Found 95 Enz. Inhib. hit(s) with all data for entry = 50042175 
Affinity DataIC50: 19nMAssay Description:In vitro binding affinity against cloned human alpha-1D-adrenoreceptor receptors expressed in rat-1 fibroblastsMore data for this Ligand-Target Pair
Affinity DataIC50: 58nMAssay Description:In vitro binding affinity against cloned human alpha-1D-adrenoreceptor receptors expressed in rat-1 fibroblastsMore data for this Ligand-Target Pair
Affinity DataIC50: 66nMAssay Description:In vitro binding affinity against cloned human alpha-1A-adrenoreceptor receptors expressed in rat-1 fibroblastsMore data for this Ligand-Target Pair
Affinity DataIC50: 78nMAssay Description:In vitro binding affinity against cloned human alpha-1A-adrenoreceptor receptors expressed in rat-1 fibroblastsMore data for this Ligand-Target Pair
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
Glaxosmithkline
Curated by ChEMBL
Glaxosmithkline
Curated by ChEMBL
Affinity DataIC50: 102nMAssay Description:Inhibition of binding of [3H]-prazosin at alpha1 adrenoceptors isolated from rat brainMore data for this Ligand-Target Pair
Affinity DataIC50: 107nMAssay Description:In vitro binding affinity against cloned human alpha-1A-adrenoreceptor receptors expressed in rat-1 fibroblastsMore data for this Ligand-Target Pair
Affinity DataIC50: 170nMAssay Description:In vitro binding affinity against cloned human alpha-1A-adrenoreceptor receptors expressed in rat-1 fibroblastsMore data for this Ligand-Target Pair
Affinity DataIC50: 219nMAssay Description:In vitro binding affinity against cloned human alpha-1B-adrenoreceptor receptors expressed in rat-1 fibroblastsMore data for this Ligand-Target Pair
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
Glaxosmithkline
Curated by ChEMBL
Glaxosmithkline
Curated by ChEMBL
Affinity DataIC50: 263nMAssay Description:Inhibition of binding of [3H]-prazosin at alpha1 adrenoceptors isolated from rat brainMore data for this Ligand-Target Pair
Affinity DataIC50: 282nMAssay Description:In vitro binding affinity against cloned human alpha-1A-adrenoreceptor receptors expressed in rat-1 fibroblastsMore data for this Ligand-Target Pair
Affinity DataIC50: 302nMAssay Description:In vitro binding affinity against cloned human alpha-1A-adrenoreceptor receptors expressed in rat-1 fibroblastsMore data for this Ligand-Target Pair
Affinity DataIC50: 513nMAssay Description:In vitro binding affinity against cloned human alpha-1D-adrenoreceptor receptors expressed in rat-1 fibroblastsMore data for this Ligand-Target Pair
Affinity DataIC50: 550nMAssay Description:In vitro binding affinity against cloned human alpha-1D-adrenoreceptor receptors expressed in rat-1 fibroblastsMore data for this Ligand-Target Pair
Affinity DataIC50: 871nMAssay Description:In vitro binding affinity against cloned human alpha-1D-adrenoreceptor receptors expressed in rat-1 fibroblastsMore data for this Ligand-Target Pair
Affinity DataIC50: 891nMAssay Description:In vitro binding affinity against cloned human alpha-1B-adrenoreceptor receptors expressed in rat-1 fibroblastsMore data for this Ligand-Target Pair
Affinity DataIC50: 933nMAssay Description:In vitro binding affinity against cloned human alpha-1D-adrenoreceptor receptors expressed in rat-1 fibroblastsMore data for this Ligand-Target Pair
Affinity DataIC50: 1.70E+3nMAssay Description:In vitro binding affinity against cloned human alpha-1B-adrenoreceptor receptors expressed in rat-1 fibroblastsMore data for this Ligand-Target Pair
Affinity DataIC50: 2.40E+3nMAssay Description:In vitro binding affinity against cloned human alpha-1B-adrenoreceptor receptors expressed in rat-1 fibroblastsMore data for this Ligand-Target Pair
Affinity DataIC50: 3.02E+3nMAssay Description:In vitro binding affinity against cloned human alpha-1B-adrenoreceptor receptors expressed in rat-1 fibroblastsMore data for this Ligand-Target Pair
Affinity DataIC50: 5.89E+3nMAssay Description:In vitro binding affinity against cloned human alpha-1B-adrenoreceptor receptors expressed in rat-1 fibroblastsMore data for this Ligand-Target Pair
Affinity DataIC50: <3.02E+4nMAssay Description:In vitro binding affinity against cloned human alpha-1D-adrenoceptor receptors expressed in rat-1 fibroblastsMore data for this Ligand-Target Pair
Affinity DataIC50: <3.02E+4nMAssay Description:In vitro binding affinity against cloned human alpha-1B-adrenoceptor receptors expressed in rat-1 fibroblastsMore data for this Ligand-Target Pair
