Compile Data Set for Download or QSAR
maximum 50k data
Found 26 Enz. Inhib. hit(s) with all data for entry = 50031254
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50309925(3-oxo-2-(4-(piperidin-4-yl)phenyl)isoindoline-4-ca...)
Affinity DataKi:  32nMAssay Description:Inhibition of PARP1 by microplate scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50309916(3-oxo-2-(piperidin-4-yl)isoindoline-4-carboxamide ...)
Affinity DataKi:  33nMAssay Description:Inhibition of PARP1 by microplate scintillation countingMore data for this Ligand-Target Pair
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50309927(2-(4-(4-methylpiperazin-1-yl)phenyl)-3-oxoisoindol...)
Affinity DataKi:  48nMAssay Description:Inhibition of PARP1 by microplate scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50309923(3-oxo-2-(4-(pyrrolidin-1-ylmethyl)phenyl)isoindoli...)
Affinity DataKi:  53nMAssay Description:Inhibition of PARP1 by microplate scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50309915(3-oxo-2-(pyrrolidin-3-yl)isoindoline-4-carboxamide...)
Affinity DataKi:  59nMAssay Description:Inhibition of PARP1 by microplate scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50309922(2-(4-(dimethylamino)phenyl)-3-oxoisoindoline-4-car...)
Affinity DataKi:  70nMAssay Description:Inhibition of PARP1 by microplate scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50309913(2-isobutyl-3-oxoisoindoline-4-carboxamide | CHEMBL...)
Affinity DataKi:  112nMAssay Description:Inhibition of PARP1 by microplate scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50309912(2-methyl-3-oxoisoindoline-4-carboxamide | CHEMBL61...)
Affinity DataKi:  123nMAssay Description:Inhibition of PARP1 by microplate scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50309917(3-oxo-2-(piperidin-3-yl)isoindoline-4-carboxamide ...)
Affinity DataKi:  140nMAssay Description:Inhibition of PARP1 by microplate scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50309920(3-oxo-2-(piperidin-3-ylmethyl)isoindoline-4-carbox...)
Affinity DataKi:  164nMAssay Description:Inhibition of PARP1 by microplate scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50309914(2-cyclohexyl-3-oxoisoindoline-4-carboxamide | CHEM...)
Affinity DataKi:  172nMAssay Description:Inhibition of PARP1 by microplate scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50309921(3-oxo-2-m-tolylisoindoline-4-carboxamide | CHEMBL5...)
Affinity DataKi:  261nMAssay Description:Inhibition of PARP1 by microplate scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50309926(3-oxo-2-(3-(piperidin-4-yl)phenyl)isoindoline-4-ca...)
Affinity DataKi:  314nMAssay Description:Inhibition of PARP1 by microplate scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50309918(3-oxo-2-(pyrrolidin-2-ylmethyl)isoindoline-4-carbo...)
Affinity DataKi:  377nMAssay Description:Inhibition of PARP1 by microplate scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50309919(3-oxo-2-(piperidin-4-ylmethyl)isoindoline-4-carbox...)
Affinity DataKi:  384nMAssay Description:Inhibition of PARP1 by microplate scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50309924(3-oxo-2-(3-(pyrrolidin-1-ylmethyl)phenyl)isoindoli...)
Affinity DataKi:  391nMAssay Description:Inhibition of PARP1 by microplate scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50309928(3-oxo-2-(pyridin-3-ylmethyl)isoindoline-4-carboxam...)
Affinity DataKi: >9.50E+3nMAssay Description:Inhibition of PARP1 by microplate scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50309916(3-oxo-2-(piperidin-4-yl)isoindoline-4-carboxamide ...)
Affinity DataEC50:  51nMAssay Description:Inhibition of PARP1 in human C41 cellsMore data for this Ligand-Target Pair
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50309923(3-oxo-2-(4-(pyrrolidin-1-ylmethyl)phenyl)isoindoli...)
Affinity DataEC50:  53nMAssay Description:Inhibition of PARP1 in human C41 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50309925(3-oxo-2-(4-(piperidin-4-yl)phenyl)isoindoline-4-ca...)
Affinity DataEC50:  120nMAssay Description:Inhibition of PARP1 in human C41 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50309914(2-cyclohexyl-3-oxoisoindoline-4-carboxamide | CHEM...)
Affinity DataEC50: >1.00E+3nMAssay Description:Inhibition of PARP1 in human C41 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50309913(2-isobutyl-3-oxoisoindoline-4-carboxamide | CHEMBL...)
Affinity DataEC50: >1.00E+3nMAssay Description:Inhibition of PARP1 in human C41 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50309927(2-(4-(4-methylpiperazin-1-yl)phenyl)-3-oxoisoindol...)
Affinity DataEC50:  22nMAssay Description:Inhibition of PARP1 in human C41 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50309922(2-(4-(dimethylamino)phenyl)-3-oxoisoindoline-4-car...)
Affinity DataEC50:  372nMAssay Description:Inhibition of PARP1 in human C41 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50309918(3-oxo-2-(pyrrolidin-2-ylmethyl)isoindoline-4-carbo...)
Affinity DataEC50:  374nMAssay Description:Inhibition of PARP1 in human C41 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50309915(3-oxo-2-(pyrrolidin-3-yl)isoindoline-4-carboxamide...)
Affinity DataEC50:  160nMAssay Description:Inhibition of PARP1 in human C41 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed