Compile Data Set for Download or QSAR
maximum 50k data
Found 21 Enz. Inhib. hit(s) with all data for entry = 50046669
TargetAldo-keto reductase family 1 member C3(Homo sapiens (Human))
Rwth Aachen University

Curated by ChEMBL
LigandPNGBDBM50124574(CHEMBL3623737)
Affinity DataIC50:  35nMAssay Description:Inhibition of recombinant AKR1C3 (unknown origin) using S-tetralol as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAldo-keto reductase family 1 member C3(Homo sapiens (Human))
Rwth Aachen University

Curated by ChEMBL
LigandPNGBDBM50124577(CHEMBL3623738)
Affinity DataIC50:  36nMAssay Description:Inhibition of recombinant AKR1C3 (unknown origin) using S-tetralol as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAldo-keto reductase family 1 member C3(Homo sapiens (Human))
Rwth Aachen University

Curated by ChEMBL
LigandPNGBDBM50124575(CHEMBL3623735)
Affinity DataIC50:  57nMAssay Description:Inhibition of recombinant AKR1C3 (unknown origin) using S-tetralol as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAldo-keto reductase family 1 member C3(Homo sapiens (Human))
Rwth Aachen University

Curated by ChEMBL
LigandPNGBDBM50124576(CHEMBL3623736)
Affinity DataIC50:  86nMAssay Description:Inhibition of recombinant AKR1C3 (unknown origin) using S-tetralol as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAldo-keto reductase family 1 member C2(Homo sapiens (Human))
Rwth Aachen University

Curated by ChEMBL
LigandPNGBDBM50124577(CHEMBL3623738)
Affinity DataIC50:  150nMAssay Description:Inhibition of recombinant AKR1C2 (unknown origin) using S-tetralol as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAldo-keto reductase family 1 member C2(Homo sapiens (Human))
Rwth Aachen University

Curated by ChEMBL
LigandPNGBDBM50124575(CHEMBL3623735)
Affinity DataIC50:  270nMAssay Description:Inhibition of recombinant AKR1C2 (unknown origin) using S-tetralol as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(Homo sapiens (Human))
Rwth Aachen University

Curated by ChEMBL
LigandPNGBDBM50124575(CHEMBL3623735)
Affinity DataIC50:  1.80E+3nMAssay Description:Inhibition of COX1 (unknown origin) using arachidonic acid substrate by colorimetric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))
Rwth Aachen University

Curated by ChEMBL
LigandPNGBDBM50124575(CHEMBL3623735)
Affinity DataIC50:  1.20E+4nMAssay Description:Inhibition of COX2 (unknown origin) using arachidonic acid substrate by colorimetric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAldo-keto reductase family 1 member C2(Homo sapiens (Human))
Rwth Aachen University

Curated by ChEMBL
LigandPNGBDBM50124576(CHEMBL3623736)
Affinity DataIC50:  1.40E+4nMAssay Description:Inhibition of recombinant AKR1C2 (unknown origin) using S-tetralol as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAldo-keto reductase family 1 member C2(Homo sapiens (Human))
Rwth Aachen University

Curated by ChEMBL
LigandPNGBDBM50124574(CHEMBL3623737)
Affinity DataIC50:  2.00E+4nMAssay Description:Inhibition of recombinant AKR1C2 (unknown origin) using S-tetralol as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(Homo sapiens (Human))
Rwth Aachen University

Curated by ChEMBL
LigandPNGBDBM50124577(CHEMBL3623738)
Affinity DataIC50:  2.20E+4nMAssay Description:Inhibition of COX1 (unknown origin) using arachidonic acid substrate by colorimetric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(Homo sapiens (Human))
Rwth Aachen University

Curated by ChEMBL
LigandPNGBDBM50124574(CHEMBL3623737)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of COX1 (unknown origin) using arachidonic acid substrate by colorimetric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))
Rwth Aachen University

Curated by ChEMBL
LigandPNGBDBM50124574(CHEMBL3623737)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of COX2 (unknown origin) using arachidonic acid substrate by colorimetric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))
Rwth Aachen University

Curated by ChEMBL
LigandPNGBDBM50124577(CHEMBL3623738)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of COX2 (unknown origin) using arachidonic acid substrate by colorimetric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))
Rwth Aachen University

Curated by ChEMBL
LigandPNGBDBM50124576(CHEMBL3623736)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of COX2 (unknown origin) using arachidonic acid substrate by colorimetric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(Homo sapiens (Human))
Rwth Aachen University

Curated by ChEMBL
LigandPNGBDBM50124576(CHEMBL3623736)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of COX1 (unknown origin) using arachidonic acid substrate by colorimetric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcid-sensing ion channel 5(Rattus norvegicus)
Rwth Aachen University

Curated by ChEMBL
LigandPNGBDBM17636(2-{[3-(trifluoromethyl)phenyl]amino}benzoic acid |...)
Affinity DataEC50:  2.60E+6nMAssay Description:Binding affinity to rat bile acid-sensitive ion channel expressed in xenopus oocytesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcid-sensing ion channel 5(Rattus norvegicus)
Rwth Aachen University

Curated by ChEMBL
LigandPNGBDBM50124575(CHEMBL3623735)
Affinity DataEC50:  1.40E+6nMAssay Description:Binding affinity to rat bile acid-sensitive ion channel expressed in xenopus oocytesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcid-sensing ion channel 5(Rattus norvegicus)
Rwth Aachen University

Curated by ChEMBL
LigandPNGBDBM50124576(CHEMBL3623736)
Affinity DataEC50:  2.90E+6nMAssay Description:Binding affinity to rat bile acid-sensitive ion channel expressed in xenopus oocytesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcid-sensing ion channel 5(Rattus norvegicus)
Rwth Aachen University

Curated by ChEMBL
LigandPNGBDBM50124574(CHEMBL3623737)
Affinity DataEC50:  2.80E+6nMAssay Description:Binding affinity to rat bile acid-sensitive ion channel expressed in xenopus oocytesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcid-sensing ion channel 5(Rattus norvegicus)
Rwth Aachen University

Curated by ChEMBL
LigandPNGBDBM50124577(CHEMBL3623738)
Affinity DataEC50:  2.60E+6nMAssay Description:Binding affinity to rat bile acid-sensitive ion channel expressed in xenopus oocytesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed