Compile Data Set for Download or QSAR
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Found 15 Enz. Inhib. hit(s) with all data for entry = 50048891
TargetAlpha-2A/Alpha-2B/Alpha-2C adrenergic receptor(Homo sapiens (Human))
Ohio State University

Curated by ChEMBL
LigandPNGBDBM50001922(2-Naphthalen-1-ylmethyl-4,5-dihydro-1H-imidazole; ...)
Affinity DataIC50:  0.00110nMAssay Description:Compound was evaluated for Adrenergic activity against Alpha-2 adrenergic receptor in human plateletsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetAlpha-2A/Alpha-2B/Alpha-2C adrenergic receptor(Homo sapiens (Human))
Ohio State University

Curated by ChEMBL
LigandPNGBDBM50230389(CHEMBL541105)
Affinity DataIC50:  0.00340nMAssay Description:Compound was tested for Adrenergic activity against Alpha-2 adrenergic receptor from rat aortaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-2A/Alpha-2B/Alpha-2C adrenergic receptor(Homo sapiens (Human))
Ohio State University

Curated by ChEMBL
LigandPNGBDBM50230393(CHEMBL553231)
Affinity DataIC50:  0.0140nMAssay Description:Compound was evaluated for Adrenergic activity against Alpha-2 adrenergic receptor in human plateletsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-2A/Alpha-2B/Alpha-2C adrenergic receptor(Homo sapiens (Human))
Ohio State University

Curated by ChEMBL
LigandPNGBDBM50230395(CHEMBL557985)
Affinity DataIC50:  0.0160nMAssay Description:Compound was evaluated for Adrenergic activity against Alpha-2 adrenergic receptor in human plateletsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-2A/Alpha-2B/Alpha-2C adrenergic receptor(Homo sapiens (Human))
Ohio State University

Curated by ChEMBL
LigandPNGBDBM50230388(CHEMBL537830)
Affinity DataIC50:  0.0340nMAssay Description:Compound was evaluated for Adrenergic activity against Alpha-2 adrenergic receptor in human plateletsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-2A/Alpha-2B/Alpha-2C adrenergic receptor(Homo sapiens (Human))
Ohio State University

Curated by ChEMBL
LigandPNGBDBM50230394(CHEMBL538801)
Affinity DataIC50:  0.120nMAssay Description:Compound was evaluated for Adrenergic activity against Alpha-2 adrenergic receptor in human plateletsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-2A/Alpha-2B/Alpha-2C adrenergic receptor(Homo sapiens (Human))
Ohio State University

Curated by ChEMBL
LigandPNGBDBM50230392(CHEMBL554581)
Affinity DataIC50:  0.260nMAssay Description:Compound was evaluated for Adrenergic activity against Alpha-2 adrenergic receptor in human plateletsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-2A/Alpha-2B/Alpha-2C adrenergic receptor(Homo sapiens (Human))
Ohio State University

Curated by ChEMBL
LigandPNGBDBM50230391(CHEMBL164540)
Affinity DataIC50:  0.610nMAssay Description:Compound was evaluated for Adrenergic activity against Alpha-2 adrenergic receptor in human plateletsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-2A/Alpha-2B/Alpha-2C adrenergic receptor(Homo sapiens (Human))
Ohio State University

Curated by ChEMBL
LigandPNGBDBM50230390(CHEBI:48556 | MEDETOMIDINE HYDROCHLORIDE | MPV-785...)
Affinity DataIC50:  3.30E+3nMAssay Description:Compound was evaluated for Adrenergic activity in Alpha-2 adrenergic receptor of human plateletsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
Ohio State University

Curated by ChEMBL
LigandPNGBDBM50001922(2-Naphthalen-1-ylmethyl-4,5-dihydro-1H-imidazole; ...)
Affinity DataEC50:  12nMAssay Description:Compound was evaluated for Adrenergic activity against Alpha-1 adrenergic receptor from rat aortaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
Ohio State University

Curated by ChEMBL
LigandPNGBDBM50230389(CHEMBL541105)
Affinity DataEC50:  200nMAssay Description:Compound was evaluated for Adrenergic activity against Alpha-1 adrenergic receptor from rat aortaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
Ohio State University

Curated by ChEMBL
LigandPNGBDBM50230392(CHEMBL554581)
Affinity DataEC50:  0.00770nMAssay Description:Compound was evaluated for Adrenergic activity against Alpha-1 adrenergic receptor from rat aortaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
Ohio State University

Curated by ChEMBL
LigandPNGBDBM50230393(CHEMBL553231)
Affinity DataEC50:  0.000540nMAssay Description:Compound was evaluated for Adrenergic activity against Alpha-1 adrenergic receptor from rat aortaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
Ohio State University

Curated by ChEMBL
LigandPNGBDBM50230390(CHEBI:48556 | MEDETOMIDINE HYDROCHLORIDE | MPV-785...)
Affinity DataEC50:  310nMAssay Description:Compound was evaluated for Adrenergic activity against Alpha-1 adrenergic receptor from rat aortaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
Ohio State University

Curated by ChEMBL
LigandPNGBDBM50230388(CHEMBL537830)
Affinity DataEC50:  200nMAssay Description:Compound was evaluated for Adrenergic activity against Alpha-1 adrenergic receptor from rat aortaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed