TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Homo sapiens (Human))
University Of Wollongong
Curated by ChEMBL
University Of Wollongong
Curated by ChEMBL
Affinity DataKi: 0.0460nMAssay Description:Binding affinity against nicotinic acetylcholine receptor alpha4-beta2 using [3H]epibatidine as radioligand expressed in HEK293 cells or tsA cellsMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-4(Homo sapiens (Human))
University Of Wollongong
Curated by ChEMBL
University Of Wollongong
Curated by ChEMBL
Affinity DataKi: 0.0720nMAssay Description:Binding affinity against nicotinic acetylcholine receptor using [3H]epibatidine as radioligand in rat brain tissueMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor; alpha2/beta4(Homo sapiens (Human))
University Of Wollongong
Curated by ChEMBL
University Of Wollongong
Curated by ChEMBL
Affinity DataKi: 0.0910nMAssay Description:Agonistic potency against nicotinic acetylcholine receptor alpha3-beta4More data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-4(Homo sapiens (Human))
University Of Wollongong
Curated by ChEMBL
University Of Wollongong
Curated by ChEMBL
Affinity DataKi: 0.457nMAssay Description:Binding affinity of the compound was determined against Nicotinic acetylcholine receptor using [3H]-(-)-nicotine radioligandMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Homo sapiens (Human))
University Of Wollongong
Curated by ChEMBL
University Of Wollongong
Curated by ChEMBL
Affinity DataKi: 7.40nMAssay Description:Binding affinity against nicotinic acetylcholine receptor alpha4-beta2 using [3H]epibatidine as radioligand expressed in HEK293 cells or tsA cellsMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Homo sapiens (Human))
University Of Wollongong
Curated by ChEMBL
University Of Wollongong
Curated by ChEMBL
Affinity DataKi: 9.10nMAssay Description:Binding affinity against nicotinic acetylcholine receptor using [3H]epibatidine as radioligand in rat brain tissueMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor; alpha2/beta4(Homo sapiens (Human))
University Of Wollongong
Curated by ChEMBL
University Of Wollongong
Curated by ChEMBL
Affinity DataKi: 31nMAssay Description:In vitro ability to displace [3H]-(-)-cytisine binding to whole rat brain membranes at Nicotinic acetylcholine receptor alpha4-beta2More data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-4(Homo sapiens (Human))
University Of Wollongong
Curated by ChEMBL
University Of Wollongong
Curated by ChEMBL
Affinity DataKi: 38nMAssay Description:Binding affinity against nicotinic acetylcholine receptor alpha2-beta4 using [3H]epibatidine as radioligand expressed in HEK293 cells or tsA cellsMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-4(Homo sapiens (Human))
University Of Wollongong
Curated by ChEMBL
University Of Wollongong
Curated by ChEMBL
Affinity DataKi: 88nMAssay Description:Binding affinity against nicotinic acetylcholine receptor alpha4-beta2 using [3H]epibatidine as radioligand expressed in HEK293 cells or tsA cellsMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor; alpha2/beta4(Homo sapiens (Human))
University Of Wollongong
Curated by ChEMBL
University Of Wollongong
Curated by ChEMBL
Affinity DataKi: 103nMAssay Description:Binding affinity against nicotinic acetylcholine receptor alpha2-beta4 using [3H]epibatidine as radioligand expressed in HEK293 cells or tsA cellsMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-4(Homo sapiens (Human))
University Of Wollongong
Curated by ChEMBL
University Of Wollongong
Curated by ChEMBL
Affinity DataKi: 129nMAssay Description:Binding affinity against nicotinic acetylcholine receptor alpha4-beta4 using [3H]epibatidine as radioligand expressed in HEK293 cells or tsA cellsMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-4(Homo sapiens (Human))
University Of Wollongong
Curated by ChEMBL
University Of Wollongong
Curated by ChEMBL
Affinity DataKi: 320nMAssay Description:Binding affinity against nicotinic acetylcholine receptor alpha3-beta4 using [3H]epibatidine as radioligand expressed in HEK293 cells or tsA cellsMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-4(Homo sapiens (Human))
University Of Wollongong
Curated by ChEMBL
University Of Wollongong
Curated by ChEMBL
Affinity DataEC50: 4.30E+3nMAssay Description:Agonistic potency against nicotinic acetylcholine receptor alpha3-beta4More data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-4(Homo sapiens (Human))
University Of Wollongong
Curated by ChEMBL
University Of Wollongong
Curated by ChEMBL
Affinity DataEC50: 19nMAssay Description:Binding affinity against nicotinic acetylcholine receptor alpha3-beta4 using [3H]epibatidine as radioligand expressed in HEK293 cells or tsA cellsMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-4(Homo sapiens (Human))
University Of Wollongong
Curated by ChEMBL
University Of Wollongong
Curated by ChEMBL
Affinity DataEC50: 2.10E+3nMAssay Description:Binding affinity of the compound was determined against Nicotinic acetylcholine receptor using [3H]-(-)-nicotine radioligandMore data for this Ligand-Target Pair