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Found 33 Enz. Inhib. hit(s) with all data for entry = 50034151
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
University Of Lisbon

Curated by ChEMBL
LigandPNGBDBM50357943(CHEMBL1916768)
Affinity DataKi:  621nMAssay Description:Mixed-type inhibition of Electrophorus electricus AChE assessed as hydrolysis of acetylthiocholine by Lineweaver-Burk plot analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Equus caballus (Horse))
University Of Lisbon

Curated by ChEMBL
LigandPNGBDBM8961(1,2,3,4-tetrahydro-9-acridinamine | 1,2,3,4-tetrah...)
Affinity DataIC50:  5.20nMAssay Description:Inhibition of equine serum BuChE using butylthiocholine iodide as substrate preincubated for 10 mins before substrate addition by Ellman's methodMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
University Of Lisbon

Curated by ChEMBL
LigandPNGBDBM8961(1,2,3,4-tetrahydro-9-acridinamine | 1,2,3,4-tetrah...)
Affinity DataIC50:  27nMAssay Description:Inhibition of Electrophorus electricus AChE using acetylthiocholine iodide as substrate preincubated for 10 mins before substrate addition by Ellman'...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Equus caballus (Horse))
University Of Lisbon

Curated by ChEMBL
LigandPNGBDBM50357943(CHEMBL1916768)
Affinity DataIC50:  74nMAssay Description:Inhibition of equine serum BuChE using butylthiocholine iodide as substrate preincubated for 10 mins before substrate addition by Ellman's methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
University Of Lisbon

Curated by ChEMBL
LigandPNGBDBM50357943(CHEMBL1916768)
Affinity DataIC50:  610nMAssay Description:Inhibition of Electrophorus electricus AChE using acetylthiocholine iodide as substrate preincubated for 10 mins before substrate addition by Ellman'...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Equus caballus (Horse))
University Of Lisbon

Curated by ChEMBL
LigandPNGBDBM50357944(CHEMBL1916769)
Affinity DataIC50:  1.10E+3nMAssay Description:Inhibition of equine serum BuChE using butylthiocholine iodide as substrate preincubated for 10 mins before substrate addition by Ellman's method in ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Equus caballus (Horse))
University Of Lisbon

Curated by ChEMBL
LigandPNGBDBM50357945(CHEMBL1916770)
Affinity DataIC50:  2.90E+3nMAssay Description:Inhibition of equine serum BuChE using butylthiocholine iodide as substrate preincubated for 10 mins before substrate addition by Ellman's methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Equus caballus (Horse))
University Of Lisbon

Curated by ChEMBL
LigandPNGBDBM50357941(CHEMBL1916766)
Affinity DataIC50:  3.60E+3nMAssay Description:Inhibition of equine serum BuChE using butylthiocholine iodide as substrate preincubated for 10 mins before substrate addition by Ellman's methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Homo sapiens (Human))
University Of Lisbon

Curated by ChEMBL
LigandPNGBDBM50357941(CHEMBL1916766)
Affinity DataIC50:  3.78E+3nMAssay Description:Inhibition of human serum BuChE using butyrylthiocholine as substrate by Ellman's assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Equus caballus (Horse))
University Of Lisbon

Curated by ChEMBL
LigandPNGBDBM50357942(CHEMBL1916767)
Affinity DataIC50:  6.00E+3nMAssay Description:Inhibition of equine serum BuChE using butylthiocholine iodide as substrate preincubated for 10 mins before substrate addition by Ellman's methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Homo sapiens (Human))
University Of Lisbon

Curated by ChEMBL
LigandPNGBDBM50357943(CHEMBL1916768)
Affinity DataIC50:  8.57E+3nMAssay Description:Inhibition of human serum BuChE using butyrylthiocholine as substrate by Ellman's assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Equus caballus (Horse))
University Of Lisbon

Curated by ChEMBL
LigandPNGBDBM50357946(CHEMBL1916926)
Affinity DataIC50:  1.30E+4nMAssay Description:Inhibition of equine serum BuChE using butylthiocholine iodide as substrate preincubated for 10 mins before substrate addition by Ellman's method in ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Equus caballus (Horse))
University Of Lisbon

Curated by ChEMBL
LigandPNGBDBM50357950(CHEMBL1916930)
Affinity DataIC50:  1.50E+4nMAssay Description:Inhibition of equine serum BuChE using butylthiocholine iodide as substrate preincubated for 10 mins before substrate addition by Ellman's method in ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Equus caballus (Horse))
University Of Lisbon

Curated by ChEMBL
LigandPNGBDBM50357947(CHEMBL1916927)
Affinity DataIC50:  2.30E+4nMAssay Description:Inhibition of equine serum BuChE using butylthiocholine iodide as substrate preincubated for 10 mins before substrate addition by Ellman's methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
University Of Lisbon

Curated by ChEMBL
LigandPNGBDBM50357950(CHEMBL1916930)
Affinity DataIC50:  2.40E+4nMAssay Description:Inhibition of Electrophorus electricus AChE using acetylthiocholine iodide as substrate preincubated for 10 mins before substrate addition by Ellman'...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Homo sapiens (Human))
University Of Lisbon

Curated by ChEMBL
LigandPNGBDBM50357947(CHEMBL1916927)
Affinity DataIC50:  2.61E+4nMAssay Description:Inhibition of human serum BuChE using butyrylthiocholine as substrate by Ellman's assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
University Of Lisbon

Curated by ChEMBL
LigandPNGBDBM50357946(CHEMBL1916926)
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of Electrophorus electricus AChE using acetylthiocholine iodide as substrate preincubated for 10 mins before substrate addition by Ellman'...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
University Of Lisbon

Curated by ChEMBL
LigandPNGBDBM50357944(CHEMBL1916769)
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of Electrophorus electricus AChE using acetylthiocholine iodide as substrate preincubated for 10 mins before substrate addition by Ellman'...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Equus caballus (Horse))
University Of Lisbon

Curated by ChEMBL
LigandPNGBDBM50357949(CHEMBL1916929)
Affinity DataIC50:  3.24E+4nMAssay Description:Inhibition of equine serum BuChE using butylthiocholine iodide as substrate preincubated for 10 mins before substrate addition by Ellman's method in ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Equus caballus (Horse))
University Of Lisbon

Curated by ChEMBL
LigandPNGBDBM50357948(CHEMBL1916928)
Affinity DataIC50:  4.30E+4nMAssay Description:Inhibition of equine serum BuChE using butylthiocholine iodide as substrate preincubated for 10 mins before substrate addition by Ellman's method in ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
University Of Lisbon

Curated by ChEMBL
LigandPNGBDBM50357943(CHEMBL1916768)
Affinity DataIC50:  4.55E+4nMAssay Description:Inhibition of human recombinant AChE using acetylthiocholine as substrate by Ellman's assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
University Of Lisbon

Curated by ChEMBL
LigandPNGBDBM50357949(CHEMBL1916929)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of human recombinant AChE using acetylthiocholine as substrate by Ellman's assay in presence of bovine serum albuminMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
University Of Lisbon

Curated by ChEMBL
LigandPNGBDBM50357947(CHEMBL1916927)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of human recombinant AChE using acetylthiocholine as substrate by Ellman's assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
University Of Lisbon

Curated by ChEMBL
LigandPNGBDBM50357945(CHEMBL1916770)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of human recombinant AChE using acetylthiocholine as substrate by Ellman's assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
University Of Lisbon

Curated by ChEMBL
LigandPNGBDBM50357941(CHEMBL1916766)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of human recombinant AChE using acetylthiocholine as substrate by Ellman's assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
University Of Lisbon

Curated by ChEMBL
LigandPNGBDBM50357949(CHEMBL1916929)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of Electrophorus electricus AChE using acetylthiocholine iodide as substrate preincubated for 10 mins before substrate addition by Ellman'...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
University Of Lisbon

Curated by ChEMBL
LigandPNGBDBM50357948(CHEMBL1916928)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of Electrophorus electricus AChE using acetylthiocholine iodide as substrate preincubated for 10 mins before substrate addition by Ellman'...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
University Of Lisbon

Curated by ChEMBL
LigandPNGBDBM50357947(CHEMBL1916927)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of Electrophorus electricus AChE using acetylthiocholine iodide as substrate preincubated for 10 mins before substrate addition by Ellman'...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
University Of Lisbon

Curated by ChEMBL
LigandPNGBDBM50357945(CHEMBL1916770)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of Electrophorus electricus AChE using acetylthiocholine iodide as substrate preincubated for 10 mins before substrate addition by Ellman'...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
University Of Lisbon

Curated by ChEMBL
LigandPNGBDBM50357941(CHEMBL1916766)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of Electrophorus electricus AChE using acetylthiocholine iodide as substrate preincubated for 10 mins before substrate addition by Ellman'...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
University Of Lisbon

Curated by ChEMBL
LigandPNGBDBM50357942(CHEMBL1916767)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of Electrophorus electricus AChE using acetylthiocholine iodide as substrate preincubated for 10 mins before substrate addition by Ellman'...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Homo sapiens (Human))
University Of Lisbon

Curated by ChEMBL
LigandPNGBDBM50357949(CHEMBL1916929)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of human serum BuChE using butyrylthiocholine as substrate by Ellman's assay in presence of bovine serum albuminMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Homo sapiens (Human))
University Of Lisbon

Curated by ChEMBL
LigandPNGBDBM50357945(CHEMBL1916770)
Affinity DataIC50:  1.19E+5nMAssay Description:Inhibition of human serum BuChE using butyrylthiocholine as substrate by Ellman's assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed