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Found 7 Enz. Inhib. hit(s) with all data for entry = 50034357
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
The Second Military Medical University

Curated by ChEMBL
LigandPNGBDBM50361151(CHEMBL1933805)
Affinity DataIC50:  1.51E+3nMAssay Description:Inhibition of GST-tagged human DYRK1A using dephosphorylated MBP as substrate after 10 mins by Kinase-Glo plus luminescent kinase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
The Second Military Medical University

Curated by ChEMBL
LigandPNGBDBM50361149(CHEMBL1933803)
Affinity DataIC50:  6.39E+3nMAssay Description:Inhibition of GST-tagged human DYRK1A using dephosphorylated MBP as substrate after 10 mins by Kinase-Glo plus luminescent kinase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
The Second Military Medical University

Curated by ChEMBL
LigandPNGBDBM50070942((-)-Epigallocatechin gallate | (-)-Epigallocatechi...)
Affinity DataIC50:  1.34E+4nMAssay Description:Inhibition of GST-tagged human DYRK1A using dephosphorylated MBP as substrate after 10 mins by Kinase-Glo plus luminescent kinase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
The Second Military Medical University

Curated by ChEMBL
LigandPNGBDBM50361150(CHEMBL1933804)
Affinity DataIC50:  1.95E+4nMAssay Description:Inhibition of GST-tagged human DYRK1A using dephosphorylated MBP as substrate after 10 mins by Kinase-Glo plus luminescent kinase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
The Second Military Medical University

Curated by ChEMBL
LigandPNGBDBM50361152(CHEMBL1933806)
Affinity DataIC50:  2.37E+4nMAssay Description:Inhibition of GST-tagged human DYRK1A using dephosphorylated MBP as substrate after 10 mins by Kinase-Glo plus luminescent kinase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
The Second Military Medical University

Curated by ChEMBL
LigandPNGBDBM50361148(CHEMBL1933802)
Affinity DataIC50:  2.47E+4nMAssay Description:Inhibition of GST-tagged human DYRK1A using dephosphorylated MBP as substrate after 10 mins by Kinase-Glo plus luminescent kinase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
The Second Military Medical University

Curated by ChEMBL
LigandPNGBDBM50361147(CHEMBL1933801)
Affinity DataIC50:  8.81E+4nMAssay Description:Inhibition of GST-tagged human DYRK1A using dephosphorylated MBP as substrate after 10 mins by Kinase-Glo plus luminescent kinase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed