Compile Data Set for Download or QSAR
maximum 50k data
Found 25 Enz. Inhib. hit(s) with all data for entry = 50029385
TargetEndothelin receptor type B(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM50284007(CHEMBL412460 | Trp-Ile-Ile-Asp-Leu-Hisc(Cys-Ser-Se...)
Affinity DataIC50:  60nMAssay Description:Binding affinity against Endothelin B receptor in rat cerebellar membrane (ET-B) from adult blue laurie ratMore data for this Ligand-Target Pair
In DepthDetails Article
TargetEndothelin receptor type B(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM50284006(CHEMBL438380 | Trp-Ile-Ile-Asp-Leu-Hisc(Cys-Ser-Ao...)
Affinity DataIC50:  240nMAssay Description:Binding affinity against Endothelin B receptor in rat cerebellar membrane (ET-B) from adult blue laurie ratMore data for this Ligand-Target Pair
In DepthDetails Article
TargetEndothelin receptor type B(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM50284008(CHEMBL265164 | Trp-Ile-Ile-Asp-Leu-Hisc(Cys-Ser-Ap...)
Affinity DataIC50:  350nMAssay Description:Binding affinity against endothelin receptor in rat cerebellar membrane (ET-B) from adult blue laurie ratMore data for this Ligand-Target Pair
In DepthDetails Article
TargetEndothelin receptor type B(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM50284011(CHEMBL438768 | Trp-Ile-Ile-Asp-Leu-Hisc(Cys-Ser-As...)
Affinity DataIC50:  1.10E+3nMAssay Description:Binding affinity against Endothelin B receptor in rat cerebellar membrane (ET-B) from adult blue laurie ratMore data for this Ligand-Target Pair
In DepthDetails Article
TargetEndothelin-1 receptor(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM50284007(CHEMBL412460 | Trp-Ile-Ile-Asp-Leu-Hisc(Cys-Ser-Se...)
Affinity DataIC50:  1.20E+3nMAssay Description:In vitro binding affinity against Endothelin A receptor by using endothelin (ET-1) as radioligand in rat heart ventricleMore data for this Ligand-Target Pair
In DepthDetails Article
TargetEndothelin receptor type B(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM50284010(CHEMBL436899 | Trp-Ile-Ile-Asp-Leu-Hisc(Cys-Ser-Se...)
Affinity DataIC50:  1.40E+3nMAssay Description:Binding affinity against Endothelin B receptor in rat cerebellar membrane (ET-B) from adult blue laurie ratMore data for this Ligand-Target Pair
In DepthDetails Article
TargetEndothelin-1 receptor(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM50284006(CHEMBL438380 | Trp-Ile-Ile-Asp-Leu-Hisc(Cys-Ser-Ao...)
Affinity DataIC50:  1.60E+3nMAssay Description:In vitro binding affinity against Endothelin A receptor by using endothelin (ET-1) as radioligand in rat heart ventricleMore data for this Ligand-Target Pair
In DepthDetails Article
TargetEndothelin receptor type B(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM50284014(CHEMBL436884 | Trp-Ile-Ile-Asp-Leu-Hisc(Cys-Val-Ty...)
Affinity DataIC50:  1.70E+3nMAssay Description:Binding affinity against Endothelin B receptor in rat cerebellar membrane (ET-B) from adult blue laurie ratMore data for this Ligand-Target Pair
In DepthDetails Article
TargetEndothelin receptor type B(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM50284009(CHEMBL408141 | Trp-Ile-Ile-Asp-Leu-Hisc(Cys-Ser-Va...)
Affinity DataIC50:  1.70E+3nMAssay Description:Binding affinity against Endothelin B receptor in rat cerebellar membrane (ET-B) from adult blue laurie ratMore data for this Ligand-Target Pair
In DepthDetails Article
TargetEndothelin-1 receptor(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM50284008(CHEMBL265164 | Trp-Ile-Ile-Asp-Leu-Hisc(Cys-Ser-Ap...)
Affinity DataIC50:  1.80E+3nMAssay Description:In vitro binding affinity against Endothelin A receptor by using endothelin (ET-1) as radioligand in rat heart ventricleMore data for this Ligand-Target Pair
In DepthDetails Article
TargetEndothelin-1 receptor(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM50284010(CHEMBL436899 | Trp-Ile-Ile-Asp-Leu-Hisc(Cys-Ser-Se...)
Affinity DataIC50:  1.80E+3nMAssay Description:In vitro binding affinity against Endothelin A receptor by using endothelin (ET-1) as radioligand in rat heart ventricleMore data for this Ligand-Target Pair
In DepthDetails Article
TargetEndothelin-1 receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50284006(CHEMBL438380 | Trp-Ile-Ile-Asp-Leu-Hisc(Cys-Ser-Ao...)
Affinity DataIC50:  1.80E+3nMAssay Description:Binding affinity against Endothelin A receptor in rabbit renal artery vascular smooth muscle membrane (ET-A)More data for this Ligand-Target Pair
In DepthDetails Article
TargetEndothelin-1 receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50284010(CHEMBL436899 | Trp-Ile-Ile-Asp-Leu-Hisc(Cys-Ser-Se...)
