Compile Data Set for Download or QSAR
maximum 50k data
Found 23 Enz. Inhib. hit(s) with all data for entry = 50011906
TargetVoltage-dependent N-type calcium channel subunit alpha-1B(Homo sapiens (Human))
Minase Research Institute

Curated by ChEMBL
LigandPNGBDBM50111944((R)-4-[(R)-2-Cyclohexylmethylsulfanyl-1-(4-phenoxy...)
Affinity DataIC50:  120nMAssay Description:In vitro inhibition of N-type calcium channels in IMR-32 cells.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent N-type calcium channel subunit alpha-1B(Homo sapiens (Human))
Minase Research Institute

Curated by ChEMBL
LigandPNGBDBM50111936((R)-3-(2-Methoxy-acetyl)-thiazolidine-4-carboxylic...)
Affinity DataIC50:  120nMAssay Description:In vitro inhibition of N-type calcium channels in IMR-32 cells.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent N-type calcium channel subunit alpha-1B(Homo sapiens (Human))
Minase Research Institute

Curated by ChEMBL
LigandPNGBDBM50111940((R)-4-[(R)-2-Cyclohexylmethylsulfanyl-1-(4-phenoxy...)
Affinity DataIC50:  140nMAssay Description:In vitro inhibition of N-type calcium channels in IMR-32 cells.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent N-type calcium channel subunit alpha-1B(Homo sapiens (Human))
Minase Research Institute

Curated by ChEMBL
LigandPNGBDBM50111945((R)-3-(2-Methoxy-ethyl)-thiazolidine-4-carboxylic ...)
Affinity DataIC50:  200nMAssay Description:In vitro inhibition of N-type calcium channels in IMR-32 cells.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent N-type calcium channel subunit alpha-1B(Homo sapiens (Human))
Minase Research Institute

Curated by ChEMBL
LigandPNGBDBM50111935((R)-Thiazolidine-4-carboxylic acid [(R)-2-cyclohex...)
Affinity DataIC50:  290nMAssay Description:In vitro inhibition of N-type calcium channels in IMR-32 cells.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent N-type calcium channel subunit alpha-1B(Homo sapiens (Human))
Minase Research Institute

Curated by ChEMBL
LigandPNGBDBM50111949((R)-4-[(R)-2-Cyclohexylmethylsulfanyl-1-(4-phenoxy...)
Affinity DataIC50:  330nMAssay Description:In vitro inhibition of N-type calcium channels in IMR-32 cells.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent N-type calcium channel subunit alpha-1B(Homo sapiens (Human))
Minase Research Institute

Curated by ChEMBL
LigandPNGBDBM50111938((R)-3-(2-Hydroxy-ethyl)-thiazolidine-4-carboxylic ...)
Affinity DataIC50:  350nMAssay Description:In vitro inhibition of N-type calcium channels in IMR-32 cells.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent N-type calcium channel subunit alpha-1B(Homo sapiens (Human))
Minase Research Institute

Curated by ChEMBL
LigandPNGBDBM50111948((R)-4-[(R)-2-Cyclohexylmethylsulfanyl-1-(4-phenoxy...)
Affinity DataIC50:  360nMAssay Description:In vitro inhibition of N-type calcium channels in IMR-32 cells.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent N-type calcium channel subunit alpha-1B(Homo sapiens (Human))
Minase Research Institute

Curated by ChEMBL
LigandPNGBDBM50111950((R)-4-[(R)-2-Cyclohexylmethylsulfanyl-1-(4-methoxy...)
Affinity DataIC50:  390nMAssay Description:In vitro inhibition of N-type calcium channels in IMR-32 cells.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent N-type calcium channel subunit alpha-1B(Homo sapiens (Human))
Minase Research Institute

Curated by ChEMBL
LigandPNGBDBM50111939((R)-4-[(R)-1-(4-Benzyloxy-benzylcarbamoyl)-2-cyclo...)
Affinity DataIC50:  500nMAssay Description:In vitro inhibition of N-type calcium channels in IMR-32 cells.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent N-type calcium channel subunit alpha-1B(Homo sapiens (Human))
Minase Research Institute

Curated by ChEMBL
LigandPNGBDBM50111947((R)-4-[(R)-2-Cyclohexylmethylsulfanyl-1-(4-nitro-b...)
Affinity DataIC50:  600nMAssay Description:In vitro inhibition of N-type calcium channels in IMR-32 cells.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent N-type calcium channel subunit alpha-1B(Homo sapiens (Human))
Minase Research Institute

Curated by ChEMBL
LigandPNGBDBM50111933((R)-4-[(R)-2-Cyclohexylmethylsulfanyl-1-(4-dimethy...)
Affinity DataIC50:  610nMAssay Description:In vitro inhibition of N-type calcium channels in IMR-32 cells.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent N-type calcium channel subunit alpha-1B(Homo sapiens (Human))
Minase Research Institute

Curated by ChEMBL
LigandPNGBDBM50111946((R)-2-tert-Butoxycarbonylamino-3-cyclohexylmethyls...)
Affinity DataIC50:  610nMAssay Description:In vitro inhibition of N-type calcium channels in IMR-32 cells.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent N-type calcium channel subunit alpha-1B(Homo sapiens (Human))
Minase Research Institute

Curated by ChEMBL
LigandPNGBDBM50102915(CHEMBL431324 | [(R)-2-Cyclopentylmethylsulfanyl-1-...)
Affinity DataIC50:  640nMAssay Description:In vitro inhibition of N-type calcium channels in IMR-32 cells.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent N-type calcium channel subunit alpha-1B(Homo sapiens (Human))
Minase Research Institute

Curated by ChEMBL
LigandPNGBDBM50111937((R)-3-Cyclohexylmethylsulfanyl-2-isobutoxycarbonyl...)
Affinity DataIC50:  720nMAssay Description:In vitro inhibition of N-type calcium channels in IMR-32 cells.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent N-type calcium channel subunit alpha-1B(Homo sapiens (Human))
Minase Research Institute

Curated by ChEMBL
LigandPNGBDBM50111941((S)-2-[(R)-2-Cyclohexylmethylsulfanyl-1-(4-methoxy...)
Affinity DataIC50:  880nMAssay Description:In vitro inhibition of N-type calcium channels in IMR-32 cells.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent N-type calcium channel subunit alpha-1B(Homo sapiens (Human))
Minase Research Institute

Curated by ChEMBL
LigandPNGBDBM50111953((R)-3-Cyclohexylmethylsulfanyl-2-(cyclopentanecarb...)
Affinity DataIC50:  920nMAssay Description:In vitro inhibition of N-type calcium channels in IMR-32 cells.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent N-type calcium channel subunit alpha-1B(Homo sapiens (Human))
Minase Research Institute

Curated by ChEMBL
LigandPNGBDBM50111943((R)-3-Cyclohexylmethylsulfanyl-2-(3-methyl-butyryl...)
Affinity DataIC50:  1.20E+3nMAssay Description:In vitro inhibition of N-type calcium channels in IMR-32 cells.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent N-type calcium channel subunit alpha-1B(Homo sapiens (Human))
Minase Research Institute

Curated by ChEMBL
LigandPNGBDBM50111954((R)-2-(Cyclohexanecarbonyl-amino)-3-cyclohexylmeth...)
Affinity DataIC50:  1.30E+3nMAssay Description:In vitro inhibition of N-type calcium channels in IMR-32 cells.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent N-type calcium channel subunit alpha-1B(Homo sapiens (Human))
Minase Research Institute

Curated by ChEMBL
LigandPNGBDBM50111951((R)-4-[(R)-2-Cyclohexylmethylsulfanyl-1-(4-hydroxy...)
Affinity DataIC50:  1.80E+3nMAssay Description:In vitro inhibition of N-type calcium channels in IMR-32 cells.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent N-type calcium channel subunit alpha-1B(Homo sapiens (Human))
Minase Research Institute

Curated by ChEMBL
LigandPNGBDBM50111952((R)-3-Cyclohexylmethylsulfanyl-2-[(thiazole-4-carb...)
Affinity DataIC50:  1.90E+3nMAssay Description:In vitro inhibition of N-type calcium channels in IMR-32 cells.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent N-type calcium channel subunit alpha-1B(Homo sapiens (Human))
Minase Research Institute

Curated by ChEMBL
LigandPNGBDBM50111942((R)-3-Cyclohexylmethylsulfanyl-2-[((R)-thiazolidin...)
Affinity DataIC50:  2.70E+3nMAssay Description:In vitro inhibition of N-type calcium channels in IMR-32 cells.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent N-type calcium channel subunit alpha-1B(Homo sapiens (Human))
Minase Research Institute

Curated by ChEMBL
LigandPNGBDBM50111934((R)-2-Amino-3-cyclohexylmethylsulfanyl-propionic a...)
Affinity DataIC50:  5.80E+3nMAssay Description:In vitro inhibition of N-type calcium channels in IMR-32 cells.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed