Compile Data Set for Download or QSAR
maximum 50k data
Found 21 Enz. Inhib. hit(s) with all data for entry = 50034733
TargetNeurotensin receptor type 1(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50281809((S)-2-{(2S,3S)-2-[(S)-2-{[(S)-1-((S)-6-Amino-2-ter...)
Affinity DataKi:  63nMAssay Description:Binding affinity against rat neurotensin receptor.More data for this Ligand-Target Pair
In DepthDetails Article
TargetNeurotensin receptor type 1(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50281812((S)-2-{(2S,3S)-2-[(S)-2-{[(S)-1-((S)-5-Amino-2-ter...)
Affinity DataKi:  82nMAssay Description:Binding affinity against rat neurotensin receptor.More data for this Ligand-Target Pair
In DepthDetails Article
TargetNeurotensin receptor type 1(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50366303(CHEMBL1790460)
Affinity DataKi:  100nMAssay Description:Binding affinity against rat neurotensin receptor.More data for this Ligand-Target Pair
In DepthDetails Article
TargetNeurotensin receptor type 1(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50281811((S)-2-{(2S,3S)-2-[(S)-2-[((S)-1-{(S)-2-[(Adamantan...)
Affinity DataKi:  120nMAssay Description:Binding affinity against rat neurotensin receptor.More data for this Ligand-Target Pair
In DepthDetails Article
TargetNeurotensin receptor type 1(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50366296(CHEMBL1790463)
Affinity DataKi:  180nMAssay Description:Binding affinity against rat neurotensin receptor.More data for this Ligand-Target Pair
In DepthDetails Article
TargetNeurotensin receptor type 1(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50366308(CHEMBL1790472)
Affinity DataKi:  190nMAssay Description:Binding affinity against rat neurotensin receptor.More data for this Ligand-Target Pair
In DepthDetails Article
TargetNeurotensin receptor type 1(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50366299(CHEMBL1790467)
Affinity DataKi:  220nMAssay Description:Binding affinity against rat neurotensin receptor.More data for this Ligand-Target Pair
In DepthDetails Article
TargetNeurotensin receptor type 1(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50366307(CHEMBL1790457)
Affinity DataKi:  290nMAssay Description:Binding affinity against rat neurotensin receptor.More data for this Ligand-Target Pair
In DepthDetails Article
TargetNeurotensin receptor type 1(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50366298(CHEMBL1790466)
Affinity DataKi:  420nMAssay Description:Binding affinity against rat neurotensin receptor.More data for this Ligand-Target Pair
In DepthDetails Article
TargetNeurotensin receptor type 1(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50366311(CHEMBL1790470)
Affinity DataKi:  520nMAssay Description:Binding affinity against rat neurotensin receptor.More data for this Ligand-Target Pair
In DepthDetails Article
TargetNeurotensin receptor type 1(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50366302(CHEMBL2369587)
Affinity DataKi:  540nMAssay Description:Binding affinity against rat neurotensin receptor.More data for this Ligand-Target Pair
In DepthDetails Article
TargetNeurotensin receptor type 1(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50366310(CHEMBL1790461)
Affinity DataKi:  680nMAssay Description:Binding affinity against rat neurotensin receptor.More data for this Ligand-Target Pair
In DepthDetails Article
TargetNeurotensin receptor type 1(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50281807((S)-2-{(2S,3S)-2-[(S)-2-{[(S)-1-((S)-2,6-Diamino-h...)
Affinity DataKi:  690nMAssay Description:Binding affinity against rat neurotensin receptor.More data for this Ligand-Target Pair
In DepthDetails Article
TargetNeurotensin receptor type 1(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50366300(CHEMBL1790465)
Affinity DataKi:  880nMAssay Description:Binding affinity against rat neurotensin receptor.More data for this Ligand-Target Pair
In DepthDetails Article
TargetNeurotensin receptor type 1(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50366304(CHEMBL2369588)
Affinity DataKi:  1.00E+3nMAssay Description:Binding affinity against rat neurotensin receptor.More data for this Ligand-Target Pair
In DepthDetails Article
TargetNeurotensin receptor type 1(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50366301(CHEMBL1790469)
Affinity DataKi:  2.10E+3nMAssay Description:Binding affinity against rat neurotensin receptor.More data for this Ligand-Target Pair
In DepthDetails Article
TargetNeurotensin receptor type 1(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50366306(CHEMBL1790473)
Affinity DataKi:  2.10E+3nMAssay Description:Binding affinity against rat neurotensin receptor.More data for this Ligand-Target Pair
In DepthDetails Article
TargetNeurotensin receptor type 1(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50366312(CHEMBL1790476)
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity against rat neurotensin receptor.More data for this Ligand-Target Pair
In DepthDetails Article
TargetMu-type opioid receptor(GUINEA PIG)
TBA

Curated by ChEMBL
LigandPNGBDBM50281811((S)-2-{(2S,3S)-2-[(S)-2-[((S)-1-{(S)-2-[(Adamantan...)
Affinity DataKi: >1.00E+4nMAssay Description:Compound was evaluated for binding affinity against mu receptor by opioid receptor binding assay: InactiveMore data for this Ligand-Target Pair
In DepthDetails Article
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
TBA

Curated by ChEMBL
LigandPNGBDBM50281811((S)-2-{(2S,3S)-2-[(S)-2-[((S)-1-{(S)-2-[(Adamantan...)
Affinity DataKi: >1.00E+4nMAssay Description:Compound was evaluated for binding affinity against Opioid receptor kappa 1 by opioid receptor binding assay: InactiveMore data for this Ligand-Target Pair
In DepthDetails Article
TargetDelta-type opioid receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50281811((S)-2-{(2S,3S)-2-[(S)-2-[((S)-1-{(S)-2-[(Adamantan...)
Affinity DataKi: >1.00E+5nMAssay Description:Compound was evaluated for binding affinity against Opioid receptor delta 1 binding assay: InactiveMore data for this Ligand-Target Pair
In DepthDetails Article