, 39 | US9908875, 39)
Affinity DataIC50:  2.30nMAssay Description:The assay measures the phosphorylation level of a biotinylated peptide substrate by the ASK1 kinase using HTRF detection. This is a competitive, time...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Gilead Sciences

US Patent
LigandPNGBDBM187390(US9169243, 38 | US9908875, 38)
Affinity DataIC50:  2.40nMAssay Description:The assay measures the phosphorylation level of a biotinylated peptide substrate by the ASK1 kinase using HTRF detection. This is a competitive, time...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Gilead Sciences

US Patent
LigandPNGBDBM187372(US9169243, 20 | US9908875, 20)
Affinity DataIC50:  2.5nMAssay Description:The assay measures the phosphorylation level of a biotinylated peptide substrate by the ASK1 kinase using HTRF detection. This is a competitive, time...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Gilead Sciences

US Patent
LigandPNGBDBM187360(US9169243, 8 | US9908875, 8)
Affinity DataIC50:  2.5nMAssay Description:The assay measures the phosphorylation level of a biotinylated peptide substrate by the ASK1 kinase using HTRF detection. This is a competitive, time...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Gilead Sciences

US Patent
LigandPNGBDBM187397(US9169243, 45 | US9908875, 45)
Affinity DataIC50:  2.60nMAssay Description:The assay measures the phosphorylation level of a biotinylated peptide substrate by the ASK1 kinase using HTRF detection. This is a competitive, time...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Gilead Sciences

US Patent
LigandPNGBDBM187368(US9169243, 16 | US9908875, 16)
Affinity DataIC50:  2.70nMAssay Description:The assay measures the phosphorylation level of a biotinylated peptide substrate by the ASK1 kinase using HTRF detection. This is a competitive, time...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Gilead Sciences

US Patent
LigandPNGBDBM187367(US9169243, 15 | US9908875, 15)
Affinity DataIC50:  2.70nMAssay Description:The assay measures the phosphorylation level of a biotinylated peptide substrate by the ASK1 kinase using HTRF detection. This is a competitive, time...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Gilead Sciences

US Patent
LigandPNGBDBM187357(US9169243, 5 | US9908875, 5)
Affinity DataIC50:  2.80nMAssay Description:The assay measures the phosphorylation level of a biotinylated peptide substrate by the ASK1 kinase using HTRF detection. This is a competitive, time...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Gilead Sciences

US Patent
LigandPNGBDBM187358(US9169243, 6 | US9908875, 6)
Affinity DataIC50:  2.80nMAssay Description:The assay measures the phosphorylation level of a biotinylated peptide substrate by the ASK1 kinase using HTRF detection. This is a competitive, time...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Gilead Sciences

US Patent
LigandPNGBDBM187371(US9169243, 19 | US9908875, 19)
Affinity DataIC50:  2.80nMAssay Description:The assay measures the phosphorylation level of a biotinylated peptide substrate by the ASK1 kinase using HTRF detection. This is a competitive, time...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Gilead Sciences

US Patent
LigandPNGBDBM187365(US9169243, 13 | US9908875, 13)
Affinity DataIC50:  2.90nMAssay Description:The assay measures the phosphorylation level of a biotinylated peptide substrate by the ASK1 kinase using HTRF detection. This is a competitive, time...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Gilead Sciences

US Patent
LigandPNGBDBM187359(US9169243, 7 | US9908875, 7)
Affinity DataIC50:  3.20nMAssay Description:The assay measures the phosphorylation level of a biotinylated peptide substrate by the ASK1 kinase using HTRF detection. This is a competitive, time...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Gilead Sciences

US Patent
LigandPNGBDBM187362(US9169243, 10 | US9908875, 10)
Affinity DataIC50:  3.20nMAssay Description:The assay measures the phosphorylation level of a biotinylated peptide substrate by the ASK1 kinase using HTRF detection. This is a competitive, time...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Gilead Sciences

US Patent
LigandPNGBDBM187366(US9169243, 14 | US9908875, 14)
Affinity DataIC50:  3.80nMAssay Description:The assay measures the phosphorylation level of a biotinylated peptide substrate by the ASK1 kinase using HTRF detection. This is a competitive, time...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Gilead Sciences

US Patent
LigandPNGBDBM187374(US9169243, 22 | US9908875, 22)
Affinity DataIC50:  4.5nMAssay Description:The assay measures the phosphorylation level of a biotinylated peptide substrate by the ASK1 kinase using HTRF detection. This is a competitive, time...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Gilead Sciences

US Patent
LigandPNGBDBM187364(US9169243, 12 | US9908875, 12)
Affinity DataIC50:  14.2nMAssay Description:The assay measures the phosphorylation level of a biotinylated peptide substrate by the ASK1 kinase using HTRF detection. This is a competitive, time...More data for this Ligand-Target Pair
In DepthDetails US Patent