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Found 71 Enz. Inhib. hit(s) with all data for entry = 139
LigandPNGBDBM189846(US9670194, Ex. 65 (S)-2-(1-((6-amino-5-(3-methyl-1...)
Affinity DataIC50:  2nMT: 2°CAssay Description:PI3K (p110α/p85α) (h) is incubated in assay buffer containing 10 μM phosphatidylinositol 4,5-bisphosphate and MgATP (concentration as ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
LigandPNGBDBM188124(US9670194, Ex. 3 (S)-2-(1-((6-amino-5-(3-methyl-1,...)
Affinity DataIC50:  2nMT: 2°CAssay Description:PI3K (p110α/p85α) (h) is incubated in assay buffer containing 10 μM phosphatidylinositol 4,5-bisphosphate and MgATP (concentration as ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
LigandPNGBDBM188116(US9670194, Ex. 1 (S)-2-(1-((6-amino-5-(5-methyl-1,...)
Affinity DataIC50:  3nMT: 2°CAssay Description:PI3K (p110α/p85α) (h) is incubated in assay buffer containing 10 μM phosphatidylinositol 4,5-bisphosphate and MgATP (concentration as ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
LigandPNGBDBM189408(US9670194, Ex. 41 (S)-2-(1-((6-amino-5-(3-methyl-1...)
Affinity DataIC50:  5nMT: 2°CAssay Description:PI3K (p110α/p85α) (h) is incubated in assay buffer containing 10 μM phosphatidylinositol 4,5-bisphosphate and MgATP (concentration as ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
LigandPNGBDBM189403(US9670194, Ex. 37 (S)-2-(1-((6-amino-5-(3-methyl-1...)
Affinity DataIC50:  6nMT: 2°CAssay Description:PI3K (p110α/p85α) (h) is incubated in assay buffer containing 10 μM phosphatidylinositol 4,5-bisphosphate and MgATP (concentration as ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
LigandPNGBDBM189838(US9670194, Ex. 57 (S)-2-(1-((6-amino-5-(3-isopropy...)
Affinity DataIC50:  6nMT: 2°CAssay Description:PI3K (p110α/p85α) (h) is incubated in assay buffer containing 10 μM phosphatidylinositol 4,5-bisphosphate and MgATP (concentration as ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
LigandPNGBDBM188145(US9670194, Ex. 4 (S)-2-(1-((6-amino-5-(3-methyl-1,...)
Affinity DataIC50:  8nMT: 2°CAssay Description:PI3K (p110α/p85α) (h) is incubated in assay buffer containing 10 μM phosphatidylinositol 4,5-bisphosphate and MgATP (concentration as ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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LigandPNGBDBM189845(US9670194, Ex. 64 (S)-2-(1-((6-amino-5-(5-methyl-1...)
Affinity DataIC50:  8nMT: 2°CAssay Description:PI3K (p110α/p85α) (h) is incubated in assay buffer containing 10 μM phosphatidylinositol 4,5-bisphosphate and MgATP (concentration as ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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LigandPNGBDBM189837(US9670194, Ex. 56 (S)-2-(1-((6-amino-5-(3-ethyl-1,...)
Affinity DataIC50:  9nMT: 2°CAssay Description:PI3K (p110α/p85α) (h) is incubated in assay buffer containing 10 μM phosphatidylinositol 4,5-bisphosphate and MgATP (concentration as ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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LigandPNGBDBM189405(US9670194, Ex. 39 (S)-2-(1-((6-amino-5-(3-methyl-1...)
Affinity DataIC50:  11nMT: 2°CAssay Description:PI3K (p110α/p85α) (h) is incubated in assay buffer containing 10 μM phosphatidylinositol 4,5-bisphosphate and MgATP (concentration as ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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LigandPNGBDBM189306(US9670194, Ex. 34 (S)-2-(1-((6-amino-5-(5-methyl-1...)
Affinity DataIC50:  12nMT: 2°CAssay Description:PI3K (p110α/p85α) (h) is incubated in assay buffer containing 10 μM phosphatidylinositol 4,5-bisphosphate and MgATP (concentration as ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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LigandPNGBDBM189404(US9670194, Ex. 38 (S)-2-(1-((6-amino-5-(5-methyl-1...)
Affinity DataIC50:  12nMT: 2°CAssay Description:PI3K (p110α/p85α) (h) is incubated in assay buffer containing 10 μM phosphatidylinositol 4,5-bisphosphate and MgATP (concentration as ...More data for this Ligand-Target Pair
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LigandPNGBDBM189298(US9670194, Ex. 27 (S)-2-(1-((6-amino-5-(3-methyl-1...)
Affinity DataIC50:  13nMT: 2°CAssay Description:PI3K (p110α/p85α) (h) is incubated in assay buffer containing 10 μM phosphatidylinositol 4,5-bisphosphate and MgATP (concentration as ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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LigandPNGBDBM189832(US9670194, Ex. 52 (S)-2-(1-((6-amino-5-(4-methylox...)
Affinity DataIC50:  15nMT: 2°CAssay Description:PI3K (p110α/p85α) (h) is incubated in assay buffer containing 10 μM phosphatidylinositol 4,5-bisphosphate and MgATP (concentration as ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
LigandPNGBDBM189303(US9670194, Ex. 31 (S)-2-(1-((6-amino-5-(5-methyl-1...)
Affinity DataIC50:  18nMT: 2°CAssay Description:PI3K (p110α/p85α) (h) is incubated in assay buffer containing 10 μM phosphatidylinositol 4,5-bisphosphate and MgATP (concentration as ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
LigandPNGBDBM189844(US9670194, Ex. 63 (S)-2-(1-((6-amino-5-(3-methyl-1...)
Affinity DataIC50:  18nMT: 2°CAssay Description:PI3K (p110α/p85α) (h) is incubated in assay buffer containing 10 μM phosphatidylinositol 4,5-bisphosphate and MgATP (concentration as ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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LigandPNGBDBM188473(US9670194, Ex. 21 (S)-2-(1-((6-amino-5-(3-methyl-1...)
Affinity DataIC50:  19nMT: 2°CAssay Description:PI3K (p110α/p85α) (h) is incubated in assay buffer containing 10 μM phosphatidylinositol 4,5-bisphosphate and MgATP (concentration as ...More data for this Ligand-Target Pair
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LigandPNGBDBM188332(US9670194, Ex. 14 (S)-2-(1-((6-amino-5-(isoxazol-3...)
Affinity DataIC50:  20nMT: 2°CAssay Description:PI3K (p110α/p85α) (h) is incubated in assay buffer containing 10 μM phosphatidylinositol 4,5-bisphosphate and MgATP (concentration as ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
LigandPNGBDBM189840(US9670194, Ex. 59 (S)-2-(1-((6-amino-5-(5-isopropy...)
Affinity DataIC50:  20nMT: 2°CAssay Description:PI3K (p110α/p85α) (h) is incubated in assay buffer containing 10 μM phosphatidylinositol 4,5-bisphosphate and MgATP (concentration as ...More data for this Ligand-Target Pair
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LigandPNGBDBM188474(US9670194, Ex. 22 (S)-2-(1-((6-amino-5-(3-methyl-1...)
Affinity DataIC50:  26nMT: 2°CAssay Description:PI3K (p110α/p85α) (h) is incubated in assay buffer containing 10 μM phosphatidylinositol 4,5-bisphosphate and MgATP (concentration as ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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LigandPNGBDBM188117(US9670194, Ex. 2 (S)-2-(1-((6-amino-5-(5-methyl-1,...)
Affinity DataIC50:  33nMT: 2°CAssay Description:PI3K (p110α/p85α) (h) is incubated in assay buffer containing 10 μM phosphatidylinositol 4,5-bisphosphate and MgATP (concentration as ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
LigandPNGBDBM189408(US9670194, Ex. 41 (S)-2-(1-((6-amino-5-(3-methyl-1...)
Affinity DataIC50:  35nMT: 2°CAssay Description:PI3K (p110β/p85α) (h) is incubated in assay buffer containing 10 μM phosphatidylinositol-4,5-bisphosphate and MgATP (concentration as ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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LigandPNGBDBM189843(US9670194, Ex. 62 2-((S)-1-((6-amino-5-(3-methyl-1...)
Affinity DataIC50:  37nMT: 2°CAssay Description:PI3K (p110α/p85α) (h) is incubated in assay buffer containing 10 μM phosphatidylinositol 4,5-bisphosphate and MgATP (concentration as ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform(Homo sapiens (Human))
Calitor Sciences

