Compile Data Set for Download or QSAR
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Found 81 Enz. Inhib. hit(s) with all data for entry = 50042186
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50421641(CHEMBL277375)
Affinity DataIC50:  25nMAssay Description:Inhibitory concentration against radioligand binding to human Alpha-1A adrenergic receptor, expressed in rat 1 fibroblast cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1D adrenergic receptor(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50421641(CHEMBL277375)
Affinity DataIC50:  40nMAssay Description:Inhibitory concentration against radioligand binding to human aAlpha-1D adrenergic receptor, expressed in rat 1 fibroblast cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1B adrenergic receptor(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50421641(CHEMBL277375)
Affinity DataIC50:  158nMAssay Description:Inhibitory concentration against radioligand binding to human Alpha-1B adrenergic receptor, expressed in rat 1 fibroblast cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50421640(CHEMBL17851)
Affinity DataIC50:  200nMAssay Description:Inhibitory concentration against radioligand binding to human Alpha-1A adrenergic receptor, expressed in rat 1 fibroblast cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1B adrenergic receptor(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50421640(CHEMBL17851)
Affinity DataIC50:  398nMAssay Description:Inhibitory concentration against radioligand binding to human Alpha-1B adrenergic receptor, expressed in rat 1 fibroblast cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1D adrenergic receptor(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50421640(CHEMBL17851)
Affinity DataIC50:  501nMAssay Description:Inhibitory concentration against radioligand binding to human Alpha-1D adrenergic receptor, expressed in rat 1 fibroblast cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50222903(CHEMBL17776)
Affinity DataEC50:  13nMAssay Description:Agonism of human alpha-1A adrenergic receptor expressed in rat 1 fibroblast cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1D adrenergic receptor(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50421641(CHEMBL277375)
Affinity DataEC50:  20nMAssay Description:Agonism of recombinant human alpha-1D adrenergic receptor, expressed in rat 1 fibroblast cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1B adrenergic receptor(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50222924(CHEMBL17819)
Affinity DataEC50: <5.01E+3nMAssay Description:Agonism of human alpha-1B adrenergic receptor, expressed in rat 1 fibroblast cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1B adrenergic receptor(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50222925(CHEMBL18303)
Affinity DataEC50: <1.00E+5nMAssay Description:Agonism of human alpha-1B adrenergic receptor, expressed in rat 1 fibroblast cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1D adrenergic receptor(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50222909(CHEMBL276733)
Affinity DataEC50: <1.00E+5nMAssay Description:Agonism of recombinant human alpha-1D adrenergic receptor, expressed in rat 1 fibroblast cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1D adrenergic receptor(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50222910(CHEMBL17491)
Affinity DataEC50:  4nMAssay Description:Agonism of recombinant human alpha-1D adrenergic receptor, expressed in rat 1 fibroblast cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1B adrenergic receptor(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50222933(CHEMBL275386)
Affinity DataEC50: <1.00E+5nMAssay Description:Agonism of human alpha-1B adrenergic receptor, expressed in rat 1 fibroblast cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1B adrenergic receptor(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50222929(CHEMBL275902)
Affinity DataEC50: <1.00E+5nMAssay Description:Agonism of human alpha-1B adrenergic receptor, expressed in rat 1 fibroblast cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1B adrenergic receptor(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50222932(CHEMBL18256)
Affinity DataEC50:  40nMAssay Description:Agonism of human alpha-1B adrenergic receptor, expressed in rat 1 fibroblast cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1B adrenergic receptor(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50222931(CHEMBL441412)
Affinity DataEC50: <1.00E+5nMAssay Description:Agonism of human alpha-1B adrenergic receptor, expressed in rat 1 fibroblast cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50219153(CHEMBL414185)
Affinity DataEC50:  0.794nMAssay Description:Effective concentration showing agonistic activity towards Human alpha-1A adrenergic receptor, expressed in rat 1 fibroblast cells was determinedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50222924(CHEMBL17819)
Affinity DataEC50:  1.00E+3nMAssay Description:Agonism of human alpha-1A adrenergic receptor expressed in rat 1 fibroblast cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50222925(CHEMBL18303)
Affinity DataEC50: <1.00E+5nMAssay Description:Agonism of human alpha-1A adrenergic receptor expressed in rat 1 fibroblast cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50222926(CHEMBL17764)
Affinity DataEC50:  79nMAssay Description:Agonism of human alpha-1A adrenergic receptor expressed in rat 1 fibroblast cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50222929(CHEMBL275902)
Affinity DataEC50:  2.5nMAssay Description:Agonism of human alpha-1A adrenergic receptor expressed in rat 1 fibroblast cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50222931(CHEMBL441412)
Affinity DataEC50:  50nMAssay Description:Agonism of human alpha-1A adrenergic receptor expressed in rat 1 fibroblast cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50222932(CHEMBL18256)
Affinity DataEC50:  6.30nMAssay Description:Agonism of human alpha-1A adrenergic receptor expressed in rat 1 fibroblast cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50222933(CHEMBL275386)
Affinity DataEC50:  251nMAssay Description:Agonism of human alpha-1A adrenergic receptor expressed in rat 1 fibroblast cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1D adrenergic receptor(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50222911(CHEMBL18436)
Affinity DataEC50:  398nMAssay Description:Agonism of recombinant human alpha-1D adrenergic receptor, expressed in rat 1 fibroblast cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1B adrenergic receptor(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50421640(CHEMBL17851)
Affinity DataEC50: <1.00E+5nMAssay Description:Agonism of human alpha-1B adrenergic receptor, expressed in rat 1 fibroblast cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50421640(CHEMBL17851)
Affinity DataEC50:  10nMAssay Description:Inhibition of T-cell proliferation was determined by a human T-cell assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1D adrenergic receptor(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50421640(CHEMBL17851)
Affinity DataEC50: <1.00E+5nMAssay Description:Inhibition of T-cell proliferation was determined by a human T-cell assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1B adrenergic receptor(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50219153(CHEMBL414185)
Affinity DataEC50:  0.398nMAssay Description:Inhibition of DiTc binding to Kv1.3 channel in human brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1D adrenergic receptor(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50222931(CHEMBL441412)
Affinity DataEC50: <1.00E+5nMAssay Description:Inhibition of T-cell proliferation was determined by a human T-cell assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1B adrenergic receptor(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50222911(CHEMBL18436)
Affinity DataEC50:  200nMAssay Description:Agonism of human alpha-1B adrenergic receptor, expressed in rat 1 fibroblast cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1D adrenergic receptor(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50222932(CHEMBL18256)
Affinity DataEC50:  200nMAssay Description:Agonism of recombinant human alpha-1D adrenergic receptor, expressed in rat 1 fibroblast cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1D adrenergic receptor(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50222933(CHEMBL275386)
Affinity DataEC50: <1.00E+5nMAssay Description:Agonism of recombinant human alpha-1D adrenergic receptor, expressed in rat 1 fibroblast cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1D adrenergic receptor(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50222929(CHEMBL275902)
Affinity DataEC50: <1.00E+5nMAssay Description:Agonism of recombinant human alpha-1D adrenergic receptor, expressed in rat 1 fibroblast cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1B adrenergic receptor(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50421641(CHEMBL277375)
Affinity DataEC50:  5nMAssay Description:Agonism of human alpha-1B adrenergic receptor, expressed in rat 1 fibroblast cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50222935(CHEMBL275844)
Affinity DataEC50:  1.30nMAssay Description:Agonism of human alpha-1A adrenergic receptor expressed in rat 1 fibroblast cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50222934(CHEMBL17492)
Affinity DataEC50:  20nMAssay Description:Agonism of human alpha-1A adrenergic receptor expressed in rat 1 fibroblast cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50222911(CHEMBL18436)
Affinity DataEC50:  200nMAssay Description:Agonism of human alpha-1A adrenergic receptor expressed in rat 1 fibroblast cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50222927(CHEMBL17657)
Affinity DataEC50:  794nMAssay Description:Agonism of human alpha-1A adrenergic receptor expressed in rat 1 fibroblast cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50222923(CHEMBL17221)
Affinity DataEC50:  63nMAssay Description:Agonism of human alpha-1A adrenergic receptor expressed in rat 1 fibroblast cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50222930(CHEMBL17151)
Affinity DataEC50:  6.30nMAssay Description:Agonism of human alpha-1A adrenergic receptor expressed in rat 1 fibroblast cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50222928(CHEMBL273312)
Affinity DataEC50:  398nMAssay Description:Agonism of human alpha-1A adrenergic receptor expressed in rat 1 fibroblast cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1D adrenergic receptor(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50222930(CHEMBL17151)
Affinity DataEC50:  3.16E+3nMAssay Description:Agonism of recombinant human alpha-1D adrenergic receptor, expressed in rat 1 fibroblast cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1B adrenergic receptor(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50222910(CHEMBL17491)
Affinity DataEC50:  5nMAssay Description:Agonism of human alpha-1B adrenergic receptor, expressed in rat 1 fibroblast cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1D adrenergic receptor(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50222924(CHEMBL17819)
Affinity DataEC50: <5.01E+3nMAssay Description:Agonism of recombinant human alpha-1D adrenergic receptor, expressed in rat 1 fibroblast cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1B adrenergic receptor(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50222909(CHEMBL276733)
Affinity DataEC50: <1.00E+5nMAssay Description:Agonism of human alpha-1B adrenergic receptor, expressed in rat 1 fibroblast cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1D adrenergic receptor(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50222925(CHEMBL18303)
Affinity DataEC50: <1.00E+5nMAssay Description:Agonism of recombinant human alpha-1D adrenergic receptor, expressed in rat 1 fibroblast cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1D adrenergic receptor(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50222926(CHEMBL17764)
Affinity DataEC50: <1.00E+5nMAssay Description:Agonism of recombinant human alpha-1D adrenergic receptor, expressed in rat 1 fibroblast cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1B adrenergic receptor(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50222926(CHEMBL17764)
Affinity DataEC50: <1.00E+5nMAssay Description:Agonism of human alpha-1B adrenergic receptor, expressed in rat 1 fibroblast cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1D adrenergic receptor(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50222935(CHEMBL275844)
Affinity DataEC50:  20nMAssay Description:Agonism of recombinant human alpha-1D adrenergic receptor, expressed in rat 1 fibroblast cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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