Compile Data Set for Download or QSAR
maximum 50k data
Found 30 Enz. Inhib. hit(s) with all data for entry = 50031275
TargetPlasminogen activator inhibitor 1(Homo sapiens (Human))
Eastern Michigan University

Curated by ChEMBL
LigandPNGBDBM50310309(CHEMBL596879 | N-(3,4-dihydroxyphenylsulfonyl)-N-h...)
Affinity DataIC50:  284nMAssay Description:Inhibition of human recombinant PAI1 assessed as rate of AMC release after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasminogen activator inhibitor 1(Homo sapiens (Human))
Eastern Michigan University

Curated by ChEMBL
LigandPNGBDBM50310311(CHEMBL601265 | N-cyclohexyl-N-(3,4-dihydroxyphenyl...)
Affinity DataIC50:  594nMAssay Description:Inhibition of human recombinant PAI1 assessed as rate of AMC release after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasminogen activator inhibitor 1(Homo sapiens (Human))
Eastern Michigan University

Curated by ChEMBL
LigandPNGBDBM50310308(CHEMBL597478 | N-(3,4-dihydroxyphenylsulfonyl)-3,4...)
Affinity DataIC50:  2.67E+3nMAssay Description:Inhibition of human recombinant PAI1 assessed as rate of AMC release after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasminogen activator inhibitor 1(Homo sapiens (Human))
Eastern Michigan University

Curated by ChEMBL
LigandPNGBDBM50310310(CHEMBL596880 | N-benzyl-N-(3,4-dihydroxyphenylsulf...)
Affinity DataIC50:  4.82E+3nMAssay Description:Inhibition of human recombinant PAI1 assessed as rate of AMC release after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasminogen activator inhibitor 1(Homo sapiens (Human))
Eastern Michigan University

Curated by ChEMBL
LigandPNGBDBM50310301(CHEMBL599742 | N,N'-(ethane-1,2-diyl)bis(N-ethyl-3...)
Affinity DataIC50:  9.32E+3nMAssay Description:Inhibition of human recombinant PAI1 assessed as rate of AMC release after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasminogen activator inhibitor 1(Homo sapiens (Human))
Eastern Michigan University

Curated by ChEMBL
LigandPNGBDBM50310307(CHEMBL596861 | N,N'-(ethane-1,2-diyl)bis(N-ethyl-3...)
Affinity DataIC50:  1.28E+5nMAssay Description:Inhibition of human recombinant PAI1 assessed as rate of AMC release after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasminogen activator inhibitor 1(Homo sapiens (Human))
Eastern Michigan University

Curated by ChEMBL
LigandPNGBDBM50310306(CHEMBL611972 | N,N'-(ethane-1,2-diyl)bis(N-ethylbe...)
Affinity DataIC50: >3.00E+5nMAssay Description:Inhibition of human recombinant PAI1 assessed as rate of AMC release after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasminogen activator inhibitor 1(Homo sapiens (Human))
Eastern Michigan University

Curated by ChEMBL
LigandPNGBDBM50310305(CHEMBL596859 | N,N'-(ethane-1,2-diyl)bis(N-ethyl-4...)
Affinity DataIC50: >3.00E+5nMAssay Description:Inhibition of human recombinant PAI1 assessed as rate of AMC release after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasminogen activator inhibitor 1(Homo sapiens (Human))
Eastern Michigan University

Curated by ChEMBL
LigandPNGBDBM50310313(CHEMBL596860 | N,N'-(ethane-1,2-diyl)bis(N-ethyl-2...)
Affinity DataIC50: >3.00E+5nMAssay Description:Inhibition of human recombinant PAI1 assessed as rate of AMC release after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAntithrombin-III(Homo sapiens (Human))
Eastern Michigan University

Curated by ChEMBL
LigandPNGBDBM50310309(CHEMBL596879 | N-(3,4-dihydroxyphenylsulfonyl)-N-h...)
Affinity DataIC50: >3.00E+5nMAssay Description:Inhibition of antithrombin-3 assessed as residual alpha-thrombin activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAntithrombin-III(Homo sapiens (Human))
Eastern Michigan University

Curated by ChEMBL
LigandPNGBDBM50310306(CHEMBL611972 | N,N'-(ethane-1,2-diyl)bis(N-ethylbe...)
Affinity DataIC50: >3.00E+5nMAssay Description:Inhibition of antithrombin-3 assessed as residual alpha-thrombin activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAntithrombin-III(Homo sapiens (Human))
Eastern Michigan University

Curated by ChEMBL
LigandPNGBDBM50310310(CHEMBL596880 | N-benzyl-N-(3,4-dihydroxyphenylsulf...)
Affinity DataIC50: >3.00E+5nMAssay Description:Inhibition of antithrombin-3 assessed as residual alpha-thrombin activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAntithrombin-III(Homo sapiens (Human))
Eastern Michigan University

Curated by ChEMBL
LigandPNGBDBM50310313(CHEMBL596860 | N,N'-(ethane-1,2-diyl)bis(N-ethyl-2...)
Affinity DataIC50: >3.00E+5nMAssay Description:Inhibition of antithrombin-3 assessed as residual alpha-thrombin activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAntithrombin-III(Homo sapiens (Human))
Eastern Michigan University

Curated by ChEMBL
LigandPNGBDBM50310299(CHEMBL599342 | N,N'-(ethane-1,2-diyl)bis(N-ethyl-3...)
Affinity DataIC50: >3.00E+5nMAssay Description:Inhibition of antithrombin-3 assessed as residual alpha-thrombin activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasminogen activator inhibitor 1(Homo sapiens (Human))
Eastern Michigan University

Curated by ChEMBL
LigandPNGBDBM50310312(CHEMBL597509 | N,N'-bis(3,4-dihydroxybenzenesulfon...)
Affinity DataIC50: >3.00E+5nMAssay Description:Inhibition of human recombinant PAI1 assessed as rate of AMC release after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAntithrombin-III(Homo sapiens (Human))
Eastern Michigan University

Curated by ChEMBL
LigandPNGBDBM50310311(CHEMBL601265 | N-cyclohexyl-N-(3,4-dihydroxyphenyl...)
Affinity DataIC50: >3.00E+5nMAssay Description:Inhibition of antithrombin-3 assessed as residual alpha-thrombin activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAntithrombin-III(Homo sapiens (Human))
Eastern Michigan University

Curated by ChEMBL
LigandPNGBDBM50310312(CHEMBL597509 | N,N'-bis(3,4-dihydroxybenzenesulfon...)
Affinity DataIC50: >3.00E+5nMAssay Description:Inhibition of antithrombin-3 assessed as residual alpha-thrombin activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasminogen activator inhibitor 1(Homo sapiens (Human))
Eastern Michigan University

Curated by ChEMBL
LigandPNGBDBM50310299(CHEMBL599342 | N,N'-(ethane-1,2-diyl)bis(N-ethyl-3...)
Affinity DataIC50: >3.00E+5nMAssay Description:Inhibition of human recombinant PAI1 assessed as rate of AMC release after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAntithrombin-III(Homo sapiens (Human))
Eastern Michigan University

Curated by ChEMBL
LigandPNGBDBM50310305(CHEMBL596859 | N,N'-(ethane-1,2-diyl)bis(N-ethyl-4...)
Affinity DataIC50: >3.00E+5nMAssay Description:Inhibition of antithrombin-3 assessed as residual alpha-thrombin activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasminogen activator inhibitor 1(Homo sapiens (Human))
Eastern Michigan University

Curated by ChEMBL
LigandPNGBDBM50310304(CHEMBL597510 | N,N'-(ethane-1,2-diyl)bis(N-ethyl-3...)
Affinity DataIC50:  3.43E+5nMAssay Description:Inhibition of human recombinant PAI1 assessed as rate of AMC release after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasminogen activator inhibitor 1(Homo sapiens (Human))
Eastern Michigan University

Curated by ChEMBL
LigandPNGBDBM50310300(CHEMBL606451 | N,N'-(ethane-1,2-diyl)bis(3,4-dihyd...)
Affinity DataIC50:  5.18E+5nMAssay Description:Inhibition of human recombinant PAI1 assessed as rate of AMC release after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAntithrombin-III(Homo sapiens (Human))
Eastern Michigan University

Curated by ChEMBL
LigandPNGBDBM50310308(CHEMBL597478 | N-(3,4-dihydroxyphenylsulfonyl)-3,4...)
Affinity DataIC50: >1.00E+6nMAssay Description:Inhibition of antithrombin-3 assessed as residual alpha-thrombin activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAntithrombin-III(Homo sapiens (Human))
Eastern Michigan University

Curated by ChEMBL
LigandPNGBDBM50310304(CHEMBL597510 | N,N'-(ethane-1,2-diyl)bis(N-ethyl-3...)
Affinity DataIC50: >1.00E+6nMAssay Description:Inhibition of antithrombin-3 assessed as residual alpha-thrombin activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAntithrombin-III(Homo sapiens (Human))
Eastern Michigan University

Curated by ChEMBL
LigandPNGBDBM50310301(CHEMBL599742 | N,N'-(ethane-1,2-diyl)bis(N-ethyl-3...)
Affinity DataIC50: >1.00E+6nMAssay Description:Inhibition of antithrombin-3 assessed as residual alpha-thrombin activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasminogen activator inhibitor 1(Homo sapiens (Human))
Eastern Michigan University

Curated by ChEMBL
LigandPNGBDBM50310303(CHEMBL599769 | N,N'-(hexane-1,6-diyl)bis(3,4-dihyd...)
Affinity DataIC50:  1.38E+6nMAssay Description:Inhibition of human recombinant PAI1 assessed as rate of AMC release after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAntithrombin-III(Homo sapiens (Human))
Eastern Michigan University

Curated by ChEMBL
LigandPNGBDBM50310303(CHEMBL599769 | N,N'-(hexane-1,6-diyl)bis(3,4-dihyd...)
Affinity DataIC50: >3.00E+6nMAssay Description:Inhibition of antithrombin-3 assessed as residual alpha-thrombin activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAntithrombin-III(Homo sapiens (Human))
Eastern Michigan University

Curated by ChEMBL
LigandPNGBDBM50310302(CHEMBL611992 | N,N'-(butane-1,4-diyl)bis(3,4-dihyd...)
Affinity DataIC50: >3.00E+6nMAssay Description:Inhibition of antithrombin-3 assessed as residual alpha-thrombin activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAntithrombin-III(Homo sapiens (Human))
Eastern Michigan University

Curated by ChEMBL
LigandPNGBDBM50310300(CHEMBL606451 | N,N'-(ethane-1,2-diyl)bis(3,4-dihyd...)
Affinity DataIC50: >3.00E+6nMAssay Description:Inhibition of antithrombin-3 assessed as residual alpha-thrombin activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasminogen activator inhibitor 1(Homo sapiens (Human))
Eastern Michigan University

Curated by ChEMBL
LigandPNGBDBM50310302(CHEMBL611992 | N,N'-(butane-1,4-diyl)bis(3,4-dihyd...)
Affinity DataIC50: >3.00E+6nMAssay Description:Inhibition of human recombinant PAI1 assessed as rate of AMC release after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAntithrombin-III(Homo sapiens (Human))
Eastern Michigan University

Curated by ChEMBL
LigandPNGBDBM50310307(CHEMBL596861 | N,N'-(ethane-1,2-diyl)bis(N-ethyl-3...)
Affinity DataIC50: >3.00E+6nMAssay Description:Inhibition of antithrombin-3 assessed as residual alpha-thrombin activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed