Compile Data Set for Download or QSAR
maximum 50k data
Found 29 Enz. Inhib. hit(s) with all data for entry = 50000113
TargetLeukotriene B4 receptor 1(Homo sapiens (Human))
Centre De Recherche De Vitry-Alfortville

Curated by ChEMBL
LigandPNGBDBM50001611((E)-3-{3-(2-Carboxy-ethyl)-4-[6-(4-methoxy-phenyl)...)
Affinity DataIC50:  2nMAssay Description:Inhibition of [3H]-LTB4 binding to Leukotriene B4 receptor in the human polymorphonuclear leukocytesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLeukotriene B4 receptor 1(Homo sapiens (Human))
Centre De Recherche De Vitry-Alfortville

Curated by ChEMBL
LigandPNGBDBM50001611((E)-3-{3-(2-Carboxy-ethyl)-4-[6-(4-methoxy-phenyl)...)
Affinity DataIC50:  3.5nMAssay Description:Inhibition of [3H]-LTB4 binding to Leukotriene B4 receptor in the human polymorphonuclear leukocytesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLeukotriene B4 receptor 1(Homo sapiens (Human))
Centre De Recherche De Vitry-Alfortville

Curated by ChEMBL
LigandPNGBDBM50001622(6-[4-(4-Methoxy-phenyl)-quinolin-2-yloxy]-2,2-dime...)
Affinity DataIC50:  10nMAssay Description:Inhibition of [3H]-LTB4 binding to Leukotriene B4 receptor in the guinea pig spleen membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLeukotriene B4 receptor 1(Homo sapiens (Human))
Centre De Recherche De Vitry-Alfortville

Curated by ChEMBL
LigandPNGBDBM50001619(6-[4-(4-Chloro-phenyl)-quinolin-2-yloxy]-2,2-dimet...)
Affinity DataIC50:  15nMAssay Description:Inhibition of [3H]-LTB4 binding to Leukotriene B4 receptor in the guinea pig spleen membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLeukotriene B4 receptor 1(Homo sapiens (Human))
Centre De Recherche De Vitry-Alfortville

Curated by ChEMBL
LigandPNGBDBM50001617(6-[4-(4-Chloro-phenyl)-quinolin-2-yloxy]-hexanoic ...)
Affinity DataIC50:  30nMAssay Description:Inhibition of [3H]-LTB4 binding to Leukotriene B4 receptor in the guinea pig spleen membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLeukotriene B4 receptor 1(Homo sapiens (Human))
Centre De Recherche De Vitry-Alfortville

Curated by ChEMBL
LigandPNGBDBM50001620(4-(4-Chloro-phenyl)-2-[5-methyl-5-(1H-tetrazol-5-y...)
Affinity DataIC50:  30nMAssay Description:Inhibition of [3H]-LTB4 binding to Leukotriene B4 receptor in the guinea pig spleen membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLeukotriene B4 receptor 1(Homo sapiens (Human))
Centre De Recherche De Vitry-Alfortville

Curated by ChEMBL
LigandPNGBDBM50001628(2,2-Dimethyl-6-(4-p-tolyl-quinolin-2-yloxy)-hexano...)
Affinity DataIC50:  30nMAssay Description:Inhibition of [3H]-LTB4 binding to Leukotriene B4 receptor in the guinea pig spleen membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLeukotriene B4 receptor 1(Homo sapiens (Human))
Centre De Recherche De Vitry-Alfortville

Curated by ChEMBL
LigandPNGBDBM50001616(6-[4-(4-Amino-phenyl)-quinolin-2-yloxy]-2,2-dimeth...)
Affinity DataIC50:  40nMAssay Description:Inhibition of [3H]-LTB4 binding to Leukotriene B4 receptor in the guinea pig spleen membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLeukotriene B4 receptor 1(Homo sapiens (Human))
Centre De Recherche De Vitry-Alfortville

Curated by ChEMBL
LigandPNGBDBM50001620(4-(4-Chloro-phenyl)-2-[5-methyl-5-(1H-tetrazol-5-y...)
Affinity DataIC50:  50nMAssay Description:Inhibition of [3H]-LTB4 binding to Leukotriene B4 receptor in the human polymorphonuclear leukocytesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLeukotriene B4 receptor 1(Homo sapiens (Human))
Centre De Recherche De Vitry-Alfortville

Curated by ChEMBL
LigandPNGBDBM50001628(2,2-Dimethyl-6-(4-p-tolyl-quinolin-2-yloxy)-hexano...)
Affinity DataIC50:  100nMAssay Description:Inhibition of [3H]-LTB4 binding to Leukotriene B4 receptor in the human polymorphonuclear leukocytesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLeukotriene B4 receptor 1(Homo sapiens (Human))
Centre De Recherche De Vitry-Alfortville

Curated by ChEMBL
LigandPNGBDBM50001622(6-[4-(4-Methoxy-phenyl)-quinolin-2-yloxy]-2,2-dime...)
Affinity DataIC50:  140nMAssay Description:Inhibition of [3H]-LTB4 binding to Leukotriene B4 receptor in the guinea pig spleen membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLeukotriene B4 receptor 1(Homo sapiens (Human))
Centre De Recherche De Vitry-Alfortville

Curated by ChEMBL
LigandPNGBDBM50001630(2,2-Dimethyl-6-[4-(4-nitro-phenyl)-quinolin-2-ylox...)
Affinity DataIC50:  150nMAssay Description:Inhibition of [3H]-LTB4 binding to Leukotriene B4 receptor in the guinea pig spleen membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLeukotriene B4 receptor 1(Homo sapiens (Human))
Centre De Recherche De Vitry-Alfortville

Curated by ChEMBL
LigandPNGBDBM50001617(6-[4-(4-Chloro-phenyl)-quinolin-2-yloxy]-hexanoic ...)
Affinity DataIC50:  150nMAssay Description:Inhibition of [3H]-LTB4 binding to Leukotriene B4 receptor in the human polymorphonuclear leukocytesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLeukotriene B4 receptor 1(Homo sapiens (Human))
Centre De Recherche De Vitry-Alfortville

Curated by ChEMBL
LigandPNGBDBM50001625(2,2-Dimethyl-6-(4-phenyl-quinolin-2-yloxy)-hexanoi...)
Affinity DataIC50:  183nMAssay Description:Inhibition of [3H]-LTB4 binding to Leukotriene B4 receptor in the guinea pig spleen membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLeukotriene B4 receptor 1(Homo sapiens (Human))
Centre De Recherche De Vitry-Alfortville

Curated by ChEMBL
LigandPNGBDBM50001616(6-[4-(4-Amino-phenyl)-quinolin-2-yloxy]-2,2-dimeth...)
Affinity DataIC50:  250nMAssay Description:Inhibition of [3H]-LTB4 binding to Leukotriene B4 receptor in the human polymorphonuclear leukocytesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLeukotriene B4 receptor 1(Homo sapiens (Human))
Centre De Recherche De Vitry-Alfortville

Curated by ChEMBL
LigandPNGBDBM50001627(2,2-Dimethyl-6-[4-(4-trifluoromethyl-phenyl)-quino...)
Affinity DataIC50:  300nMAssay Description:Inhibition of [3H]-LTB4 binding to Leukotriene B4 receptor in the guinea pig spleen membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLeukotriene B4 receptor 1(Homo sapiens (Human))
Centre De Recherche De Vitry-Alfortville

Curated by ChEMBL
LigandPNGBDBM50001629(6-[4-(3-Methoxy-phenyl)-quinolin-2-yloxy]-2,2-dime...)
Affinity DataIC50:  300nMAssay Description:Inhibition of [3H]-LTB4 binding to Leukotriene B4 receptor in the guinea pig spleen membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLeukotriene B4 receptor 1(Homo sapiens (Human))
Centre De Recherche De Vitry-Alfortville

Curated by ChEMBL
LigandPNGBDBM50001623(2-[5-Methyl-5-(1H-tetrazol-5-yl)-hexyloxy]-4-pheny...)
Affinity DataIC50:  400nMAssay Description:Inhibition of [3H]-LTB4 binding to Leukotriene B4 receptor in the guinea pig spleen membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLeukotriene B4 receptor 1(Homo sapiens (Human))
Centre De Recherche De Vitry-Alfortville

Curated by ChEMBL
LigandPNGBDBM50001631(4-Phenyl-2-[5-(1H-tetrazol-5-yl)-pentyloxy]-quinol...)
Affinity DataIC50:  500nMAssay Description:Inhibition of [3H]-LTB4 binding to Leukotriene B4 receptor in the guinea pig spleen membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLeukotriene B4 receptor 1(Homo sapiens (Human))
Centre De Recherche De Vitry-Alfortville

