TargetCalcium-dependent protein kinase 4(Plasmodium falciparum (isolate 3D7))
Montclair State University
Curated by ChEMBL
Montclair State University
Curated by ChEMBL
Affinity DataIC50: 4nMAssay Description:Inhibition of CDPK4 in Plasmodium falciparum 3D7 microgametesMore data for this Ligand-Target Pair
TargetCell division related protein kinase 2(Leishmania major)
Montclair State University
Curated by ChEMBL
Montclair State University
Curated by ChEMBL
Affinity DataIC50: 5nMAssay Description:Inhibition of Leishmania major CRK3 expressed in Escherichia coli BL21 (DE3) using 5FAM-GGGRSPGRRRRK-OH as substrate after 60 mins by IMAP assayMore data for this Ligand-Target Pair
TargetcGMP-dependent protein kinase(Plasmodium falciparum)
Montclair State University
Curated by ChEMBL
Montclair State University
Curated by ChEMBL
Affinity DataIC50: 8nMAssay Description:Inhibition of PKG in Plasmodium falciparum 3D7 microgametesMore data for this Ligand-Target Pair
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform(Homo sapiens (Human))
Montclair State University
Curated by ChEMBL
Montclair State University
Curated by ChEMBL
Affinity DataIC50: <10nMAssay Description:Inhibition of PI3KgammaMore data for this Ligand-Target Pair
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform(Homo sapiens (Human))
Montclair State University
Curated by ChEMBL
Montclair State University
Curated by ChEMBL
Affinity DataIC50: <10nMAssay Description:Inhibition of PI3KdeltaMore data for this Ligand-Target Pair
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit beta isoform(Homo sapiens (Human))
Montclair State University
Curated by ChEMBL
Montclair State University
Curated by ChEMBL
Affinity DataIC50: <10nMAssay Description:Inhibition of PI3KbetaMore data for this Ligand-Target Pair
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform(Homo sapiens (Human))
Montclair State University
Curated by ChEMBL
Montclair State University
Curated by ChEMBL
Affinity DataIC50: <10nMAssay Description:Inhibition of PI3KalphaMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase mTOR(Homo sapiens (Human))
Montclair State University
Curated by ChEMBL
Montclair State University
Curated by ChEMBL
TargetCell division related protein kinase 2(Leishmania major)
Montclair State University
Curated by ChEMBL
Montclair State University
Curated by ChEMBL
Affinity DataIC50: 20nMAssay Description:Inhibition of Leishmania major CRK3 expressed in Escherichia coli BL21 (DE3) using 5FAM-GGGRSPGRRRRK-OH as substrate after 60 mins by IMAP assayMore data for this Ligand-Target Pair
TargetCell division related protein kinase 2(Leishmania major)
Montclair State University
Curated by ChEMBL
Montclair State University
Curated by ChEMBL
Affinity DataIC50: 60nMAssay Description:Inhibition of Leishmania major CRK3 expressed in Escherichia coli BL21 (DE3) using 5FAM-GGGRSPGRRRRK-OH as substrate after 60 mins by IMAP assayMore data for this Ligand-Target Pair
TargetCalcium-dependent protein kinase 4(Plasmodium falciparum (isolate 3D7))
Montclair State University
Curated by ChEMBL
Montclair State University
Curated by ChEMBL
Affinity DataIC50: 177nMAssay Description:Inhibition of CDPK4 in Plasmodium falciparum 3D7 microgametesMore data for this Ligand-Target Pair
TargetCell division related protein kinase 2(Leishmania major)
Montclair State University
Curated by ChEMBL
Montclair State University
Curated by ChEMBL
Affinity DataIC50: 240nMAssay Description:Inhibition of Leishmania major CRK3 expressed in Escherichia coli BL21 (DE3) using 5FAM-GGGRSPGRRRRK-OH as substrate after 60 mins by IMAP assayMore data for this Ligand-Target Pair
TargetCell division related protein kinase 2(Leishmania major)
Montclair State University
Curated by ChEMBL
Montclair State University
Curated by ChEMBL
Affinity DataIC50: 260nMAssay Description:Inhibition of Leishmania major CRK3 expressed in Escherichia coli BL21 (DE3) using 5FAM-GGGRSPGRRRRK-OH as substrate after 60 mins by IMAP assayMore data for this Ligand-Target Pair
TargetCell division related protein kinase 2(Leishmania major)
Montclair State University
Curated by ChEMBL
Montclair State University
Curated by ChEMBL
Affinity DataIC50: 510nMAssay Description:Inhibition of Leishmania major CRK3 expressed in Escherichia coli BL21 (DE3) using 5FAM-GGGRSPGRRRRK-OH as substrate after 60 mins by IMAP assayMore data for this Ligand-Target Pair
TargetCell division related protein kinase 2(Leishmania major)
Montclair State University
Curated by ChEMBL
Montclair State University
Curated by ChEMBL
Affinity DataIC50: 1.50E+3nMAssay Description:Inhibition of Leishmania major CRK3 expressed in Escherichia coli BL21 (DE3) using 5FAM-GGGRSPGRRRRK-OH as substrate after 60 mins by IMAP assayMore data for this Ligand-Target Pair
TargetCell division related protein kinase 2(Leishmania major)
Montclair State University
Curated by ChEMBL
Montclair State University
Curated by ChEMBL
Affinity DataIC50: 5.30E+3nMAssay Description:Inhibition of Leishmania major CRK3 expressed in Escherichia coli BL21 (DE3) using 5FAM-GGGRSPGRRRRK-OH as substrate after 60 mins by IMAP assayMore data for this Ligand-Target Pair
TargetCell division related protein kinase 2(Leishmania major)
Montclair State University
Curated by ChEMBL
Montclair State University
Curated by ChEMBL
Affinity DataIC50: 1.10E+4nMAssay Description:Inhibition of Leishmania major CRK3 expressed in Escherichia coli BL21 (DE3) using 5FAM-GGGRSPGRRRRK-OH as substrate after 60 mins by IMAP assayMore data for this Ligand-Target Pair
Affinity DataIC50: >2.00E+4nMAssay Description:Inhibition of human CDK1More data for this Ligand-Target Pair
Affinity DataIC50: >2.00E+4nMAssay Description:Inhibition of human CDK2More data for this Ligand-Target Pair
Affinity DataIC50: >2.00E+4nMAssay Description:Inhibition of human CDK6More data for this Ligand-Target Pair
Affinity DataIC50: >2.00E+4nMAssay Description:Inhibition of human CDK7More data for this Ligand-Target Pair