US Patent
LigandPNGBDBM189846(US9670194, Ex. 65 (S)-2-(1-((6-amino-5-(3-methyl-1...)
Affinity DataIC50:  37nMT: 2°CAssay Description:PI3K (p110α/p85α) (h) is incubated in assay buffer containing 10 μM phosphatidylinositol 4,5-bisphosphate and MgATP (concentration as ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
LigandPNGBDBM189842(US9670194, Ex. 61 (S)-2-(1-((6-amino-5-(5-ethyl-1,...)
Affinity DataIC50:  44nMT: 2°CAssay Description:PI3K (p110α/p85α) (h) is incubated in assay buffer containing 10 μM phosphatidylinositol 4,5-bisphosphate and MgATP (concentration as ...More data for this Ligand-Target Pair
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LigandPNGBDBM188330(US9670194, Ex. 12 (S)-2-(1-((6-amino-5-(5-methyl-1...)
Affinity DataIC50:  48nMT: 2°CAssay Description:PI3K (p110α/p85α) (h) is incubated in assay buffer containing 10 μM phosphatidylinositol 4,5-bisphosphate and MgATP (concentration as ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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LigandPNGBDBM188338(US9670194, Ex. 20 (S)-2-(1-((6-amino-5-(5-methyl-1...)
Affinity DataIC50:  49nMT: 2°CAssay Description:PI3K (p110α/p85α) (h) is incubated in assay buffer containing 10 μM phosphatidylinositol 4,5-bisphosphate and MgATP (concentration as ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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LigandPNGBDBM188475(US9670194, Ex. 23 (S)-2-(1-((6-amino-5-(3-methyl-1...)
Affinity DataIC50:  52nMT: 2°CAssay Description:PI3K (p110α/p85α) (h) is incubated in assay buffer containing 10 μM phosphatidylinositol 4,5-bisphosphate and MgATP (concentration as ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform(Homo sapiens (Human))
Calitor Sciences