Affinity DataIC50: <3.02E+4nMAssay Description:In vitro binding affinity against cloned human alpha-1A-adrenoceptor receptors expressed in rat-1 fibroblastsMore data for this Ligand-Target Pair
Affinity DataIC50: <3.02E+4nMAssay Description:In vitro binding affinity against cloned human alpha-1A-adrenoceptor receptors expressed in rat-1 fibroblastsMore data for this Ligand-Target Pair
Affinity DataIC50: <3.02E+4nMAssay Description:In vitro binding affinity against cloned human alpha-1B-adrenoceptor receptors expressed in rat-1 fibroblastsMore data for this Ligand-Target Pair
Affinity DataIC50: <3.02E+4nMAssay Description:In vitro binding affinity against cloned human alpha-1D-adrenoceptor receptors expressed in rat-1 fibroblastsMore data for this Ligand-Target Pair
Affinity DataEC50: <1.00E+5nMAssay Description:Activation of human Alpha-1D adrenergic receptors expressed in rat-1 fibroblastsMore data for this Ligand-Target Pair
Affinity DataEC50: 32nMAssay Description:Activation of human alpha-1A adrenergic receptor expressed in rat-1 fibroblastsMore data for this Ligand-Target Pair
Affinity DataEC50: 63nMAssay Description:Activation of human alpha-1A adrenergic receptor expressed in rat-1 fibroblastsMore data for this Ligand-Target Pair
Affinity DataEC50: 6.30nMAssay Description:Activation of human alpha-1A adrenergic receptor expressed in rat-1 fibroblastsMore data for this Ligand-Target Pair
Affinity DataEC50: 50nMAssay Description:Activation of human alpha-1A adrenergic receptor expressed in rat-1 fibroblastsMore data for this Ligand-Target Pair
Affinity DataEC50: 50nMAssay Description:Activation of human alpha-1A adrenergic receptor expressed in rat-1 fibroblastsMore data for this Ligand-Target Pair
Affinity DataEC50: 20nMAssay Description:Activation of human alpha-1A adrenergic receptor expressed in rat-1 fibroblastsMore data for this Ligand-Target Pair
Affinity DataEC50: 4nMAssay Description:Activation of human alpha-1A adrenergic receptor expressed in rat-1 fibroblastsMore data for this Ligand-Target Pair
Affinity DataEC50: 316nMAssay Description:Activation of human alpha-1B adrenergic receptors expressed in rat-1 fibroblastsMore data for this Ligand-Target Pair
Affinity DataEC50: <1.00E+5nMAssay Description:Activation of human alpha-1B adrenergic receptors expressed in rat-1 fibroblastsMore data for this Ligand-Target Pair
Affinity DataEC50: <1.00E+5nMAssay Description:Activation of human alpha-1B adrenergic receptors expressed in rat-1 fibroblastsMore data for this Ligand-Target Pair
Affinity DataEC50: <1.00E+5nMAssay Description:Activation of human alpha-1A adrenergic receptor expressed in rat-1 fibroblastsMore data for this Ligand-Target Pair
Affinity DataEC50: 13nMAssay Description:Activation of human alpha-1A adrenergic receptor expressed in rat-1 fibroblastsMore data for this Ligand-Target Pair
Affinity DataEC50: 2.00E+3nMAssay Description:Activation of human alpha-1B adrenergic receptors expressed in rat-1 fibroblastsMore data for this Ligand-Target Pair
Affinity DataEC50: <1.00E+5nMAssay Description:Activation of human Alpha-1D adrenergic receptors expressed in rat-1 fibroblastsMore data for this Ligand-Target Pair
Affinity DataEC50: 126nMAssay Description:Activation of human alpha-1A adrenergic receptor expressed in rat-1 fibroblastsMore data for this Ligand-Target Pair
Affinity DataEC50: <5.01E+3nMAssay Description:Activation of human Alpha-1D adrenergic receptors expressed in rat-1 fibroblastsMore data for this Ligand-Target Pair
Affinity DataEC50: 13nMAssay Description:Activation of human alpha-1A adrenergic receptor expressed in rat-1 fibroblastsMore data for this Ligand-Target Pair
Affinity DataEC50: <5.01E+3nMAssay Description:Activation of human alpha-1B adrenergic receptors expressed in rat-1 fibroblastsMore data for this Ligand-Target Pair
Affinity DataEC50: <1.00E+5nMAssay Description:Activation of human alpha-1B adrenergic receptors expressed in rat-1 fibroblastsMore data for this Ligand-Target Pair
Affinity DataEC50: <1.00E+5nMAssay Description:Activation of human alpha-1B adrenergic receptors expressed in rat-1 fibroblastsMore data for this Ligand-Target Pair
Affinity DataEC50: <1.00E+5nMAssay Description:Activation of human Alpha-1D adrenergic receptors expressed in rat-1 fibroblastsMore data for this Ligand-Target Pair
Affinity DataEC50: 63nMAssay Description:Activation of human alpha-1B adrenergic receptors expressed in rat-1 fibroblastsMore data for this Ligand-Target Pair
Affinity DataEC50: <5.01E+3nMAssay Description:Activation of human Alpha-1D adrenergic receptors expressed in rat-1 fibroblastsMore data for this Ligand-Target Pair
