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Found 34 Enz. Inhib. hit(s) with all data for entry = 50006459
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
University Of Ferrara

Curated by ChEMBL
LigandPNGBDBM50049378(1-((S)-2-{(S)-2-[(S)-2-Amino-3-(4-hydroxy-phenyl)-...)
Affinity DataKi:  0.0450nMAssay Description:Displacement of [3H]-DPDPE (0.63 nM) from Opioid receptor delta 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
University Of Ferrara

Curated by ChEMBL
LigandPNGBDBM50049377(1-((S)-2-{(S)-2-[(S)-2-Amino-3-(4-hydroxy-phenyl)-...)
Affinity DataKi:  0.0540nMAssay Description:Displacement of [3H]-DPDPE (0.63 nM) from Opioid receptor delta 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
University Of Ferrara

Curated by ChEMBL
LigandPNGBDBM50049376(1-((S)-2-{(S)-2-[(S)-2-Amino-3-(4-hydroxy-phenyl)-...)
Affinity DataKi:  0.0540nMAssay Description:Displacement of [3H]-DPDPE (0.63 nM) from Opioid receptor delta 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
University Of Ferrara

Curated by ChEMBL
LigandPNGBDBM50001468((S)-3-((S)-2-{(R)-2-[(S)-2-Amino-3-(4-hydroxy-phen...)
Affinity DataKi:  0.150nMAssay Description:Displacement of [3H]-DPDPE (0.63 nM) from Opioid receptor delta 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
University Of Ferrara

Curated by ChEMBL
LigandPNGBDBM50049377(1-((S)-2-{(S)-2-[(S)-2-Amino-3-(4-hydroxy-phenyl)-...)
Affinity DataKi:  0.270nMAssay Description:Displacement of [3H]-DAGO (1.28 nM) from Opioid receptor mu 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
University Of Ferrara

Curated by ChEMBL
LigandPNGBDBM50049376(1-((S)-2-{(S)-2-[(S)-2-Amino-3-(4-hydroxy-phenyl)-...)
Affinity DataKi:  0.580nMAssay Description:Displacement of [3H]-DAGO (1.28 nM) from Opioid receptor mu 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
University Of Ferrara

Curated by ChEMBL
LigandPNGBDBM50049378(1-((S)-2-{(S)-2-[(S)-2-Amino-3-(4-hydroxy-phenyl)-...)
Affinity DataKi:  2.45nMAssay Description:Displacement of [3H]-DAGO (1.28 nM) from Opioid receptor mu 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
University Of Ferrara

Curated by ChEMBL
LigandPNGBDBM50049379((S)-3-[(S)-2-({1-[(S)-2-Amino-3-(4-hydroxy-phenyl)...)
Affinity DataKi:  2.48nMAssay Description:Displacement of [3H]-DPDPE (0.63 nM) from Opioid receptor delta 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
University Of Ferrara

Curated by ChEMBL
LigandPNGBDBM50049382((S)-3-[(1-{(S)-2-[(S)-2-Amino-3-(4-hydroxy-phenyl)...)
Affinity DataKi:  3.28nMAssay Description:Displacement of [3H]-DPDPE (0.63 nM) from Opioid receptor delta 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
University Of Ferrara

Curated by ChEMBL
LigandPNGBDBM50049381((S)-3-[(1-{(S)-2-[(S)-2-Amino-3-(4-hydroxy-phenyl)...)
Affinity DataKi:  15.4nMAssay Description:Displacement of [3H]-DPDPE (0.63 nM) from Opioid receptor delta 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
University Of Ferrara

Curated by ChEMBL
LigandPNGBDBM50049375((S)-3-[(1-{(S)-2-[(S)-2-Amino-3-(4-hydroxy-phenyl)...)
Affinity DataKi:  19nMAssay Description:Displacement of [3H]-DPDPE (0.63 nM) from Opioid receptor delta 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
University Of Ferrara

Curated by ChEMBL
LigandPNGBDBM50049383((S)-3-{[1-({1-[(S)-2-Amino-3-(4-hydroxy-phenyl)-pr...)
Affinity DataKi:  87.8nMAssay Description:Displacement of [3H]-DPDPE (0.63 nM) from Opioid receptor delta 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
University Of Ferrara

Curated by ChEMBL
LigandPNGBDBM50001468((S)-3-((S)-2-{(R)-2-[(S)-2-Amino-3-(4-hydroxy-phen...)
Affinity DataKi:  147nMAssay Description:Displacement of [3H]-DAGO (1.28 nM) from Opioid receptor mu 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
University Of Ferrara

Curated by ChEMBL
LigandPNGBDBM50049379((S)-3-[(S)-2-({1-[(S)-2-Amino-3-(4-hydroxy-phenyl)...)
Affinity DataKi:  3.11E+3nMAssay Description:Displacement of [3H]-DAGO (1.28 nM) from Opioid receptor mu 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
University Of Ferrara

Curated by ChEMBL
LigandPNGBDBM50049380((S)-3-({1-[(S)-2-Amino-3-(4-hydroxy-phenyl)-propio...)
Affinity DataKi:  5.26E+3nMAssay Description:Displacement of [3H]-DPDPE (0.63 nM) from Opioid receptor delta 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
University Of Ferrara

Curated by ChEMBL
LigandPNGBDBM50049382((S)-3-[(1-{(S)-2-[(S)-2-Amino-3-(4-hydroxy-phenyl)...)
Affinity DataKi:  5.47E+3nMAssay Description:Displacement of [3H]-DAGO (1.28 nM) from Opioid receptor mu 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
University Of Ferrara

Curated by ChEMBL
LigandPNGBDBM50049381((S)-3-[(1-{(S)-2-[(S)-2-Amino-3-(4-hydroxy-phenyl)...)
Affinity DataKi:  6.82E+3nMAssay Description:Displacement of [3H]-DAGO (1.28 nM) from Opioid receptor mu 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
University Of Ferrara

Curated by ChEMBL
LigandPNGBDBM50049375((S)-3-[(1-{(S)-2-[(S)-2-Amino-3-(4-hydroxy-phenyl)...)
Affinity DataKi:  1.02E+4nMAssay Description:Displacement of [3H]-DAGO (1.28 nM) from Opioid receptor mu 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
University Of Ferrara

Curated by ChEMBL
LigandPNGBDBM50049383((S)-3-{[1-({1-[(S)-2-Amino-3-(4-hydroxy-phenyl)-pr...)
Affinity DataKi:  1.48E+4nMAssay Description:Displacement of [3H]-DAGO (1.28 nM) from Opioid receptor mu 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
University Of Ferrara

Curated by ChEMBL
LigandPNGBDBM50049380((S)-3-({1-[(S)-2-Amino-3-(4-hydroxy-phenyl)-propio...)
Affinity DataKi:  4.41E+5nMAssay Description:Displacement of [3H]-DAGO (1.28 nM) from Opioid receptor mu 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(MOUSE)
University Of Ferrara

Curated by ChEMBL
LigandPNGBDBM50049376(1-((S)-2-{(S)-2-[(S)-2-Amino-3-(4-hydroxy-phenyl)-...)
Affinity DataIC50:  0.190nMAssay Description:Inhibitory activity against Opioid receptor delta 1 of mouse vas deferens (MVD)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(MOUSE)
University Of Ferrara

Curated by ChEMBL
LigandPNGBDBM50049377(1-((S)-2-{(S)-2-[(S)-2-Amino-3-(4-hydroxy-phenyl)-...)
Affinity DataIC50:  0.430nMAssay Description:Inhibitory activity against Opioid receptor delta 1 of mouse vas deferens (MVD)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(MOUSE)
University Of Ferrara

Curated by ChEMBL
LigandPNGBDBM50001468((S)-3-((S)-2-{(R)-2-[(S)-2-Amino-3-(4-hydroxy-phen...)
Affinity DataIC50:  0.460nMAssay Description:Inhibitory activity against Opioid receptor delta 1 of mouse vas deferens (MVD)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(MOUSE)
University Of Ferrara

Curated by ChEMBL
LigandPNGBDBM50049378(1-((S)-2-{(S)-2-[(S)-2-Amino-3-(4-hydroxy-phenyl)-...)
Affinity DataIC50:  0.520nMAssay Description:Inhibitory activity against Opioid receptor delta 1 of mouse vas deferens (MVD)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
University Of Ferrara

Curated by ChEMBL
LigandPNGBDBM50049377(1-((S)-2-{(S)-2-[(S)-2-Amino-3-(4-hydroxy-phenyl)-...)
Affinity DataIC50:  15nMAssay Description:Compound was evaluated for its inhibitory activity towards Opioid receptor mu 1 of guinea pig ileum (GPI)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
University Of Ferrara

Curated by ChEMBL
LigandPNGBDBM50049376(1-((S)-2-{(S)-2-[(S)-2-Amino-3-(4-hydroxy-phenyl)-...)
Affinity DataIC50:  140nMAssay Description:Compound was evaluated for its inhibitory activity towards Opioid receptor mu 1 of guinea pig ileum (GPI)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
University Of Ferrara

Curated by ChEMBL
LigandPNGBDBM50001468((S)-3-((S)-2-{(R)-2-[(S)-2-Amino-3-(4-hydroxy-phen...)
Affinity DataIC50:  337nMAssay Description:Compound was evaluated for its inhibitory activity towards Opioid receptor mu 1 of guinea pig ileum (GPI)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(MOUSE)
University Of Ferrara

Curated by ChEMBL
LigandPNGBDBM50049375((S)-3-[(1-{(S)-2-[(S)-2-Amino-3-(4-hydroxy-phenyl)...)
Affinity DataIC50:  458nMAssay Description:Inhibitory activity against Opioid receptor delta 1 of mouse vas deferens (MVD)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(MOUSE)
University Of Ferrara

Curated by ChEMBL
LigandPNGBDBM50049382((S)-3-[(1-{(S)-2-[(S)-2-Amino-3-(4-hydroxy-phenyl)...)
Affinity DataIC50:  540nMAssay Description:Inhibitory activity against Opioid receptor delta 1 of mouse vas deferens (MVD)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
University Of Ferrara

Curated by ChEMBL
LigandPNGBDBM50049378(1-((S)-2-{(S)-2-[(S)-2-Amino-3-(4-hydroxy-phenyl)-...)
Affinity DataIC50:  558nMAssay Description:Compound was evaluated for its inhibitory activity towards Opioid receptor mu 1 of guinea pig ileum (GPI)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(MOUSE)
University Of Ferrara

Curated by ChEMBL
LigandPNGBDBM50049381((S)-3-[(1-{(S)-2-[(S)-2-Amino-3-(4-hydroxy-phenyl)...)
Affinity DataIC50:  1.64E+3nMAssay Description:Inhibitory activity against Opioid receptor delta 1 of mouse vas deferens (MVD)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
University Of Ferrara

Curated by ChEMBL
LigandPNGBDBM50049382((S)-3-[(1-{(S)-2-[(S)-2-Amino-3-(4-hydroxy-phenyl)...)
Affinity DataIC50: >1.00E+4nMAssay Description:Compound was evaluated for its inhibitory activity towards Opioid receptor mu 1 of guinea pig ileum (GPI)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
University Of Ferrara

Curated by ChEMBL
LigandPNGBDBM50049375((S)-3-[(1-{(S)-2-[(S)-2-Amino-3-(4-hydroxy-phenyl)...)
Affinity DataIC50: >1.00E+4nMAssay Description:Compound was evaluated for its inhibitory activity towards Opioid receptor mu 1 of guinea pig ileum (GPI)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
University Of Ferrara

Curated by ChEMBL
LigandPNGBDBM50049381((S)-3-[(1-{(S)-2-[(S)-2-Amino-3-(4-hydroxy-phenyl)...)
Affinity DataIC50: >1.00E+4nMAssay Description:Compound was evaluated for its inhibitory activity towards Opioid receptor mu 1 of guinea pig ileum (GPI)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed