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Found 60 Enz. Inhib. hit(s) with all data for entry = 50048350
TargetAlpha-2B adrenergic receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50212995(CHEMBL75030)
Affinity DataKi:  2.10nMAssay Description:Binding affinity towards human Alpha-2B adrenergic receptor by the displacement of [3H]rauwolscineMore data for this Ligand-Target Pair
In DepthDetails
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50212995(CHEMBL75030)
Affinity DataKi:  2.30nMAssay Description:Binding affinity towards human Alpha-2A adrenergic receptor by the displacement of [3H]rauwolscineMore data for this Ligand-Target Pair
In DepthDetails
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50212997(CHEMBL310335)
Affinity DataKi:  3nMAssay Description:Binding affinity towards human Alpha-2A adrenergic receptor by the displacement of [3H]rauwolscineMore data for this Ligand-Target Pair
In DepthDetails
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50212993(CHEMBL305928)
Affinity DataKi:  5.40nMAssay Description:Binding affinity towards human Alpha-2A adrenergic receptor by the displacement of [3H]rauwolscineMore data for this Ligand-Target Pair
In DepthDetails
TargetAlpha-2B adrenergic receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50212997(CHEMBL310335)
Affinity DataKi:  5.90nMAssay Description:Binding affinity towards human Alpha-2B adrenergic receptor by the displacement of [3H]rauwolscineMore data for this Ligand-Target Pair
In DepthDetails
TargetAlpha-2B adrenergic receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50016897(2-(2,6-dichloroanilino)-1,3-diazacyclopentene-(2) ...)
Affinity DataKi:  6.20nMAssay Description:Binding affinity towards human Alpha-2B adrenergic receptor by the displacement of [3H]rauwolscineMore data for this Ligand-Target Pair
In DepthDetails
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50016897(2-(2,6-dichloroanilino)-1,3-diazacyclopentene-(2) ...)
Affinity DataKi:  7.90nMAssay Description:Binding affinity towards human Alpha-2A adrenergic receptor by the displacement of [3H]rauwolscineMore data for this Ligand-Target Pair
In DepthDetails
TargetAlpha-2B adrenergic receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50212993(CHEMBL305928)
Affinity DataKi:  9.80nMAssay Description:Binding affinity towards human Alpha-2B adrenergic receptor by the displacement of [3H]rauwolscineMore data for this Ligand-Target Pair
In DepthDetails
TargetAlpha-2C adrenergic receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50212995(CHEMBL75030)
Affinity DataKi:  12nMAssay Description:Binding affinity towards human Alpha-2C adrenergic receptor by the displacement of [3H]rauwolscineMore data for this Ligand-Target Pair
In DepthDetails
TargetAlpha-2C adrenergic receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50212997(CHEMBL310335)
Affinity DataKi:  25nMAssay Description:Binding affinity towards human Alpha-2C adrenergic receptor by the displacement of [3H]rauwolscineMore data for this Ligand-Target Pair
In DepthDetails
TargetAlpha-2B adrenergic receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50212996(CHEMBL306377)
Affinity DataKi:  25nMAssay Description:Binding affinity towards human Alpha-2B adrenergic receptor by the displacement of [3H]rauwolscineMore data for this Ligand-Target Pair
In DepthDetails
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50212996(CHEMBL306377)
Affinity DataKi:  26nMAssay Description:Binding affinity towards human Alpha-2A adrenergic receptor by the displacement of [3H]rauwolscineMore data for this Ligand-Target Pair
In DepthDetails
TargetAlpha-2C adrenergic receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50212993(CHEMBL305928)
Affinity DataKi:  33nMAssay Description:Binding affinity towards human Alpha-2C adrenergic receptor by the displacement of [3H]rauwolscineMore data for this Ligand-Target Pair
In DepthDetails
TargetAlpha-2C adrenergic receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50016897(2-(2,6-dichloroanilino)-1,3-diazacyclopentene-(2) ...)
Affinity DataKi:  56nMAssay Description:Binding affinity towards human Alpha-2C adrenergic receptor by the displacement of [3H]rauwolscineMore data for this Ligand-Target Pair
In DepthDetails
TargetAlpha-2B adrenergic receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50070328(CHEBI:8862 | Rilmenidine)
Affinity DataKi:  71nMAssay Description:Binding affinity towards human Alpha-2B adrenergic receptor by the displacement of [3H]rauwolscineMore data for this Ligand-Target Pair
In DepthDetails
TargetAlpha-2C adrenergic receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50212996(CHEMBL306377)
Affinity DataKi:  85nMAssay Description:Binding affinity towards human Alpha-2C adrenergic receptor by the displacement of [3H]rauwolscineMore data for this Ligand-Target Pair
In DepthDetails
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50212995(CHEMBL75030)
Affinity DataKi:  126nMAssay Description:Binding affinity towards human Alpha-1C adrenergic receptor by the displacement of [3H]prazosinMore data for this Ligand-Target Pair
In DepthDetails
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50212997(CHEMBL310335)
Affinity DataKi:  141nMAssay Description:Binding affinity towards human Alpha-1C adrenergic receptor by the displacement of [3H]prazosinMore data for this Ligand-Target Pair
In DepthDetails
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50070328(CHEBI:8862 | Rilmenidine)
Affinity DataKi:  182nMAssay Description:Binding affinity towards human Alpha-2A adrenergic receptor by the displacement of [3H]rauwolscineMore data for this Ligand-Target Pair
In DepthDetails
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50212995(CHEMBL75030)
Affinity DataKi:  204nMAssay Description:Binding affinity towards human Alpha-1A adrenergic receptor by the displacement of [3H]prazosinMore data for this Ligand-Target Pair
In DepthDetails
TargetAlpha-2C adrenergic receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50070328(CHEBI:8862 | Rilmenidine)
Affinity DataKi:  288nMAssay Description:Binding affinity towards human Alpha-2C adrenergic receptor by the displacement of [3H]rauwolscineMore data for this Ligand-Target Pair
In DepthDetails
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50016897(2-(2,6-dichloroanilino)-1,3-diazacyclopentene-(2) ...)
Affinity DataKi:  513nMAssay Description:Binding affinity towards human Alpha-1A adrenergic receptor by the displacement of [3H]prazosinMore data for this Ligand-Target Pair
In DepthDetails
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50212997(CHEMBL310335)
Affinity DataKi:  562nMAssay Description:Binding affinity towards human Alpha-1A adrenergic receptor by the displacement of [3H]prazosinMore data for this Ligand-Target Pair
In DepthDetails
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50016897(2-(2,6-dichloroanilino)-1,3-diazacyclopentene-(2) ...)
Affinity DataKi:  977nMAssay Description:Binding affinity towards human Alpha-1C adrenergic receptor by the displacement of [3H]prazosinMore data for this Ligand-Target Pair
In DepthDetails
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50212996(CHEMBL306377)
Affinity DataKi:  1.95E+3nMAssay Description:Binding affinity towards human Alpha-1C adrenergic receptor by the displacement of [3H]prazosinMore data for this Ligand-Target Pair
In DepthDetails
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50212993(CHEMBL305928)
Affinity DataKi:  2.00E+3nMAssay Description:Binding affinity towards human Alpha-1C adrenergic receptor by the displacement of [3H]prazosinMore data for this Ligand-Target Pair
In DepthDetails
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50212996(CHEMBL306377)
Affinity DataKi:  2.19E+3nMAssay Description:Binding affinity towards human Alpha-1A adrenergic receptor by the displacement of [3H]prazosinMore data for this Ligand-Target Pair
In DepthDetails
TargetAlpha-1B adrenergic receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50016897(2-(2,6-dichloroanilino)-1,3-diazacyclopentene-(2) ...)
Affinity DataKi:  2.40E+3nMAssay Description:Binding affinity towards human Alpha-1B adrenergic receptor by the displacement of [3H]prazosinMore data for this Ligand-Target Pair
In DepthDetails
TargetAlpha-1B adrenergic receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50212995(CHEMBL75030)
Affinity DataKi:  2.45E+3nMAssay Description:Binding affinity towards human Alpha-1B adrenergic receptor by the displacement of [3H]prazosinMore data for this Ligand-Target Pair
In DepthDetails
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50212993(CHEMBL305928)
Affinity DataKi:  3.80E+3nMAssay Description:Binding affinity towards human Alpha-1A adrenergic receptor by the displacement of [3H]prazosinMore data for this Ligand-Target Pair
In DepthDetails
TargetAlpha-1B adrenergic receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50212997(CHEMBL310335)
Affinity DataKi:  3.98E+3nMAssay Description:Binding affinity towards human Alpha-1B adrenergic receptor by the displacement of [3H]prazosinMore data for this Ligand-Target Pair
In DepthDetails
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50070328(CHEBI:8862 | Rilmenidine)
Affinity DataKi:  6.03E+3nMAssay Description:Binding affinity towards human Alpha-1C adrenergic receptor by the displacement of [3H]prazosinMore data for this Ligand-Target Pair
In DepthDetails
TargetAlpha-1B adrenergic receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50212996(CHEMBL306377)
Affinity DataKi:  6.76E+3nMAssay Description:Binding affinity towards human Alpha-1B adrenergic receptor by the displacement of [3H]prazosinMore data for this Ligand-Target Pair
In DepthDetails
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50070328(CHEBI:8862 | Rilmenidine)
Affinity DataKi:  8.91E+3nMAssay Description:Binding affinity towards human Alpha-1A adrenergic receptor by the displacement of [3H]prazosinMore data for this Ligand-Target Pair
In DepthDetails
TargetAlpha-2B adrenergic receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50212994(CHEMBL75201)
Affinity DataKi:  1.17E+4nMAssay Description:Binding affinity towards human Alpha-2B adrenergic receptor by the displacement of [3H]rauwolscineMore data for this Ligand-Target Pair
In DepthDetails
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50212994(CHEMBL75201)
Affinity DataKi:  1.66E+4nMAssay Description:Binding affinity towards human Alpha-2A adrenergic receptor by the displacement of [3H]rauwolscineMore data for this Ligand-Target Pair
In DepthDetails
TargetAlpha-2C adrenergic receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50212994(CHEMBL75201)
Affinity DataKi:  1.66E+4nMAssay Description:Binding affinity towards human Alpha-2C adrenergic receptor by the displacement of [3H]rauwolscineMore data for this Ligand-Target Pair
In DepthDetails
TargetAlpha-1B adrenergic receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50070328(CHEBI:8862 | Rilmenidine)
Affinity DataKi:  2.14E+4nMAssay Description:Binding affinity towards human Alpha-1B adrenergic receptor by the displacement of [3H]prazosinMore data for this Ligand-Target Pair
In DepthDetails
TargetAlpha-1B adrenergic receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50212993(CHEMBL305928)
Affinity DataKi:  2.82E+4nMAssay Description:Binding affinity towards human Alpha-1B adrenergic receptor by the displacement of [3H]prazosinMore data for this Ligand-Target Pair
In DepthDetails
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50212994(CHEMBL75201)
Affinity DataKi:  1.07E+5nMAssay Description:Binding affinity towards human Alpha-1C adrenergic receptor by the displacement of [3H]prazosinMore data for this Ligand-Target Pair
In DepthDetails
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50212994(CHEMBL75201)
Affinity DataKi:  1.20E+5nMAssay Description:Binding affinity towards human Alpha-1A adrenergic receptor by the displacement of [3H]prazosinMore data for this Ligand-Target Pair
In DepthDetails
TargetAlpha-1B adrenergic receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50212994(CHEMBL75201)
Affinity DataKi:  1.00E+6nMAssay Description:Binding affinity towards human Alpha-1B adrenergic receptor by the displacement of [3H]prazosinMore data for this Ligand-Target Pair
In DepthDetails
TargetAlpha-2C adrenergic receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50016897(2-(2,6-dichloroanilino)-1,3-diazacyclopentene-(2) ...)
Affinity DataEC50:  55nMAssay Description:Agonistic activity towards human Alpha-2C adrenergic receptor was measured as ability to inhibit forskolin-stimulated synthesis of cyclic adenosine m...More data for this Ligand-Target Pair
In DepthDetails
TargetAlpha-2B adrenergic receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50016897(2-(2,6-dichloroanilino)-1,3-diazacyclopentene-(2) ...)
Affinity DataEC50:  166nMAssay Description:Agonistic activity towards human Alpha-2B adrenergic receptor was measured as ability to inhibit forskolin-stimulated synthesis of cyclic adenosine m...More data for this Ligand-Target Pair
In DepthDetails
TargetAlpha-2C adrenergic receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50212995(CHEMBL75030)
Affinity DataEC50:  2.20nMAssay Description:Agonistic activity towards human Alpha-2C adrenergic receptor was measured as ability to inhibit forskolin-stimulated synthesis of cyclic adenosine m...More data for this Ligand-Target Pair
In DepthDetails
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50212996(CHEMBL306377)
Affinity DataEC50:  229nMAssay Description:Agonistic activity towards human Alpha-2A adrenergic receptor was measured as ability to inhibit forskolin-stimulated synthesis of cyclic adenosine m...More data for this Ligand-Target Pair
In DepthDetails
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50212997(CHEMBL310335)
Affinity DataEC50:  1.60nMAssay Description:Agonistic activity towards human Alpha-2A adrenergic receptor was measured as ability to inhibit forskolin-stimulated synthesis of cyclic adenosine m...More data for this Ligand-Target Pair
In DepthDetails
TargetAlpha-2B adrenergic receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50212993(CHEMBL305928)
Affinity DataEC50:  214nMAssay Description:Agonistic activity towards human Alpha-2B adrenergic receptor was measured as ability to inhibit forskolin-stimulated synthesis of cyclic adenosine m...More data for this Ligand-Target Pair
In DepthDetails
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50070328(CHEBI:8862 | Rilmenidine)
Affinity DataEC50:  275nMAssay Description:Agonistic activity towards human Alpha-2A adrenergic receptor was measured as ability to inhibit forskolin-stimulated synthesis of cyclic adenosine m...More data for this Ligand-Target Pair
In DepthDetails
TargetAlpha-2B adrenergic receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50212995(CHEMBL75030)
Affinity DataEC50:  3.5nMAssay Description:Agonistic activity towards human Alpha-2B adrenergic receptor was measured as ability to inhibit forskolin-stimulated synthesis of cyclic adenosine m...More data for this Ligand-Target Pair
In DepthDetails
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