US Patent
LigandPNGBDBM188124(US9670194, Ex. 3 (S)-2-(1-((6-amino-5-(3-methyl-1,...)
Affinity DataIC50:  66nMT: 2°CAssay Description:PI3K (p110α/p85α) (h) is incubated in assay buffer containing 10 μM phosphatidylinositol 4,5-bisphosphate and MgATP (concentration as ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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LigandPNGBDBM189305(US9670194, Ex. 33 (S)-2-(1-((6-amino-5-(5-methyl-1...)
Affinity DataIC50:  67nMT: 2°CAssay Description:PI3K (p110α/p85α) (h) is incubated in assay buffer containing 10 μM phosphatidylinositol 4,5-bisphosphate and MgATP (concentration as ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
LigandPNGBDBM189304(US9670194, Ex. 32 (S)-2-(1-((6-amino-5-(1-methyl-1...)
Affinity DataIC50:  70nMT: 2°CAssay Description:PI3K (p110α/p85α) (h) is incubated in assay buffer containing 10 μM phosphatidylinositol 4,5-bisphosphate and MgATP (concentration as ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
LigandPNGBDBM189406(US9670194, Ex. 40 (S)-2-(1-((6-amino-5-(5-methyl-1...)
Affinity DataIC50:  93nMT: 2°CAssay Description:PI3K (p110α/p85α) (h) is incubated in assay buffer containing 10 μM phosphatidylinositol 4,5-bisphosphate and MgATP (concentration as ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
LigandPNGBDBM188324(US9670194, Ex. 6 2-((S)-1((6-amino-5-((S)-4-methyl...)
Affinity DataIC50:  99nMT: 2°CAssay Description:PI3K (p110α/p85α) (h) is incubated in assay buffer containing 10 μM phosphatidylinositol 4,5-bisphosphate and MgATP (concentration as ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform(Homo sapiens (Human))
Calitor Sciences

US Patent
LigandPNGBDBM189845(US9670194, Ex. 64 (S)-2-(1-((6-amino-5-(5-methyl-1...)
Affinity DataIC50:  112nMT: 2°CAssay Description:PI3K (p110α/p85α) (h) is incubated in assay buffer containing 10 μM phosphatidylinositol 4,5-bisphosphate and MgATP (concentration as ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
LigandPNGBDBM188145(US9670194, Ex. 4 (S)-2-(1-((6-amino-5-(3-methyl-1,...)
Affinity DataIC50:  113nMT: 2°CAssay Description:PI3K (p110β/p85α) (h) is incubated in assay buffer containing 10 μM phosphatidylinositol-4,5-bisphosphate and MgATP (concentration as ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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LigandPNGBDBM189829(US9670194, Ex. 51 (S)-2-(1-((6-amino-5-(1-methyl-1...)
Affinity DataIC50:  135nMT: 2°CAssay Description:PI3K (p110α/p85α) (h) is incubated in assay buffer containing 10 μM phosphatidylinositol 4,5-bisphosphate and MgATP (concentration as ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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LigandPNGBDBM188124(US9670194, Ex. 3 (S)-2-(1-((6-amino-5-(3-methyl-1,...)
Affinity DataIC50:  142nMT: 2°CAssay Description:PI3K (p110β/p85α) (h) is incubated in assay buffer containing 10 μM phosphatidylinositol-4,5-bisphosphate and MgATP (concentration as ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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LigandPNGBDBM189846(US9670194, Ex. 65 (S)-2-(1-((6-amino-5-(3-methyl-1...)
Affinity DataIC50:  154nMT: 2°CAssay Description:PI3K (p110β/p85α) (h) is incubated in assay buffer containing 10 μM phosphatidylinositol-4,5-bisphosphate and MgATP (concentration as ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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LigandPNGBDBM188117(US9670194, Ex. 2 (S)-2-(1-((6-amino-5-(5-methyl-1,...)
Affinity DataIC50:  168nMT: 2°CAssay Description:PI3K (p110β/p85α) (h) is incubated in assay buffer containing 10 μM phosphatidylinositol-4,5-bisphosphate and MgATP (concentration as ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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LigandPNGBDBM189833(US9670194, Ex. 53 (S)-2-(1-((6-amino-5-(1-methyl-1...)
Affinity DataIC50:  239nMT: 2°CAssay Description:PI3K (p110α/p85α) (h) is incubated in assay buffer containing 10 μM phosphatidylinositol 4,5-bisphosphate and MgATP (concentration as ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
LigandPNGBDBM188325(US9670194, Ex. 7 (S)-2-(1-((6-amino-5-(5-methyloxa...)
Affinity DataIC50:  246nMT: 2°CAssay Description:PI3K (p110α/p85α) (h) is incubated in assay buffer containing 10 μM phosphatidylinositol 4,5-bisphosphate and MgATP (concentration as ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform(Homo sapiens (Human))
Calitor Sciences

US Patent
LigandPNGBDBM188145(US9670194, Ex. 4 (S)-2-(1-((6-amino-5-(3-methyl-1,...)
Affinity DataIC50:  258nMT: 2°CAssay Description:PI3K (p110α/p85α) (h) is incubated in assay buffer containing 10 μM phosphatidylinositol 4,5-bisphosphate and MgATP (concentration as ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform(Homo sapiens (Human))
Calitor Sciences

US Patent
LigandPNGBDBM189408(US9670194, Ex. 41 (S)-2-(1-((6-amino-5-(3-methyl-1...)
Affinity DataIC50:  261nMT: 2°CAssay Description:PI3K (p110α/p85α) (h) is incubated in assay buffer containing 10 μM phosphatidylinositol 4,5-bisphosphate and MgATP (concentration as ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform(Homo sapiens (Human))
Calitor Sciences

US Patent
LigandPNGBDBM189844(US9670194, Ex. 63 (S)-2-(1-((6-amino-5-(3-methyl-1...)
Affinity DataIC50:  269nMT: 2°CAssay Description:PI3K (p110α/p85α) (h) is incubated in assay buffer containing 10 μM phosphatidylinositol 4,5-bisphosphate and MgATP (concentration as ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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LigandPNGBDBM189295(US9670194, Ex. 25 (S)-2-(1-((6-amino-5-(5-methyl-1...)
Affinity DataIC50:  298nMT: 2°CAssay Description:PI3K (p110α/p85α) (h) is incubated in assay buffer containing 10 μM phosphatidylinositol 4,5-bisphosphate and MgATP (concentration as ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
LigandPNGBDBM189795(US9670194, Ex. 44 (S)-2-(1-((6-amino-5-(1-methyl-1...)
Affinity DataIC50:  358nMT: 2°CAssay Description:PI3K (p110α/p85α) (h) is incubated in assay buffer containing 10 μM phosphatidylinositol 4,5-bisphosphate and MgATP (concentration as ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform(Homo sapiens (Human))
Calitor Sciences

US Patent
LigandPNGBDBM188116(US9670194, Ex. 1 (S)-2-(1-((6-amino-5-(5-methyl-1,...)
Affinity DataIC50:  384nMT: 2°CAssay Description:PI3K (p110α/p85α) (h) is incubated in assay buffer containing 10 μM phosphatidylinositol 4,5-bisphosphate and MgATP (concentration as ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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LigandPNGBDBM188124(US9670194, Ex. 3 (S)-2-(1-((6-amino-5-(3-methyl-1,...)
Affinity DataIC50:  442nMT: 2°CAssay Description:PI3K (p110α/p85α) (h) is incubated in assay buffer containing 10 μM phosphatidylinositol 4,5-bisphosphate and MgATP (concentration as ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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LigandPNGBDBM189405(US9670194, Ex. 39 (S)-2-(1-((6-amino-5-(3-methyl-1...)
Affinity DataIC50:  502nMT: 2°CAssay Description:PI3K (p110β/p85α) (h) is incubated in assay buffer containing 10 μM phosphatidylinositol-4,5-bisphosphate and MgATP (concentration as ...More data for this Ligand-Target Pair
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LigandPNGBDBM189845(US9670194, Ex. 64 (S)-2-(1-((6-amino-5-(5-methyl-1...)
Affinity DataIC50:  674nMT: 2°CAssay Description:PI3K (p110β/p85α) (h) is incubated in assay buffer containing 10 μM phosphatidylinositol-4,5-bisphosphate and MgATP (concentration as ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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