Affinity DataIC50:  2.00E+3nMAssay Description:Binding affinity against Endothelin A receptor in rabbit renal artery vascular smooth muscle membrane (ET-A)More data for this Ligand-Target Pair
In DepthDetails Article
TargetEndothelin-1 receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50284007(CHEMBL412460 | Trp-Ile-Ile-Asp-Leu-Hisc(Cys-Ser-Se...)
Affinity DataIC50:  2.50E+3nMAssay Description:Binding affinity against Endothelin A receptor in rabbit renal artery vascular smooth muscle membrane (ET-A)More data for this Ligand-Target Pair
In DepthDetails Article
TargetEndothelin-1 receptor(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM50284012(CHEMBL414448 | Trp-Ile-Ile-Asp-Leu-Hisc(Cys-Ser-Ah...)
Affinity DataIC50:  2.50E+3nMAssay Description:In vitro binding affinity against Endothelin A receptor by using endothelin (ET-1) as radioligand in rat heart ventricleMore data for this Ligand-Target Pair
In DepthDetails Article
TargetEndothelin-1 receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50284008(CHEMBL265164 | Trp-Ile-Ile-Asp-Leu-Hisc(Cys-Ser-Ap...)
Affinity DataIC50:  2.50E+3nMAssay Description:Binding affinity against Endothelin A receptor in rabbit renal artery vascular smooth muscle membrane (ET-A)More data for this Ligand-Target Pair
In DepthDetails Article
TargetEndothelin-1 receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50284014(CHEMBL436884 | Trp-Ile-Ile-Asp-Leu-Hisc(Cys-Val-Ty...)
Affinity DataIC50:  2.60E+3nMAssay Description:Binding affinity against Endothelin A receptor in rabbit renal artery vascular smooth muscle membrane (ET-A)More data for this Ligand-Target Pair
In DepthDetails Article
TargetEndothelin-1 receptor(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM50284009(CHEMBL408141 | Trp-Ile-Ile-Asp-Leu-Hisc(Cys-Ser-Va...)
Affinity DataIC50:  2.80E+3nMAssay Description:In vitro binding affinity against Endothelin A receptor by using endothelin (ET-1) as radioligand in rat heart ventricleMore data for this Ligand-Target Pair
In DepthDetails Article
TargetEndothelin-1 receptor(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM50284011(CHEMBL438768 | Trp-Ile-Ile-Asp-Leu-Hisc(Cys-Ser-As...)
Affinity DataIC50:  3.50E+3nMAssay Description:In vitro binding affinity against Endothelin A receptor by using endothelin (ET-1) as radioligand in rat heart ventricleMore data for this Ligand-Target Pair
In DepthDetails Article
TargetEndothelin-1 receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50284009(CHEMBL408141 | Trp-Ile-Ile-Asp-Leu-Hisc(Cys-Ser-Va...)
Affinity DataIC50:  3.80E+3nMAssay Description:Binding affinity against Endothelin A receptor in rabbit renal artery vascular smooth muscle membrane (ET-A)More data for this Ligand-Target Pair
In DepthDetails Article
TargetEndothelin-1 receptor(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM50284014(CHEMBL436884 | Trp-Ile-Ile-Asp-Leu-Hisc(Cys-Val-Ty...)
Affinity DataIC50:  6.50E+3nMAssay Description:In vitro binding affinity against Endothelin A receptor by using endothelin (ET-1) as radioligand in rat heart ventricleMore data for this Ligand-Target Pair
In DepthDetails Article
TargetEndothelin-1 receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50284011(CHEMBL438768 | Trp-Ile-Ile-Asp-Leu-Hisc(Cys-Ser-As...)
Affinity DataIC50:  7.10E+3nMAssay Description:Binding affinity against Endothelin A receptor in rabbit renal artery vascular smooth muscle membrane (ET-A)More data for this Ligand-Target Pair
In DepthDetails Article
TargetEndothelin-1 receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50284013(CHEMBL409777 | Trp-Ile-Ile-Asp-Leu-Hisc(Cys-Ser-Se...)
Affinity DataIC50: >1.00E+4nMAssay Description:Binding affinity against Endothelin A receptor in rabbit renal artery vascular smooth muscle membrane (ET-A)More data for this Ligand-Target Pair
In DepthDetails Article
TargetEndothelin receptor type B(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM50284013(CHEMBL409777 | Trp-Ile-Ile-Asp-Leu-Hisc(Cys-Ser-Se...)
Affinity DataIC50: >1.00E+4nMAssay Description:Binding affinity against endothelin receptor in rat cerebellar membrane (ET-B) from adult blue laurie ratMore data for this Ligand-Target Pair
In DepthDetails Article
TargetEndothelin-1 receptor(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM50284013(CHEMBL409777 | Trp-Ile-Ile-Asp-Leu-Hisc(Cys-Ser-Se...)
Affinity DataIC50:  4.90E+4nMAssay Description:In vitro binding affinity against Endothelin A receptor by using endothelin (ET-1) as radioligand in rat heart ventricleMore data for this Ligand-Target Pair
In DepthDetails Article