Compile Data Set for Download or QSAR
maximum 50k data
Found 8 Enz. Inhib. hit(s) with all data for entry = 50017737
TargetAmyloid-beta precursor protein(Homo sapiens (Human))
Nagasaki University

Curated by ChEMBL
LigandPNGBDBM50185948(5-hydroxy-2-(4-methylaminophenyl)benzofuran | CHEM...)
Affinity DataKi:  0.700nMAssay Description:Displacement of [125I]IMPY from beta amyloid in human corpse AD brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmyloid-beta precursor protein(Homo sapiens (Human))
Nagasaki University

Curated by ChEMBL
LigandPNGBDBM50185947(5-methoxy-2-(4-methylaminophenyl)benzofuran | CHEM...)
Affinity DataKi:  1.30nMAssay Description:Displacement of [125I]IMPY from beta amyloid in human corpse AD brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmyloid-beta precursor protein(Homo sapiens (Human))
Nagasaki University

Curated by ChEMBL
LigandPNGBDBM50185946(5-methoxy-2-(4-aminophenyl)benzofuran | CHEMBL2052...)
Affinity DataKi:  2.30nMAssay Description:Displacement of [125I]IMPY from beta amyloid in human corpse AD brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmyloid-beta precursor protein(Homo sapiens (Human))
Nagasaki University

Curated by ChEMBL
LigandPNGBDBM50185950(5-hydroxy-2-(4-dimethylaminophenyl)benzofuran | CH...)
Affinity DataKi:  2.80nMAssay Description:Displacement of [125I]IMPY from beta amyloid in human corpse AD brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmyloid-beta precursor protein(Homo sapiens (Human))
Nagasaki University

Curated by ChEMBL
LigandPNGBDBM50129793(2-(4''-methylaminophenyl)-6-hydroxybenzothiazole |...)
Affinity DataKi:  4.30nMAssay Description:Binding affinity to beta amyloid in human corpse AD brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmyloid-beta precursor protein(Homo sapiens (Human))
Nagasaki University

Curated by ChEMBL
LigandPNGBDBM50173647((E)-4-(4-(methylamino)styryl)phenol | 4-(4-(methyl...)
Affinity DataKi:  6nMAssay Description:Binding affinity to beta amyloid in human corpse AD brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmyloid-beta precursor protein(Homo sapiens (Human))
Nagasaki University

Curated by ChEMBL
LigandPNGBDBM50185949(5-hydroxy-2-(4-aminophenyl)benzofuran | CHEMBL3804...)
Affinity DataKi:  11.5nMAssay Description:Displacement of [125I]IMPY from beta amyloid in human corpse AD brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmyloid-beta precursor protein(Homo sapiens (Human))
Nagasaki University

Curated by ChEMBL
LigandPNGBDBM50185945(5-methoxy-2-(4-dimethylaminophenyl)benzofuran | CH...)
Affinity DataKi:  12nMAssay Description:Displacement of [125I]IMPY from beta amyloid in human corpse AD brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed