Found 84 Enz. Inhib. hit(s) with all data for entry = 50005934 
Affinity DataKi: 0.0750nMAssay Description:The binding affinity of the compound was measured on histamine H1 receptor using [3H]- mepyramine as radioligand.More data for this Ligand-Target Pair
Affinity DataKi: 0.190nMAssay Description:The binding affinity was measured on 5-hydroxytryptamine 3 receptor using [3H]GR-65630 as radioligand.More data for this Ligand-Target Pair
Affinity DataKi: 0.190nMAssay Description:The binding affinity of the compound was measured on alpha2-adrenergic receptor using [3H]- clonidine as radioligand.More data for this Ligand-Target Pair
Affinity DataKi: 0.230nMAssay Description:Displacement of [3H]GR-65630 binding to 5-hydroxytryptamine 3 receptor in rat brain cortical membranesMore data for this Ligand-Target Pair
Affinity DataKi: 0.25nMAssay Description:Displacement of [3H]- GR-65,630 binding to 5-hydroxytryptamine 3 receptor in rat brain cortical membranesMore data for this Ligand-Target Pair
Affinity DataKi: 0.280nMAssay Description:The binding affinity of the compound was measured on glycine receptor using [3H]- strychnine as radioligand.More data for this Ligand-Target Pair
Affinity DataKi: 0.330nMAssay Description:The binding affinity of the compound was measured on muscarine M1 receptor using [3H]- pirenzepine as radioligand.More data for this Ligand-Target Pair
Affinity DataKi: 0.640nMAssay Description:The binding affinity of the compound was measured on dopamine receptor D1 using [3H]- dopamine as radioligand.More data for this Ligand-Target Pair
Affinity DataKi: 0.640nMAssay Description:The binding affinity of the compound was measured on 5-hydroxytryptamine 1C receptor using [3H]- serotonin as radioligand.More data for this Ligand-Target Pair
Affinity DataKi: 0.75nMAssay Description:Displacement of [3H]- GR-65,630 binding to 5-hydroxytryptamine 3 receptor in rat brain cortical membranesMore data for this Ligand-Target Pair
Affinity DataKi: 0.770nMAssay Description:Displacement of [3H]- GR-65,630 binding to 5-hydroxytryptamine 3 receptor in rat brain cortical membranesMore data for this Ligand-Target Pair
Affinity DataKi: 0.780nMAssay Description:Displacement of [3H]- GR-65,630 binding to 5-hydroxytryptamine 3 receptor in rat brain cortical membranesMore data for this Ligand-Target Pair
3D Structure (crystal)Affinity DataKi: 1.10nMAssay Description:The binding affinity of the compound was measured on mu-opiate receptor using [3H]- naloxone as radioligand.More data for this Ligand-Target Pair
Affinity DataKi: 1.10nMAssay Description:The binding affinity of the compound was measured on 5-hydroxytryptamine 3 receptor using [3H]- GR-65,630 as radioligand.More data for this Ligand-Target Pair
Affinity DataKi: 1.10nMAssay Description:The binding affinity of the compound was measured on kappa-opiate receptor using [3H]- EKC as radioligand.More data for this Ligand-Target Pair
Affinity DataKi: 1.30nMAssay Description:Displacement of [3H]GR-65630 binding to 5-hydroxytryptamine 3 receptor in rat brain cortical membranesMore data for this Ligand-Target Pair
Affinity DataKi: 1.60nMAssay Description:The binding affinity was measured on muscarine M2 receptor using [3H]- N-Me-SCOPOL as radioligand.More data for this Ligand-Target Pair
Affinity DataKi: 1.60nMAssay Description:The binding affinity of the compound was measured on imidazoline I2 receptor using [3H]- indazoxan as radioligand.More data for this Ligand-Target Pair
Affinity DataKi: 1.60nMAssay Description:Displacement of [3H]- GR-65,630 binding to 5-hydroxytryptamine 3 receptor in rat brain cortical membranesMore data for this Ligand-Target Pair
Affinity DataKi: 340nMAssay Description:The binding affinity of the compound was measured on delta-opiate receptor using [3H]- dadle as radioligand.More data for this Ligand-Target Pair
Affinity DataKi: 680nMAssay Description:The binding affinity of the compound was measured on sigma receptor using [3H]- (+)-3-PPP as radioligand.More data for this Ligand-Target Pair
Affinity DataKi: 680nMAssay Description:The binding affinity of the compound was measured on cholecystokinin type B receptor using [3H]- CCK-8 as radioligand.More data for this Ligand-Target Pair
Affinity DataKi: 910nMAssay Description:The binding affinity was measured on muscarine M1 receptor using [3H]- pirenzepine as radioligand.More data for this Ligand-Target Pair
Affinity DataKi: 960nMAssay Description:Displacement of [3H]- GR-65,630 binding to 5-hydroxytryptamine 3 receptor in rat brain cortical membranesMore data for this Ligand-Target Pair
Affinity DataKi: 1.20E+3nMAssay Description:The binding affinity of the compound was measured on 5-hydroxytryptamine 4 receptor using [3H]- GR-113,808 as radioligand.More data for this Ligand-Target Pair
Affinity DataKi: 2.90E+3nMAssay Description:The binding affinity of the compound was measured on mu-opiate receptor using [3H]- naloxone as radioligand.More data for this Ligand-Target Pair
Affinity DataKi: 3.70E+3nMAssay Description:The binding affinity of the compound was measured on 5-hydroxytryptamine 1B receptor using [3H]- serotonin as radioligand.More data for this Ligand-Target Pair
Affinity DataKi: 4.90E+3nMAssay Description:The binding affinity of the compound was measured on dopamine receptor D3 using [3H]- dopamine as radioligand.More data for this Ligand-Target Pair
Affinity DataKi: 5.00E+3nMAssay Description:The binding affinity of the compound was measured on 5-hydroxytryptamine 1C receptor using [3H]- serotonin as radioligand.More data for this Ligand-Target Pair
TargetVoltage-dependent L-type calcium channel subunit alpha-1C/alpha-1D/alpha-1S(Rattus norvegicus)
Solvay Duphar
Curated by ChEMBL
Solvay Duphar
Curated by ChEMBL
Affinity DataKi: 5.40E+3nMAssay Description:The binding affinity of the compound was measured on dopamine receptor D2 using [3H]- spiperone as radioligand.More data for this Ligand-Target Pair
Affinity DataKi: 5.60E+3nMAssay Description:The binding affinity of the compound was measured on sigma receptor using [3H]- (+)-3-PPP as radioligand.More data for this Ligand-Target Pair
Affinity DataKi: 6.50E+3nMAssay Description:Displacement of [3H]- GR-65,630 binding to 5-hydroxytryptamine 3 receptor in rat brain cortical membranesMore data for this Ligand-Target Pair
Affinity DataKi: 7.80E+3nMAssay Description:Compound was evaluated for binding affinity against 5-hydroxytryptamine 3 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 8.50E+3nMAssay Description:The binding affinity of the compound was measured on tryptamine receptor using [3H]- tryptamine as radioligand.More data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:The binding affinity of the compound was measured on imidazoline I2 receptor using [3H]- indazoxan as radioligand.More data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:The binding affinity of the compound was measured on dopamine receptor D1 using [3H]- dopamine as radioligand.More data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:The binding affinity of the compound was measured on dopamine receptor D2 using [3H]- spiperone as radioligand.More data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:The binding affinity of the compound was measured on histamine H1 receptor using [3H]- mepyramine as radioligand.More data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:The binding affinity of the compound was measured on glycine receptor using [3H]- strychnine as radioligand.More data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:The binding affinity of the compound was measured on delta-opiate receptor using [3H]- dadle as radioligand.More data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:The binding affinity of the compound was measured on tryptamine receptor using [3H]- tryptamine as radioligand.More data for this Ligand-Target Pair
Affinity DataKi: 1.00E+4nMAssay Description:The binding affinity of the compound was measured on muscarine M1 receptor using [3H]- pirenzepine as radioligand.More data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:The binding affinity of the compound was measured on kappa-opiate receptor using [3H]- EKC as radioligand.More data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:The binding affinity of the compound was measured on cholecystokinin type A receptor using [3H]- CCK-8 as radioligand.More data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:The binding affinity of the compound was measured on muscarine M3 receptor using [3H]- N-Me-SCOPOL as radioligand.More data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:The binding affinity of the compound was measured on leukotriene-D4 receptor using [3H]- LTD4 as radioligand.More data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:The binding affinity of the compound was measured on alpha2-adrenergic receptor using [3H]- clonidine as radioligand.More data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:The binding affinity of the compound was measured on NMDA receptor using [3H]- CGS-19,755 as radioligand.More data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:The binding affinity of the compound was measured on 5-hydroxytryptamine 1A receptor using [3H]- 8-OH-DPAT as radioligand.More data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:The binding affinity of the compound was measured on TRH receptor using [3H]- MeTRH as radioligand.More data for this Ligand-Target Pair
