Affinity DataIC50: 89nMAssay Description:Concentration required for 50% inhibition of binding against human Alpha-1D adrenergic receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 214nMAssay Description:Concentration required for 50% inhibition of binding against Alpha-1A adrenergic receptor in humanMore data for this Ligand-Target Pair
Affinity DataIC50: 224nMAssay Description:Concentration required for 50% inhibition of binding against Alpha-1A adrenergic receptor in humanMore data for this Ligand-Target Pair
Affinity DataIC50: 468nMAssay Description:Concentration required for 50% inhibition of binding against Alpha-1A adrenergic receptor in humanMore data for this Ligand-Target Pair
Affinity DataIC50: 692nMAssay Description:Concentration required for 50% inhibition of binding against human Alpha-1B adrenergic receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 851nMAssay Description:Concentration required for 50% inhibition of binding against Alpha-1A adrenergic receptor in humanMore data for this Ligand-Target Pair
Affinity DataIC50: 1.05E+3nMAssay Description:Concentration required for 50% inhibition of binding against Alpha-1A adrenergic receptor in humanMore data for this Ligand-Target Pair
Affinity DataIC50: 1.48E+3nMAssay Description:Concentration required for 50% inhibition of binding against human Alpha-1D adrenergic receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 1.70E+3nMAssay Description:Concentration required for 50% inhibition of binding against human Alpha-1D adrenergic receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 1.78E+3nMAssay Description:Concentration required for 50% inhibition of binding against human Alpha-1B adrenergic receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 1.95E+3nMAssay Description:Concentration required for 50% inhibition of binding against human Alpha-1B adrenergic receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 2.00E+3nMAssay Description:Concentration required for 50% inhibition of binding against human Alpha-1D adrenergic receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 2.04E+3nMAssay Description:Concentration required for 50% inhibition of binding against Alpha-1A adrenergic receptor in humanMore data for this Ligand-Target Pair
Affinity DataIC50: 2.24E+3nMAssay Description:Concentration required for 50% inhibition of binding against human Alpha-1B adrenergic receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 5.89E+3nMAssay Description:Concentration required for 50% inhibition of binding against human Alpha-1B adrenergic receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 6.61E+3nMAssay Description:Concentration required for 50% inhibition of binding against human Alpha-1D adrenergic receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 6.76E+3nMAssay Description:Concentration required for 50% inhibition of binding against human Alpha-1D adrenergic receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 1.05E+4nMAssay Description:Concentration required for 50% inhibition of binding against human Alpha-1B adrenergic receptorMore data for this Ligand-Target Pair
Affinity DataEC50: 79nMAssay Description:Potency against cloned human alpha 1B adrenoceptor expressed in rat-1 fibroblasts.More data for this Ligand-Target Pair
Affinity DataEC50: 40nMAssay Description:Agonist potency against cloned human alpha 1A adrenoceptor expressed in rat-1 fibroblasts.More data for this Ligand-Target Pair
Affinity DataEC50: 200nMAssay Description:Potency against cloned human alpha 1B adrenoceptor expressed in rat-1 fibroblasts.More data for this Ligand-Target Pair
Affinity DataEC50: <5.01E+3nMAssay Description:Agonist potency against cloned human alpha 1A adrenoceptor expressed in rat-1 fibroblasts.More data for this Ligand-Target Pair
Affinity DataEC50: 63nMAssay Description:Potency against cloned human alpha 1B adrenoceptor expressed in rat-1 fibroblasts.More data for this Ligand-Target Pair
Affinity DataEC50: <5.01E+3nMAssay Description:Potency against cloned human alpha 1D-adrenoceptor expressed in rat-1 fibroblasts.More data for this Ligand-Target Pair
Affinity DataEC50: 501nMAssay Description:Agonist potency against cloned human alpha 1A adrenoceptor expressed in rat-1 fibroblasts.More data for this Ligand-Target Pair
Affinity DataEC50: <5.01E+3nMAssay Description:Potency against cloned human alpha 1B adrenoceptor expressed in rat-1 fibroblasts.More data for this Ligand-Target Pair
Affinity DataEC50: 13nMAssay Description:Agonist potency against cloned human alpha 1A adrenoceptor expressed in rat-1 fibroblasts.More data for this Ligand-Target Pair
Affinity DataEC50: <5.01E+3nMAssay Description:Potency against cloned human alpha 1B adrenoceptor expressed in rat-1 fibroblasts.More data for this Ligand-Target Pair
Affinity DataEC50: <5.01E+3nMAssay Description:Potency against cloned human alpha 1B adrenoceptor expressed in rat-1 fibroblasts.More data for this Ligand-Target Pair
Affinity DataEC50: 2.5nMAssay Description:Agonist potency against cloned human alpha 1A adrenoceptor expressed in rat-1 fibroblasts.More data for this Ligand-Target Pair
Affinity DataEC50: 63nMAssay Description:Potency against cloned human alpha 1D-adrenoceptor expressed in rat-1 fibroblasts.More data for this Ligand-Target Pair
Affinity DataEC50: 0.794nMAssay Description:Agonist potency against cloned human alpha 1A adrenoceptor expressed in rat-1 fibroblasts.More data for this Ligand-Target Pair
Affinity DataEC50: 251nMAssay Description:Potency against cloned human alpha 1B adrenoceptor expressed in rat-1 fibroblasts.More data for this Ligand-Target Pair
Affinity DataEC50: 13nMAssay Description:Agonist potency against cloned human alpha 1A adrenoceptor expressed in rat-1 fibroblasts.More data for this Ligand-Target Pair
Affinity DataEC50: <5.01E+3nMAssay Description:Potency against cloned human alpha 1B adrenoceptor expressed in rat-1 fibroblasts.More data for this Ligand-Target Pair
Affinity DataEC50: 10nMAssay Description:Agonist potency against cloned human alpha 1A adrenoceptor expressed in rat-1 fibroblasts.More data for this Ligand-Target Pair
Affinity DataEC50: 3.20nMAssay Description:Agonist potency against cloned human alpha 1A adrenoceptor expressed in rat-1 fibroblasts.More data for this Ligand-Target Pair
Affinity DataEC50: <5.01E+3nMAssay Description:Potency against cloned human alpha 1D-adrenoceptor expressed in rat-1 fibroblasts.More data for this Ligand-Target Pair
Affinity DataEC50: <5.01E+3nMAssay Description:Potency against cloned human alpha 1B adrenoceptor expressed in rat-1 fibroblasts.More data for this Ligand-Target Pair
Affinity DataEC50: 63nMAssay Description:Agonist potency against cloned human alpha 1A adrenoceptor expressed in rat-1 fibroblasts.More data for this Ligand-Target Pair
Affinity DataEC50: <5.01E+3nMAssay Description:Potency against cloned human alpha 1B adrenoceptor expressed in rat-1 fibroblasts.More data for this Ligand-Target Pair
Affinity DataEC50: 32nMAssay Description:Agonist potency against cloned human alpha 1A adrenoceptor expressed in rat-1 fibroblasts.More data for this Ligand-Target Pair
Affinity DataEC50: 631nMAssay Description:Potency against cloned human alpha 1D-adrenoceptor expressed in rat-1 fibroblasts.More data for this Ligand-Target Pair
Affinity DataEC50: 200nMAssay Description:Potency against cloned human alpha 1D-adrenoceptor expressed in rat-1 fibroblasts.More data for this Ligand-Target Pair
Affinity DataEC50: <5.01E+3nMAssay Description:Potency against cloned human alpha 1D-adrenoceptor expressed in rat-1 fibroblasts.More data for this Ligand-Target Pair
Affinity DataEC50: <5.01E+3nMAssay Description:Potency against cloned human alpha 1D-adrenoceptor expressed in rat-1 fibroblasts.More data for this Ligand-Target Pair
Affinity DataEC50: <5.01E+3nMAssay Description:Potency against cloned human alpha 1D-adrenoceptor expressed in rat-1 fibroblasts.More data for this Ligand-Target Pair
Affinity DataEC50: <5.01E+3nMAssay Description:Potency against cloned human alpha 1D-adrenoceptor expressed in rat-1 fibroblasts.More data for this Ligand-Target Pair
Affinity DataEC50: 50nMAssay Description:Agonist potency against cloned human alpha 1A adrenoceptor expressed in rat-1 fibroblasts.More data for this Ligand-Target Pair
Affinity DataEC50: 20nMAssay Description:Agonist potency against cloned human alpha 1A adrenoceptor expressed in rat-1 fibroblasts.More data for this Ligand-Target Pair