Affinity DataIC50: 60nMAssay Description:Binding affinity against Endothelin B receptor in rat cerebellar membrane (ET-B) from adult blue laurie ratMore data for this Ligand-Target Pair
Affinity DataIC50: 240nMAssay Description:Binding affinity against Endothelin B receptor in rat cerebellar membrane (ET-B) from adult blue laurie ratMore data for this Ligand-Target Pair
Affinity DataIC50: 350nMAssay Description:Binding affinity against endothelin receptor in rat cerebellar membrane (ET-B) from adult blue laurie ratMore data for this Ligand-Target Pair
Affinity DataIC50: 1.10E+3nMAssay Description:Binding affinity against Endothelin B receptor in rat cerebellar membrane (ET-B) from adult blue laurie ratMore data for this Ligand-Target Pair
Affinity DataIC50: 1.20E+3nMAssay Description:In vitro binding affinity against Endothelin A receptor by using endothelin (ET-1) as radioligand in rat heart ventricleMore data for this Ligand-Target Pair
Affinity DataIC50: 1.40E+3nMAssay Description:Binding affinity against Endothelin B receptor in rat cerebellar membrane (ET-B) from adult blue laurie ratMore data for this Ligand-Target Pair
Affinity DataIC50: 1.60E+3nMAssay Description:In vitro binding affinity against Endothelin A receptor by using endothelin (ET-1) as radioligand in rat heart ventricleMore data for this Ligand-Target Pair
Affinity DataIC50: 1.70E+3nMAssay Description:Binding affinity against Endothelin B receptor in rat cerebellar membrane (ET-B) from adult blue laurie ratMore data for this Ligand-Target Pair
Affinity DataIC50: 1.70E+3nMAssay Description:Binding affinity against Endothelin B receptor in rat cerebellar membrane (ET-B) from adult blue laurie ratMore data for this Ligand-Target Pair
Affinity DataIC50: 1.80E+3nMAssay Description:In vitro binding affinity against Endothelin A receptor by using endothelin (ET-1) as radioligand in rat heart ventricleMore data for this Ligand-Target Pair
Affinity DataIC50: 1.80E+3nMAssay Description:In vitro binding affinity against Endothelin A receptor by using endothelin (ET-1) as radioligand in rat heart ventricleMore data for this Ligand-Target Pair
Affinity DataIC50: 1.80E+3nMAssay Description:Binding affinity against Endothelin A receptor in rabbit renal artery vascular smooth muscle membrane (ET-A)More data for this Ligand-Target Pair
Affinity DataIC50: 2.00E+3nMAssay Description:Binding affinity against Endothelin A receptor in rabbit renal artery vascular smooth muscle membrane (ET-A)More data for this Ligand-Target Pair
Affinity DataIC50: 2.50E+3nMAssay Description:Binding affinity against Endothelin A receptor in rabbit renal artery vascular smooth muscle membrane (ET-A)More data for this Ligand-Target Pair
Affinity DataIC50: 2.50E+3nMAssay Description:In vitro binding affinity against Endothelin A receptor by using endothelin (ET-1) as radioligand in rat heart ventricleMore data for this Ligand-Target Pair
Affinity DataIC50: 2.50E+3nMAssay Description:Binding affinity against Endothelin A receptor in rabbit renal artery vascular smooth muscle membrane (ET-A)More data for this Ligand-Target Pair
Affinity DataIC50: 2.60E+3nMAssay Description:Binding affinity against Endothelin A receptor in rabbit renal artery vascular smooth muscle membrane (ET-A)More data for this Ligand-Target Pair
Affinity DataIC50: 2.80E+3nMAssay Description:In vitro binding affinity against Endothelin A receptor by using endothelin (ET-1) as radioligand in rat heart ventricleMore data for this Ligand-Target Pair
Affinity DataIC50: 3.50E+3nMAssay Description:In vitro binding affinity against Endothelin A receptor by using endothelin (ET-1) as radioligand in rat heart ventricleMore data for this Ligand-Target Pair
Affinity DataIC50: 3.80E+3nMAssay Description:Binding affinity against Endothelin A receptor in rabbit renal artery vascular smooth muscle membrane (ET-A)More data for this Ligand-Target Pair
Affinity DataIC50: 6.50E+3nMAssay Description:In vitro binding affinity against Endothelin A receptor by using endothelin (ET-1) as radioligand in rat heart ventricleMore data for this Ligand-Target Pair
Affinity DataIC50: 7.10E+3nMAssay Description:Binding affinity against Endothelin A receptor in rabbit renal artery vascular smooth muscle membrane (ET-A)More data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+4nMAssay Description:Binding affinity against Endothelin A receptor in rabbit renal artery vascular smooth muscle membrane (ET-A)More data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+4nMAssay Description:Binding affinity against endothelin receptor in rat cerebellar membrane (ET-B) from adult blue laurie ratMore data for this Ligand-Target Pair
Affinity DataIC50: 4.90E+4nMAssay Description:In vitro binding affinity against Endothelin A receptor by using endothelin (ET-1) as radioligand in rat heart ventricleMore data for this Ligand-Target Pair