Compile Data Set for Download or QSAR
maximum 50k data
Found 38 Enz. Inhib. hit(s) with all data for entry = 50046498
TargetATP-dependent translocase ABCB1(Homo sapiens (Human))
The First Affiliated Hospital Of Dalian Medical University

Curated by ChEMBL
LigandPNGBDBM50115973(CHEMBL3612151)
Affinity DataKi:  120nMAssay Description:Inhibition of P-glycoprotein in human drug-resistant K562/ADR cells assessed as reduction in P-gp mediated rhodamine 123 efflux by spectrofluorometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-dependent translocase ABCB1(Homo sapiens (Human))
The First Affiliated Hospital Of Dalian Medical University

Curated by ChEMBL
LigandPNGBDBM50115974(CHEMBL3612170)
Affinity DataKi:  120nMAssay Description:Inhibition of P-glycoprotein in human drug-resistant K562/ADR cells assessed as reduction in P-gp mediated rhodamine 123 efflux by spectrofluorometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-dependent translocase ABCB1(Homo sapiens (Human))
The First Affiliated Hospital Of Dalian Medical University

Curated by ChEMBL
LigandPNGBDBM50115978(CHEMBL3612172)
Affinity DataKi:  220nMAssay Description:Inhibition of P-glycoprotein in human drug-resistant K562/ADR cells assessed as reduction in P-gp mediated rhodamine 123 efflux by spectrofluorometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-dependent translocase ABCB1(Homo sapiens (Human))
The First Affiliated Hospital Of Dalian Medical University

Curated by ChEMBL
LigandPNGBDBM50115977(CHEMBL3612153)
Affinity DataKi:  220nMAssay Description:Inhibition of P-glycoprotein in human drug-resistant K562/ADR cells assessed as reduction in P-gp mediated rhodamine 123 efflux by spectrofluorometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-dependent translocase ABCB1(Homo sapiens (Human))
The First Affiliated Hospital Of Dalian Medical University

Curated by ChEMBL
LigandPNGBDBM50115972(CHEMBL3612169)
Affinity DataKi:  320nMAssay Description:Inhibition of P-glycoprotein in human drug-resistant K562/ADR cells assessed as reduction in P-gp mediated rhodamine 123 efflux by spectrofluorometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-dependent translocase ABCB1(Homo sapiens (Human))
The First Affiliated Hospital Of Dalian Medical University

Curated by ChEMBL
LigandPNGBDBM50115971(CHEMBL3612150)
Affinity DataKi:  320nMAssay Description:Inhibition of P-glycoprotein in human drug-resistant K562/ADR cells assessed as reduction in P-gp mediated rhodamine 123 efflux by spectrofluorometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-dependent translocase ABCB1(Homo sapiens (Human))
The First Affiliated Hospital Of Dalian Medical University

Curated by ChEMBL
LigandPNGBDBM50115976(CHEMBL3612171)
Affinity DataKi:  470nMAssay Description:Inhibition of P-glycoprotein in human drug-resistant K562/ADR cells assessed as reduction in P-gp mediated rhodamine 123 efflux by spectrofluorometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-dependent translocase ABCB1(Homo sapiens (Human))
The First Affiliated Hospital Of Dalian Medical University

Curated by ChEMBL
LigandPNGBDBM50115975(CHEMBL3612152)
Affinity DataKi:  470nMAssay Description:Inhibition of P-glycoprotein in human drug-resistant K562/ADR cells assessed as reduction in P-gp mediated rhodamine 123 efflux by spectrofluorometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-dependent translocase ABCB1(Homo sapiens (Human))
The First Affiliated Hospital Of Dalian Medical University

Curated by ChEMBL
LigandPNGBDBM50116014(CHEMBL3612160)
Affinity DataKi:  480nMAssay Description:Inhibition of P-glycoprotein in human drug-resistant K562/ADR cells assessed as reduction in P-gp mediated rhodamine 123 efflux by spectrofluorometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-dependent translocase ABCB1(Homo sapiens (Human))
The First Affiliated Hospital Of Dalian Medical University

Curated by ChEMBL
LigandPNGBDBM50116013(CHEMBL3612141)
Affinity DataKi:  480nMAssay Description:Inhibition of P-glycoprotein in human drug-resistant K562/ADR cells assessed as reduction in P-gp mediated rhodamine 123 efflux by spectrofluorometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-dependent translocase ABCB1(Homo sapiens (Human))
The First Affiliated Hospital Of Dalian Medical University

Curated by ChEMBL
LigandPNGBDBM50115962(CHEMBL3612149)
Affinity DataKi:  730nMAssay Description:Inhibition of P-glycoprotein in human drug-resistant K562/ADR cells assessed as reduction in P-gp mediated rhodamine 123 efflux by spectrofluorometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-dependent translocase ABCB1(Homo sapiens (Human))
The First Affiliated Hospital Of Dalian Medical University

Curated by ChEMBL
LigandPNGBDBM50115968(CHEMBL3612168)
Affinity DataKi:  730nMAssay Description:Inhibition of P-glycoprotein in human drug-resistant K562/ADR cells assessed as reduction in P-gp mediated rhodamine 123 efflux by spectrofluorometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-dependent translocase ABCB1(Homo sapiens (Human))
The First Affiliated Hospital Of Dalian Medical University

Curated by ChEMBL
LigandPNGBDBM50116015(CHEMBL3612142)
Affinity DataKi:  940nMAssay Description:Inhibition of P-glycoprotein in human drug-resistant K562/ADR cells assessed as reduction in P-gp mediated rhodamine 123 efflux by spectrofluorometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-dependent translocase ABCB1(Homo sapiens (Human))
The First Affiliated Hospital Of Dalian Medical University

Curated by ChEMBL
LigandPNGBDBM50116016(CHEMBL3612161)
Affinity DataKi:  940nMAssay Description:Inhibition of P-glycoprotein in human drug-resistant K562/ADR cells assessed as reduction in P-gp mediated rhodamine 123 efflux by spectrofluorometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-dependent translocase ABCB1(Homo sapiens (Human))
The First Affiliated Hospital Of Dalian Medical University

Curated by ChEMBL
LigandPNGBDBM50115960(CHEMBL3612148)
Affinity DataKi:  1.01E+3nMAssay Description:Inhibition of P-glycoprotein in human drug-resistant K562/ADR cells assessed as reduction in P-gp mediated rhodamine 123 efflux by spectrofluorometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-dependent translocase ABCB1(Homo sapiens (Human))
The First Affiliated Hospital Of Dalian Medical University

Curated by ChEMBL
LigandPNGBDBM50115961(CHEMBL3612167)
Affinity DataKi:  1.01E+3nMAssay Description:Inhibition of P-glycoprotein in human drug-resistant K562/ADR cells assessed as reduction in P-gp mediated rhodamine 123 efflux by spectrofluorometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-dependent translocase ABCB1(Homo sapiens (Human))
The First Affiliated Hospital Of Dalian Medical University

Curated by ChEMBL
LigandPNGBDBM50115979(CHEMBL3612154)
Affinity DataKi:  1.34E+3nMAssay Description:Inhibition of P-glycoprotein in human drug-resistant K562/ADR cells assessed as reduction in P-gp mediated rhodamine 123 efflux by spectrofluorometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-dependent translocase ABCB1(Homo sapiens (Human))
The First Affiliated Hospital Of Dalian Medical University

Curated by ChEMBL
LigandPNGBDBM50115980(CHEMBL3612173)
Affinity DataKi:  1.34E+3nMAssay Description:Inhibition of P-glycoprotein in human drug-resistant K562/ADR cells assessed as reduction in P-gp mediated rhodamine 123 efflux by spectrofluorometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-dependent translocase ABCB1(Homo sapiens (Human))
The First Affiliated Hospital Of Dalian Medical University

Curated by ChEMBL
LigandPNGBDBM50115958(CHEMBL3612158)
Affinity DataKi:  1.71E+3nMAssay Description:Inhibition of P-glycoprotein in human drug-resistant K562/ADR cells assessed as reduction in P-gp mediated rhodamine 123 efflux by spectrofluorometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-dependent translocase ABCB1(Homo sapiens (Human))
The First Affiliated Hospital Of Dalian Medical University

Curated by ChEMBL
LigandPNGBDBM50115829(CHEMBL3612139)
Affinity DataKi:  1.71E+3nMAssay Description:Inhibition of P-glycoprotein in human drug-resistant K562/ADR cells assessed as reduction in P-gp mediated rhodamine 123 efflux by spectrofluorometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-dependent translocase ABCB1(Homo sapiens (Human))
The First Affiliated Hospital Of Dalian Medical University

Curated by ChEMBL
LigandPNGBDBM50116021(CHEMBL3612145)
Affinity DataKi:  1.78E+3nMAssay Description:Inhibition of P-glycoprotein in human drug-resistant K562/ADR cells assessed as reduction in P-gp mediated rhodamine 123 efflux by spectrofluorometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-dependent translocase ABCB1(Homo sapiens (Human))
The First Affiliated Hospital Of Dalian Medical University

Curated by ChEMBL
LigandPNGBDBM50116022(CHEMBL3612164)
Affinity DataKi:  1.78E+3nMAssay Description:Inhibition of P-glycoprotein in human drug-resistant K562/ADR cells assessed as reduction in P-gp mediated rhodamine 123 efflux by spectrofluorometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-dependent translocase ABCB1(Homo sapiens (Human))
The First Affiliated Hospital Of Dalian Medical University

Curated by ChEMBL
LigandPNGBDBM50116069(CHEMBL3612147)
Affinity DataKi: >2.23E+3nMAssay Description:Inhibition of P-glycoprotein in human drug-resistant K562/ADR cells assessed as reduction in P-gp mediated rhodamine 123 efflux by spectrofluorometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-dependent translocase ABCB1(Homo sapiens (Human))
The First Affiliated Hospital Of Dalian Medical University

Curated by ChEMBL
LigandPNGBDBM50116060(CHEMBL3612165)
Affinity DataKi: >2.23E+3nMAssay Description:Inhibition of P-glycoprotein in human drug-resistant K562/ADR cells assessed as reduction in P-gp mediated rhodamine 123 efflux by spectrofluorometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-dependent translocase ABCB1(Homo sapiens (Human))
The First Affiliated Hospital Of Dalian Medical University

Curated by ChEMBL
LigandPNGBDBM50116023(CHEMBL3612146)
Affinity DataKi: >2.23E+3nMAssay Description:Inhibition of P-glycoprotein in human drug-resistant K562/ADR cells assessed as reduction in P-gp mediated rhodamine 123 efflux by spectrofluorometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-dependent translocase ABCB1(Homo sapiens (Human))
The First Affiliated Hospital Of Dalian Medical University

Curated by ChEMBL
LigandPNGBDBM50116020(CHEMBL3612163)
Affinity DataKi: >2.23E+3nMAssay Description:Inhibition of P-glycoprotein in human drug-resistant K562/ADR cells assessed as reduction in P-gp mediated rhodamine 123 efflux by spectrofluorometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-dependent translocase ABCB1(Homo sapiens (Human))
The First Affiliated Hospital Of Dalian Medical University

Curated by ChEMBL
LigandPNGBDBM50116019(CHEMBL3612144)
Affinity DataKi: >2.23E+3nMAssay Description:Inhibition of P-glycoprotein in human drug-resistant K562/ADR cells assessed as reduction in P-gp mediated rhodamine 123 efflux by spectrofluorometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-dependent translocase ABCB1(Homo sapiens (Human))
The First Affiliated Hospital Of Dalian Medical University

Curated by ChEMBL
LigandPNGBDBM50116018(CHEMBL3612162)
Affinity DataKi: >2.23E+3nMAssay Description:Inhibition of P-glycoprotein in human drug-resistant K562/ADR cells assessed as reduction in P-gp mediated rhodamine 123 efflux by spectrofluorometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-dependent translocase ABCB1(Homo sapiens (Human))
The First Affiliated Hospital Of Dalian Medical University

Curated by ChEMBL
LigandPNGBDBM50116017(CHEMBL3612143)
Affinity DataKi: >2.23E+3nMAssay Description:Inhibition of P-glycoprotein in human drug-resistant K562/ADR cells assessed as reduction in P-gp mediated rhodamine 123 efflux by spectrofluorometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-dependent translocase ABCB1(Homo sapiens (Human))
The First Affiliated Hospital Of Dalian Medical University

Curated by ChEMBL
LigandPNGBDBM50116011(CHEMBL3612159)
Affinity DataKi: >2.23E+3nMAssay Description:Inhibition of P-glycoprotein in human drug-resistant K562/ADR cells assessed as reduction in P-gp mediated rhodamine 123 efflux by spectrofluorometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-dependent translocase ABCB1(Homo sapiens (Human))
The First Affiliated Hospital Of Dalian Medical University

Curated by ChEMBL
LigandPNGBDBM50115987(CHEMBL3612140)
Affinity DataKi: >2.23E+3nMAssay Description:Inhibition of P-glycoprotein in human drug-resistant K562/ADR cells assessed as reduction in P-gp mediated rhodamine 123 efflux by spectrofluorometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-dependent translocase ABCB1(Homo sapiens (Human))
The First Affiliated Hospital Of Dalian Medical University

Curated by ChEMBL
LigandPNGBDBM50115986(CHEMBL3612236)
Affinity DataKi: >2.23E+3nMAssay Description:Inhibition of P-glycoprotein in human drug-resistant K562/ADR cells assessed as reduction in P-gp mediated rhodamine 123 efflux by spectrofluorometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-dependent translocase ABCB1(Homo sapiens (Human))
The First Affiliated Hospital Of Dalian Medical University

Curated by ChEMBL
LigandPNGBDBM50115985(CHEMBL3612157)
Affinity DataKi: >2.23E+3nMAssay Description:Inhibition of P-glycoprotein in human drug-resistant K562/ADR cells assessed as reduction in P-gp mediated rhodamine 123 efflux by spectrofluorometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-dependent translocase ABCB1(Homo sapiens (Human))
The First Affiliated Hospital Of Dalian Medical University

Curated by ChEMBL
LigandPNGBDBM50115984(CHEMBL3612175)
Affinity DataKi: >2.23E+3nMAssay Description:Inhibition of P-glycoprotein in human drug-resistant K562/ADR cells assessed as reduction in P-gp mediated rhodamine 123 efflux by spectrofluorometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-dependent translocase ABCB1(Homo sapiens (Human))
The First Affiliated Hospital Of Dalian Medical University

Curated by ChEMBL
LigandPNGBDBM50116079(CHEMBL3612166)
Affinity DataKi: >2.23E+3nMAssay Description:Inhibition of P-glycoprotein in human drug-resistant K562/ADR cells assessed as reduction in P-gp mediated rhodamine 123 efflux by spectrofluorometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-dependent translocase ABCB1(Homo sapiens (Human))
The First Affiliated Hospital Of Dalian Medical University

Curated by ChEMBL
LigandPNGBDBM50115982(CHEMBL3612174)
Affinity DataKi: >2.23E+3nMAssay Description:Inhibition of P-glycoprotein in human drug-resistant K562/ADR cells assessed as reduction in P-gp mediated rhodamine 123 efflux by spectrofluorometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-dependent translocase ABCB1(Homo sapiens (Human))
The First Affiliated Hospital Of Dalian Medical University

Curated by ChEMBL
LigandPNGBDBM50115981(CHEMBL3612155)
Affinity DataKi: >2.23E+3nMAssay Description:Inhibition of P-glycoprotein in human drug-resistant K562/ADR cells assessed as reduction in P-gp mediated rhodamine 123 efflux by spectrofluorometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-dependent translocase ABCB1(Homo sapiens (Human))
The First Affiliated Hospital Of Dalian Medical University

Curated by ChEMBL
LigandPNGBDBM50115983(CHEMBL3612156)
Affinity DataKi: >2.23E+3nMAssay Description:Inhibition of P-glycoprotein in human drug-resistant K562/ADR cells assessed as reduction in P-gp mediated rhodamine 123 efflux by spectrofluorometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed