Compile Data Set for Download or QSAR
maximum 50k data
Found 49 Enz. Inhib. hit(s) with all data for entry = 50000960
TargetTyrosine-protein kinase Lck(Homo sapiens (Human))
Purdue University

Curated by ChEMBL
LigandPNGBDBM50011418(2-(4-Amino-phenyl)-6-hydroxy-chromen-4-one | 2-(4-...)
Affinity DataIC50:  1.20E+3nMAssay Description:Ability to inhibit protein-tyrosine kinase activity of p56lck (isolated from bovine thymus) in vitro.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase Lck(Homo sapiens (Human))
Purdue University

Curated by ChEMBL
LigandPNGBDBM50011429(2-(4-Amino-phenyl)-5,7-dihydroxy-chromen-4-one | 2...)
Affinity DataIC50:  7.40E+3nMAssay Description:Ability to inhibit protein-tyrosine kinase activity of p56lck (isolated from bovine thymus) in vitro.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase Lck(Homo sapiens (Human))
Purdue University

Curated by ChEMBL
LigandPNGBDBM7460(2-(3,4-dihydroxyphenyl)-3,5,7-trihydroxy-4H-chrome...)
Affinity DataIC50:  1.30E+4nMAssay Description:Ability to inhibit protein-tyrosine kinase activity of p56lck (isolated from bovine thymus) in vitro.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase Lck(Homo sapiens (Human))
Purdue University

Curated by ChEMBL
LigandPNGBDBM50011424(2-(4-Hydroxy-3,5-dimethoxy-phenyl)-chromen-4-one |...)
Affinity DataIC50:  2.60E+4nMAssay Description:Ability to inhibit protein-tyrosine kinase activity of p56lck (isolated from bovine thymus) in vitro.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase Lck(Homo sapiens (Human))
Purdue University

Curated by ChEMBL
LigandPNGBDBM50011438(2-(4-Amino-phenyl)-7-hydroxy-chromen-4-one | 2-(4-...)
Affinity DataIC50:  1.38E+5nMAssay Description:Ability to inhibit protein-tyrosine kinase activity of p56lck (isolated from bovine thymus) in vitro.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase Lck(Homo sapiens (Human))
Purdue University

Curated by ChEMBL
LigandPNGBDBM50011437(2-(4-Amino-phenyl)-chromen-4-one | 2-(4-aminopheny...)
Affinity DataIC50:  2.10E+5nMAssay Description:Ability to inhibit protein-tyrosine kinase activity of p56lck (isolated from bovine thymus) in vitro.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase Lck(Homo sapiens (Human))
Purdue University

Curated by ChEMBL
LigandPNGBDBM50011455(2-(4-Hydroxy-phenyl)-4-oxo-4H-chromene-3-carboxyli...)
Affinity DataIC50:  4.39E+5nMAssay Description:Ability to inhibit protein-tyrosine kinase activity of p56lck (isolated from bovine thymus) in vitro.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase Lck(Homo sapiens (Human))
Purdue University

Curated by ChEMBL
LigandPNGBDBM50011446(2-(4-Hydroxy-phenyl)-chromen-4-one | 2-(4-hydroxyp...)
Affinity DataIC50:  5.04E+5nMAssay Description:Ability to inhibit protein-tyrosine kinase activity of p56lck (isolated from bovine thymus) in vitro.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase Lck(Homo sapiens (Human))
Purdue University

Curated by ChEMBL
LigandPNGBDBM50011416(2-(4-Amino-phenyl)-4-oxo-4H-chromene-3-carboxylic ...)
Affinity DataIC50:  8.10E+5nMAssay Description:Ability to inhibit protein-tyrosine kinase activity of p56lck (isolated from bovine thymus) in vitro.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase Lck(Homo sapiens (Human))
Purdue University

Curated by ChEMBL
LigandPNGBDBM50011422(2-(4-Hydroxy-phenyl)-7-methoxy-4-oxo-4H-chromene-3...)
Affinity DataIC50:  1.03E+6nMAssay Description:Ability to inhibit protein-tyrosine kinase activity of p56lck (isolated from bovine thymus) in vitro.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase Lck(Homo sapiens (Human))
Purdue University

Curated by ChEMBL
LigandPNGBDBM50011451(3-(2-Hydroxy-4-methoxy-phenyl)-3-oxo-propionic aci...)
Affinity DataIC50:  1.16E+6nMAssay Description:Ability to inhibit protein-tyrosine kinase activity of p56lck (isolated from bovine thymus) in vitro.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase Lck(Homo sapiens (Human))
Purdue University

Curated by ChEMBL
LigandPNGBDBM50011458(2-(4-Hydroxy-phenyl)-4-oxo-4H-chromene-3-carboxyli...)
Affinity DataIC50:  1.60E+6nMAssay Description:Ability to inhibit protein-tyrosine kinase activity of p56lck (isolated from bovine thymus) in vitro.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase Lck(Homo sapiens (Human))
Purdue University

Curated by ChEMBL
LigandPNGBDBM50011428(2-(3,4,5-Trimethoxy-phenyl)-chromen-4-one | 2-(3,4...)
Affinity DataIC50: >2.00E+6nMAssay Description:Ability to inhibit protein-tyrosine kinase activity of p56lck (isolated from bovine thymus) in vitro.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase Lck(Homo sapiens (Human))
Purdue University

Curated by ChEMBL
LigandPNGBDBM50011420(7-Methoxy-2-(4-nitro-phenyl)-4-oxo-4H-chromene-3-c...)
Affinity DataIC50: >2.00E+6nMAssay Description:Ability to inhibit protein-tyrosine kinase activity of p56lck (isolated from bovine thymus) in vitro.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase Lck(Homo sapiens (Human))
Purdue University

Curated by ChEMBL
LigandPNGBDBM50011431(2-(4-Acetylamino-phenyl)-6-methoxy-4-oxo-4H-chrome...)
Affinity DataIC50: >2.00E+6nMAssay Description:Ability to inhibit protein-tyrosine kinase activity of p56lck (isolated from bovine thymus) in vitro.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase Lck(Homo sapiens (Human))
Purdue University

Curated by ChEMBL
LigandPNGBDBM50011430(4-Oxo-2-(3,4,5-trimethoxy-phenyl)-4H-chromene-3-ca...)
Affinity DataIC50: >2.00E+6nMAssay Description:Ability to inhibit protein-tyrosine kinase activity of p56lck (isolated from bovine thymus) in vitro.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase Lck(Homo sapiens (Human))
Purdue University

Curated by ChEMBL
LigandPNGBDBM50011432(2-(3,4-Dimethoxy-phenyl)-4-oxo-4H-chromene-3-carbo...)
Affinity DataIC50: >2.00E+6nMAssay Description:Ability to inhibit protein-tyrosine kinase activity of p56lck (isolated from bovine thymus) in vitro.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase Lck(Homo sapiens (Human))
Purdue University

Curated by ChEMBL
LigandPNGBDBM50011433(3-(2,4-Bis-benzyloxy-6-hydroxy-phenyl)-3-oxo-propi...)
Affinity DataIC50: >2.00E+6nMAssay Description:Ability to inhibit protein-tyrosine kinase activity of p56lck (isolated from bovine thymus) in vitro.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase Lck(Homo sapiens (Human))
Purdue University

Curated by ChEMBL
LigandPNGBDBM50011434(2-(4-Bromo-phenyl)-4-oxo-4H-chromene-3-carboxylic ...)
Affinity DataIC50: >2.00E+6nMAssay Description:Ability to inhibit protein-tyrosine kinase activity of p56lck (isolated from bovine thymus) in vitro.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase Lck(Homo sapiens (Human))
Purdue University

Curated by ChEMBL
LigandPNGBDBM50011436(5,7-Dihydroxy-2-(4-nitro-phenyl)-4-oxo-4H-chromene...)
Affinity DataIC50: >2.00E+6nMAssay Description:Ability to inhibit protein-tyrosine kinase activity of p56lck (isolated from bovine thymus) in vitro.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase Lck(Homo sapiens (Human))
Purdue University

Curated by ChEMBL
LigandPNGBDBM50011435(3-(2-Hydroxy-5-methoxy-phenyl)-3-oxo-propionic aci...)
Affinity DataIC50: >2.00E+6nMAssay Description:Ability to inhibit protein-tyrosine kinase activity of p56lck (isolated from bovine thymus) in vitro.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase Lck(Homo sapiens (Human))
Purdue University

Curated by ChEMBL
LigandPNGBDBM50011419(6-Methoxy-2-(4-nitro-phenyl)-4-oxo-4H-chromene-3-c...)
Affinity DataIC50: >2.00E+6nMAssay Description:Ability to inhibit protein-tyrosine kinase activity of p56lck (isolated from bovine thymus) in vitro.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase Lck(Homo sapiens (Human))
Purdue University

Curated by ChEMBL
LigandPNGBDBM50011439(2-(3,5-Dimethoxy-phenyl)-4-oxo-4H-chromene-3-carbo...)
Affinity DataIC50: >2.00E+6nMAssay Description:Ability to inhibit protein-tyrosine kinase activity of p56lck (isolated from bovine thymus) in vitro.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase Lck(Homo sapiens (Human))
Purdue University

Curated by ChEMBL
LigandPNGBDBM50011440(2-(4-Nitro-phenyl)-4-oxo-4H-chromene-3-carboxylic ...)
Affinity DataIC50: >2.00E+6nMAssay Description:Ability to inhibit protein-tyrosine kinase activity of p56lck (isolated from bovine thymus) in vitro.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase Lck(Homo sapiens (Human))
Purdue University

Curated by ChEMBL
LigandPNGBDBM50011441(2-(4-Methoxy-phenyl)-4-oxo-4H-chromene-3-carboxyli...)
Affinity DataIC50: >2.00E+6nMAssay Description:Ability to inhibit protein-tyrosine kinase activity of p56lck (isolated from bovine thymus) in vitro.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase Lck(Homo sapiens (Human))
Purdue University

Curated by ChEMBL
LigandPNGBDBM50011415(3-(2-Hydroxy-phenyl)-3-oxo-propionic acid ethyl es...)
Affinity DataIC50: >2.00E+6nMAssay Description:Ability to inhibit protein-tyrosine kinase activity of p56lck (isolated from bovine thymus) in vitro.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase Lck(Homo sapiens (Human))
Purdue University

Curated by ChEMBL
LigandPNGBDBM50011442(6-Hydroxy-2-(4-nitro-phenyl)-chromen-4-one | 6-hyd...)
Affinity DataIC50: >2.00E+6nMAssay Description:Ability to inhibit protein-tyrosine kinase activity of p56lck (isolated from bovine thymus) in vitro.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase Lck(Homo sapiens (Human))
Purdue University

Curated by ChEMBL
LigandPNGBDBM50011443(2-(3,5-Dimethoxy-phenyl)-4-oxo-4H-chromene-3-carbo...)
Affinity DataIC50: >2.00E+6nMAssay Description:Ability to inhibit protein-tyrosine kinase activity of p56lck (isolated from bovine thymus) in vitro.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase Lck(Homo sapiens (Human))
Purdue University

Curated by ChEMBL
LigandPNGBDBM50011444(7-Methoxy-2-(4-nitro-phenyl)-4-oxo-4H-chromene-3-c...)
Affinity DataIC50: >2.00E+6nMAssay Description:Ability to inhibit protein-tyrosine kinase activity of p56lck (isolated from bovine thymus) in vitro.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase Lck(Homo sapiens (Human))
Purdue University

Curated by ChEMBL
LigandPNGBDBM50011445(2-(4-Benzyloxy-phenyl)-7-methoxy-4-oxo-4H-chromene...)
Affinity DataIC50: >2.00E+6nMAssay Description:Ability to inhibit protein-tyrosine kinase activity of p56lck (isolated from bovine thymus) in vitro.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase Lck(Homo sapiens (Human))
Purdue University

Curated by ChEMBL
LigandPNGBDBM50011453(3-Oxo-3-(2,3,4-trihydroxy-phenyl)-propionic acid m...)
Affinity DataIC50: >2.00E+6nMAssay Description:Ability to inhibit protein-tyrosine kinase activity of p56lck (isolated from bovine thymus) in vitro.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase Lck(Homo sapiens (Human))
Purdue University

Curated by ChEMBL
LigandPNGBDBM50011454(2-(4-Benzyloxy-phenyl)-6-methoxy-4-oxo-4H-chromene...)
Affinity DataIC50: >2.00E+6nMAssay Description:Ability to inhibit protein-tyrosine kinase activity of p56lck (isolated from bovine thymus) in vitro.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase Lck(Homo sapiens (Human))
Purdue University

Curated by ChEMBL
LigandPNGBDBM50011452(2-(4-Methoxy-phenyl)-4-oxo-4H-chromene-3-carboxyli...)
Affinity DataIC50: >2.00E+6nMAssay Description:Ability to inhibit protein-tyrosine kinase activity of p56lck (isolated from bovine thymus) in vitro.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase Lck(Homo sapiens (Human))
Purdue University

Curated by ChEMBL
LigandPNGBDBM50011447(4-Oxo-2-(3,4,5-trimethoxy-phenyl)-4H-chromene-3-ca...)
Affinity DataIC50: >2.00E+6nMAssay Description:Ability to inhibit protein-tyrosine kinase activity of p56lck (isolated from bovine thymus) in vitro.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase Lck(Homo sapiens (Human))
Purdue University

Curated by ChEMBL
LigandPNGBDBM50011449(3-(2-Hydroxy-phenyl)-3-oxo-propionic acid methyl e...)
Affinity DataIC50: >2.00E+6nMAssay Description:Ability to inhibit protein-tyrosine kinase activity of p56lck (isolated from bovine thymus) in vitro.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase Lck(Homo sapiens (Human))
Purdue University

Curated by ChEMBL
LigandPNGBDBM50011448(4-Oxo-2-[4-(3,4,5-trimethoxy-benzoylamino)-phenyl]...)
Affinity DataIC50: >2.00E+6nMAssay Description:Ability to inhibit protein-tyrosine kinase activity of p56lck (isolated from bovine thymus) in vitro.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase Lck(Homo sapiens (Human))
Purdue University

Curated by ChEMBL
LigandPNGBDBM50011450(2-(4-Bromo-phenyl)-4-oxo-4H-chromene-3-carboxylic ...)
Affinity DataIC50: >2.00E+6nMAssay Description:Ability to inhibit protein-tyrosine kinase activity of p56lck (isolated from bovine thymus) in vitro.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase Lck(Homo sapiens (Human))
Purdue University

Curated by ChEMBL
LigandPNGBDBM50011456(2-(4-Hydroxy-phenyl)-6-methoxy-4-oxo-4H-chromene-3...)
Affinity DataIC50: >2.00E+6nMAssay Description:Ability to inhibit protein-tyrosine kinase activity of p56lck (isolated from bovine thymus) in vitro.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase Lck(Homo sapiens (Human))
Purdue University

Curated by ChEMBL
LigandPNGBDBM50011460(2-(4-Acetylamino-phenyl)-7-methoxy-4-oxo-4H-chrome...)
Affinity DataIC50: >2.00E+6nMAssay Description:Ability to inhibit protein-tyrosine kinase activity of p56lck (isolated from bovine thymus) in vitro.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase Lck(Homo sapiens (Human))
Purdue University

Curated by ChEMBL
LigandPNGBDBM50011461(2-(4-Benzyloxy-phenyl)-4-oxo-4H-chromene-3-carboxy...)
Affinity DataIC50: >2.00E+6nMAssay Description:Ability to inhibit protein-tyrosine kinase activity of p56lck (isolated from bovine thymus) in vitro.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase Lck(Homo sapiens (Human))
Purdue University

Curated by ChEMBL
LigandPNGBDBM50011457(2-(4-Nitro-phenyl)-4-oxo-4H-chromene-3-carboxylic ...)
Affinity DataIC50: >2.00E+6nMAssay Description:Ability to inhibit protein-tyrosine kinase activity of p56lck (isolated from bovine thymus) in vitro.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase Lck(Homo sapiens (Human))
Purdue University

Curated by ChEMBL
LigandPNGBDBM50011459(6-Methoxy-2-(4-nitro-phenyl)-4-oxo-4H-chromene-3-c...)
Affinity DataIC50: >2.00E+6nMAssay Description:Ability to inhibit protein-tyrosine kinase activity of p56lck (isolated from bovine thymus) in vitro.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase Lck(Homo sapiens (Human))
Purdue University

Curated by ChEMBL
LigandPNGBDBM50011462(3-(2,4-Bis-benzyloxy-6-hydroxy-phenyl)-3-oxo-propi...)
Affinity DataIC50: >2.00E+6nMAssay Description:Ability to inhibit protein-tyrosine kinase activity of p56lck (isolated from bovine thymus) in vitro.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase Lck(Homo sapiens (Human))
Purdue University

Curated by ChEMBL
LigandPNGBDBM50011427(7-Hydroxy-2-(4-nitro-phenyl)-chromen-4-one | 7-hyd...)
Affinity DataIC50: >2.00E+6nMAssay Description:Ability to inhibit protein-tyrosine kinase activity of p56lck (isolated from bovine thymus) in vitro.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase Lck(Homo sapiens (Human))
Purdue University

Curated by ChEMBL
LigandPNGBDBM50011426(2-(4-Hydroxy-phenyl)-7-methoxy-4-oxo-4H-chromene-3...)
Affinity DataIC50: >2.00E+6nMAssay Description:Ability to inhibit protein-tyrosine kinase activity of p56lck (isolated from bovine thymus) in vitro.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase Lck(Homo sapiens (Human))
Purdue University

Curated by ChEMBL
LigandPNGBDBM50011417(5,7-Dihydroxy-2-(4-nitro-phenyl)-chromen-4-one | 5...)
Affinity DataIC50: >2.00E+6nMAssay Description:Ability to inhibit protein-tyrosine kinase activity of p56lck (isolated from bovine thymus) in vitro.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase Lck(Homo sapiens (Human))
Purdue University

Curated by ChEMBL
LigandPNGBDBM50011425(2-(3,4-Dimethoxy-phenyl)-4-oxo-4H-chromene-3-carbo...)
Affinity DataIC50: >2.00E+6nMAssay Description:Ability to inhibit protein-tyrosine kinase activity of p56lck (isolated from bovine thymus) in vitro.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase Lck(Homo sapiens (Human))
Purdue University

Curated by ChEMBL
LigandPNGBDBM50011421(2-(4-Nitro-phenyl)-chromen-4-one | CHEMBL64780)
Affinity DataIC50: >2.00E+6nMAssay Description:Ability to inhibit protein-tyrosine kinase activity of p56lck (isolated from bovine thymus) in vitro.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase Lck(Homo sapiens (Human))
Purdue University

Curated by ChEMBL
LigandPNGBDBM50011423(5,7-Bis-benzyloxy-2-(4-nitro-phenyl)-4-oxo-4H-chro...)
Affinity DataIC50: >2.00E+6nMAssay Description:Ability to inhibit protein-tyrosine kinase activity of p56lck (isolated from bovine thymus) in vitro.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed