Compile Data Set for Download or QSAR
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Found 21 Enz. Inhib. hit(s) with all data for entry = 50047841
TargetNischarin(RAT)
University Of Camerino

Curated by ChEMBL
LigandPNGBDBM50000214(CHEMBL337862)
Affinity DataKi:  1.40nMAssay Description:Displacement of [125I]-p-iodoclonidine from I1 receptor imidazoline binding site in Sprague-Dawley rat kidney cell membranes after 30 mins by liquid ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNischarin(RAT)
University Of Camerino

Curated by ChEMBL
LigandPNGBDBM50193034(CHEMBL3904276)
Affinity DataKi:  2nMAssay Description:Displacement of [125I]-p-iodoclonidine from I1 receptor imidazoline binding site in Sprague-Dawley rat kidney cell membranes after 30 mins by liquid ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNischarin(RAT)
University Of Camerino

Curated by ChEMBL
LigandPNGBDBM50193035(CHEMBL3961335)
Affinity DataKi:  4nMAssay Description:Displacement of [125I]-p-iodoclonidine from I1 receptor imidazoline binding site in Sprague-Dawley rat kidney cell membranes after 30 mins by liquid ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNischarin(RAT)
University Of Camerino

Curated by ChEMBL
LigandPNGBDBM50027031((2-Chloro-phenyl)-(4,5-dihydro-1H-imidazol-2-ylmet...)
Affinity DataKi:  7.60nMAssay Description:Displacement of [125I]-p-iodoclonidine from I1 receptor imidazoline binding site in Sprague-Dawley rat kidney cell membranes after 30 mins by liquid ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNischarin(RAT)
University Of Camerino

Curated by ChEMBL
LigandPNGBDBM50193036(CHEMBL3892351)
Affinity DataKi:  8.30nMAssay Description:Displacement of [125I]-p-iodoclonidine from I1 receptor imidazoline binding site in Sprague-Dawley rat kidney cell membranes after 30 mins by liquid ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNischarin(RAT)
University Of Camerino

Curated by ChEMBL
LigandPNGBDBM50193039(CHEMBL1439667)
Affinity DataKi:  18nMAssay Description:Displacement of [125I]-p-iodoclonidine from I1 receptor imidazoline binding site in Sprague-Dawley rat kidney cell membranes after 30 mins by liquid ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNischarin(RAT)
University Of Camerino

Curated by ChEMBL
LigandPNGBDBM50138500(2-((E)-Styryl)-4,5-dihydro-1H-imidazole | 2-styryl...)
Affinity DataKi:  19nMAssay Description:Displacement of [125I]-p-iodoclonidine from I1 receptor imidazoline binding site in rat PC12 cell membranes after 30 mins by gamma counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNischarin(RAT)
University Of Camerino

Curated by ChEMBL
LigandPNGBDBM50193037(CHEMBL3920069)
Affinity DataKi:  24nMAssay Description:Displacement of [125I]-p-iodoclonidine from I1 receptor imidazoline binding site in Sprague-Dawley rat kidney cell membranes after 30 mins by liquid ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNischarin(RAT)
University Of Camerino

Curated by ChEMBL
LigandPNGBDBM50193041(CHEMBL3939078)
Affinity DataKi:  69nMAssay Description:Displacement of [125I]-p-iodoclonidine from I1 receptor imidazoline binding site in Sprague-Dawley rat kidney cell membranes after 30 mins by liquid ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNischarin(RAT)
University Of Camerino

Curated by ChEMBL
LigandPNGBDBM50193038(CHEMBL3911124)
Affinity DataKi:  98nMAssay Description:Displacement of [125I]-p-iodoclonidine from I1 receptor imidazoline binding site in Sprague-Dawley rat kidney cell membranes after 30 mins by liquid ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-2C adrenergic receptor(Homo sapiens (Human))
University Of Camerino

Curated by ChEMBL
LigandPNGBDBM50193034(CHEMBL3904276)
Affinity DataEC50:  22nMAssay Description:Agonist activity at human alpha2c-AR expressed in CHO cells assessed as rate of acidification after 240 mins by cytosensor microphysiometric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-2C adrenergic receptor(Homo sapiens (Human))
University Of Camerino

Curated by ChEMBL
LigandPNGBDBM50193036(CHEMBL3892351)
Affinity DataEC50:  115nMAssay Description:Agonist activity at human alpha2c-AR expressed in CHO cells assessed as rate of acidification after 240 mins by cytosensor microphysiometric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))
University Of Camerino

Curated by ChEMBL
LigandPNGBDBM50000214(CHEMBL337862)
Affinity DataEC50:  63nMAssay Description:Agonist activity at human alpha2a-AR expressed in CHO cells assessed as rate of acidification after 240 mins by cytosensor microphysiometric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-2C adrenergic receptor(Homo sapiens (Human))
University Of Camerino

Curated by ChEMBL
LigandPNGBDBM50027031((2-Chloro-phenyl)-(4,5-dihydro-1H-imidazol-2-ylmet...)
Affinity DataEC50:  224nMAssay Description:Agonist activity at human alpha2c-AR expressed in CHO cells assessed as rate of acidification after 240 mins by cytosensor microphysiometric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-2B adrenergic receptor(Homo sapiens (Human))
University Of Camerino

Curated by ChEMBL
LigandPNGBDBM50027031((2-Chloro-phenyl)-(4,5-dihydro-1H-imidazol-2-ylmet...)
Affinity DataEC50:  776nMAssay Description:Agonist activity at human alpha2b-AR expressed in CHO cells assessed as rate of acidification after 240 mins by cytosensor microphysiometric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-2B adrenergic receptor(Homo sapiens (Human))
University Of Camerino

Curated by ChEMBL
LigandPNGBDBM50193034(CHEMBL3904276)
Affinity DataEC50:  3.16E+3nMAssay Description:Agonist activity at human alpha2b-AR expressed in CHO cells assessed as rate of acidification after 240 mins by cytosensor microphysiometric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-2C adrenergic receptor(Homo sapiens (Human))
University Of Camerino

Curated by ChEMBL
LigandPNGBDBM50000214(CHEMBL337862)
Affinity DataEC50:  148nMAssay Description:Agonist activity at human alpha2c-AR expressed in CHO cells assessed as rate of acidification after 240 mins by cytosensor microphysiometric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-2C adrenergic receptor(Homo sapiens (Human))
University Of Camerino

Curated by ChEMBL
LigandPNGBDBM50193035(CHEMBL3961335)
Affinity DataEC50:  158nMAssay Description:Agonist activity at human alpha2c-AR expressed in CHO cells assessed as rate of acidification after 240 mins by cytosensor microphysiometric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-2B adrenergic receptor(Homo sapiens (Human))
University Of Camerino

Curated by ChEMBL
LigandPNGBDBM50193035(CHEMBL3961335)
Affinity DataEC50:  2.51E+3nMAssay Description:Agonist activity at human alpha2b-AR expressed in CHO cells assessed as rate of acidification after 240 mins by cytosensor microphysiometric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-2B adrenergic receptor(Homo sapiens (Human))
University Of Camerino

Curated by ChEMBL
LigandPNGBDBM50193036(CHEMBL3892351)
Affinity DataEC50:  4.57E+3nMAssay Description:Agonist activity at human alpha2b-AR expressed in CHO cells assessed as rate of acidification after 240 mins by cytosensor microphysiometric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-2B adrenergic receptor(Homo sapiens (Human))
University Of Camerino

Curated by ChEMBL
LigandPNGBDBM50000214(CHEMBL337862)
Affinity DataEC50:  955nMAssay Description:Agonist activity at human alpha2b-AR expressed in CHO cells assessed as rate of acidification after 240 mins by cytosensor microphysiometric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed