Found 48 Enz. Inhib. hit(s) with all data for entry = 50007045 TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Oregon State University
Curated by ChEMBL
Oregon State University
Curated by ChEMBL
Affinity DataKi: 0.310nMAssay Description:Binding affinity to Opioid receptor kappa 1 by competitive inhibition of radioligand [3H]-diprenorphine using cloned receptors transiently expressed ...More data for this Ligand-Target Pair
Affinity DataKi: 0.920nMAssay Description:Binding affinity to Opioid receptor mu 1 by competitive inhibition of radioligand [3H]-DAMGO using cloned receptors transiently expressed on CHO cell...More data for this Ligand-Target Pair
Affinity DataKi: 1.20nMAssay Description:Binding affinity to Opioid receptor mu 1 by competitive inhibition of radioligand [3H]-DAMGO using cloned receptors transiently expressed on CHO cell...More data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Oregon State University
Curated by ChEMBL
Oregon State University
Curated by ChEMBL
Affinity DataKi: 1.5nMAssay Description:Binding affinity to Opioid receptor kappa 1 by competitive inhibition of radioligand [3H]-diprenorphine using cloned receptors transiently expressed ...More data for this Ligand-Target Pair
Affinity DataKi: 1.5nMAssay Description:Binding affinity to Opioid receptor mu 1 by competitive inhibition of radioligand [3H]-DAMGO using cloned receptors transiently expressed on CHO cell...More data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Oregon State University
Curated by ChEMBL
Oregon State University
Curated by ChEMBL
Affinity DataKi: 2.5nMAssay Description:Binding affinity to Opioid receptor kappa 1 by competitive inhibition of radioligand [3H]-diprenorphine using cloned receptors transiently expressed ...More data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Oregon State University
Curated by ChEMBL
Oregon State University
Curated by ChEMBL
Affinity DataKi: 2.60nMAssay Description:Binding affinity to Opioid receptor kappa 1 by competitive inhibition of radioligand [3H]-diprenorphine using cloned receptors transiently expressed ...More data for this Ligand-Target Pair
Affinity DataKi: 3.20nMAssay Description:Binding affinity to Opioid receptor mu 1 by competitive inhibition of radioligand [3H]-DAMGO using cloned receptors transiently expressed on CHO cell...More data for this Ligand-Target Pair
Affinity DataKi: 4.40nMAssay Description:Binding affinity to Opioid receptor mu 1 by competitive inhibition of radioligand [3H]-DAMGO using cloned receptors transiently expressed on CHO cell...More data for this Ligand-Target Pair
Affinity DataKi: 4.80nMAssay Description:Binding affinity to Opioid receptor mu 1 by competitive inhibition of radioligand [3H]-DAMGO using cloned receptors transiently expressed on CHO cell...More data for this Ligand-Target Pair
Affinity DataKi: 6.10nMAssay Description:Binding affinity to Opioid receptor mu 1 by competitive inhibition of radioligand [3H]-DAMGO using cloned receptors transiently expressed on CHO cell...More data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Oregon State University
Curated by ChEMBL
Oregon State University
Curated by ChEMBL
Affinity DataKi: 8nMAssay Description:Binding affinity to Opioid receptor kappa 1 by competitive inhibition of radioligand [3H]-diprenorphine using cloned receptors transiently expressed ...More data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Oregon State University
Curated by ChEMBL
Oregon State University
Curated by ChEMBL
Affinity DataKi: 8nMAssay Description:Binding affinity to Opioid receptor kappa 1 by competitive inhibition of radioligand [3H]-diprenorphine using cloned receptors transiently expressed ...More data for this Ligand-Target Pair
Affinity DataKi: 8.20nMAssay Description:Binding affinity to Opioid receptor delta 1 by competitive inhibition of radioligand [3H]-DPDPE using cloned receptors transiently expressed on CHO c...More data for this Ligand-Target Pair
Affinity DataKi: 8.30nMAssay Description:Binding affinity to Opioid receptor mu 1 by competitive inhibition of radioligand [3H]-DAMGO using cloned receptors transiently expressed on CHO cell...More data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Oregon State University
Curated by ChEMBL
Oregon State University
Curated by ChEMBL
Affinity DataKi: 12nMAssay Description:Binding affinity to Opioid receptor kappa 1 by competitive inhibition of radioligand [3H]-diprenorphine using cloned receptors transiently expressed ...More data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Oregon State University
Curated by ChEMBL
Oregon State University
Curated by ChEMBL
Affinity DataKi: 12nMAssay Description:Binding affinity to Opioid receptor kappa 1 by competitive inhibition of radioligand [3H]-diprenorphine using cloned receptors transiently expressed ...More data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Oregon State University
Curated by ChEMBL
Oregon State University
Curated by ChEMBL
Affinity DataKi: 14nMAssay Description:Binding affinity to Opioid receptor kappa 1 by competitive inhibition of radioligand [3H]-diprenorphine using cloned receptors transiently expressed ...More data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Oregon State University
Curated by ChEMBL
Oregon State University
Curated by ChEMBL
Affinity DataKi: 20nMAssay Description:Binding affinity to Opioid receptor kappa 1 by competitive inhibition of radioligand [3H]-diprenorphine using cloned receptors transiently expressed ...More data for this Ligand-Target Pair
Affinity DataKi: 22nMAssay Description:Binding affinity to Opioid receptor delta 1 by competitive inhibition of radioligand [3H]-DPDPE using cloned receptors transiently expressed on CHO c...More data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Oregon State University
Curated by ChEMBL
Oregon State University
Curated by ChEMBL
Affinity DataKi: 28nMAssay Description:Binding affinity to Opioid receptor kappa 1 by competitive inhibition of radioligand [3H]-diprenorphine using cloned receptors transiently expressed ...More data for this Ligand-Target Pair
Affinity DataKi: 28nMAssay Description:Binding affinity to Opioid receptor delta 1 by competitive inhibition of radioligand [3H]-DPDPE using cloned receptors transiently expressed on CHO c...More data for this Ligand-Target Pair
Affinity DataKi: 28nMAssay Description:Binding affinity to Opioid receptor delta 1 by competitive inhibition of radioligand [3H]-DPDPE using cloned receptors transiently expressed on CHO c...More data for this Ligand-Target Pair
Affinity DataKi: 40nMAssay Description:Binding affinity to Opioid receptor mu 1 by competitive inhibition of radioligand [3H]-DAMGO using cloned receptors transiently expressed on CHO cell...More data for this Ligand-Target Pair
Affinity DataKi: 48nMAssay Description:Binding affinity to Opioid receptor delta 1 by competitive inhibition of radioligand [3H]-DPDPE using cloned receptors transiently expressed on CHO c...More data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Oregon State University
Curated by ChEMBL
Oregon State University
Curated by ChEMBL
Affinity DataKi: 58nMAssay Description:Binding affinity to Opioid receptor kappa 1 by competitive inhibition of radioligand [3H]-diprenorphine using cloned receptors transiently expressed ...More data for this Ligand-Target Pair
Affinity DataKi: 62nMAssay Description:Binding affinity to Opioid receptor mu 1 by competitive inhibition of radioligand [3H]-DAMGO using cloned receptors transiently expressed on CHO cell...More data for this Ligand-Target Pair
Affinity DataKi: 75nMAssay Description:Binding affinity to Opioid receptor mu 1 by competitive inhibition of radioligand [3H]-DAMGO using cloned receptors transiently expressed on CHO cell...More data for this Ligand-Target Pair
Affinity DataKi: 100nMAssay Description:Binding affinity of compound was measured on Opioid receptor mu 1 by competitive inhibition of radioligand [3H]-DAMGO using cloned receptors transien...More data for this Ligand-Target Pair
Affinity DataKi: 180nMAssay Description:Binding affinity to Opioid receptor mu 1 by competitive inhibition of radioligand [3H]-DAMGO using cloned receptors transiently expressed on CHO cell...More data for this Ligand-Target Pair
Affinity DataKi: 180nMAssay Description:Binding affinity to Opioid receptor delta 1 by competitive inhibition of radioligand [3H]-DPDPE using cloned receptors transiently expressed on CHO c...More data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Oregon State University
Curated by ChEMBL
Oregon State University
Curated by ChEMBL
Affinity DataKi: 200nMAssay Description:Binding affinity of compound was measured on Opioid receptor kappa 1 by competitive inhibition of radioligand [3H]-diprenorphine using cloned recepto...More data for this Ligand-Target Pair
Affinity DataKi: 210nMAssay Description:Binding affinity of compound was measured on Opioid receptor mu 1 by competitive inhibition of radioligand [3H]-DAMGO using cloned receptors transien...More data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Oregon State University
Curated by ChEMBL
Oregon State University
Curated by ChEMBL
Affinity DataKi: 270nMAssay Description:Binding affinity of compound was measured on Opioid receptor kappa 1 by competitive inhibition of radioligand [3H]-diprenorphine using cloned recepto...More data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Oregon State University
Curated by ChEMBL
Oregon State University
Curated by ChEMBL
Affinity DataKi: 300nMAssay Description:Binding affinity of compound was measured on Opioid receptor kappa 1 by competitive inhibition of radioligand [3H]-diprenorphine using cloned recepto...More data for this Ligand-Target Pair
Affinity DataKi: 320nMAssay Description:Binding affinity of compound was measured on Opioid receptor delta 1 by competitive inhibition of radioligand [3H]-DPDPE using cloned receptors trans...More data for this Ligand-Target Pair
Affinity DataKi: 320nMAssay Description:Binding affinity of compound was measured on Opioid receptor mu 1 by competitive inhibition of radioligand [3H]-DAMGO using cloned receptors transien...More data for this Ligand-Target Pair
Affinity DataKi: 430nMAssay Description:Binding affinity to Opioid receptor delta 1 by competitive inhibition of radioligand [3H]-DPDPE using cloned receptors transiently expressed on CHO c...More data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Oregon State University
Curated by ChEMBL
Oregon State University
Curated by ChEMBL
Affinity DataKi: 480nMAssay Description:Binding affinity of compound was measured on Opioid receptor kappa 1 by competitive inhibition of radioligand [3H]-diprenorphine using cloned recepto...More data for this Ligand-Target Pair
Affinity DataKi: 910nMAssay Description:Binding affinity of compound was measured on Opioid receptor mu 1 by competitive inhibition of radioligand [3H]-DAMGO using cloned receptors transien...More data for this Ligand-Target Pair
Affinity DataKi: 1.00E+3nMAssay Description:Binding affinity of compound was measured on Opioid receptor delta 1 by competitive inhibition of radioligand [3H]-DPDPE using cloned receptors trans...More data for this Ligand-Target Pair
Affinity DataKi: 1.30E+3nMAssay Description:Binding affinity of compound was measured on Opioid receptor delta 1 by competitive inhibition of radioligand [3H]-DPDPE using cloned receptors trans...More data for this Ligand-Target Pair
Affinity DataKi: 1.30E+3nMAssay Description:Binding affinity to Opioid receptor delta 1 by competitive inhibition of radioligand [3H]-DPDPE using cloned receptors transiently expressed on CHO c...More data for this Ligand-Target Pair
Affinity DataKi: 1.60E+3nMAssay Description:Binding affinity to Opioid receptor delta 1 by competitive inhibition of radioligand [3H]-DPDPE using cloned receptors transiently expressed on CHO c...More data for this Ligand-Target Pair
Affinity DataKi: 1.90E+3nMAssay Description:Binding affinity to Opioid receptor delta 1 by competitive inhibition of radioligand [3H]-DPDPE using cloned receptors transiently expressed on CHO c...More data for this Ligand-Target Pair
Affinity DataKi: 2.80E+3nMAssay Description:Binding affinity of compound was measured on Opioid receptor delta 1 by competitive inhibition of radioligand [3H]-DPDPE using cloned receptors trans...More data for this Ligand-Target Pair
Affinity DataKi: 3.30E+3nMAssay Description:Binding affinity to Opioid receptor delta 1 by competitive inhibition of radioligand [3H]-DPDPE using cloned receptors transiently expressed on CHO c...More data for this Ligand-Target Pair
Affinity DataKi: 4.10E+3nMAssay Description:Binding affinity to Opioid receptor delta 1 by competitive inhibition of radioligand [3H]-DPDPE using cloned receptors transiently expressed on CHO c...More data for this Ligand-Target Pair