Curated by ChEMBL
LigandPNGBDBM50001615(2-Methyl-6-(4-phenyl-quinolin-2-yloxy)-hexanoic ac...)
Affinity DataIC50:  550nMAssay Description:Inhibition of [3H]-LTB4 binding to Leukotriene B4 receptor in the guinea pig spleen membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLeukotriene B4 receptor 1(Homo sapiens (Human))
Centre De Recherche De Vitry-Alfortville

Curated by ChEMBL
LigandPNGBDBM50001632(6-(4-Phenyl-quinolin-2-yloxy)-hexanoic acid | CHEM...)
Affinity DataIC50:  700nMAssay Description:Inhibition of [3H]-LTB4 binding to Leukotriene B4 receptor in the guinea pig spleen membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLeukotriene B4 receptor 1(Homo sapiens (Human))
Centre De Recherche De Vitry-Alfortville

Curated by ChEMBL
LigandPNGBDBM50001624(6-[4-(2-Fluoro-phenyl)-quinolin-2-yloxy]-2,2-dimet...)
Affinity DataIC50:  800nMAssay Description:Inhibition of [3H]-LTB4 binding to Leukotriene B4 receptor in the guinea pig spleen membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLeukotriene B4 receptor 1(Homo sapiens (Human))
Centre De Recherche De Vitry-Alfortville

Curated by ChEMBL
LigandPNGBDBM50001626(6-[4-(3-Chloro-phenyl)-quinolin-2-yloxy]-2,2-dimet...)
Affinity DataIC50:  1.10E+3nMAssay Description:Inhibition of [3H]-LTB4 binding to Leukotriene B4 receptor in the guinea pig spleen membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLeukotriene B4 receptor 1(Homo sapiens (Human))
Centre De Recherche De Vitry-Alfortville

Curated by ChEMBL
LigandPNGBDBM50001613(7-(4-Phenyl-quinolin-2-yloxy)-heptanoic acid | CHE...)
Affinity DataIC50:  1.80E+3nMAssay Description:Inhibition of [3H]-LTB4 binding to Leukotriene B4 receptor in the guinea pig spleen membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLeukotriene B4 receptor 1(Homo sapiens (Human))
Centre De Recherche De Vitry-Alfortville

Curated by ChEMBL
LigandPNGBDBM50001633(8-(4-Phenyl-quinolin-2-yloxy)-octanoic acid | CHEM...)
Affinity DataIC50:  2.00E+3nMAssay Description:Inhibition of [3H]-LTB4 binding to Leukotriene B4 receptor in the guinea pig spleen membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLeukotriene B4 receptor 1(Homo sapiens (Human))
Centre De Recherche De Vitry-Alfortville

Curated by ChEMBL
LigandPNGBDBM50001621(6-(7-Chloro-4-phenyl-quinolin-2-yloxy)-2,2-dimethy...)
Affinity DataIC50:  2.00E+3nMAssay Description:Inhibition of [3H]-LTB4 binding to Leukotriene B4 receptor in the guinea pig spleen membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLeukotriene B4 receptor 1(Homo sapiens (Human))
Centre De Recherche De Vitry-Alfortville

Curated by ChEMBL
LigandPNGBDBM50001618(6-(6-Chloro-4-phenyl-quinolin-2-yloxy)-2,2-dimethy...)
Affinity DataIC50:  2.50E+3nMAssay Description:Inhibition of [3H]-LTB4 binding to Leukotriene B4 receptor in the guinea pig spleen membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLeukotriene B4 receptor 1(Homo sapiens (Human))
Centre De Recherche De Vitry-Alfortville

Curated by ChEMBL
LigandPNGBDBM50001625(2,2-Dimethyl-6-(4-phenyl-quinolin-2-yloxy)-hexanoi...)
Affinity DataIC50:  4.00E+3nMAssay Description:Inhibition of [3H]-LTB4 binding to Leukotriene B4 receptor in the human polymorphonuclear leukocytesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLeukotriene B4 receptor 1(Homo sapiens (Human))
Centre De Recherche De Vitry-Alfortville

Curated by ChEMBL
LigandPNGBDBM50001614(2,2-Dimethyl-6-(3-methyl-4-phenyl-quinolin-2-yloxy...)
Affinity DataIC50:  8.00E+3nMAssay Description:Inhibition of [3H]-LTB4 binding to Leukotriene B4 receptor in the guinea pig spleen membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed